Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
09/1999
09/30/1999WO1999048890A1 Herbicidal tetrazolinones
09/30/1999WO1999048889A1 Halimide, a cytotoxic marine natural product, and derivatives thereof
09/30/1999WO1999048888A1 Imidazolone anorectic agents: ii. phenyl derivatives
09/30/1999WO1999048887A1 Imidazolone anorectic agents: iii. heteroaryl derivatives
09/30/1999WO1999048873A1 Imidazolone anorectic agents: i. acyclic derivatives
09/30/1999WO1999048868A2 Heterocyclic classes of compounds for the modulating tyrosine protein kinase
09/30/1999WO1999037638A8 2-(2'-hydroxyphenyl) benzotriazoles containing a 2,4-imidazolidinedione group and process for their preparation
09/30/1999WO1999036410A9 Triazine antiviral compounds
09/30/1999CA2325935A1 Heterocyclic families of compounds for the modulation of tyrosine protein kinase
09/30/1999CA2325588A1 Imidazolone anorectic agents: i. acyclic derivatives
09/30/1999CA2325587A1 Imidazolone anorectic agents: ii. phenyl derivatives
09/30/1999CA2325472A1 Imidazolone anorectic agents: iii. heteroaryl derivatives
09/30/1999CA2325417A1 Halimide, a cytotoxic marine natural product, and derivatives thereof
09/29/1999EP0945447A1 Trisubstituted 1,3,5-triazine derivatives for treatment of HIV infections
09/29/1999EP0945445A1 1,5-benzodiazepine derivatives
09/29/1999EP0945438A1 Pyrazole derivatives
09/29/1999EP0945437A1 Pyrazolyl acrylic acid- and pyrazolyl oximino-acetic acid derivatives, their preparation and their use as fungicides
09/29/1999EP0944624A1 Insoluble s-triazine derivatives and their use as uv filters
09/29/1999EP0944621A1 2-imidazolinylaminoindole compounds useful as alpha-2 adrenoceptor agonists
09/29/1999EP0944620A1 2-imidazolinylaminoindazole compounds useful as alpha-2 adrenoceptor agonists
09/29/1999EP0944616A1 Bicyclic aryl carboxamides and their therapeutic use
09/29/1999EP0944606A1 4,5-diaminopyrimidine derivatives and a method for the preparation thereof
09/29/1999EP0944603A1 Process for making 2-amino-2-imidazoline, guanidine, and 2-amino-3,4,5,6-tetrahydropyrimidine derivatives
09/29/1999EP0944596A1 Seco precursors of cyclopropylindolines and their use as prodrugs
09/29/1999EP0944594A1 Inhibitors of the enzymatic activity of psa
09/29/1999EP0944590A2 Aminoguanidines and alkoxyguanidines as protease inhibitors
09/29/1999EP0944386A1 Sulfonic acid or sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
09/29/1999EP0944322A1 Quarternary ammonium salts and their use in agricultural formulations
09/29/1999EP0944314A1 Methyl substituted fungicides and arthropodicides
09/29/1999EP0778825B1 Improved process for making sulfonyl isocyanates
09/29/1999EP0553107B1 Protein kinase c modulators with anti-inflammatory and antiviral activity
09/29/1999CN1230110A Cell adhesion inhibitors
09/29/1999CN1045294C Method for prepn. of indole derivatives
09/28/1999US5959123 Reacating substituted amino acid with 3-amino-4-substituted-azetidine-2-one compound to form 3, 4-disubstituted-azetidine-2-one compound; useful for treating muscular dystrophy, arthritis, viral and parasitic infections
09/28/1999US5959120 Acetate ester compounds
09/28/1999US5959109 Compounds and methods for increasing endogenous levels of corticotropin-releasing factor
09/28/1999US5958968 Cardiovascular disorders; kidney dieases
09/28/1999US5958926 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
09/28/1999US5958918 Substituted (sulfinic acid, sulfonic acid, sulfonylamino or sulfinylamino) N- (aminominomethyl)phenylalkyl!-azaheterocyclylamide compounds
09/28/1999US5958664 Coupler capable of releasing a development accelerator
09/28/1999CA2014457C Pyrimidine derivatives
09/23/1999WO1999047518A1 Substituted bisindolymaleimides for the inhibition of cell proliferation
09/23/1999WO1999047517A1 Novel heterocyclic compounds
09/23/1999WO1999047516A1 3-(2-pyrrolidinylmethyl)-indole compounds having 5-ht6 affinity
09/23/1999CA2322742A1 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
09/22/1999EP0943616A1 Substituted imidazole derivatives and their use as cytokine inhibitors
09/22/1999EP0943008A1 Metal mediated serine protease inhibitors
09/22/1999EP0942904A1 3-thiocarbamoylpyrazole derivatives as pesticides
09/22/1999CN1229412A Inhibitors of interleukin-1'beta' converting emzyme
09/22/1999CN1229080A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229079A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229078A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/21/1999US5955611 Cyclization of diamidepyrazole to form pyrimidone of pyrazole
09/21/1999US5955501 Derived from phorboids of the diterpene- and benzolactam-classes.
