Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
01/2008
01/03/2008CA2658362A1 Metalloprotease inhibitors
01/03/2008CA2655444A1 New compounds 385
01/03/2008CA2655441A1 New compounds 384
01/03/2008CA2654915A1 Tetrazole-substituted arylamides
01/03/2008CA2647601A1 Pyrrole derivatives and their methods of use
01/02/2008EP1871769A2 Process for the preparation of 4-(6-chloro-2,3-methylenedioxyanilino)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-tetrahydropyran-4-yloxyquinazoline,their intermediates and crystalline salts thereof
01/02/2008EP1871766A1 Antifungal triazole derivatives
01/02/2008EP1871762A2 Subtituted heteroaryl cb1 antagonists
01/02/2008EP1871758A1 Aminoalkyl-amidomethyl-substituted 2- (4-sulphonylamino) -3-hydroxy-3 , 4-dihydro-2h-cromen-6-yl derivatives and their use as potassium channel blockers
01/02/2008EP1871749A1 1h-quinaz0line-2,4-diones and their use as ampa-receptor ligands
01/02/2008EP1871741A2 Substituted azetidinones
01/02/2008EP1871374A2 2,3 substituted pyrazine sulfonamides as inhibitors of crth2
01/02/2008EP1416933B1 Substituted piperidines as modulators of the melanocortin receptor
01/02/2008EP1414797B1 Hepatitis c virus polymerase inhibitors with a heterobicylic structure
01/02/2008EP1414441B1 Hepatitis c virus polymerase inhibitors with heterobicyclic structure
01/02/2008EP1335915B1 Tetrahydrobenzazepine derivatives useful as modulators of dopamine d3 receptors (antipsychotic agents)
01/02/2008EP1282605B1 Thioimidazolidine derivatives as light stabilisers for polymers
01/02/2008CN101099286A Method and installation means for installing an electrical machine
01/02/2008CN101098865A 1h-indole-3-carboxylic acid derivatives and their use as PPAR agonists
01/02/2008CN101098858A 吲唑磺酰胺衍生物 Indazole sulfonamide derivative
01/02/2008CN100358875C Fluoro-contained 1H-1,2,3-triazaazole compounds, preparation method thereof and their use
01/02/2008CN100358870C Aminotetralin derivatives as muscarinic receptor antagonists
01/01/2008USRE39991 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/01/2008US7314938 Immune and/or inflammatory disorders; autoimmune disorders; disorders mediated by the CD11/CD18 family of cellular adhesion molecules (e.g., LFA-1); antagonize CD11/CD18 receptors associated with leukocytes.
01/01/2008US7314937 Non-imidazole aryl alkylamines compounds as histamine H3 receptor antagonists, preparation and therapeutic uses
01/01/2008US7314885 (4-(4-(2,3-difluorophenyl)-4H-1,2,4-triazol-3-yl)-1H-pyrrol-2-yl)(2H-pyrrol-1(5H)-yl)methanone; anticarcinogenic, antiproliferative and antimetastasis agent; inhibitors of c-Met protein kinase
01/01/2008US7314884 non-insulin dependent diabetes mellitus, and impaired glucose tolerance; dipeptidyl peptidase IV (DPP-IV) inhibitors eg (2S)-1-{[(1S)-2-(5-cyano-2-methyl-indol-1-yl)-1-methyl-ethylamino]-acetyl}-pyrrolidine-2-carbonitrile
01/01/2008US7314883 (+-)-3-(1H-Indazol-5-yl)-2-{[4-(2-oxo-1,4-dihydro-2H-quinazolin-3-yl)-piperidine-1-carbonyl]-amino}-propionic acid to treat neurogenic vasodilation, neurogenic inflammaton, thermal injury, circulatory shock, flushing associated with menopause, airway inflammatory diseases
01/01/2008US7314879 N-Acylpiperazine derivatives for obesity, diabetes, and erectile dysfunction treatment; sexual disorders
01/01/2008US7314877 Benzofuran derivative
12/2007
12/27/2007WO2007149512A2 Peptide epoxyketones for pr0teas0me inhibition
12/27/2007WO2007149478A2 Pyrazine derivatives with extended conjugation and uses thereof
12/27/2007WO2007149031A1 Isoquinoline derivatives and their use as inhibitors of cytokine mediated diseases
12/27/2007WO2007148738A1 Pest control agent containing novel pyridyl-methanamine derivative or salt thereof
12/27/2007WO2007148676A1 Therapeutic or prophylactic agent for leukemia
12/27/2007WO2007148648A1 Therapeutic or prophylactic agent for multiple sclerosis
12/27/2007WO2007148185A2 Substituted 3 -amino- pyrrolidino-4 -lactams as dpp inhibitors
12/27/2007WO2007148158A1 Enantiomerically pure flavone derivatives for the treatment of poliferative disorders and processes for their preparation
12/27/2007WO2007147874A1 Pyridine and pyrazine derivatives as mnk kinase inhibitors
12/27/2007WO2007147841A1 Azolylmethyloxiranes, their use for controlling phytopathogenic fungi and compositions comprising them
12/27/2007WO2007147778A1 Azolylmethyloxiranes, their use for controlling phytopathogenic fungi and compositions comprising them
12/27/2007WO2007147769A1 Azolylmethyloxiranes, their use for controlling phytopathogenic fungi and compositions comprising them
12/27/2007WO2007147746A1 2-pyrazinecarboxamide derivatives
12/27/2007WO2007116230A8 Azetidine derivatives as g-protein coupled receptor (gpr119 ) agonists
12/27/2007WO2007047306A8 Methods of treating amyloidosis using aryl-cyclopropyl derivative aspartyl protease inhibitors
12/27/2007US20070299104 Tetrahydropyranyl Cyclopentyl 1-Substituted and 1,1-Disubstituted Tetrahydroisoquinoline Modulators of Chemokine Receptor Activity
