Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
02/2005
02/08/2005US6852736 Phenoxypropanolamines, preparation and therapeutic use thereof
02/08/2005US6852734 Indole wherein A is an oxygen atom or a nitrogen atom which nitrogen atom is optionally substituted with an alkyl group, and (i) R1 and R2 each stand for a hydrogen atom or an alkyl group, independently, or (ii) R1 and R2 as taken together form
02/08/2005US6852733 Sodium-hydrogen exchanger type 1 inhibitor
02/08/2005US6852732 A tetrahydropyridino or piperidino heterocyclic derivative represented by the formula (I): has a high affinity for CRF receptors and is effective against diseases in which CRF is considered to be involved. (Corticotropin releasing factor
02/08/2005US6852730 Substituted fused pyrazolecarboxylic acid arylamides and related compounds
02/08/2005US6852725 Imidazolyl derivatives
02/08/2005US6852717 Inhibit the release of inflammatory cytokines such as interleukin-1 and tumor necrosis factor; for use in therapy of diseases and pathological conditions involving inflammation such as chronic inflammatory disease
02/08/2005US6852673 Herbicidal pyridine compounds
02/08/2005CA2322900C 2-(hetero)aryl-substituted purin-6-ones as phosphodiesterase inhibitors
02/08/2005CA2130754C Amine derivatives of oxo- and hydroxy-substituted hydrocarbons
02/08/2005CA2112081C Imidazole compounds, their preparation and use
02/08/2005CA2096525C Retroviral protease inhibitors
02/08/2005CA2096409C Retroviral protease inhibitors
02/08/2005CA2096408C Retroviral protease inhibitors
02/03/2005WO2005010001A1 Nicotinamide derivatives useful as pdea4 inhibitors
02/03/2005WO2005009997A1 3,5 disubstituted indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation
02/03/2005WO2005009991A1 Process for producing 1,2,4-triazole compound and intermediate therefor
02/03/2005WO2005009989A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005WO2005009988A1 Heteroaryl-tetrahydropiperidyl compounds useful for treating or preventing pain
02/03/2005WO2005009987A1 Piperidine compounds and pharmaceutical compositions containing them
02/03/2005WO2005009980A1 Substituted pyridin-2-ylamine analogues
02/03/2005WO2005009978A1 2-aminopyrimidine and 2-aminopyridine-4-carbamates for use in the treatment of autoimmune diseases
02/03/2005WO2005009977A1 Substituted pyrimidin-4-ylamina analogues as vanilloid receptor ligands
02/03/2005WO2005009974A1 Imidazole compounds and uses thereof
02/03/2005WO2005009973A1 5-membered heterocycle-based p38 kinase inhibitors
02/03/2005WO2005009967A2 Quinolinone derivatives as inhibitors of c-fms kinase
02/03/2005WO2005009966A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005WO2005009965A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005WO2005009964A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005WO2005009959A1 Piperidine derivatives as ccr5 receptor modulators
02/03/2005WO2005009958A1 Ppar active compounds
02/03/2005WO2005009957A1 Tyrosine kinase inhibitors
02/03/2005WO2005009435A1 Aminopyrazole compounds and use as chk1 inhibitors
02/03/2005WO2005009373A2 Tyrosine kinase inhibitors
02/03/2005WO2004106307A3 Novel imidazole derivatives, the production thereof, and the use of the same as a medicament
02/03/2005WO2004075840A3 Selective non-steroidal glucocorticoid receptor modulators
02/03/2005WO2004072102A3 Benzene acetamide compounds useful as serine protease inhibitors
02/03/2005WO2004054581A3 Cyclohexyl compounds as ccr5 antagonists
02/03/2005WO2003106450A8 Phenylaminopyrimidines and their use as rho-kinase inhibitors
02/03/2005US20050027129 Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
02/03/2005US20050027121 Heterocyclic carboxy amines such as (2R)-1-[3,5-Bis(trifluoromethyl)benzoyl]-4-[4-((3S)-3-ethylmorpholino)-2-butynyl]-2-[(1H-indol-3-yl)methyl]piperazine, used as substance P and neurokinin antagonist for prophylaxis of diseases
02/03/2005US20050027007 Allylamides useful in the treatment of alzheimer's disease
02/03/2005US20050026991 mono-N-substituted amide monohydroxyamide derivatives, e.g., 1-Benzyl-3-(3,4-dichloro-benzyloxy)-1H-pyrrole-2,4-dicarboxylic acid 2-[(1-benzyl-piperidin-4-yl)-amide]4-hydroxyamide, that modulate levels of gene expression in cellular systems, including cancer cells
02/03/2005US20050026990 N-[(3S)-1-hydroxy-2-oxopyrrolidinyl]-N-methyl-4'-(trifluoromethyl)[1,1'-biphenyl]-4-sulfonamide or derivatives to treat Respiratory system disorders; arthritis, and bone disorders
02/03/2005US20050026989 treatment or prophylaxis of cardiovascular disease, metabolic disease, cancerous disease, or fibrotic disease; arrhythmias, life-threatening cardiac ventricular fibrillation, myocardial infarction, angina pectoris; ischemic states of the heart, diabetes
02/03/2005US20050026988 Cyclopenta'b! indole derivatives as spla inhibitors
02/03/2005US20050026985 Such as N-{5-[1-(4-tert-butylphenyl)-3-pyridin-2-yl-1H-pyrazol-5-yl]pentanoyl}tyrosinamide; useful for the treatment of mammalian infertility
02/03/2005US20050026983 Imidazole compounds and uses thereof
02/03/2005US20050026976 Isoindolinone kinase inhibitors
02/03/2005US20050026975 Such as ethyl 4-chloroacetamido-N-(3,4-dichlorobenzyl)indole-2-carboxylate use in the treatment of disease mediated by monocyte chemoattractant protein-1
