Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
03/2000
03/22/2000EP0986302A1 A method of treating cancer
03/22/2000CN1248255A 3-heterocyclyl-substituted benzoyl derivatives
03/22/2000CN1248251A Disubstituted bicyclic heterocycles, their production and use as medicaments
03/22/2000CN1050603C Prepn. of intermediate product used in process for diastereoselective synthesis of nucleosides
03/21/2000US6040454 Process for preparation of a 1-(tetrazolylbiphenylmethyl)-imidazole derivative
03/21/2000US6040451 Used as analgesic, sedative and anaesthetic agents
03/21/2000US6040329 Substituted indazole analogs
03/21/2000US6040327 Benzimidazole, benzoxazole and benzothiazole compounds
03/21/2000US6040324 Prophylactic or therapeutic drug for renal diseases
03/21/2000US6040317 Sulfonamide fibrinogen receptor antagonists
03/21/2000US6040311 Treating bone disorders for preventing osteoporosis or inhibiting bone resorption in a mammal; treating tumor growth in a mammal
03/21/2000US6040302 1,4-disubstituted piperazines
03/21/2000CA2282885A1 New cationic 4-hydroxyindoles, their application in keratin fibre oxidation dye, dye compositions and dyeing methods
03/16/2000WO2000014073A1 Benzodiazepinone derivatives, preparation method and intermediates therefor, use as medicines and compositions
03/16/2000WO2000014065A1 Kappa agonist compounds and pharmaceutical formulations thereof
03/16/2000WO2000013708A1 Methods for treating or preventing viral infections and associated diseases
03/16/2000WO2000013707A1 Preventives/remedies for multiple organ failure
03/16/2000WO2000013683A2 Novel nitrophenylaziridine compounds and their use as prodrugs
03/16/2000WO2000005206A8 Arylpiperazine derivatives useful as uro-selective alpha-1-adrenoceptor blockers
03/16/2000CA2343522A1 Methods for treating or preventing viral infections and associated diseases
03/16/2000CA2342994A1 Kappa agonist compounds and pharmaceutical formulations thereof
03/16/2000CA2342943A1 Novel nitrophenylaziridine compounds and their use as prodrugs
03/16/2000CA2342796A1 Preventives/remedies for multiple organ failure
03/15/2000EP0984960A1 N-triazolyl-2-indolecarboxamides and their use as cck-a agonists
03/15/2000EP0984944A1 Substituted 4-(3-alkenyl-benzoyl)-pyrazoles
03/15/2000EP0984930A1 2-indolinone derivatives as modulators of protein kinase activity
03/15/2000EP0984777A1 Arylsubstituted piperazines useful in the treatement of benign prostatic hyperlasia
03/15/2000EP0619805B1 5-(hetero- or carbocyclylamino)-indole derivatives, their preparation and their use as 5-ht1 agonists
03/15/2000CN1247533A Heterocyclic carboxylic acid derivatives, prodn. and use thereof as endothelin receptor antagonists
03/14/2000US6037475 Reacting optionally substituted, n-protected indol-3-yl-acetamide with an alkyl oxalate and a strong organic base in a polar aprotic solvent forming optionally substituted 4-(indol-3-yl)-3-hydroxy pyrrole-2,5-dione
03/14/2000US6037354 Administering phenyl-substituted thiazolidin-4-one or oxazolidin-2-one derivative to treat benign prostate hyperplasia; side effect reduction
03/14/2000US6037352 N-substituted piperidine derivatives; treating alzheimer*s disease, nervous system disorders; acetylcholinesterase inhibitors
03/09/2000WO2000012500A2 2-aryl-4-(1-[4-heteroaryl]piperazin-1-yl) methylimidazoles: dopamine d4 receptor subtype ligands
03/09/2000WO2000012497A2 Quinazoline derivatives as medicaments
03/09/2000WO2000012489A1 1, 2, 4-triazole-3-thione compounds
03/09/2000WO2000012485A1 Pyrimidine compounds
03/09/2000WO2000012484A1 Tan-1057 derivatives
03/09/2000WO2000012089A1 Novel angiogenesis inhibitors
03/09/2000WO2000012084A1 Geometrically restricted 2-indolinone derivatives as modulators of protein kinase activity
03/09/2000WO2000012076A1 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
03/09/2000WO2000012067A1 Novel pharmaceutical salt form
03/09/2000WO2000005230A8 Pyrazole derivatives and salts thereof
03/09/2000WO1999051215A3 Immunosuppressive imidazole derivatives and their combination preparations with tacrolimus or cyclosporins
03/09/2000DE19838998A1 Neue Naturstoffderivate New natural product derivatives
03/09/2000CA2342250A1 Quinazoline derivatives as medicaments
03/09/2000CA2342222A1 Geometrically restricted 2-indolinone derivatives as modulators of protein kinase activity
03/09/2000CA2341522A1 Novel pharmaceutical salt form
03/09/2000CA2341409A1 Novel angiogenesis inhibitors
03/09/2000CA2339189A1 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
