Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
10/2000
10/17/2000US6133276 A ligand inhibitor of a crf/crf-binding protein complex to effect increased levels of crf; 2,4-dioxo- or 2-thiocarbonyl-4-oxo-5-(hydrocarbyl(thio)carbonylaminomethyl)-6-hydroxy-hexa-hexahydropyrimidines; alzheimer's, obesity; low side effects
10/17/2000US6133275 3-phenylpyrrolidine alpha-1 adrenergic compounds
10/17/2000US6133272 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
10/17/2000US6133268 1,4-disubstituted piperazines
10/17/2000US6133257 Fused polycyclic 2-aminopyrimidine derivatives
10/17/2000CA2114300C Quinoline or quinazoline derivatives, their production and use
10/15/2000CA2305940A1 Aminotriazol compounds, the process for preparing them and the pharmaceutical compositions containing them
10/12/2000WO2000059904A2 Compounds and methods to treat cardiac failure and other disorders
10/12/2000WO2000059901A1 Substituted 1,4-dihydroindeno[1,2-c]pyrazoles as inhibitors of tyrosine kinase
10/12/2000WO2000059886A2 Benzimidazole abd imidazolophyridine derivaties, their preparation and their use as selective modulators of bradykinin b2 (=bk-2) receptors
10/12/2000WO2000059884A1 Pharmaceutically active compounds and methods of use thereof
10/12/2000WO2000059881A1 Substituted azetidin-2-ones as cysteine protease inhibitors
10/12/2000WO2000059510A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors
10/12/2000WO2000059506A1 HETEROCYCLIC CONTAINING BIPHENYL aP2 INHIBITORS AND METHOD
10/12/2000WO2000059502A1 Pyrrolidine modulators of chemokine receptor activity
10/12/2000WO2000009106A3 Carboxylic acids and isosteres of heterocyclic ring compounds having multiple heteroatoms for vision and memory disorders
10/12/2000CA2484282A1 Pyrimidine derivatives intermediates for producing aminopyrimidines as sorbitol dehydrogenase inhibitors
10/12/2000CA2373717A1 Pyrrolidine modulators of chemokine receptor activity
10/12/2000CA2369544A1 Aryl and heteroaryl fused aminoalkyl-imidazole derivatives:selective modulators of bradykinin b2 receptors
10/12/2000CA2369446A1 Substituted azetidin-2-ones as cysteine protease inhibitors
10/12/2000CA2368686A1 Substituted 1,4-dihydroindeno[1,2-c]pyrazoles as inhibitors of tyrosine kinase
10/12/2000CA2366858A1 Sorbitol dehydrogenase inhibitors
10/12/2000CA2361734A1 Pharmaceutically active compounds and methods of use thereof
10/11/2000EP1043365A1 Polymerizable 1,2-dipyrazolylethenes as dyes for ophthalmic plastic lenses
10/11/2000EP1042320A1 New compounds which are p2-purinoceptor 7-transmembrane (tm) g-protein coupled receptor antagonists
10/11/2000EP1042317A1 New pharmaceutically active compounds
10/11/2000EP1042299A1 Nitrogen containing heteroaromatics with ortho-substituted p1's as factor xa inhibitors
10/11/2000EP1042293A1 Substituted pyridine and pyridazine compounds and their pharmaceutical use
10/11/2000EP1042287A1 Indole derivatives as inhibitors of factor xa
10/11/2000EP1042279A1 Substituted beta-alanines
10/11/2000CN1269806A Piptides containing arginine mimetic for treatment of bone metabolic disorders, their production and drugs containing these compounds
10/11/2000CN1269794A 6,7-asymmetrically disubstituted quinoxalinecarboxylic acid derivatives, addition salts thereof and process for preparation of both
10/11/2000CN1269363A Method for proparing heterocyclic compound
10/11/2000CN1057297C Waterless crystallization of quinolone derivative and crystallization method of its 3/2 hydrate
10/10/2000US6130239 Inhibit cyclin-dependent kinases
10/10/2000US6130235 Piperidine moieties coupled to indole, benzimidazole or benzotriazole.
10/10/2000US6130215 Central nervous system
10/05/2000WO2000058306A1 Substituted benzoylpyrazoles as herbicides
10/05/2000WO2000058304A1 Heterocyclic sulfonamide derivatives
10/05/2000WO2000058295A2 Compounds and methods for treatment of asthma, allergy and inflammatory disorders
10/05/2000WO2000057877A1 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof
10/05/2000WO2000042026B1 Non-peptide glp-1 agonists
10/05/2000CA2368631A1 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof
10/05/2000CA2368459A1 Substituted benzoylpyrazoles as herbicides
10/05/2000CA2368090A1 Compounds and methods for treatment of asthma, allergy and inflammatory disorders
10/04/2000EP1041064A2 N-substituted alpha aminoacid amides as calcium channel modulators
10/04/2000EP1040101A1 Substituted 2-aryl-4-amino-chinazolines, method for the production and use thereof as medicaments
10/04/2000EP1019040A4 INHIBITION OF p38 KINASE ACTIVITY BY ARYL UREAS
10/04/2000CN1268352A Method for preparing medicinal prepns. contg. 6-heterocycle-4-amino-1,3,4,5-tetrabenzo [cd] indole
10/04/2000CN1057086C Phenylsulfonyl ureas, process for preparing same, and use as herbicide, herbicide composition contg. same
10/04/2000CN1057085C Heterocyclically substituted phenyl-cyclohexane carboxylcic acid derivatives
10/03/2000US6127547 Halobenzimidazoles and their use as microbicides
10/03/2000US6127404 Tissue selective compounds in the treatment of endometrial proliferation
10/03/2000US6127403 An enzyme inhibitor for treating arteriosclerotic lesions of arteriosclerosis, hyperlipemia and diabetes, as well as ischemic diseases of brain, heart
10/03/2000US6127376 Aryl and heterocyclyl substituted pyrimidine derivatives as anti-coagulants
10/03/2000US6127375 A 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthiones for treating viral infection
10/03/2000US6127360 Antihistamines, antileukotrienes, antiinflammatory agents, antiasthmatic agents
10/03/2000US6127357 N-((phenyl, benzodioxinyl or N-heteroarylpiperazinyl)alkyl)-N-(N-heteroaryl)substituted carboxamides
10/03/2000US6126932 Insoluble polymer bearing pendant side chains, said side chains each terminating with the 1-(3-(1-pyrrolidinyl)-propyl)-3-ethylcarbodiimide moiety.