12/27/2007US20070299092 Quinone Substituted Quinazoline and Quinoline Kinase Inhibitors
12/27/2007US20070299073 Imidazolyl derivatives
12/27/2007US20070299069 Methods for treating hepatitis C
12/27/2007US20070299068 viricides comprising (3-cyano-indol-2-yl)phenyl derivatives, used for for treating viral diseases and infections or for affecting viral internal ribosome entry site (IRES) activity
12/27/2007US20070299065 Tetrahydropyran Derivatives as Antidiabetics
12/27/2007US20070299063 N3 alkylated benzimidazole derivatives as mek inhibitors
12/27/2007US20070299060 (1R,2R,3S,4S)-5-fluoro-N4-[3- methylaminocarbonylbicyclo[2.2.1]hept-5- en-2-yl)-N2-[1-methylsulfonyl-2,3- dihydroindol-5-yl]-2,4-pyrimidinediamine, used to inhibit cellular proliferation and to treat proliferate diseases such as tumorigenic cancers
12/27/2007US20070299057 Heterocyclic piperidines as modulators of chemokine receptor activity
12/27/2007US20070299056 Benzazepine derivatives for the treatment of neurological disorders
12/27/2007US20070299039 Substituted benz-azoles and methods of their use as inhibitors of Raf kinase
12/27/2007DE102006028649A1 New 5-quinoline derivatives are topoisomerase inhibitors useful to treat bacterial infections
12/27/2007CA2657213A1 Peptide epoxyketones for proteasome inhibition
12/27/2007CA2655857A1 Pyrazine derivatives with extended conjugation and uses thereof
12/27/2007CA2655801A1 Therapeutic or prophylactic agent for leukemia
12/27/2007CA2655789A1 Enantiomerically pure flavone derivatives for the treatment of poliferative disorders and processes for their preparation
12/27/2007CA2655573A1 Therapeutic or prophylactic agent for multiple sclerosis
12/27/2007CA2654781A1 2-pyrazinecarboxamide derivatives
12/27/2007CA2654689A1 Azolylmethyloxiranes, their use for controlling phytopathogenic fungi and compositions comprising them
12/27/2007CA2654358A1 Pyridine and pyrazine derivatives as mnk kinase inhibitors
12/26/2007EP1870409A1 Benzimidazole compound
12/26/2007EP1870402A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as VLA-4 inhibitors
12/26/2007EP1870399A1 Hydroxamate derivatives useful as deacetylase inhibitors
12/26/2007EP1869040A1 Dna-pk inhibitors
12/26/2007EP1869022A1 Naphthalamide derivatives having antiproliferative activity
12/26/2007EP1869021A1 Dna-pk inhibitors
12/26/2007EP1869006A1 Pyrimidindione derivatives as prokineticin 2 receptor antagonists
12/26/2007EP1869003A1 Indazoles as glucocorticoid receptor ligands
12/26/2007EP1869000A1 Cyclopentapyridine and tetrahydroquinoline derivatives
12/26/2007EP1868997A1 Hydroxamates as histone deacetylase inhibitors and pharmaceutical formulations containing them
12/26/2007EP1556390A4 Functionalized ionic liquids, and methods of use thereof
12/26/2007EP1539708B1 Benzimidazolones and their use as cytokine inhibitors
12/26/2007EP1233769B1 Imidazole derivatives
12/26/2007EP0804428B1 Bis-sulfonamide hydroxyethylamino retroviral protease inhibitors
12/26/2007CN101094861A Agonists and antagonists of the somatostatin receptor
12/26/2007CN101094848A Organic compounds
12/26/2007CN101094846A 1-(hetero)aryl-3-amino-pyrollidine derivatives for use as mglur3 receptor antagonists
12/26/2007CN101094836A Methods for preparing indazole compounds
12/26/2007CN101092415A Compound of new benzo heterocycle categories, preparation method and application
12/26/2007CN101092414A Preparation and application of a category of 6 ¿C aryl ¿C 3 ¿C cycroamido methyl pyrone derviation
12/26/2007CN101092384A A category of compound of alpha ¿C amido - N ¿C substituent amide, its composition, and application
12/26/2007CN100357290C Pesticidal 3-(substituted phenyl)-5-(thienyl or furyl)-1,2,4-triazoles
12/26/2007CN100357289C Process for preparing 5-(4-fluorophenyl)-1-[2-((2r,4r)-4-hydroxy -6-oxo-tetrahydro-pyran-2-yl)ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide
12/26/2007CN100357278C Substituted triazole diamine derivatives as kinase inhibitors
12/26/2007CN100357277C 1,2,4-triazole derivative, method for preparing the same, and pharmaceutical composition containing the same
12/26/2007CN100357276C Quinoline and quinoxaline compounds as PDGF-R and/or LCD tyrosine kinase inhibitors
12/26/2007CN100357275C N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases
12/26/2007CN100357273C Process for the production of substituted nicotinic acid esters
12/26/2007CN100357270C D-proline derivative
12/26/2007CN100356979C Integrin expression inhibitors
12/25/2007US7312336 Ligands for the delta opiod receptor; novel compounds which possess a piperidine ring with an exocyclic double bond do not show significant convulsive effects when administered systemically
12/25/2007US7312245 controlling harmful drug resistant fungi at lower concentrations; safe for crops; rice blast
12/25/2007US7312235 Anticoagulants
12/25/2007US7312230 Carboxylic acid derivatives as IP antagonists
12/25/2007US7312227 Autoimmune diseases; Alzheimer's disease; Parkinson's disease; bone disorders; liver disorders; rheumatic disease; amythrophiic lateral sclerosis