Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
06/1999
06/17/1999CA2312720A1 Retinoic acid mimetic anilides
06/16/1999EP0922697A1 Substituted Pyrazolyl benzenesulfonamides and their use as cyclooxygenase II inhibitors
06/16/1999EP0922042A1 Novel piperazine containing compounds
06/16/1999EP0922036A1 Arylalkanoyl pyridazines
06/16/1999EP0922035A1 Tetrahydroisoquinoline derivatives and their pharmaceutical use
06/16/1999EP0921801A1 Inhibitors of farnesyl-protein transferase
06/16/1999EP0711283B1 Tetrahydro-1h-benzazepinones and hexahydroazepinones as selective cholecystokinin-b receptor antagonists
06/16/1999EP0553218B1 Indole derivatives
06/16/1999CN1219932A Aromatic amidine derivatives useful as selective thrombin inhibitors
06/16/1999CN1219841A DNA-binding indole derivatives, their prodrugs and immunoconjugates as anticancer agents
06/16/1999CN1219538A Antifungal agent and its preparing process and intermediate
06/15/1999US5912260 Gastrin and CCK antagonists
06/15/1999US5912244 Muscle disorders, breathing disorders and urinary incontinence
06/15/1999US5912110 Photographic coupler capable of releasing a photographically useful group
06/12/1999CA2224752A1 5-alkenyl and 5-alkynyl indole compounds
06/10/1999WO1999028315A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof
06/10/1999WO1999028313A1 Inhibitors of farnesyl-protein transferase
06/10/1999WO1999028305A1 Fungicidal cyclic amides
06/10/1999WO1999028304A2 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
06/10/1999WO1999028301A1 Substituted pyrimidine and pyridine herbicides
06/10/1999WO1999028300A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
06/10/1999WO1999028297A1 Substituted indoles, having a thrombin inhibiting effect
06/10/1999DE19753522A1 Substituierte Indole, ihre Herstellung und ihre Verwendung als Arzneimittel Substituted indoles, their preparation and their use as medicaments
06/10/1999CA2312749A1 Pdgf receptor kinase inhibitory compounds and compositions, method for synthesis of same and use of same for treatment of proliferate disorders
06/10/1999CA2312366A1 Inhibitors of farnesyl-protein transferase
06/10/1999CA2312334A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
06/10/1999CA2310629A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof
06/09/1999EP0921120A1 Selective beta 3 adrenergic agonists
06/09/1999EP0921119A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them
06/09/1999EP0920424A1 Non-peptide bombesin receptor antagonists
06/09/1999EP0920419A1 Compounds, compositions and methods for treating influenza
06/09/1999CN1219172A Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
06/09/1999CN1218801A Tri-substituted imidazoles, and process of their preparation and using the same and having their pharmic composition
06/08/1999CA1340588C Amino acid derivatives
06/03/1999WO1999026944A1 New compounds which are p2-purinoceptor 7-transmembrane (tm) g-protein coupled receptor antagonists
06/03/1999WO1999026942A1 5-(2-imidazolinylamino)-benzimidazole derivatives, their preparation and their use as .alpha.-adrenoceptor agonists with improved metabolic stability
06/03/1999WO1999026941A1 Substituted amidinoaryl derivatives and their use as anticoagulants
06/03/1999WO1999026935A1 Trisaryl-1,3,5-triazine ultraviolet light absorbers
06/03/1999WO1999026932A1 By amidino group substituted heterocyclic derivatives and their use as anticoagulants
06/03/1999WO1999026930A2 Benzylidene pyrazolones and use as herbicide
06/03/1999WO1999026922A1 Substituted pyrrole derivatives as cell adhesion inhibitors
06/03/1999WO1999026921A1 SUBSTITUTED β-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS
06/03/1999WO1999026659A1 Combination of an aldose reductase inhibitor and a glycogen phosphorylase inhibitor
06/03/1999CA2311538A1 Trisaryl-1,3,5-triazine ultraviolet light absorbers
06/03/1999CA2310087A1 Benzylidene pyrazolones and use as herbicide
06/03/1999CA2310069A1 Combination of an aldose reductase inhibitor and a glycogen phosphorylase inhibitor
06/03/1999CA2309341A1 Substituted .beta.-alanine derivatives as cell adhesion inhibitors
06/02/1999EP0919554A1 Imidazole-substituted quinoxalinedione derivatives
06/02/1999EP0918768A1 Aromatic amidine derivatives useful as selective thrombin inhibitors
06/02/1999EP0918758A1 Process for preparing 1-substituted 4-cyano-1,2,3-triazoles
