Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
02/2005
02/02/2005EP1501807A1 Sulfonylquinoxalone acetamide derivatives and related compounds as bradykinin antagonists
02/02/2005EP1501805A1 Substituted pyrazolyl compounds for the treatment of inflammation
02/02/2005EP1501803A2 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
02/02/2005EP1501801A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as vla-4 inhibitors
02/02/2005EP1501800A1 Bombesin antagonists
02/02/2005EP1501798A2 SULFONYLAMINOVALEROLAC TAMS AND DERIVATIVES THEREOF AS FACTOR Xa INHIBITORS
02/02/2005EP1501797A1 3-substituted amino-1h-indole-2-carboxylic acid and 3-substituted amino-benzo[b]thiophene-2-carboxylic acid derivatives as interleukin-4 gene expression inhibitors
02/02/2005EP1501796A1 3-substituted amino-1h-indole-2-carboxylic acid and 3-substituted amino-benzo[b]thiophene-2-carboxylic acid derivatives as interleukin-4 gene expression inhibitors
02/02/2005EP1501795A1 Cinnamic acid amides
02/02/2005EP1501514A2 Protein kinase modulators and methods of use
02/02/2005EP1501513A2 Compositions and methods for combating lower urinary tract dysfunctions with delta opioid receptor agonists
02/02/2005EP1501508A1 Inhibitors of histone deacetylase
02/02/2005EP1501504A1 1-substituted imidazole derivatives as nos inhibitors
02/02/2005EP1501467A2 Heterocyclo inhibitors of potassium channel function
02/02/2005EP1501360A1 2,6 substituted pyridine-3-carbonyl derivatives serving as plant protection agents having herbicidal action
02/02/2005EP1414814B1 6-aryl-4-aminopicolinates and their use as herbicides
02/02/2005EP1379587B1 Long chain hindered amines and compositions stabilized therewith
02/02/2005EP1303506B1 6-heteroarylphenanthridines
02/02/2005EP1292591B1 Substituted bicyclic derivatives for the treatment of abnormal cell growth
02/02/2005EP1286955B1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides
02/02/2005EP0828754B1 Dipeptides which promote release of growth hormone
02/02/2005CN1575291A Derivatives of 4-(thio- or selenoxanthene-9-ylidene)-piperidine or acridine and its use as a selective 5-ht2b receptor antagonist
02/02/2005CN1575290A Pyrimidine derivatives and pharmaceutical compositions containing that compounds
02/02/2005CN1575284A Substituted triazole diamine derivatives as kinase inhibitors
02/02/2005CN1575283A Piperazine derivatives with CCRI receptor antagonist activity
02/02/2005CN1575177A Cxcr3 antagonists
02/02/2005CN1575176A Process for making substituted pyrazoles
02/02/2005CN1575174A Pharmaceutically active isoindoline derivatives
02/02/2005CN1575172A Substituted ideno[1, 2-c]isoquinoline derivatives and methods of use thereof
02/02/2005CN1575171A Novel anti-diabetic agents
02/02/2005CN1572792A Pyrazolo [4, 3-d] pyrimidine derivatives
02/02/2005CN1572299A Agents for improving excretory potency of urinary bladder
02/02/2005CN1187342C Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
02/02/2005CN1187338C 5-phenyl-pyrimidine derivatives
02/02/2005CN1187333C Certain substituted caprolactams, pharmaceutical compositions containing them and their use in treating tumors
02/02/2005CN1187331C Esters of 3-hydroxy-piperidinemethanol derivatives, pharmaceutical composition containing same and their preparation method and uses
02/02/2005CN1187326C Novel compounds
02/02/2005CN1187325C Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
02/01/2005US6849740 Antimicrobial quinolones, their compositions and uses
02/01/2005US6849739 N-heterocyclic derivatives as NOS inhibitors
02/01/2005US6849732 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses, and methods and intermediates useful for their preparation
02/01/2005US6849713 Topisomerase inhibitor
02/01/2005US6849660 Antimicrobial biaryl compounds
02/01/2005US6849653 Substituted pyrazolyl benzenesulfamide compounds for the treatment of inflammation
02/01/2005US6849648 Phenylene alkyne matrix metalloproteinase inhibitors
02/01/2005US6849647 Amide compounds and medications containing the same technical field
02/01/2005US6849644 For example, 7-(Indole-1-sulfonyl)-1,2,3,4-tetrahydro-isoquinoline; treatment of depression, anxiety, Alzheimers disease, age related cognitive decline, Attention Deficit Disorder
02/01/2005US6849643 Indazolyl-substituted pyrroline compounds as kinase inhibitors
02/01/2005US6849639 Anticancer agents, antiinflamatory agents, osteoporosis, atherosclerosis
02/01/2005US6849636 Useful for treatment of noninsulin-dependent diabetes, hyperglycemia, obesity, insulin resistance, dyslipidemia, hyperlipidemia, hypertension, Metabolic Syndrome
02/01/2005US6849633 Pyrazole derivative, production process thereof, and pest control agent containing the same as active ingredient
02/01/2005US6849631 Semicarbazides and their uses
02/01/2005US6849629 Heteroaromatic substituted sulfonyl or sulfoxide or thio-pyridazinone derivatives, useful for treating diabetic complications and cardiovascular disorders
