Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
09/1999
09/07/1999CA2098944C Novel pyrazole derivatives, method of preparing them and pharmaceutical compositions in which they are present
09/07/1999CA2014008C Benzimidazoles, medicaments containing these compounds and processes for their preparation
09/02/1999WO1999043672A1 Inhibitors of phospholipase a2
09/02/1999WO1999043663A1 N-[(substituted five-membered di- or triaza diunsaturated ring)carbonyl] guanidine derivatives for the treatment of ischemia
09/02/1999WO1999043654A2 Inhibitors of phospholipase enzymes
09/02/1999WO1999043651A2 Inhibitors of phospholipase enzymes
09/02/1999WO1999043642A1 Phenylalanine derivatives as inhibitors of alpha4 integrins
09/02/1999WO1999024460A3 Dipeptide nitriles
09/02/1999CA2322163A1 Inhibitors of phospholipase a2
09/02/1999CA2322162A1 Inhibitors of phospholipase enzymes
09/02/1999CA2322161A1 Inhibitors of phospholipase enzymes
09/02/1999CA2321642A1 N-¬(substituted five-membered di- or triaza diunsaturated ring)carbonyl|guanidine derivatives for the treatment of ischemia
09/01/1999EP0939078A2 Substituted phthalimido-cinnamic acid derivatives with herbicidal activity
09/01/1999EP0939077A2 3-Substituted 1-arylindole compounds as 5-HT2 antagonists
09/01/1999EP0938479A1 Quaternary nitrogen heterocycles, method for their production and their use as pesticides
09/01/1999EP0938474A2 Cyclopropylindole compounds and their use as prodrugs
09/01/1999CN1227551A N-sulfonylimidazoles used as fungicides
09/01/1999CN1227547A Arylalkanoyl pyridazines
09/01/1999CN1227546A Substituted 1-(3-pyrazolyl)-pyrazoles with herbicide activity and intermediate for its preparation
09/01/1999CN1044906C 3(2H)-pyridazinono derivatives, its preparing method and its composition
08/1999
08/31/1999US5945443 Kappa agonist compounds and pharmaceutical formulations thereof
08/31/1999US5945425 Method of using (H+ /K+)ATPase inhibitors as antiviral agents
08/31/1999US5945413 Treating human immunodeficiency virus infections
08/31/1999US5945118 Indole derivative for the treatment of migraine
08/31/1999CA2173328C Hiv protease inhibitors
08/31/1999CA2145835C Hydroxamic acid derivatives with tricyclic substitution
08/26/1999WO1999042463A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
08/26/1999WO1999042461A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
08/26/1999WO1999042458A1 Histamine h3 receptor ligands
08/26/1999WO1999042453A1 5-substituted pyrimidine-2-yloxy carboxylic acid derivatives, the production of the same and their utilization as endothelin antagonists
08/26/1999WO1999042452A1 Phthalazine derivatives and remedies for erectile dysfunction
08/26/1999WO1999042100A1 Cell death inhibitors
08/26/1999WO1999042092A2 Compounds and methods of use for treatment of neurogenic inflammation
08/26/1999WO1999031060A3 Piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides as cytostatics and immunesuppressants
08/26/1999WO1999024421A8 Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom
08/26/1999CA2321182A1 5-substituted pyrimidine-2-yloxy carboxylic acid derivatives, the production of the same and their utilization as endothelin antagonists
08/26/1999CA2318836A1 Histamine h3 receptor ligands
08/25/1999EP0937722A1 Benzimidazole derivatives as cyclooxygenase-2 inhibitors
08/25/1999EP0937715A1 Tetrahydrobenzindole compounds
08/25/1999EP0937070A1 Benzoheterocyclic distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agents
08/25/1999EP0937069A1 Piperazino derivatives as neurokinin antagonists
08/25/1999EP0937068A1 Process for the crystallization of losartan
08/25/1999EP0937067A1 1-(3-aminoindazol-5-yl)-3-phenylmethyl-cyclic ureas useful as hiv protease inhibitors
08/25/1999EP0937066A1 (4r,5s,6s,7r)-hexahydro-1- 5-(3-aminoinazole)methyl] -3-butyl-5,6-dihydroxy-4,7-bis phenylmethyl] -2h-1,3-diazepin-2-one, its preparation and its use as hiv protease inhibitor
08/25/1999EP0937051A1 Fungicidal cyclic amides
08/25/1999EP0937046A2 Substituted 3-benzylpyrazoles and their use as herbicides and for lowering the sugar content in blood
08/25/1999EP0937042A1 Heteroaryl succinamides and their use as metalloproteinase inhibitors
08/25/1999EP0937040A2 N-substituted 2-cyanopyrrolidines
08/24/1999US5942536 Useful for treating migraine
08/24/1999US5942532 Inhibitors of histidine protein kinase; bacteria resistant to other antibiotics
08/24/1999US5942524 Serotonin(5-ht-1) agonists
08/24/1999US5942517 Antagonist of alpha(1c) receptors; treatment of benign prostatic hyperplasia
