Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
01/2005
01/18/2005US6844446 Catalysts containing per-ortho aryl substituted aryl or heteroaryl substituted nitrogen donors
01/18/2005US6844439 Process for the preparation of imidazole compounds
01/18/2005US6844367 Benzamides and related inhibitors of factor Xa
01/18/2005US6844357 Anticarcinogenic agents
01/18/2005US6844350 Febrifugine, isofebrifugine and method for producing the same
01/18/2005US6844349 Salt forms of E-2-methoxy-N-(3-{4-[3 methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide and method of production
01/18/2005US6844347 Substituted 4-amino-2aryl-pyrimidines, their production and use and pharmaceutical preparations containing same
01/18/2005US6844342 Heterocyclic substituted 2-methyl-benzimidazole antiviral agents
01/18/2005US6844338 Piperidyindoles as serotonin receptor ligands
01/18/2005US6844335 2-amino-3-(alkyl)-pyrimidone derivatives as GSK3.β.inhibitors
01/18/2005CA2142463C Herbicidal pyrazolyloxy-picolinamides
01/16/2005WO2005000281A2 Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
01/16/2005CA2529436A1 Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
01/13/2005WO2005003127A1 Bicyclic heteroaromatic derivatives as modulators of cxcr3 function
01/13/2005WO2005003120A2 Metabolites of tricyclic amides useful for inhibition of g-protein function and methods of treatment of proliferative diseases
01/13/2005WO2005003119A1 2,4-bis(trifluoroethoxy)pyridine compound and medicine containing the same
01/13/2005WO2005003118A1 Amide-substituted 1,2,4-triazin-5(2h)-ones for the treatment of chronically inflammatory diseases
01/13/2005WO2005003117A1 Imidazole derivatives iii
01/13/2005WO2005003103A2 2, 4, 6-tri-substituted 6-membered heterocycles and their use in the treatment of neurodegenerative diseases
01/13/2005WO2005003102A1 Methods of preparation of dehydro-diketopiperazines in liquid phase or of solid supported phase
01/13/2005WO2005003101A2 Pyrazine and pyridine derivatives as rho kinase inhibitors
01/13/2005WO2005003100A2 4-arylamino-quinazolines as activators of caspases and inducers of apoptosis
01/13/2005WO2005003099A2 Pyrimidines useful as modulators of voltage-gated ion channels
01/13/2005WO2005003097A1 Cis-2,4,5-triaryl-imidazolines
01/13/2005WO2005003086A2 Sulfonic acid derivatives of polycyclic dyes used for analytical applications
01/13/2005WO2005002577A1 Dual nk1/nk3 antagonists for treating schizophrenia
01/13/2005WO2005002575A1 Cis-imidazolines as mdm2 inhibitors
01/13/2005WO2005002574A1 Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
01/13/2005WO2005002552A2 Benzimidazole derivatives and their use as protein kinases inhibitors
01/13/2005WO2005002503A2 Asymmetric benzimidazoles and related compounds as potassium channel modulators
01/13/2005WO2004099192A3 Heterocycle substituted carboxylic acids as inhibitors of protein tyrosine phosphatase-1b
01/13/2005WO2004092130A3 N-containing heteroaromatic compounds as modulators of ppars and methods of treating metabolic disorders
01/13/2005WO2004082623A3 Substituted piperidine compounds
01/13/2005WO2004078744A3 Urea derivatives and their use as vanilloid receptor antagonists in the treatment of pain
01/13/2005WO2004072047A8 Indoles, benzimidazoles or naphhimidazoles as histone deacetylase (hdac) inhibitors
01/13/2005WO2004064764A3 Substituted alkyl amido piperidines
01/13/2005WO2004050035A3 Benzimidazoles and analogs thereof as antivirals
01/13/2005WO2004022055B1 1, 4, 5-substituted 1, 2-dihydro-pyrazol-3-one and 3-alkoxy-1h-pyrazole derivatives s tnf-alpha and interleukin lowering agents for the treatment of inflammations
