Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
02/2000
02/17/2000WO2000007542A2 Utilization of aryl(or heteroaryl)azolylcarbinol derivatives in the preparation of a medicament for the treatment of troubles mediated by an excess of substance p
02/17/2000DE19836697A1 New substituted 4-amino-2-aryl-pyrimidines, are soluble guanylate cyclase activators useful e.g. for treating atherosclerosis, hypertension, angina pectoris, thrombosis, asthma or diabetes
02/17/2000DE19836404A1 New benzimidazolonyl-substituted 3-azabicyclo (3.2.0) heptane derivatives, useful e.g. as neuroleptics, antidepressants, hypnotics and sedatives
02/17/2000DE19836044A1 New 2-(hetero)aryl-alkanoic acid derivatives, useful as mixed endothelin receptor antagonists, e.g. for treating cardiac insufficiency, restenosis, hypertension or prostate cancer
02/17/2000DE19834325A1 New benzo-condensed heterocyclic compounds useful in treatment of thrombosis and prevention of vascular occlusion
02/17/2000CA2383623A1 3-methylidenyl-2-indolinone modulators of protein kinase
02/17/2000CA2339270A1 Triazolone derivatives, use thereof, and intermediate therefor
02/17/2000CA2338944A1 Succinoylamino lactams as inhibitors of a.beta. protein production
02/17/2000CA2338594A1 Imidazoles and related compounds as .alpha.1a agonists
02/16/2000CN1244864A 2-imidazolinylaminoindazole compounds useful as alpha-2 adrenoceptor agonists
02/16/2000CN1244798A Sulfonic acid or sulfonylamino N-(heteroaralkyl)-azaheterocyclylamide compounds
02/16/2000CN1049434C Aromatic amidine derivatives and method for preparing medicinal salts thereof
02/16/2000CN1049430C Sulfonamides and its preparing method and use thereof
02/15/2000US6025478 High reactivity and fixing capacity, good low temperature dyeing, good color intensity, lightfastness, washfastness
02/15/2000US6025374 Migraine
02/15/2000US6025355 Substituted indolinyl and derivatives thereof, neurological injury and neurodegenerative disorders.
02/15/2000CA2152792C Novel 3,4-diaryl thiophenes and analogs thereof having use as antiinflammatory agents
02/15/2000CA2109585C Isoxazole and isothiazole compounds that enhance cognitive function
02/10/2000WO2000006597A2 Endogenous constitutively activated g protein-coupled orphan receptors
02/10/2000WO2000006568A1 Substituted pyrazole derivatives
02/10/2000WO2000006564A1 Disubstituted maleimide compounds and medicinal utilization thereof
02/10/2000WO2000006563A1 Substituted imidazoles having cytokine inhibitory activity
02/10/2000WO2000006541A1 Sulfurated distamycin derivatives, process for preparing them, and their use as antitumor agents
02/10/2000WO2000006531A2 Nitric esters and nitrate salts of specific drugs
02/10/2000WO2000006169A1 Integrin receptor antagonists
02/10/2000WO1999063944A3 Novel therapeutic agents that modulate estrogen receptors
02/10/2000CA2338866A1 Disubstituted maleimide compound and pharmaceutical use thereof
02/10/2000CA2338275A1 Integrin receptor antagonists
02/09/2000EP0978515A2 1-(substituted phenyl)-4-biphenylmethyl-imidazol-2-one derivatives, their preparation and their use as angiotensin II antagonists
02/09/2000EP0978392A1 Optical recording media
02/09/2000EP0977750A1 Farnesyltransferase inhibiting quinazolinones
02/09/2000CN1049215C Pharmaceutical compounds
02/09/2000CN1049116C Process for treating cardiovascular hypertrophy and hyperplasia
02/08/2000US6022967 Heterocyclic compounds
02/08/2000US6022883 Heterocyclyloxybenzoylguanidines
02/08/2000US6022875 Use of substituted 2,4-imidazolidinedione compounds as analgesics
02/08/2000US6022870 4-(heterocycle-substituted-phenyl)-1,2,4-triazol-3-ones
02/08/2000CA2150016C Pyrrolopyrimidines as crf antagonists
02/08/2000CA2095587C Process for preparing aryl piperazinyl-hetero-cyclic compounds
02/08/2000CA2090942C Anti-tumour compounds containing quinazoline and tetrazole rings
02/08/2000CA2014467C 3-substituted-2-oxindole derivatives
02/03/2000WO2000005230A1 Pyrazole derivatives and salts thereof
02/03/2000WO2000005229A1 Phenylindole derivatives as 5-ht2a receptor ligands
02/03/2000WO2000005225A1 Biphenyl derivatives
02/03/2000WO2000005222A1 Dihydrotriazolone derivatives as pesticides
02/03/2000WO2000005217A1 Imidazole compounds and their use as adenosine deaminase inhibitors
02/03/2000WO2000005210A1 N,n-substituted cyclic amine derivatives
02/03/2000WO2000005206A1 Arylpiperazine derivatives useful as uro-selective alpha-1-adrenoceptor blockers