09/21/1999US5955487 Treating high blood pressure, cardiac insufficiency, glaucoma
09/21/1999US5955464 4-anilinoquinazoline derivatives bearing a heteroaryl substituted at the 6-position and possessing anti-cell-proliferation properties
09/21/1999US5955463 Antitumor, antiinflammatory, and antiarthritic agents
09/21/1999US5955462 Antiinflammatory agents for neurogenic inflammation and administering bisindole or compounds
09/21/1999US5955461 Quinoxalinedione derivatives, their production and use in pharmaceutical agents
09/21/1999US5955060 Cosmetics and veterinary medicine
09/21/1999CA2192975C Benzimidazolone derivatives
09/16/1999WO1999046264A1 New compounds
09/16/1999WO1999046260A1 New compounds
09/16/1999WO1999046248A1 1,2-diazepane derivatives as interleukin-1beta converting enzyme inhibitors
09/16/1999WO1999046246A1 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
09/16/1999WO1999028304A9 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
09/15/1999EP0941086A1 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
09/15/1999EP0652752B1 Water-dispersible tablets
09/15/1999EP0637242B1 Agents for treating substance abuse disorders
09/15/1999CN1228773A Heterocyclic metalloprotease inhibitors
09/15/1999CN1228772A Heterocyclic metalloprotease inhibitors
09/15/1999CN1228770A Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties
09/15/1999CN1228767A Bidentate metalloprotease inhibitors
09/14/1999US5952497 N.sup.α -Bpoc amino acid pentafluorophenyl (Pfp) esters and 3,4-dihydro-4-oxo-1,2,3-benzotriazin-3-yl (ODhbt) esters
09/14/1999US5952362 2-imidazoline, 2-oxazoline, 2-thiazoline, and 4-imidazole derivatives of methylphenyl, methoxyphenyl, and aminophenyl alkylsulfonamides and ureas and their use
09/14/1999US5952343 HIV protease inhibitors
09/14/1999US5952331 Aryl pyrimidine derivatives
09/14/1999US5952321 Substituted azetidinones as anti-inflammatory and antidegenerative agents
09/14/1999CA2150483C Pyrazoles and pyrazolopyrimidines
09/14/1999CA2098478C Preparation of substituted isoserine esters using metal alkoxides and .beta.-lactams
09/10/1999WO1999044999A1 Optically active substituted 2,4-diamino-1,3,5-triazines as herbicides
09/10/1999WO1999044613A1 Pharmaceutical compositions containing in combination two antagonists selective of arginine-vassopressin v receptors, even of v1a and v2 receptors
09/10/1999WO1999026932A8 By amidino group substituted heterocyclic derivatives and their use as anticoagulants
09/10/1999WO1999023078A3 Novel carboxylic acid derivatives which carry amide side chains, production of said carboxylic acid derivatives and their use as endothelin receptor antagonists
09/10/1999CA2322482A1 Optically active substituted 2,4-diamino-1,3,5-triazines as herbicides
09/09/1999DE19809360A1 Optisch aktive substituierte 2,4-Diamino-1,3,5-triazine Optically active substituted 2,4-diamino-1,3,5-triazines
09/08/1999EP0939757A1 Novel integrin receptor antagonists
09/08/1999CN1228094A Palladium catalyzed indolization
09/08/1999CN1228088A Arylsulfonylimidazolone derivatives as antimumor agent
09/08/1999CN1228082A Synthesis of bisindolylmalimides
09/07/1999US5948913 Hydrate for drug use
09/07/1999US5948912 Therapy for psychological, nervous system disorders
09/07/1999US5948907 Synthesis of bisindolylmaleimides
09/07/1999US5948804 Anaesthetic premedication
09/07/1999US5948793 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling neurotransmitter release
09/07/1999US5948782 Antiinflammatory agent; rheumatic diseases
09/07/1999US5948600 Method and material for the formation of a heat mode image
09/07/1999US5948593 Optical recording medium
09/07/1999US5948487 Anisotropic retardation layers for display devices
09/07/1999CA2168563C Benzopyrans and pharmaceutical compositions containing them