01/13/2005US20050010048 Aza-and polyaza-naphthalenly ketones useful as hiv integrase inhibitors
01/13/2005US20050010031 2-(S)-{3-(S)-allyl-4-[2-(R)-amino-3-(4-fluorophenyl)propionyl]-2-oxo-piperazin-1-yl}-N-methyl-3-naphthalen-2-yl-propionamide for example; various diseases and disorders including controlling appetite and treating diabetes
01/13/2005US20050009898 New substituted indolinones, their manufacture and their use as medicaments
01/13/2005US20050009894 Benzimidazole derivatives and their use as KDR kinase protein inhibitors
01/13/2005US20050009890 E.g., 1) (2R)-N-(4-phenoxybenzyl)-3-cyclohexylmethylthio-2-((4R)-3-methoxymethylcarbonylthiazolidin-4-ylcarbonylamino)propanamide; treatment of cerebral infarct, transient ischemic attack, encephalomyelopathy, spinal angiopathy, hypertension with stress, neurosis, epilepsy, asthma, pollakiuria, and pain
01/13/2005US20050009889 Synergistic fungicide compositions containing at least one n-(2-pyridinyl) 1-3-pyridinecarboxamide derivative and one or more further fungicides useful for controlling fungal plant diseases
01/13/2005US20050009883 Fipronil and chloropyridine or chlorothiazole derivatives as antagonists of nicotinic acetylcholine receptors; protection of industrial materials and plants.
01/13/2005US20050009879 N-substituted-2-oxodihydropyridine derivatives
01/13/2005US20050009878 4-(1,2-Dimethyl-1H-imidazol-4-ylethynyl)-2-methyl-pyridine compounds; treating chronic neurological disorders
01/13/2005US20050009876 Indazole compounds, compositions thereof and methods of treatment therewith
01/13/2005US20050009874 Tetrahydropyridin or piperidino heterocyclic derivatives
01/13/2005US20050009871 Ubiquitin ligase inhibitors
01/13/2005US20050009870 3-(amino)sulfonylamino-substituted, e.g., N-(1,6-Dibenzyl-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)-benzenesulfonamide and N-(1-Benzyl-2-oxo-6-(thiophen-3-yl)-1,2,3,4-tetrahydroquinolin-3-yl)benzenesulfonamide; eating, metabolic, obesity, cognitive, neurological, pain, inflammatory and psychiatric disorders
01/13/2005US20050009867 Quinoline derivatives and their use as tyrosine kinase inhibitors
01/13/2005US20050009864 Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them
01/13/2005US20050009853 Pyrimidine derivatives for the treatment of abnormal cell growth
01/13/2005US20050009844 Inhibitors of p38
01/13/2005US20050009841 N-phenylamides and ureas containing both a pyridine, pyrazine, pyrimidine, 1,2,4-triazine, imidazone or oxazine ring and a piperidine or 3,8-diazabicyclo[3.2.1]octane ring, e.g., N-(4-tert-butylphenyl)-3'-chloro-3,6-dihydro-2H-1,2'-bipyridine-4-carboxamide
01/13/2005US20050009840 2-amino- pyridines and pyrazines additionally substituted witn one or more carbocyclic or heterocyclic groups, e.g., 4-[6-amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-phenol, for treating many kinds of cancer
01/13/2005US20050009839 Novel azoles having an insecticidal action
01/13/2005US20050009838 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
01/13/2005US20050009834 E.g., 3-(2-chloro-6-fluorophenyl)-1-[4-(3,5-dichloropyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole and 3-(3-chloropyridin-2-yl)-1-[4-(3-chloro-5-trifluoromethylpyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole; for use as pesticides, especially insecticides and acaricides
01/13/2005US20050009829 1-Substituted 2-carboxamide derivatives of fused ring imidazoles, e.g., -[5-(5-Chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-1H-benzoimidazole-2-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide
