Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
12/2004
12/29/2004WO2004112793A1 Guanidino-substituted quinazolinone compounds as mc4-r agonists
12/29/2004WO2004112719A2 Chemical compounds
12/29/2004WO2004112709A2 Inhibitors of cathepsin s
12/29/2004WO2004112704A2 Substituted piperidine compounds and methods of their use
12/29/2004WO2004086050A3 Labelling agents for mass spectrometry comprising tertiary amines
12/29/2004WO2004076412A3 Aminoheteroaryl compounds as protein kinase inhibitors
12/29/2004WO2004066951A3 Quinoline derivatives as nk-2 and nk-3 receptor antagonists
12/29/2004WO2003103671A8 Basic non-peptide bradykinin antagonists and pharmaceutical compositions therefrom
12/29/2004WO2003102097A8 The hydrochloride of (s)-(+)-3-[1-[2-(1-acetyl-2,3-dihydro-1h-indol-3-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl]-6-chloro-1h-indole
12/29/2004WO2003099793A8 1,2-azole derivatives with hypoglycemic and hypolipidemic activity
12/29/2004EP1491541A1 Pyridazinone aldose reductase inhibitors
12/29/2004EP1491540A1 Pyridazinone aldose reductase inhibitors
12/29/2004EP1491539A1 1-n-aminobenzimidazole derivatives
12/29/2004EP1491533A2 Quinoline-and naphthalenecarboxamides, pharmaceutical compositions thereof and their use as calpain inhibitors
12/29/2004EP1491532A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetyloholine receptors
12/29/2004EP1491212A1 Remedy for sleep disturbance
12/29/2004EP1490362A2 (homo)piperazine substituted quinolines for inhibiting the phosphorylation of kinases
12/29/2004EP1490358A1 6-(4-substituted-anilino)pyrimidine derivatives, method for the preparation thereof and antiviral pharmaceutical composition comprising the same
12/29/2004EP1490355A1 Indolylmaleimide derivatives
12/29/2004EP1490353A1 Method for manufacture of sertindole
12/29/2004EP1490352A1 Synthesis of piperidine and piperazine compounds as ccr5 antagonists
12/29/2004EP1490344A2 Anxiolytic agents with reduced sedative and ataxic effects
12/29/2004EP1490343A1 New aryl imidazoles and related compounds as c5a receptor modulators
12/29/2004EP1490341A1 Novel adamantane derivatives
12/29/2004EP1490340A1 Heteroaromatic urea derivatives as vr-1 receptor modulators for treating pain
12/29/2004EP1490336A1 Piperidine or 8-aza-bicyclo(3.2.1)oct-3-yl derivatives useful as modulators of chemokine receptor activity (especially ccr5)
12/29/2004EP1490334A1 Phthalimido derivatives as inhibitors of monoamine oxidase b
12/29/2004EP1490067A2 Use of tyrosine kinase inhibitors for treating substance use disorders
12/29/2004EP1490065A1 Benzylimidazolyl substituted 2-quinolinone and quinazolinone derivatives for use as farnesyl transferase inhibitors
12/29/2004EP1490064A1 Substituted pyridinones as modulators of p38 map kinase
12/29/2004EP1490062A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
12/29/2004EP1490056A1 N-'4-(2-imino-pyrrolidin-1-yl)phenyl)-acetamide and corresponding piperidine derivatives as factor xa inhibitors for the treatment of thrombo-embolic diseases
12/29/2004EP1490054A2 Hemiasterlin derivatives and uses thereof in the treatment of cancer
12/29/2004EP1490043A2 Spirocyclic amides as cannabinoid receptor modulators
12/29/2004EP1373259B1 Pyridazinone aldose reductase inhibitors
12/29/2004EP1285917B1 Process for producing carbostyril derivative
12/29/2004EP1282612B1 Alkynyl phenyl heteroaromatic glucokinase activators
12/29/2004EP1257539B1 Amino pyrazole derivatives useful for the treatment of obesity and other disorders
12/29/2004EP1233769A4 Novel compounds
12/29/2004EP1230224B1 Substituted 5-benzyl-2,4-diaminopyrimidines
12/29/2004EP1226138B1 Fab i inhibitors
12/29/2004EP1226136B1 Tyrosine kinase inhibitors
12/29/2004EP1216234B1 Mediators of hedgehog signaling pathways, compositions and uses related thereto
12/29/2004EP1177178B1 Heterocyclically substituted benzimidazoles, the production and application thereof
12/29/2004EP1176140B1 Amide compounds and medicinal use thereof
12/29/2004EP1123274B1 Substituted phenyl derivatives, their preparation and use
12/29/2004EP1119551B1 Naphthalenecarboxamides as tachykinin receptor antagonists
12/29/2004EP1056729B1 N-[(substituted five-membered di- or triaza diunsaturated ring)carbonyl]guanidine derivatives for the treatment of ischemia
12/29/2004EP0934303B1 Compounds useful for inhibition of farnesyl protein transferase
12/29/2004EP0929545B1 Tricyclic inhibitors of farnesyl protein transferase
