Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
09/2000
09/20/2000EP1036066A1 Substituted pyrimidine and pyridine herbicides
09/20/2000EP1036065A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
09/20/2000EP0696288B1 Quinoxalindione derivatives, their preparation and their use in drugs
09/20/2000CN1267296A Barbituric acid derivs with antimetastatic and antitumor activity
09/20/2000CN1267286A 2-{3-[4-(2-t-butyl-6-trifluoromethylpyridin-4-yl) piperazin-1-yl] propylmercapto} pyrimidin-4-ol-fumarate
09/20/2000CN1056609C Benzoyl guanidines, their production and their use in medicinal compositions
09/19/2000US6121456 2-(2'Hydroxyphenyl) benzotriazoles and process for their preparation
09/19/2000US6121325 Naphthyl compounds promote release of growth hormone
09/19/2000US6121280 Azabicyclic rotomase inhibitors
09/19/2000US6121272 Bidentate metalloprotease inhibitors
09/19/2000US6121266 Pyridazines as interleukin-1β converting enzyme inhibitors
09/19/2000US6121264 Glutamate receptor antagonist, ampa receptor antagonist, nmda-glycine receptor antagonist, kainic acid neurotoxicity inhibitor, antiischemic agent, psychotropic agent
09/19/2000US6121260 Appetite stimulation with dosage of neuropeptide y (npy) receptor agonist
09/19/2000US6121258 For treatment of arthritis, cancer, cardiovascular disorders, skin disorders, ocular disorders, inflammation, gum disease
09/19/2000CA2018563C N-heteroaryl-purin-6-amines, a process for their preparation and their use as medicaments
09/15/2000CA2301679A1 Medication for treatment of functional distrubances or illnesses of the lower intestinal tract, particularly abdominal visceral pain which accompanies them
09/14/2000WO2000053596A2 Imidazole compounds as histamine h3 ligands
09/14/2000WO2000053595A1 Pyrimidine compounds
09/14/2000WO2000053582A1 HETEROCYCLIC COMPOUNDS HAVING EFFECT OF ACTIVATING NICOTINIC ACETYLCHOLINE α4β2 RECEPTOR
09/14/2000WO2000053579A2 Solid phase synthesis of 4-aminoproline derivatives and/or combinatorial libraries thereof
09/14/2000WO2000044722A8 Chondrongenesis promotors and indolin-2-one derivatives
09/14/2000WO1999063999A8 H1-histamine receptor antagonists
09/14/2000CA2366668A1 Pyrimidine compounds
09/14/2000CA2366260A1 Heterocyclic compounds having effect of activating .alpha.4.beta.2 nicotinic acetylcholine receptors
09/14/2000CA2362319A1 Imidazole compounds as histamine h3 ligands
09/13/2000EP1035114A2 Nitrogen-heterocyclic compounds and process for production thereof
09/13/2000EP1034174A1 Azaring-ether derivatives and their use as nicotinic ach receptor modulators
09/13/2000EP1034169A1 Trisaryl-1,3,5-triazine ultraviolet light absorbers
09/13/2000EP1034167A1 Alpha-alkylthio substituted pyrimidine ethers and thioethers as viral reverse transcriptase inhibitors
09/13/2000EP1034164A1 Substituted beta-alanine derivatives as cell adhesion inhibitors
09/13/2000EP1034162A1 9,10-dihydro-9,10-ethanoanthracene derivatives as phospholipase inhibitors
09/13/2000EP0607193B1 Triazole antifungal agents
09/13/2000CN1266431A Aroyl-piperazine derivatives, their preparation and their use as tachykinin antagonists
09/13/2000CN1266428A Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
09/13/2000CN1266057A Novel cyano-indole serotonin reextracted inhibitor compound, its preparation process and medicinal compositions having same
09/13/2000CN1056370C 4-aryloxy (arylthio or arylamino) pyrimidine derivative with herbicide active, and preparation process thereof
09/12/2000US6117940 Solid phase synthesis of compounds such as the imidazoles, benzodiazepines, pyrazines, and steroid mimics.
