Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
12/2004
12/15/2004EP1485167A1 1,2-dihydropyrazol-3-ones as cytokine mediators
12/15/2004EP1485100A1 Azinylaminoazoles as inhibitors of protein kinases
12/15/2004EP1485099A1 Inhibitors of histone deacetylase
12/15/2004EP1485094A1 FORM OF PRESENTATION FOR 3- (2-{ 4-(HEXYLOXYCARBONYLAMINO-IMINO-METHYL)-PHENYLAMINO -METHYL}-1-METHYL-1iH /i -BENZIMIDAZOL-5-CARBONYL)-PYRIDIN-2-YL-AMINO PROPIONIC ACID ETHYL ESTER TO BE ADMINISTERED ORALLY
12/15/2004EP1485093A1 Di-aryl substituted tetrazole modulators of metabotropic glutamate receptor-5
12/15/2004EP1484971A1 4-aminopyrimidines and their use for the antimicrobial treatment of surfaces
12/15/2004EP1484969A1 Synergistic fungicide compositions containing at least one n-[(2-pyridinyl)methyl]-3-pyridinecarboxamide derivative and one or more further fungicides useful for controlling fungal plant diseases
12/15/2004EP1430033A4 Anti-inflammatory and protein kinase inhibitor composition and method of use
12/15/2004EP1387840B1 3,5-diamino-1,2,4-triazoles as kinase inhibitors
12/15/2004EP1373216B1 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity
12/15/2004EP1337520B1 Substituted 5-aryl and 5-heteroaryl-2-(2-hydroxyphenyl)-2h-benzotriazole derivatives as uv absorbers
12/15/2004EP1307447B1 3-indolyl-4-phenyl-1h-pyrrole-2,5-dione derivatives as inhibitors of glycogen synthase kinase-3beta
12/15/2004EP1226137B8 Phenyl- and pyridyl-tetrahydro-pyridines having tnf inhibiting activity
12/15/2004EP1226125B1 Method for producing therapeutic agents for ulcers
12/15/2004EP1226122B1 Bicyclic vasopressin agonists
12/15/2004EP1176963B1 Use of dopamine d 3 receptor antagonists for producing medicaments for treating kidney disorders
12/15/2004EP1091957B1 Pyrimidin-aminomethyl-pyridine derivatives, their preparation and their use in the control of helicobacter bacteria
12/15/2004CN1555367A 3-substituted-4-pyrimidone derivatives
12/15/2004CN1555364A Insecticidal diamides
12/15/2004CN1555262A Novel 4,5-dihydro-1H-pyrazole derivatives having CB*-antagonistic activity
12/15/2004CN1555260A Aminoalkyl-substituted aromatic bicyclic compounds, methods for their preparation and their use as pharmaceuticals
12/15/2004CN1554656A Yunnan tolal biological coronaridine and its salts and preparing method and use
12/15/2004CN1179960C Indole derivatives and their use for treamtent of osteoporosis amongst other applications
12/15/2004CN1179954C Substd. heterocyclic compounds, preparing process thereof and pharmaceutical composition contg. them
12/15/2004CN1179952C Pyrimidine-4-one derivatives as LDL-PLA2 inhibitors
12/15/2004CN1179948C HIV protease inhibitors
12/15/2004CN1179945C Indole derivatives, process for preparation of same and use thereof
12/15/2004CN1179944C 2-oxo-1-pyrrolidine derivatives, process for preparing them and their uses
12/14/2004US6831199 Pyrimidine compounds and derivatives thereof
12/14/2004US6831175 Such as N,N-dimethyl-N-(2-((5-((E)-2-pyridin-4-ylvinyl) pyridin-3-yl)oxy)ethyl)amine
12/14/2004US6831096 Effective against both A and B forms of influenza; oral bioavailability
12/14/2004US6831094 For therapy of central nervous system disorders such as anxiety, depression, motor disorders
12/14/2004US6831089 1,4-di-substituted piperidines, some of which have M2 selectivity even higher than that of 3-alpha-chloroimperialine for treating cognitive disorders such as Alzheimer's disease
