Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
01/2000
01/19/2000EP0971901A1 Phthalazinones
01/19/2000EP0971588A1 Novel cannabinoid receptor modulators
01/19/2000EP0726899B1 Novel pyrazine carboxamide derivatives, their production and their use in medicaments
01/19/2000CN1242004A Process for making 2-amino-2-imidazoline, guanidine, and 2-amino-3,4,5,6-tetrahydropyrimidine derivatives
01/19/2000CN1242000A Farnesyl transferase inhibitors
01/19/2000CN1048490C Cyclic derivatives, pharmacecctical compositions containg the same derivatives and their use
01/19/2000CN1048486C Method for preparing benzimidazole derivatives
01/19/2000CN1048484C A process for preparing a composition containing benzoheterocycles
01/18/2000US6015825 Triazole antifungal agents
01/18/2000US6015812 N-(arylsulphonyl)amino acid derivatives having bradykinin receptor affinity
01/18/2000US6015800 Substituted quinoxaline-2-ones as glutamate receptor antagonists
01/18/2000US6015774 Pyrazin-2-one derivatives, their use, and intermediates for their production
01/18/2000CA2035314C Triazole antifungal agents
01/13/2000WO2000001704A2 Benzimidazoles, production thereof and use thereof as medicaments
01/13/2000WO2000001691A1 Process for making farnesyl-protein transferase inhibitors
01/13/2000WO2000001678A1 Process for the synthesis of substituted piperazinones via mitsunobu reaction
01/13/2000WO2000001676A1 Potassium channel blocking agents
01/13/2000WO2000001675A1 Novel benzimidazoles as corticotropin release factor antagonists
01/13/2000WO2000001389A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
01/13/2000WO2000001376A2 Pharmaceutical compositions and their uses for treatment of demyelinating disorders
01/13/2000CA2336714A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
01/13/2000CA2335779A1 Novel benzimidazoles as corticotropin release factor antagonists
01/12/2000EP0970070A1 Phthalazines with angiogenesis inhibiting activity
01/12/2000EP0970056A1 Substituted 2-anilinopyrimidines useful as protein kinase inhibitors
01/12/2000EP0969840A1 Thrombin inhibitors
01/12/2000EP0934269A4 Analogs of cc-1065 and the duocarmycins
01/12/2000CN1241188A Heterocyclylmethyl-substed pyrazol derivs.
01/12/2000CN1241187A Piperazino derivs as neurokinin antagonists
01/12/2000CN1241186A Process for crystallization of losartan
01/12/2000CN1241184A Indole derivs. for treatment of osteoporosis
01/12/2000CN1241116A Methyl substed fungicides and arthropodicides
01/12/2000CN1048159C Method for preparing pharmaceutical composition contg. imidazolyl-alkenoic acid
01/11/2000US6013808 Purifying (6-chloro-2-carbazolyl)methyl-malonic acid di(c.sub.1-c.sub.6 alkyl) ester by phase separating impurities using acetic as solvent
01/11/2000US6013797 Curing agent which crosslinks resins by decyclization without releasing volatile organic compounds; formaldehyde-free
01/11/2000US6013662 Farnesyl transferase inhibitors, their preparation, the pharmaceutical compositions which contain them and their use in the preparation of medicaments
01/11/2000CA2195027C Hiv protease inhibitors useful for the treatment of aids
01/06/2000WO2000000477A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000WO2000000473A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000CA2336625A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000CA2335921A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/05/2000EP0968207A1 Cycloimido-substituted benzofused heterocyclic herbicides
01/05/2000EP0968206A1 N-heterocyclic derivatives as nos inhibitors
01/05/2000EP0968186A1 Improved polyamides for binding in the minor groove of double stranded dna
01/05/2000EP0539420B1 substituted thiazolyl and substituted pyridinyl derivatives
01/05/2000DE19829964A1 New benzimidazolyl amidine or nitrile compounds, used as thrombin inhibitors, antithrombotic agents or intermediates
01/05/2000CN1240446A Insoluble s-triazine derivatives and their use as UV filters
01/05/2000CN1240442A Heterocyclyl uracils
01/05/2000CN1240426A Novel tetrahydrobenzindolone derivatives
01/04/2000US6011150 Synthetic intermediate of a 1 beta-methylcarbapenem derivative
01/04/2000US6011053 Substituted indole-1-carbothioic acid amides as novel antiatherosclerotic agents
01/04/2000US6011033 Phenylene derivatives
01/04/2000US6011029 Benzodiazepine compounds
01/04/2000US6011028 Cyclic amidino agents useful as nitric oxide synthase inhibitors
12/1999
12/29/1999WO1999067237A1 4,5,6 and 7-indole and indoline derivatives, their preparation and use