06/02/1999EP0918755A1 1-alkyl-4-benzoyl-5-hydroxypyrazole compounds and their use as herbicides
06/02/1999EP0918752A2 Dna-binding indole derivatives, their prodrugs and immunoconjugates as anticancer agents
06/02/1999EP0581939B1 N-sulphonyl-2-oxoindole derivatives having affinity for vasopressin and/or ocytocin receptors
06/02/1999CN1218464A 2,3 disulbstituted-4 (3H)-quinazolinones
06/02/1999CN1218456A Irreversible inhibitors of tyrosine kinases
06/02/1999CN1218052A New indole and indazole compounds, process for their preparation and pharmaceutical compositions containing them
06/02/1999CN1218046A Imide derivatives
06/02/1999CN1218044A Urea derivatives
06/02/1999CN1043532C The sulphate salt of a substituted triazole, pharmaceutical compositions thereof, and their use in therapy
06/02/1999CN1043531C Pyrimidine derivatives and a process for production thereof
06/01/1999US5908931 Preorganized hexadentate ligands useful in radiographic imaging agents
06/01/1999US5908844 Neuroleptic agent
06/01/1999US5908843 Thrombosis, antiinflammatory agent, arteriosclerosis, antitumor agents
06/01/1999CA2056334C Process for producing benzylphthalazinone derivatives and salts thereof
06/01/1999CA1340567C Heterocyclic amide derivatives
05/1999
05/27/1999WO1999025686A1 Cyclic amine derivatives and their use as drugs
05/26/1999EP0917462A1 Cell adhesion inhibitors
05/26/1999CN1217723A Tricyclic diazepines, its production and use
05/26/1999CN1217711A Aryl substituted cyclic amines as selective dopamine D3 ligands
05/26/1999CN1217327A D-proline derivative
05/20/1999WO1999024460A2 Dipeptide nitriles
05/20/1999WO1999024425A1 Benzimidazole derivatives and pharmaceutically acceptable salts thereof
05/20/1999WO1999024424A1 Pyrazole compounds and medicinal use thereof
05/20/1999WO1999024422A1 Azaring-ether derivatives and their use as nicotinic ach receptor modulators
05/20/1999WO1999024421A1 Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom
05/20/1999WO1999024420A1 Pyrimidinone compounds and pharmaceutical compositions containing them
05/20/1999WO1999024406A1 Phenyl-alkyl-imidazoles as h3 receptor antagonists
05/20/1999CA2309609A1 Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom
05/20/1999CA2309177A1 Pyrimidinone compounds and pharmaceutical compositions containing them
05/20/1999CA2309121A1 Phenyl-alkyl-imidazoles as h3 receptor antagonists
05/20/1999CA2306477A1 Azaring-ether derivatives and their use as nicotinic ach receptor modulators
05/19/1999EP0916675A2 Process for preparing sildenafil
05/19/1999EP0916658A1 Assays utilizing improved chemiluminescent esters, thioesters and amides
05/19/1999EP0915872A1 Substituted bisindolylmaleimides for the inhibition of cell proliferation
05/19/1999EP0915871A1 Substituted bisindolylmaleimides for the inhibition of cell proliferation
05/19/1999EP0915870A1 Substituted bisindolylmaleimides for the inhibition of cell proliferation
05/19/1999EP0915868A1 Carbanilides used as pesticides
05/19/1999EP0915848A1 1,2-diarylindole as cox-2 inhibitors
05/19/1999EP0915847A1 Substituted sulfonamides as selective beta3 agonists for the treatment of diabetes and obesity
05/19/1999EP0915846A2 2- and 2,5-substituted phenylketoenols
05/19/1999EP0915845A1 Acryloyl substituted distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agents
05/19/1999CN1216762A 2-(arylphenyl) amino-imidazoline derivatives
05/18/1999US5905152 Preparation of aminomethyl-phenylimidazoles
05/14/1999WO1999023093A1 2-(2'-hydroxyphenyl)benzotriazoles used as u.v. stabilisers
05/14/1999WO1999023079A1 Carbamoylphenylsulfonyl ureas, method for their production and their application as herbicides and plant growth regulators
05/14/1999WO1999023078A2 Novel carboxylic acid derivatives which carry amide side chains, production of said carboxylic acid derivatives and their use as endothelin receptor antagonists
05/14/1999WO1999007352A3 Method for promoting expression of ldl receptor gene
05/14/1999WO1998058915A3 Pyrimidin-2,4,6-trion derivatives and their use as metalloprotease-inhibitors
05/14/1999CA2309438A1 Carbamoylphenylsulfonylureas, processes for their preparation and their use as herbicides and plant growth regulators
05/14/1999CA2307770A1 Novel carboxylic acid derivatives which carry amide side chains, production of said carboxylic acid derivatives and their use as endothelin receptor antagonists