09/12/2000US6117822 Substituted phthalimidocinnamic acid derivatives and intermediates for their preparation
09/08/2000WO2000052134A2 Inhibitors of prenyl-protein transferase
09/08/2000WO2000052032A1 Heterocyclic compounds, intermediates thereof and elastase inhibitors
09/08/2000WO2000051991A1 4-AMINO-QUINAZOLINE AND QUINOLINE DERIVATIVES HAVING AN INHIBITORY EFFECT ON SIGNAL TRANsSDUCTION MEDIATED BY TYROSINE KINASES
09/08/2000WO2000051984A1 2-aryl indole derivatives as antagonists of tachykinins
09/08/2000WO2000051547A2 Inhibitors of prenyl-protein transferase
09/08/2000WO2000029404A8 Pyrimidinylbenzimidazole and triazinylbenzimidazole derivatives and agricultura/horticultural bactericides
09/08/2000WO2000012497B1 Quinazoline derivatives as medicaments
09/08/2000CA2363169A1 Inhibitors of prenyl-protein transferase
09/08/2000CA2362911A1 Heterocyclic compounds, intermediates thereof and elastase inhibitors
09/08/2000CA2362778A1 Inhibitors of prenyl-protein transferase
09/06/2000EP1032424A1 Combination of an aldose reductase inhibitor and a glycogen phosphorylase inhibitor
09/06/2000CN1265660A 2-(4-aryl or heteroaryl-piperazin-1-ylmethyl)-1H-indole derivatives
09/06/2000CN1265657A Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4
09/06/2000CN1265654A 1-(N-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of phenyl ring
09/06/2000CN1265394A Compound as intermediates for use in preparation of optically active 2-imidazoline-5-one or 2-imidazoline-5-thionone derivatives
09/06/2000CN1056144C New use of 6-heterocyclic-4-amino-3,4,5-tetrahydrobenz (CD) indoles compound
09/06/2000CN1056141C 哌嗪衍生物 Piperazine derivatives
09/06/2000CN1056140C Biphenyl derivatives, their preparation and theirt use for treatment of hypertension and cardiac disease
09/05/2000US6114532 Anticoagulant
09/05/2000US6114374 2-and 2,5-substituted phenylketoenols
09/05/2000US6114360 Pyrrole compounds
09/05/2000US6114335 Benzoylguanidine derivatives, process for their preparation their use in the preparation of medicines
09/05/2000US6114330 Substituted 2,4-diaminopyrimidines
09/05/2000CA2039399C Dual functioning excipient for metal chelate contrast agents
08/2000
08/31/2000WO2000050420A1 6-substituted-7- heteroquinoxaline carboxylic acid derivatives and addition salts thereof and processes for the preparation of both
08/31/2000WO2000050419A1 Substituted bicyclic heterocycles and the use thereof as thrombin inhibitors
08/31/2000WO2000050417A1 Anti-cancer dihydroquinazoline derivatives
08/31/2000WO2000050408A1 Pyridazin-3-one derivatives and medicines containing the same
08/31/2000WO2000050395A1 Sulfonamide-containing indole compounds
08/31/2000WO2000007996A3 Pyrazoles as estrogen receptor modulators
08/31/2000DE19908567A1 New 4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors, polyps or respiratory or gastrointestinal diseases
08/31/2000DE19907813A1 Substituierte bicyclische Heterocyclen, deren Herstellung und deren Verwendung als Arzneimittel Substituted bicyclic heterocycles, their preparation and their use as medicaments
08/31/2000CA2364749A1 6-substituted-7-heteroquinoxaline carboxylic acid derivatives and addition salts thereof and processes for the preparation of both
08/31/2000CA2364708A1 Anti-cancer dihydroquinazoline derivatives
08/30/2000EP1031571A1 Sulfamoyl compounds and agricultural or horticultural bactericide
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000EP0769010B1 2-[1',2',4'-triazol-3'-yloxymethylene]-anilides and their use as pest-control agents
08/30/2000CN1265033A Certain diarylimidaozle derivatives, new class of NPY speific ligands
08/29/2000US6110956 N-aryloxyethylamine derivatives for the treatment of depression
08/29/2000US6110940 Salts of an anti-migraine indole derivative
08/29/2000US6110939 As a substance p antagonists treating tachykinin-mediated disease, asthma, central nervous system disorder
08/29/2000US6110938 1-(arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-4-(heteroaryl)piperidines and related compounds useful as antipsychotics and analgesics
08/29/2000US6110924 Barbituric acid derivatives, processes for their production and pharmaceutical agents containing these compounds
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/29/2000CA2012628C New fluoro-4 benzoic derivatives, process for their preparation and pharmaceutical compositions containing them
08/24/2000WO2000049001A2 Phenoxy-, phenylthio-, phenylamino-, benzyloxy-, benzylthio- or benzylaminopyrimidine insectidices and acaricides
08/24/2000WO2000048597A1 Systemic use of 5-ht3 receptor antagonists against rheumatic inflammatory processes
08/24/2000WO2000031051B1 Quinoline and quinoxaline compounds as pdgf-receptor and/or lck tyrosine kinase inhibitors
08/23/2000EP1029861A1 Benzisothiazol-piperazinyl derivative and its use as neuroleptic
08/23/2000EP1029859A1 N,N'-Disubstituted unsymmetrical cyclic urea and its use in therapy
08/23/2000EP1029853A1 Heteroaromatic bicyclic derivatives useful as anticancer agents
08/23/2000EP1029851A1 Piperazine compounds and medicinal use thereof
08/23/2000EP1029541A1 Therapeutic or prophylactic agent for glomerulopathy
08/23/2000EP1028956A1 Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom
08/23/2000EP1028955A1 Pyrimidinone compounds and pharmaceutical compositions containing them
08/23/2000EP1028954A1 Substituted imidazoles useful in the treatment of inflammatory diseases
08/23/2000EP1028950A1 Novel 7-substituted quinazolin-2,4-diones useful as antibacterial agents
08/23/2000EP1028949A1 Carbamoylphenylsulfonyl ureas, method for their production and their application as herbicides and plant growth regulators
08/23/2000EP1028948A1 Phenyl-alkyl-imidazoles as h3 receptor antagonists
08/23/2000EP1028942A2 Dipeptide nitriles
08/23/2000CN1264385A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same
08/23/2000CN1264377A Substituted pyrazoles as P38 kinase inhabitors