02/03/2005US20050026968 Heterocyclic amides with anti-tuberculosis activity
02/03/2005US20050026964 4-(2-Fluoro-4-iodoanilino)-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydro-3-pyridinecarboxamide for treating cancer, restenosis, psoriasis, autoimmune disease, atherosclerosis, rheumatoid arthritis, heart failure, chronic pain, neuropathic pain, or osteoarthritis
02/03/2005US20050026963 Pyrazole substituted directly, or by a bridge, with a heteroaryl group containing N adjacent to the point of connection of the heteroaryl useful in the treatment of psychiatric and mood disorders such as, schizophrenia, anxiety, depression, bipolar disorder, circadian rhythm and sleep disorders
02/03/2005US20050026960 3-((mono- or di-fluoro-benzimidazol-2-yl))-5-(4-methyl-5-(ethylaminomethyl)pyrid-3-yl)indazole; inhibitors of cyclin dependent kinases(CDK) for use treating cancer and other proliferative disorders such as retinopathy, rheumatoid arthritis
02/03/2005US20050026956 Carbinols for the treatment of neuropathic dysfunction
02/03/2005US20050026955 Radiolabeled piperidine derivatives; chelate compounds; complexes with technetium
02/03/2005US20050026954 Muscarinic receptor antagonists; overactive bladder, irritable bowel syndrome, chronic obstructive pulmonary disease, and asthma
02/03/2005US20050026952 Nicotinamide derivatives useful as PDE4 inhibitors
02/03/2005US20050026942 Chemokine receptor binding heterocyclic compounds
02/03/2005US20050026940 Processes for the preparation of substituted bicyclic derivatives
02/03/2005US20050026929 2-Phenyl-4-(piperidin-1-ylcarbonyl)-oxazole derivatives; capsase activators; cancer, autoimmune diseases, rheumatoid arthritis, inflammatory bowel disease, or psoriasis
02/03/2005US20050026928 Chemical compounds
02/03/2005US20050026927 Pyrazole derivatives as psychopharmaceuticals
02/03/2005US20050026923 For therapy of viral diseases
02/03/2005US20050026918 Novel pyridazinone derivatives as pharmaceuticals and pharmaceutical compositions containing them
02/03/2005US20050026917 Tricyclic indanyls as integrin inhibitors
02/03/2005US20050026916 Heterocyclic compounds as P2X7 ion channel blockers
02/03/2005US20050026915 As melanin concentrating hormone (MCH)receptor antagonists, for prevention or treatment of obesity or eating disorders; (2E)-3-(4-chlorophenyl)-N-[2-(dimethylamino)quinolin-6-yl]prop-2-enamide
02/03/2005US20050026914 Pyrimidine or pyridine carbamate compounds as for example 1,1-dimethylethyl 4-(4-((4-((((2,6-dimethylphenyl)oxy)carbonyl)(4-(methyloxy)phenyl)amino)-2-pyrimidinyl)amino)phenyl)-1-piperazinecarboxylate; for the treatment of protein tyrosine kinase-associated disorders
02/03/2005US20050026911 Benzotriazapinone salts and methods for using same
02/03/2005US20050026903 Pyrazole compound; gastrointestinal disorders; central nervous system disorders
02/03/2005US20050026810 Treatment of male sexual dysfunction
02/03/2005US20050025774 Such as N-(2-ethoxybenzyl)-5-hydroxy-1-methyl-2-(4-methylphenyl)-6-oxo-1,6-dihydropyrimidine-4-carboxamide; for preventing, treating or delaying AIDS
02/03/2005US20050025702 radiotherapeutic or chemotherapeutic agents comprising metalloenzyme inhibitors and chelation compounds capable of conjugating to cytotoxic radioisotopes; anticarcinogenic agents
02/03/2005CA2744317A1 Substituted tetracycline compounds
02/03/2005CA2534262A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2533681A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2533663A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2533662A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2533626A1 Quinolinone derivatives as inhibitors of c-fms kinase
02/03/2005CA2533603A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2533397A1 Substituted pyridin-2-ylamine analogues
02/03/2005CA2532980A1 2-aminopyrimidine and 2-aminopyridine-4-carbamates for use in the treatment of autoimmune diseases
02/03/2005CA2532908A1 3,5 disubstituted indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation
02/03/2005CA2532443A1 Tyrosine kinase inhibitors
02/03/2005CA2532403A1 Ppar active compounds
02/03/2005CA2532400A1 Tyrosine kinase inhibitors
02/03/2005CA2532231A1 Aminopyrazole compounds and use as chk1 inhibitors
02/03/2005CA2531912A1 Process for producing 1,2,4-triazole compound and intermediate therefor
02/03/2005CA2531490A1 Substituted pyrimidin-4-ylamina analogues as vanilloid receptor ligands
02/03/2005CA2530352A1 Quinolone derivative or salt thereof
02/02/2005EP1502916A1 Piperidine derivatives having ccr3 antagonism
02/02/2005EP1501841A2 Non nucleoside reverse transcriptase inhibitors
02/02/2005EP1501827A2 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acid and their use as protease inhibitors
02/02/2005EP1501825A2 Substituted imidazolylmethyl pyridine and pyrazine derivatives: gaba a receptor ligands
02/02/2005EP1501824A1 A method for the purification of lansoprazole
02/02/2005EP1501823A1 New piperidinyl-alkylamino-pyridazinone derivatives, a process for the preparation thereof and pharmaceutical compositions containing said compounds
02/02/2005EP1501822A1 Phthalazinone derivatives
02/02/2005EP1501809A1 Triazole derivatives as tachykinin receptor antagonists
02/02/2005EP1501808A1 Tachykinin receptor antagonists