Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
02/2005
02/17/2005US20050038072 Nitrogeneous cyclic ketone derivative, process for producing the same, and use
02/17/2005US20050038069 Tumor necrosis factor antagonist; antiinflammatory agents; such as 2-Cyclopropyl-4-(3,5-dimethyl-4-pyridylmethoxy)-7-methoxy-3H-benzimidazole
02/17/2005US20050038067 A compound with azo containing mono and a bicyclic rings attached with an aryl or heteroaryl ring; both therapeutic and diagnostic
02/17/2005US20050038060 Spiropoperidine compounds as ligands for orl-1 receptor
02/17/2005US20050038050 Therapeutic treatment of autoimmune disease, transplant rejection, rheumatoid arthritis, by administering 4-(6-chloro-2,3-methylenedioxyanilino)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-tetrahydropyran-4-yloxyquinazoline
02/17/2005US20050038041 Fungicide for agriculture, horticulture
02/17/2005US20050038040 Corticotropin releasing factor antagonist; antiinflammatory agents; drug abuse; analgesics; antihistamines; skin disorders; neurodegenerative disease; eating disorders;eating disorders; antiepileptic agents; cardiovascular disorders
02/17/2005US20050038037 N-(naphth-2-ylaminocarbonylacetyl)- or N-(naphth-2-ylcarbonylamino- acetyl)- piperazine derivatives, e.g., 2-[((4-(ethoxycarbonyl)piperazin-1-yl)carbonylmethyl)carbonyl]aminonaphthalene; useful as antithrombotic agents
02/17/2005US20050038035 Heterocyclic amide compounds as apolipoprotein b inhibitors
02/17/2005US20050038033 use in treating respiratory system disorders such as asthma, incipient asthma and wheezy infant syndrome, chronic or acute bronchoconstriction, chronic bronchitis, small airways obstruction, emphysema, chronic eosinophilic pneumonia, chronic obstructive pulmonary disease, allergies
02/17/2005US20050038032 Quinoxaline compounds
02/17/2005US20050038031 Novel bicyclic urea derivatives useful in the treatment of cancer and other disorders
02/17/2005US20050038027 Melanocortin-4 receptor agonists; obesity, type II diabetes; such as N-(2-(2-(2,4-dichlorophenyl)ethyl)-1-oxo-2,3-dihydro-1H-isoindol-5-yl) -3-methyl-N'-(2,6,6-trimethylbicyclo(3.1.1)hept-3yl)piperazine-1-carboximidamide
02/17/2005US20050038023 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
02/17/2005US20050038016 Arylamine-substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonists
02/17/2005US20050038010 Substituted heterocyclic compounds and methods of use
02/17/2005US20050038002 Bactericides; antitumor agents; moderators of gene expression; viricides; parasiticides; malaria therapy
02/17/2005US20050037925 Mixture with other herbicides
02/17/2005DE10328533A1 New 6-amino-substituted indolinone derivatives, useful e.g. for treating tumours and angiogenesis, are inhibitors of receptor tyrosine kinases
02/17/2005DE10326918A1 Substituierte Alkylamide Substituted alkyl amides
02/17/2005CA2554566A1 Condensed pyramidine compounds as inhibitors of voltage-gated ion channels
02/17/2005CA2539227A1 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
02/17/2005CA2534975A1 Anthelmintic and insecticide pyrimidine derivatives
02/17/2005CA2534905A1 Pyridyl piperazinyl ureas
02/17/2005CA2534811A1 Quinazoline derivatives as angiogenesis inhibitors
02/17/2005CA2534528A1 3-(indol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones,3-(benzimidazol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones, and 3-(indolin-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones; their preparationand use as modulators of apoptosis
02/17/2005CA2534496A1 Pyrimidylpyrrole derivatives active as kinase inhibitors
02/17/2005CA2534494A1 Pyrrole-based hmg-coa reductase inhibitors
02/17/2005CA2534422A1 Quinazoline derivatives as inhibitors of vegf receptor tyrosine kinases
02/17/2005CA2534240A1 Treatment for alzheimer's disease and related conditions
02/17/2005CA2534101A1 2-`4-(hydroxymethyl-phenylamino) -piperidine-1-yl!-n- (9h-carbazol-3-yl) - acetamine derivatives and related compounds as neuropeptide y5 (npy5) ligands for the treatment of obesity
02/17/2005CA2534096A1 2-`4(phenylamino)-piperidin-1-yl!-n-phenyl-acetamine derivatives and related compounds as neuropeptide y5 (npy5) ligands for the treatement of obesity
02/17/2005CA2534057A1 Novel gamma-secretase inhibitors
02/17/2005CA2533996A1 1-sulfonylindole derivatives, their preparation and their use as 5-ht6 ligands
02/17/2005CA2533976A1 Indol-5-yl sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
02/17/2005CA2533698A1 Lanthanide complexes preparation and uses thereof
02/17/2005CA2533433A1 Novel n-substituted indolyl-3-glyoxylic acid amides, use thereof as a medicament, and method for the production thereof
02/17/2005CA2533335A1 Substituted lactams and their use as anti-cancer agents
02/17/2005CA2533182A1 Dry syrup containing loratadine
02/17/2005CA2532910A1 4,5-dihydro-imidazole as p2x7 ion channel blockers
02/17/2005CA2532452A1 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors
02/16/2005EP1506967A1 Dipeptidyl peptidase inhibitors
02/16/2005EP1506966A2 Process for the preparation of tetrasubstituted imidazole derivatives and novel crystaline structures thereof