12/29/2004CN1558934A Water-color ink
12/29/2004CN1558933A Novel anthrapyridone compounds, water-base magenta ink compositions, and ink-jet recording process
12/29/2004CN1558907A Substituted imidazoles as dual histamine h1 and h3 agonists or antagonists
12/29/2004CN1558904A Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same
12/29/2004CN1558902A Insecticidal and acaricidal 3-substituted pyrazoles
12/29/2004CN1558898A Antiviral agent
12/29/2004CN1558897A Antidiabetic agents
12/29/2004CN1558764A Substituted urea neuropeptide Y Y5 receptor antagonists
12/29/2004CN1558761A Substituted benzimidazole compounds and their use for the treatment of cancer
12/29/2004CN1558759A 病毒聚合酶抑制剂 Viral polymerase inhibitors
12/29/2004CN1558758A Novel pyrroles having hypolipidemic hypocholesteremic activities, process for their preparation and pharmaceutical compositions containing them and their use in medicine
12/29/2004CN1558719A Nicotinic acid-heterocyclyl-amides and analogous pyrimidine derivatives serving as pesticides
12/29/2004CN1557808A 3-substituted piperazine triadimenol antifungal compounds and their salts
12/29/2004CN1182135C Method for producing heterocyclic compounds
12/29/2004CN1182134C Quinolinyl-piperidin-4-ylidene-methyl-benzamide derivatives for treatment of pain
12/29/2004CN1182123C Substituted bicyclic derivatives useful as anticancer agents
12/29/2004CN1182114C Piperazine derivatives used as CCR5 antagonist
12/29/2004CA2530461A1 6-arylamino-5-cyano-4-pyrimidinones as pde9a inhibitors
12/29/2004CA2530058A1 Mucin synthesis inhibitors
12/29/2004CA2529524A1 Substituted piperidine compounds and methods of their use
12/29/2004CA2529250A1 Chinazoline derivatives as aurora kinase inhibitors
12/29/2004CA2529161A1 Quinolyl amide derivatives as ccr-5 antagonists
12/29/2004CA2529154A1 Novel compounds that modulate ppar.gamma. type receptors, and use thereof in cosmetic or pharmaceutical compositions
12/29/2004CA2528538A1 Dual function compounds and uses thereof
12/29/2004CA2524700A1 N-substituted 6,8-dialkoxy-1,2,3,4-tetrahydro-1h-isoquinoline as potassium channels modulators
12/29/2004CA2523015A1 Guanidino-substituted quinazolinone compounds as mc4-r agonists
12/28/2004US6835832 Catalytic hydrogenation
12/28/2004US6835744 3,3-substituted indoline derivatives
12/28/2004US6835741 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
12/28/2004US6835739 Benzamides and related inhibitors of factor Xa
12/28/2004US6835737 Quinoline inhibitors of cGMP phosphodiesterase
12/28/2004US6835731 Chemokine receptor binding heterocyclic compounds
12/28/2004US6835728 Drug combination for the treatment of depression and related disorders comprising mirtazapine
12/28/2004CA2281426C Substituted indole compounds as anti-inflammatory and analgesic agents
12/28/2004CA2105923C 7-isoindolinyl-quinolone derivatives and 7-isoindolinyl-naphthyridone derivatives
12/23/2004WO2004111193A2 Prodrugs of mitotic kinesin inhibitors
12/23/2004WO2004111040A1 Heteroaryl-substituted imdazole derivatives as glutamate receptor antagonists
12/23/2004WO2004111038A1 5,6-bis (4-chlorophenyl)-n-piperidin1-yl-3-(piperidin-1-yl-carbonyl)pyrazine-2-carboxamide
12/23/2004WO2004111036A1 4- (heterocyclyl- fused phenyl)- 3- (phenyl or pyrid -2- yl) pyrazoles as inhibitors of the alk-5- receptor
12/23/2004WO2004111035A1 Bicyclic indolyl derivatives and methods of their use as serotonergic agents
12/23/2004WO2004111034A1 3-substituted 5,6-diaryl-pyrazine-2-carboxamide and -2-sulfonamide derivatives as cb1 modulators
12/23/2004WO2004111033A1 2-substitued 5, 6-diaryl-pyrazine derivatives as cb1 modulator.
12/23/2004WO2004111032A1 Substituted piperidine carbamates for use as inhibitors of hormone sensitive lipase
12/23/2004WO2004111031A1 Pyridinyl carbamates as hormone-sensitive lipase inhibitors
12/23/2004WO2004111030A1 Method for preparing fused oxazinones
12/23/2004WO2004111029A2 Process for preparing 2-[(pyridinyl)methyl]sulfinyl-substituted benzimidazoles and novel chlorinated derivatives of pantoprazole
12/23/2004WO2004111014A1 Pyrimidine derivatives as modulators of atp-binding cassette transporters
12/23/2004WO2004111013A1 Hepatitis c virus inhibitors
12/23/2004WO2004111009A1 Fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor
12/23/2004WO2004111007A1 1-aryl-4-(aryloxycarbonyl)-piperazine derivatives for use as inhibitors of hormone sensitive lipase