12/29/1999WO1999067236A1 Novel form of irbesartan, methods for obtaining said form and pharmaceutical compositions containing same
12/29/1999WO1999067231A1 Nitrate salts of antihypertensive medicines
12/29/1999WO1999067215A1 Amidino and guanidino azetidinone tryptase inhibitors
12/29/1999WO1999066944A1 Methods for identifying novel multimeric agents that modulate receptors
12/29/1999WO1999066934A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING β-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS
12/29/1999EP0967212A1 Pyrazoline compounds and use as plant disease control agent
12/29/1999EP0967210A1 Process for preparing biologically active derivatives of 1,2,4-triazol and intermediaries useful in this process
12/29/1999EP0967207A1 Nitrone derivatives, process for their preparation and pharmaceutical compositions containing them
12/29/1999EP0966476A1 Quinazolinone compounds
12/29/1999EP0966475A1 Preparation of phosphonium compounds as intermediates for glycine antagonists
12/29/1999EP0966464A1 Substituted 2,4-diaminopyrimidines
12/29/1999EP0966463A1 Crystalline hydrated sodium salt of (e)-4,6-dichloro-3-(2-oxo-1-phenylpyrrolidin-3-ylidene methyl)-1h-indole-2-carboxylic acid
12/29/1999EP0966454A1 Disubstituted bicyclic heterocycles, their production and use as medicaments
12/29/1999EP0966447A1 Small molecules useful in the treatment of inflammatory disease
12/29/1999EP0966443A1 Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of mip-1-alpha binding to its ccr1 receptor
12/29/1999EP0966282A1 Use of angiotensin ii antagonists to treat symptomatic heart failure
12/29/1999EP0785932B1 Pyrrolyl tetrahydrobenzoquinoxaline diones, their preparation and use as glutamate receptor antagonists
12/29/1999EP0654031B1 Stereoselective synthesis of nucleoside analogues using bicyclic intermediate
12/29/1999CN1239957A Substituting 2-amino-4-alkylamino-1,3,5-triazine as herbicide
12/29/1999CN1239956A Substituted 2-amino-4-alkylamino-1,3,5-triazines as herbicides
12/29/1999CN1239955A Substituted 2,4-diamino-1,3,5-triazine as herbicide
12/29/1999CN1239953A 3-thiocarbamoylpyrazole derivatives as pesticides
12/29/1999CA2336003A1 Amidino and guanidino azetidinone tryptase inhibitors
12/29/1999CA2335711A1 4,5,6 and 7-indole and indoline derivatives, their preparation and use
12/29/1999CA2335545A1 Novel form of irbesartan, methods for obtaining said form and pharmaceutical compositions containing same
12/29/1999CA2335356A1 Nitrate salts of antihypertensive medicines
12/29/1999CA2324475A1 Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds
12/29/1999CA2319650A1 Methods for identifying novel multimeric agents that modulate receptors
12/28/1999US6008368 Pharmaceutical compositions for treatment of circulatory disorders using N-substituted (α-imidazolyl-toluyl) pyrrole aniotensin II antagonists
12/28/1999US6008353 Pesticide, insecticide, nematocide, paracitiside
12/28/1999US6008350 Process for the production of cyanine dyes
12/28/1999US6008243 An enzyme inhibitor for preventing the degradation and remodeling of connective tissues
12/28/1999US6008240 2-(1H-4(5)-imidazoyl) cyclopropyl derivatives
12/28/1999US6008230 Treating bone diseases caused by abnormal bone metabolism in human being or animals as the inhibitors of bone resorption or the inhibitors of bone metastasis
12/28/1999US6008229 Treating allergy, inflammation, autoimmune disease, shock, pain
12/28/1999US6008160 Substituted 1-amino-3-phenyluracil derivatives, their preparation and their use as herbicides
12/23/1999WO1999065898A1 Imidazolyl derivatives
12/23/1999WO1999065897A1 Inhibitors of glycogen synthase kinase 3
12/23/1999WO1999065882A1 2,4-diamino-1,3,5-triazine, method for the production and use of the same as herbicides and plant growth regulators
12/23/1999WO1999055156A3 The use of derivatives of iminotriazole as crop protection agents and novel iminotriazoles
12/23/1999DE19925329A1 New triazine derivatives useful as selective herbicides and plant growth regulators
12/23/1999CA2335435A1 Imidazolyl derivatives
12/23/1999CA2335327A1 2,4-diamino-1,3,5-triazines, their preparation, and their use as herbicides and plant growth regulators
12/22/1999EP0965586A1 Method of purifying carbazole ester precursors of 6-chloro-alpha-methyl-carbazole-2-acetic acid
12/22/1999EP0964864A2 Pyrido 2,3-d] pyrimidines and 4-aminopyrimidines as inhibitors of cellular proliferation
12/22/1999EP0731795B1 Substituted pyrazolyl benzenesulfonamides for the treatment of inflammation