02/16/2005EP1506962A2 Nitrogen-containing aromatic heterocycles
02/16/2005EP1506960A1 Indole compounds as inhibitors of tubulin polymerisation for the treatment of angiogenesis-related disorders
02/16/2005EP1506779A1 (3-(4-(Pyridin-2-ylamino)-butyryl)-2,3,4,4a,9,9a-hexahydro-1H-3-aza-fluoren-9-yl)-acetic acid derivatives and related tricyclic indanyls as alphaVbeta3 and alphaVbeta5 integrin inhibitors for the treatment of cancer and unstable angina
02/16/2005EP1506189A1 Pyrrole derivatives as inhibitors of erk2 and uses thereof
02/16/2005EP1506188A1 Process for the preparation of a hydrate of an anthranilic acid derivative
02/16/2005EP1506187A1 2-thio-substituted imidazole derivatives and their use in pharmaceutics
02/16/2005EP1506186A1 Substituted heterocyclic compounds and methods of use
02/16/2005EP1506185A1 Novel compounds and their use
02/16/2005EP1506176A1 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
02/16/2005EP1506175A1 N-substituted tricyclic 3-aminopyrazoles as pdgf receptor inhibitors
02/16/2005EP1506174A2 Opioid and opioid-like compounds and uses thereof
02/16/2005EP1506166A1 Aminotetralin-derived urea modulators of vanilloid vr1 receptor
02/16/2005EP1506040A2 Selective inos inhibitors for the treatment of respiratory diseases and conditions
02/16/2005EP1505973A2 Methods and compositions using immunomodulatory compounds for treatment and management of cancers and other diseases
02/16/2005EP1505966A1 1,1-disubstituted cycloalkyl derivatives as factor xa inhibitors
02/16/2005EP1505963A1 Hepatitis c virus inhibitors
02/16/2005EP1505945A2 Substituted cycloalkyl p1' hepatitis c virus inhibitors
02/16/2005EP1281709B1 Novel heterocyclic compounds with anti-inflammatory activity
02/16/2005CN1582286A Novel 4-2-furoylaminopiperidines, intermediates in synthesizing the same, process for producing the same and medicinal use of the same
02/16/2005CN1582285A Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (GSK3 inhibitors)
02/16/2005CN1582284A Aminopyrimidines and pyridines
02/16/2005CN1582281A Mch受体拮抗剂 Mch receptor antagonist
02/16/2005CN1582280A 3, 4-di-substituted pyridazinediones as CXC chemokine receptor antagonists
02/16/2005CN1582279A Peroxisome proliferator activated receptor agonists
02/16/2005CN1582277A Amide derivatives as glycogen synthase kinase 3-beta inhibitors
02/16/2005CN1582276A Phenylalanine enamide derivatives
02/16/2005CN1582274A Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade
02/16/2005CN1582271A Inhibitors of integrin alpha v beta 6
02/16/2005CN1582166A Vitronectin receptor antagonist pharmaceuticals for use in combination therapy
02/16/2005CN1580179A White electroluminescent polymer material and its preparing method
02/16/2005CN1580056A Heterocyclic derivatives their preparing methods and uses
02/16/2005CN1580055A Quinolone carboxylic acid derivatives and their salts
02/16/2005CN1189466C New direct chain or cyclic urea, its preparing method and medicinal composition containing them
02/16/2005CN1189465C Vitamin D3 analogs with bis C-20 side chains
02/16/2005CN1189461C Method of producing imidacloprid
02/15/2005US6855823 Selective iGluR5 receptor antagonists
02/15/2005US6855730 3-methylidenyl-2-indolinone modulators of protein kinase
02/15/2005US6855726 Heterocyclic amides such as 3-(1-5-((2R,6S)-2,6-dimethyltetra-hydro-1(2H)-pyridinyl)pentyl-2-oxo-1,2 -dihydro-3-quinolinyl) benzenecarboximidamide, administered as anticoagulants or for prophylaxis of cardiovascular disorders
02/15/2005US6855725 Excitatory amino acid receptor antagonists
02/15/2005US6855722 Substituted indoles and their use as integrin antagonists
02/15/2005US6855717 A 2(2-(4-benzamido-cyclohexyl)ethyl)-1,2,3,4-tetrahydroisoquinol ine derivatives, for use in psychotherapy
02/15/2005US6855716 Dihydropyrimidine compounds and compositions containing the same
02/15/2005US6855715 Drugs such as 1-(3-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4-(4-fluoro-2 -methylsulphonylphenyl)piperazine, used as anticoagulants
02/15/2005US6855714 For therapy of inflammatory, allergic, infectious or autoimmune diseases
02/15/2005US6855713 Benzimidazole derivatives, a process for their manufacture and use as a medicine
02/15/2005US6855710 Antiproliferative agents; antitumor agents
02/15/2005US6855709 Psychological disorders; central nervous system disorders
02/15/2005US6855708 N-arylsulfonyl aza-bicyclic derivatives as potent cell adhesion inhibitors
02/15/2005CA2251927C Cycloalkylaminomethylpyrrolidine derivatives
02/10/2005WO2005012297A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005WO2005012296A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005WO2005012292A1 Gyrase inhibitors and uses thereof
02/10/2005WO2005012290A1 Piperidyl-quinazoline derivatives as tyrosine kinase inhibitors
02/10/2005WO2005012289A1 Novel salt of (r) - pantoprazole
02/10/2005WO2005012288A1 Bicyclic imidazol derivatives against flaviviridae
02/10/2005WO2005012286A1 Substituted pyridones and pyrimidinones with antiinflammatory properties
02/10/2005WO2005012285A1 An improved process for the preparation of moxifloxacin hydrochloride