01/13/2005US20050009818 Therapeutic heterocyclic compounds
01/13/2005US20050009817 Substituted heteroaryls
01/13/2005US20050009816 Potassium channel modulators
01/13/2005US20050009815 4-Aminoquinoline compounds
01/13/2005US20050009812 Remedies for stress diseases comprising mitochondrial benzodiazepine receptor antagonists
01/13/2005US20050009809 Acridine derivatives and their use as medicaments
01/13/2005US20050009808 Azabicyclo compound matrix metalloprotease inibitor and skin preparation
01/13/2005US20050009807 Preventing the deposits of amyloid protein, treating neurodegenerative disease, Alzheimer's disease and Down's Syndrome; {[carbamoyl]cycloalkyl}-N-(2-oxo-5-phenyl((S)-3H-benzo[f]1,4-diazepin-3-yl))- or (2-oxo-5-phenyl((S)-3H-benzo[f]1,4-diazepin-3-yl))-carboxamide
01/13/2005US20050009784 2-(p-oxyphenyl)-6-oxyquinolines, e.g., 2-(3-Fluoro-4-hydroxyphenyl)-4-phenylquinolin-6-ol
01/13/2005US20050009755 (74)(3S)-3-amino-1-(1-benzyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)-5-methyl-2-heptanone for example; cysteine protease inhibitors; treating bone resorption diseases such as osteoporosis
01/13/2005US20050009054 Compounds having a fused, bicyclic moiety for binding to the minor groove of dsDNA
01/13/2005DE10328479A1 6-Arylamino-5-cyano-4-pyrimidinone 6-arylamino-5-cyano-4-pyrimidinones
01/13/2005CA2531327A1 Compounds and therapeutical use thereof
01/13/2005CA2531061A1 Pyrimidines useful as modulators of voltage-gated ion channels
01/13/2005CA2531050A1 Pharmaceutical compounds
01/13/2005CA2530886A1 Dual nk1/nk3 antagonists for treating schizophrenia
01/13/2005CA2530816A1 Amide-substituted 1,2,4-triazin-5(2h)-ones for the treatment of chronic inflammatory diseases
01/13/2005CA2530389A1 Pyrazine and pyridine derivatives as rho kinase inhibitors
01/13/2005CA2528119A1 Cis-2,4,5-triaryl-imidazolines
01/13/2005CA2525968A1 Metabolites of tricyclic amides useful for inhibition of g-protein function and methods of treatment of proliferative diseases
01/13/2005CA2525580A1 Asymmetric benzimidazoles and related compounds as potassium channel modulators
01/12/2005EP1496052A1 Novel aminobenzamide derivative
01/12/2005EP1495017A2 Novel heteroaryl alkylamide derivatives useful as bradykinin receptor modulators
01/12/2005EP1495016A2 Heterocyclic compounds and their use as modulators of p38 map kinase
01/12/2005EP1495005A1 Pyrazole compounds as anti-inflammatory and analgesic agents
01/12/2005EP1495003A1 Fredericamycin derivatives
01/12/2005EP1495002A1 Benzamide derivatives useful as histone deacetylase inhibitors
01/12/2005EP1495001A1 Antibacterial agents
01/12/2005EP1494997A1 Substituted aryl amides
01/12/2005EP1494676A1 Fused quinoxaline derivatives as inhibitors of akt activity
01/12/2005EP1494672A1 Aminocarbonyl substituted pyridines, pyridazines, pyrimidines, pyrazines and triazines having antiangiogenic activity
01/12/2005EP1494671A1 1-(4-piperidinyl)benzimidazolones as histamine h3 antagonists
01/12/2005EP1494670A1 Medicine for treating cancer
01/12/2005EP1494668A2 Use of benzimidazole analogs in the treatment of cell proliferation
01/12/2005EP1494667A1 Imidazole compounds as anti-inflammatory and analgesic agents
01/12/2005EP1494663A1 Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin k inhibitors for the treatment of bone loss
01/12/2005EP1494645A2 Method of treating mucus hypersecretion
01/12/2005EP1434773A4 Heteroaryl substituted tetrazole modulators of metabotropic glutamate receptor-5
01/12/2005EP1299383B1 Sulfonyl-pyrrolidine derivatives useful for the treatment of neurological disorders