03/08/2000EP0984010A1 Use in hair dyes of quinolin-5,8-diones or quinoxalin-5,8-diones condensed with substituted pyrroles, anilines or indoles
03/08/2000EP0983251A1 Anti-inflammatory piperazinyl-benzyl-tetrazole derivatives and intermediates thereof
03/08/2000CN1246858A Substituted pyrimidine compounds and their use
03/08/2000CN1246850A 1,5-benzodiazepine derivatives
03/08/2000CN1246847A Nitrogen containing heteroaromatics as factor Xa inhibitors
03/08/2000CN1050126C Tri-substituted imidazoles compound, process for preparing it and use and pharmaceutical compositions containing them
03/08/2000CN1050122C Benzimidazoles, pharmaceutical compositions containing these compounds and process for preparing them
03/08/2000CN1050121C Preparation method of substituted aryl-haloalkylpyrazoles compound
03/07/2000US6034250 Nitrone compounds
03/07/2000US6034248 Fungicides
03/07/2000US6034216 Low molecular weight peptidomimetic growth hormone secretagogues
03/07/2000US6034093 Anticoagulants
03/07/2000CA2030401C Inhibition of the abstinence syndrome
03/02/2000WO2000010975A1 Oxindole derivatives as growth hormone releasers
03/02/2000WO2000010565A1 Growth hormone secretagogues
03/02/2000WO2000010563A1 Novel substituted triazole compounds
03/02/2000WO1999064043A9 Muscarinic receptor antagonists
03/02/2000CA2341370A1 Novel substituted triazole compounds
03/01/2000EP0981728A2 Radiolabeled farnesyl-protein transferase inhibitors
03/01/2000EP0981521A2 Novel macrocyclic compounds as metalloprotease inhibitors
03/01/2000EP0981519A1 Methods of modulating serine/threonine protein kinase function with quinazoline-based compounds
03/01/2000CA2281177A1 Use in hair dye of condensates of quinoline-5,8-diones or quinoxaline-5,8-diones and substitute indoles, pyrroles or anilines
02/2000
02/29/2000US6031110 Ortho-substituted 2-methoxyiminophenyl-N-methylacetamides
02/29/2000US6031097 1-(N-(arylalkylaminoalkyl) aminoisoquinolines; a new class of dopamine receptor subtype specific ligands
02/29/2000US6031094 Beta-lactam substrates and uses thereof
02/29/2000US6030994 Substituted pyrroles compositions
02/29/2000US6030976 Use of sulfonamides
02/29/2000US6030966 Heterocyclic compound and their use
02/29/2000CA2169179C 5-arylindole derivatives
02/24/2000WO2000009499A1 N-substituted azabicycloheptane derivatives, production and use thereof
02/24/2000WO2000009496A1 Substituted 4-amino-2-aryl-pyrimidines, their production and use and pharmaceutical preparations containing same
02/24/2000WO2000009489A1 New carboxylic acid derivatives carrying keto side-chains, their production and their use as endothelin-receptor antagonists
02/24/2000WO2000009488A1 Pyridazinone derivatives
02/24/2000WO2000009106A2 Carboxylic acids and isosteres of heterocyclic ring compounds having multiple heteroatoms for vision and memory disorders
02/24/2000WO2000009103A2 N-linked sulfonamides of n-heterocyclic carboxylic acids or isosteres for vision and memory disorders
02/24/2000WO1999048868A3 Heterocyclic classes of compounds for the modulating tyrosine protein kinase
02/24/2000CA2340168A1 N-substituted azabicycloheptane derivatives, production and use thereof
02/24/2000CA2340167A1 New carboxylic acid derivatives carrying keto side-chains, their production and their use as endothelin-receptor antagonists
02/24/2000CA2336154A1 Carboxylic acids and isosteres of heterocyclic ring compounds having multiple heteroatoms for vision and memory disorders
02/24/2000CA2336147A1 N-linked sulfonamides of n-heterocyclic carboxylic acids or isosteres for vision and memory disorders
02/23/2000CN1245169A Nitroketone compound, its preparing process and pharmaceutical composition containing same
02/23/2000CN1049654C Piperazine derivatives and medicine composition containing same and use thereof
02/22/2000US6028073 For treating psychoses
02/22/2000US6028072 For treating inflammation and inflammation related disorders
02/22/2000US6028063 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
02/17/2000WO2000008202A2 3-methylidenyl-2-indolinone modulators of protein kinase
02/17/2000WO2000008041A1 Structural analogs of amine bases and nucleosides
02/17/2000WO2000007999A1 Triazolone derivatives, use thereof, and intermediate therefor
02/17/2000WO2000007997A1 IMIDAZOLES AND RELATED COMPOUNDS AS α1A AGONISTS
02/17/2000WO2000007996A2 Pyrazoles as estrogen receptor modulators
02/17/2000WO2000007995A1 SUCCINOYLAMINO LACTAMS AS INHIBITORS OF Aβ PROTEIN PRODUCTION