09/2000
09/28/2000WO2000056722A1 2,4-diamino-1,3,5-triazines, method for producing them and their use as herbicides and plant growth regulators
09/28/2000WO2000056710A1 3-(anilinomethylene) oxindoles as protein tyrosine kinase and protein serine/threonine kinase inhibitors
09/28/2000WO2000056709A1 Indolinone compounds as kinase inhibitors
09/28/2000WO2000056337A1 Agents for relieving side effects
09/28/2000DE19914140A1 Substituierte Benzoylpyrazole Substituted benzoylpyrazoles
09/28/2000CA2368041A1 Indolinone compounds as kinase inhibitors
09/28/2000CA2367920A1 2,4-diamino-1,3,5-triazines, processes for their preparation and their use as herbicides and plant growth regulators
09/27/2000EP1038873A2 Benzo(3,4)cyclobuta(1,2-c)pyrrole derivatives as inhibitors of serotonine reuptake
09/27/2000EP1038526A1 Treatment of functional disorders of the lower intestinal tract and subsequent visceral pain with moxonidine
09/27/2000EP1037887A1 5-(2-imidazolinylamino)-benzimidazole derivatives, their preparation and their use as .alpha.-adrenoceptor agonists with improved metabolic stability
09/27/2000EP1037886A1 Triazine angiogenesis inhibitors
09/27/2000EP1037880A1 Retinoic acid mimetic anilides
09/27/2000EP1037639A1 Compounds of heteroaryl substituted imidazole, their pharmaceutical compositions and uses
09/27/2000EP0733052B1 Bicyclene derivatives, their production and use
09/27/2000CN1268134A Bis-indole derivatives having antimetastatic activity, A process for their preparation and pharmaceutical compositions containing them
09/27/2000CN1268126A Pyrimidin-2,4,6-trion derivatives and their use as metalloprotease-inhibitors
09/27/2000CN1268124A Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments
09/27/2000CN1267671A Process for producing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative
09/27/2000CN1056842C Amino acid derivative having anti CCK activity
09/26/2000US6124463 Treatment of affective disorder, anxiety or depression
09/26/2000US6124331 Selective NPY (Y5) antagonists (tricyclics)
09/26/2000US6124330 N-[4-(Heteroarylmethyl)phenyl]-heteroarylamines
09/26/2000US6124325 Triazole antifungal agents
09/26/2000US6124306 Treating human immunodeficiency virus infections
09/26/2000US6124294 Compounds having high affinity for dopamine d3 receptor; used to treat disorders which respond to dopamine d3 ligands
09/26/2000CA2168016C Benzimidazole derivatives
09/26/2000CA2024572C N-substituted-4-pyrimidinamines and-pyrimidinediamines, a process for their preparation and their use as medicaments
09/21/2000WO2000055156A1 Substituted aromatic amidine derivative and medicinal composition comprising the same
09/21/2000WO2000055155A2 Heterocyclic compounds as adenosine deaminase inhibitors
09/21/2000WO2000055153A1 Amide derivatives
09/21/2000WO2000055141A1 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, and processes for preparing them
09/21/2000WO2000055139A2 Heterocyclic urea and related compounds useful as anti-inflammatory agents
09/21/2000WO2000054729A2 Heterocyclic aromatic compounds useful as growth hormone secretagogues
09/21/2000DE19912690A1 New benzimidazolyl amidine or nitrile compounds, useful as thrombin inhibitors or antithrombotic agents, for treating deep leg vein thrombosis
09/21/2000DE19912637A1 2,4-Diamino-1,3,5-triazine, Verfahren zur Herstellung und Verwendung als Herbizide und Pflanzenwachstumsregulatoren 2,4-diamino-1,3,5-triazines, to processes for preparation and use as herbicides and plant growth regulators
09/21/2000DE19911509A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
09/21/2000DE19911371A1 Arzneimittel zur Behandlung von funktionellen Störungen und Erkrankungen der unteren Darmwege, insbesondere von damit einhergehenden abdominalen visceralen Schmerzen Drugs for the treatment of functional disorders and diseases of the lower intestinal tracts, especially of associated abdominal visceral pain
09/21/2000DE19911366A1 New 4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors, polyps or respiratory or gastrointestinal diseases
09/21/2000CA2367461A1 Heterocyclic aromatic compounds useful as growth hormone secretagogues
09/20/2000EP1036793A2 A process for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative
09/20/2000EP1036067A2 Pdgf receptor kinase inhibitory compounds, their preparation and compositions