02/03/2000WO2000004900A1 Substituted benzimidazole antiviral agents
02/03/2000WO2000004893A2 Imidazoline receptor binding compounds
02/03/2000WO2000004892A2 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
02/03/2000WO1999063936A3 Novel therapeutic agents that modulate endothelin receptors
02/03/2000WO1999063933A3 Multivalent agonists, partial agonists and antagonists of the gaba receptors
02/03/2000WO1999058504A9 Novel 1,2,5-trisubstituted 1,2-dihydro-indazol-3-ones with anti-asthmatic, anti-allergic, anti-inflammatory, immuno-modulating and neuro-protective effect, method for the production and use thereof as a medicament
02/03/2000DE19834047A1 Substituierte Pyrazolderivate Substituted pyrazole derivatives
02/03/2000CA2338305A1 Imidazole compounds
02/03/2000CA2338279A1 Imidazoline receptor binding compounds
02/03/2000CA2338209A1 Biphenyl derivatives
02/03/2000CA2338147A1 Substituted benzimidazole antiviral agents
02/03/2000CA2337941A1 N,n-substituted cyclic amine compounds
02/03/2000CA2335062A1 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
02/03/2000CA2332589A1 Dihydrotriazolone derivatives as pesticides
02/02/2000EP0976737A1 Pyrazole derivatives, process for preparing the same, intermediates, and pest control agent containing the same as active ingredient
02/02/2000EP0976732A1 1,4-substituted cyclic amine derivatives
02/02/2000EP0975627A1 5-(2-imidazolinylamino)benzimidazole compounds useful as alpha-2 adrenoceptor agonists
02/02/2000EP0975602A1 Imidazole and imidazoline derivatives and uses thereof
02/02/2000EP0975594A1 Process for the production of indole derivatives
02/02/2000EP0975593A1 Indole derivatives having combined 5ht1a, 5ht1b and 5ht1d receptor antagonist activity
02/01/2000US6020357 Nitrogen containing heteroaromatics as factor Xa inhibitors
02/01/2000US6020354 Fungicides, bactericides
02/01/2000US6020336 Indole and indazole compounds
01/2000
01/27/2000WO2000003737A2 Water-soluble drugs and methods for their production
01/27/2000WO1999063930A3 Novel angiotensin receptor modulators and their uses
01/26/2000EP0974589A1 Benzimidazole derivatives and pharmaceutically acceptable salts thereof
01/26/2000EP0973798A1 Inhibition of major groove dna binding proteins by modified polyamides
01/26/2000EP0973788A1 Tricyclic base analogues
01/26/2000EP0973768A1 Azole compounds, their production and their use
01/26/2000EP0973767A1 Indazoles of cyclic ureas useful as hiv protease inhibitors
01/26/2000EP0973765A1 Substituted aryluracils
01/26/2000EP0973763A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same
01/26/2000EP0973753A2 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinones useful as hiv reverse transcriptase inhibitors
01/26/2000EP0973750A1 Substituted benzimidazoles and their use for treating retroviral infection
01/26/2000EP0973740A1 Design, synthesis and use of specific polyamide dna-binding ligands
01/26/2000EP0973513A1 Compositions and methods for treating bone deficit conditions
01/26/2000EP0973396A1 A method of treating cancer
01/26/2000EP0973395A1 Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them
01/26/2000CN1242767A Fungicidal cyclic amides
01/26/2000CN1242365A Azole alcohol derivatives, prepn. method and pharmaceutical use thereof
01/26/2000CN1242362A Method of purifying carbazole ester precursors of 6-chloro-alpha-methyl-carbazole-2-acetic acid
01/25/2000US6017941 Method of combatting infectious diseases using dicationic bis-benzimidazoles
01/25/2000US6017909 Salts of azelastine having improved solubility effective at treating psoriasis and providing a cytoprotective effect
01/25/2000CA2021005C Uracil derivatives and herbicides containing the same as active ingredient
01/20/2000WO2000002877A2 New pharmaceutically active compounds
01/20/2000WO2000002870A1 Antiviral macrocyclic compounds
01/20/2000WO2000002865A1 Pharmaceutical agents
01/20/2000WO2000002558A1 Use of prenyltransferase inhibitors for preparing a medicine for treating pathologies resulting from heterotrimeric g protein membrane fixation
01/20/2000WO1999055672A3 Antipsychotic indolyl derivatives
01/20/2000WO1999042092A3 Compounds and methods of use for treatment of neurogenic inflammation
01/20/2000CA2337795A1 Pharmaceutical agents
01/20/2000CA2337261A1 Use of prenyltransferase inhibitors for preparing a medicine for treating pathologies resulting from heterotrimeric g protein membrane fixation