08/24/1999US5942509 2-(triazinyloxy(or thio)phenyl)-substituted methyl 3-methoxy-2-propenoate
08/24/1999US5942506 1- 2-(substituted vinyl)!-5H-2,3-benzodiazepine derivatives
08/19/1999WO1999041367A1 Heteroaromatic oligoamides as affinity ligands
08/19/1999WO1999041253A1 Anti-viral pyrimidine derivatives
08/19/1999WO1999041242A1 Di-substituted naphthyl derivatives, preparation thereof, pharmaceutical compositions containing them
08/19/1999WO1999041235A1 Farnesyl transferase inhibitors
08/19/1999WO1999040931A1 Cyclic dipeptides and azetidinone compounds and their use in treating cns injury and neurodegenerative disorders
08/19/1999WO1999026930A3 Benzylidene pyrazolones and use as herbicide
08/19/1999DE19806438A1 New pyrimidinyloxy-propionic acid derivatives useful as endothelin receptor antagonists in treatment of e.g. cardiac insufficiency, restenosis, hypertension, kidney failure, asthma and prostate cancer
08/19/1999CA2321153A1 Anti-viral pyrimidine derivatives
08/19/1999CA2320378A1 Cyclic dipeptides and azetidinone compounds and their use in treating cns injury and neurodegenerative disorders
08/18/1999EP0936221A1 Novel 2,4-dioxopyrrolidine and 2,4-dioxotetrahydrofuran derivatives and medicines containing the same as the active ingredient
08/18/1999EP0936218A1 Novel benzimidazole derivatives
08/18/1999EP0935463A2 Anti-neurogenic inflammatory compounds and compositions and methods of use thereof
08/18/1999CN1226249A Substituted bisindolylmaleimides for inhibition of cell proliferation
08/18/1999CN1226248A Substituted bisindolylmaleimides for inhibition of cell proliferation
08/18/1999CN1226247A Substituted bisindolyl maleimides for inhibition of cell proliferation
08/18/1999CN1226244A Carbanilides used as pesticides
08/18/1999CN1226232A Acryloyl substituted distamycin derivative, process for preparing them, and use as antitumor and antiviral agents
08/18/1999CN1226166A Formulation and method for treating congestive heart failure
08/18/1999CN1044702C Ozonide reducing method
08/17/1999US5939587 N-protected/N-substituted-beta-amino hydroxy sulfonates
08/17/1999US5939560 Inhibitors of DP-mediated processes, compositions and therapeutic methods thereof
08/17/1999US5939557 Inhibitors of farnesyl-protein transferase
08/17/1999US5939451 Use of sulfonamides
08/17/1999US5939449 Novel compounds having high affinity for the neurotensin receptors
08/17/1999US5939443 Selective β3 adrenergic agonists
08/17/1999US5939440 Fungicides and bactericides
08/17/1999US5939439 Enzyme inhibitors in carriers for ras proteins
08/17/1999US5939424 Compounds for treating disorders of lipid metabolism and their preparation
08/17/1999US5939414 Benzodiazepine hydrazide derivatives as inhibitors of HIV integrase
08/17/1999US5939413 Tachykinin mediated diseases in humans for respiratory system disorders like asthma, bronchitis, rhinitis or eye diseases or skin disorders
08/17/1999US5939268 Diels-alder reaction product of a diene and a dienophile; chemical intermediates for drugs, solid phase synthesis
08/17/1999CA2179008C 5-(2-imidazolinylamino)benzimidazole derivatives, their preparation and their use as alpha-2 adrenoceptor agonists
08/12/1999WO1999040089A1 Benzothiadiazoles and derivatives
08/12/1999WO1999040075A1 Sulfonamide derivatives, process for producing the same and utilization thereof
08/12/1999WO1999040072A1 Five-membered, benzo-condensed heterocycles used as antithrombotic agents
08/12/1999WO1999040071A1 Urocanic acid derivatives
08/12/1999WO1999040064A1 Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament
08/12/1999WO1999028304A3 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
08/12/1999DE19805431A1 Heteroaromatische Oligoamide als Affinitätsliganden Heteroaromatic oligoamides as affinity ligands
08/12/1999CA2319555A1 Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament
08/12/1999CA2319494A1 5-membered heterocyclic condensed benzoderivatives, the preparation thereof and their use as pharmaceuticals
08/12/1999CA2319060A1 Urocanic acid derivatives
08/12/1999CA2318977A1 Derivatives of benzoxadiazoles, benzothiadiazoles, benzotriazoles and quinoxalines
08/12/1999CA2317017A1 Sulfonamide derivatives, their production and use
08/11/1999EP0934935A1 Heterocyclic substituted phenyl compounds, process and intermediates for their preparation and their use as fungicides and pesticides
08/11/1999EP0934931A2 3-Benzylidene-2-indolinones and their analogues as tyrosine kinase activity modulators