02/01/2005US6849625 Use in manufacture of a medicament for use as an anti-invasive agent in containment and/or treatment of solid tumor disease
02/01/2005US6849622 May be useful for the prophylaxis and treatment of diabetes, particularly type 2 diabetes, and for prophylaxis and treatment of other diseases induced or exacerbated by impaired glucose tolerance
02/01/2005US6849621 Treating: allergy, allergy-induced airway responses, congestion, hypotension, cardiovascular disease, hypotension, diseases of the GI tract, hyper and hypo motility and acidic secretion of the gastrointestinal tract, obesity, sleep
02/01/2005US6849367 Photoconductive layer containing azo compound; electrostaticlatent image
02/01/2005US6849116 Containing 1 or 2 phthalimido groups
02/01/2005CA2166326C Pyridazinone derivatives
01/2005
01/27/2005WO2005007652A2 Substituted quinolin-4-ylamine analogues
01/27/2005WO2005007648A2 Biaryl piperazinyl-pyridine analogues
01/27/2005WO2005007647A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
01/27/2005WO2005007646A1 Substituted heterocyclic diarylamine analogues
01/27/2005WO2005007645A1 Substituted 4-amino-1-benzylpiperidine compounds
01/27/2005WO2005007643A1 Novel acridine derivatives and use thereof as medicaments
01/27/2005WO2005007642A2 Novel azaheterocyclic amides useful for treating pain
01/27/2005WO2005007641A1 2-pyridine alkyne derivatives useful for treating pain
01/27/2005WO2005007629A1 Piperidine or 8-aza-bicyclo[3.2.1]oct-3-yl derivatives useful as modulators of chemokine receptor activity
01/27/2005WO2005007628A1 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
01/27/2005WO2005007625A2 Heterocyclic amides with anti-tuberculosis activity
01/27/2005WO2005007621A2 Ubiquitin ligase inhibitors
01/27/2005WO2005007164A1 Pyrimidine-2,4-dione derivatives as gonadotropin-releasing hormone receptor antagonists
01/27/2005WO2005007157A1 Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases
01/27/2005WO2005007111A2 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
01/27/2005WO2004101512A3 Naphthyridine integrase inhibitors
01/27/2005WO2004100949A3 Solid-state forms of 5-(difluoromethoxy)-2-((3,4-dimethoxy-2-pyridinyl)methyl)sulfinyl)-1h-benzimidazole (pantoprazole) sodium aqua complexes
01/27/2005WO2004099130A3 1,2-diarylimidazoles useful as inhibitors of cox
01/27/2005WO2004098518A3 Pyrazole-amide compounds useful as kinase inhibitors
01/27/2005WO2004087647A3 4-substituted quinolein derivatives with antimicrobial activity
01/27/2005WO2004085418A3 Xanthones, thioxanthones and acridinones as dna-pk inhibitors
01/27/2005WO2004069794B1 New arylpiperazinyl compounds
01/27/2005WO2004064972A3 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
01/27/2005US20050020849 via non-racemic cinchona-alkaloid-type catalyst (quinidine) for addition of nucleophile
01/27/2005US20050020836 For therapy of hyperproliferative disorder in a mammal
01/27/2005US20050020832 For therapy of atherosclerosis
01/27/2005US20050020659 Substituted pyrazole derivatives and related compounds as bradykinin B1 receptor antagonists
01/27/2005US20050020652 For example, 2-(4-{2-[1-(4-tert-Butyl-benzyl)-3-methyl-2-oxo-imidazolidin-4-yl]-ethoxy}-2-methyl-phenoxy)-2-methyl-propionic acid, 2-(4-{3-[1-(4-tert-Butyl-benzyl)-3-methyl-2-oxo-imidazolidin-4-yl]-propyl}-2-methyl-phenoky)-2-methyl-propionic acid; for treating diabetes mellitus
01/27/2005US20050020648 "PGI2-preferring" (IP) receptors; p-(imidazolin-2-ylamino-optional alkyl)phenyl p'-substituted ethers or sulfides, e.g., 4,5-Dihydro-1H-imidazol-2-yl)-[4-(4-isopropoxy-phenylsulfanyl)-phenyl]-amine, used to induce hyperalgesia
01/27/2005US20050020644 Bicyclic fused pyridinyl amides and advantagesous compositons thereof for use as fungicides
01/27/2005US20050020638 Method of stabilizing lansoprazole
01/27/2005US20050020636 Antitumor agents
01/27/2005US20050020629 Pain management
01/27/2005US20050020626 9- or 10-membered bicyclic N-heteroaryl carboxamides, N-substituted with 4-[2-(o-methylthiophenoxy)pyridin-3-ylcarbonylamino]cyclohexyl groups, e.g., Pyrazolo[1,5-a]pyridine-2-carboxylic acid(4-{[5-fluoro-2-(3-methylsulfanyl-phenoxy)-pyridine-3-carbonyl]-amino}-cyclohexyl)-amide; respiratory disorders
01/27/2005US20050020625 Blocking starting compound with metal alkoxide; anticancer agents
01/27/2005US20050020606 2,4-Bis (trifluoroethoxy)pyridine compound and drug containing the compound
01/27/2005US20050020605 Quinolyl amide derivatives as CCR-5 antagonists
01/27/2005US20050020604 5-HT receptor ligands and uses thereof
01/27/2005US20050020602 Bone disorders; reduction concentration of parathyroid hormone in blood
01/27/2005US20050020601 Novel pyrazinones as CRF1 receptor antagonists
01/27/2005US20050020597 Attention deficit disorders; hyperactivity; post-trauma stress disorders; anxiolytic agents; obsessive compulsive disorders; analgesics; Parkinson's disease