12/14/2004US6831087 2-(Pyrid-2- or 4-yl)-1,2,3,4-tetrahydroisoquinoline and derivatives; a good affinity to the NMDA receptor (N-methyl-D-asparate); acute/cronic neurodegenerative diseases; bacterial/viral infections; antidepressants; analgesics
12/14/2004US6831085 Methods and compositions utilizing quinazolinones
12/14/2004US6831083 Pyrazoline derivative or tetrahydropyridazine derivative and medicinal use thereof
12/14/2004US6831082 Method of using soluble epoxide hydrolase inhibitors
12/14/2004US6831078 3-aryl substituted having halo or alkylhalo groups; anxiety, epilepsy; presurgery muscle relaxant
12/14/2004US6831075 Heterocyclic substituted pyrazolones
12/14/2004CA2136075C Heterocyclic ether compounds that enhance cognitive function
12/10/2004WO2004108677A1 Antithrombotic ethers
12/09/2004WO2004106493A2 Chemokine receptor binding heterocyclic compounds with enhanced efficacy
12/09/2004WO2004106326A1 Novel polymorphs of imatinib mesylate
12/09/2004WO2004106325A1 Prodrugs of 1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazine
12/09/2004WO2004106324A1 Azolecarboxamide herbicides
12/09/2004WO2004106323A1 Method for producing cyclic diamine derivative or salt thereof
12/09/2004WO2004106322A2 Polymorphs of aripiprazole
12/09/2004WO2004106310A1 Novel 3-substituted-1,4-benzodiazepines
12/09/2004WO2004106308A1 Quinazolines and pyrido [3,4-d] pyrimidines as receptor tyrosine kinase inhibitors
12/09/2004WO2004106307A2 Novel imidazole derivatives, the production thereof, and the use of the same as a medicament
12/09/2004WO2004106305A1 New p2x7 receptor antagonists and their use
12/09/2004WO2004106302A1 Novel substituted 3-sulfur indoles
12/09/2004WO2004106299A2 Substituted pyrrole derivatives and their use as hmg-co inhibitors
12/09/2004WO2004106296A2 Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators
12/09/2004WO2004106289A1 Protease inhibitors
12/09/2004WO2004105757A2 Use of rho-kinase inhibitors in the treatment of aneurysm and cardiac hypertrophy
12/09/2004WO2004105752A1 Substituted pyrrole derivatives as hmg-coa reductase inhibitors
12/09/2004WO2004094388A3 Indazole derivatives as jnk inhibitors
12/09/2004WO2004089901A3 Phospholipase c inhibitors for use in treating inflammatory disorders
12/09/2004WO2004089892A3 Diarylmethyl and related compounds having beta2 andrenergic receptor agonist and muscarinic receptor antagonist activity
12/09/2004WO2004075863A3 Cxcr3 antagonists
12/09/2004WO2004069794A9 New arylpiperazinyl compounds
12/09/2004WO2004061084A8 Modulation of protein functionalities
12/09/2004WO2003104206A3 Herbicidally active heterocyclylalkynes
12/09/2004WO2003102588A3 Diagnostic agent, method for detecting a carcinoma, and means for the treatment thereof
12/09/2004WO2003080582A3 Fredericamycin derivatives
12/09/2004US20040249185 Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate
12/09/2004US20040249161 Biphenyl-derivatives as p38-kinase inhibitors
12/09/2004US20040249155 1-(omego-substituted-2-[(hetero)arylcarbonylamino]alkanoyl)-4-(1-methylpiperidin-4-yl)piperidine derivatives; e.g., 1-[N-(Indole-6-carbonyl)-D-serinyl]-4-(1-methylpiperidin-4-yl)piperidine Hydrochloride
12/09/2004US20040249153 For therapy of inflammation, rheumatoid arthritis, osteoarthritis, osteoporosis and tumors
12/09/2004US20040249151 Chemical compounds
12/09/2004US20040248961 Oxidation base compound has the nitrogen-based quaternary onium group; oxidation dye precursors; hair coloring with oxidizer; multi-compartment kit; chromatic, fast coloration
12/09/2004US20040248944 Novel 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity
12/09/2004US20040248941 such as 4-[2-[[[3-Methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl]methyl]sulfinyl]-1H-benzimidazol-1-yl]-1,3-dioxolan-2-one, used as prodrugs to lansoprazole; proton pump inhibitors; antiulcer agents
12/09/2004US20040248940 enantiomorphs of pantoprazole magnesium hydrate, used for prevention of gastrointestinal disorders
12/09/2004US20040248938 Substituted piperidines
12/09/2004US20040248936 such as (R)-1-{4-[4-(4-Phenoxy-2-propyl-phenoxy)-butoxy]-benzenesulfonyl}-azetidine-2-carboxylic acid, used as peroxisome proliferator-activated receptor agonists; hypoglycemic agents
12/09/2004US20040248932 Use of aryl- and heteroaryl-substituted tetrahydroisoquinolines in the treatment of chronic and neuropathic pain, migraine headaches, and urge, stress and mixed urinary incontinence
12/09/2004US20040248931 Poly(ADP-ribose)polymerase inhibitors; cerebral infarction; such as 3-[2-(3-hydroxypyrrolidin-1-yl)ethyl]-5-methyl-2H-isoquinolin-1-one; synthesis
12/09/2004US20040248923 Novel 4-anilinoquinoline-3-carboxamides
12/09/2004US20040248922 Lavendamycin analogs, quinoline-5,8-diones and methods of using them
12/09/2004US20040248920 Spiro-hydantoin compounds useful as anti-inflammatory agents
12/09/2004US20040248918 Anticancer agents
12/09/2004US20040248914 Method for the treatment of overactive bladder
12/09/2004US20040248907 reacting 4,6-dichloro-5-nitropyrimidine with acyclic carboxy amines, then cyclization of the intermediates to form cellular adhesion inhibitors
12/09/2004US20040248902 Central nervous system, gastrointestinal and psycological disorders; such as 3-(4-chlorobenzenesulfonyl)-2-methyl-7-piperazin-1-yl-1H-indole; synthesis
12/09/2004US20040248899 Fused bicyclic-substituted amines as histamine-3 receptor ligands
12/09/2004US20040248895 Novel guanidino compounds
12/09/2004US20040248890 Voltage gated sodium and calcium channel inhibitors
12/09/2004US20040248888 Metabotropic glutamate (mGluR5) receptor mediated disorders; psychosis, epilepsy, schizophrenia, Alzheimer' disease, cognititve disorders, memory deficits, chronic and acute pain; containing pyridin-4-ylethynyl functionality
12/09/2004US20040248884 Protein kinase inhibitors; antitumor agents; such as 5-methyl-1-quinol-4-ylmethyl-3-(4-trifluoromethanesulfonylphenyl)imidazolidine-2,4-dione trifluoroacetate
12/09/2004US20040248883 Novel heteroaryl derivatives, their preparation and use
12/09/2004US20040248882 Noninsulin dependent diabetes, obesity, hypercholesterolemia, inflammatory disorders; reduced side effects; such as 5-(4-acetylbenzenesulfonamido-2-fluorophenoxy)-3-chloropyridine
12/09/2004US20040248877 Inducing apoptosis in tumor cells
12/09/2004US20040248872 Safe for agricultural or gardening use; effective against insects and mammals
12/09/2004US20040248853 Antiinflammatory agents; antihistamines; adult respiratory distress syndrome; antidiabetic agents; inflammatory bowel disorders
12/09/2004US20040248820 Administering 2-phthalimidoglutaric acid; vision defects; antitumor agents; anticancer agents
12/09/2004US20040248740 for controlling undesirable plants
12/09/2004US20040248225 Luciferin hydrazides
12/09/2004US20040247523 Diagnosing and localizing sites of inflammation and perfusion abnormalities (e.g. reperfusion injury, vulnerable plaque, bacterial endocarditis or cardiac transplant rejection) in a single dual isotope imaging procedure, particularly CT imaging, ultrasound, or scintigraphy.