Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
03/2005
03/01/2005US6861071 Highly absorptive solid preparation
03/01/2005CA2288334C Method of manufacturing sertindole
03/01/2005CA2138287C N-substituted azabicycloheptane derivatives, the preparation and use thereof
02/2005
02/24/2005WO2005016918A2 Heterocyclic n-aryl carboxamides as cytokine inhibitors
02/24/2005WO2005016917A1 Process for preparing isomerically pure prodrugs of proton pump inhibitors
02/24/2005WO2005016916A2 Substituted quinolines serving as antimicrobial agents
02/24/2005WO2005016915A1 Piperidine/cyclohexane carboxamide derivatives for use as vanilloid receptor modulators
02/24/2005WO2005016914A1 Chemical compounds
02/24/2005WO2005016913A1 Tetrahydroisoquinoline or isochroman compounds as orl-1 receptor ligands for the treatment of pain and cns disorders
02/24/2005WO2005016912A1 An efficient microbial preparation of capravirine metabolites m4 and m5
02/24/2005WO2005016911A1 4-pyrimidone derivatives and their use as peptidyl peptidase inhibitors
02/24/2005WO2005016910A1 Pyridyltetrahydropyridines, pyridylpiperidines, and process for the production of both
02/24/2005WO2005016897A1 Process for the preparation of 2- (quinoxalin-5-ylsulfonylamino) -benzamide compounds
02/24/2005WO2005016896A1 2- (quinoxalin-5-ylsulfonylamino) -benzamide compounds as cck2 modulators
02/24/2005WO2005016894A1 2, 4-pyrimidinediamines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders
02/24/2005WO2005016892A1 Gabanergic modulators
02/24/2005WO2005016890A1 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor
02/24/2005WO2005016885A2 COMPOUNDS WITH COMBINED CALCIUM CHANNEL BLOCKER AND β-ADRENERGIC ANTAGONIST OR PARTIAL AGONIST ACTIVITIES FOR TREATMENT OF HEART DISEASE
02/24/2005WO2005016883A2 Acrylamide derivatives as vla-1 integrin antagonists and uses thereof
02/24/2005WO2005016879A2 Cyclic pyrazinoylguanidine sodium channel blockers
02/24/2005WO2005016876A2 Cyclic amine bace-1 inhibitors having a benzamide substituent
02/24/2005WO2005016862A1 Substituted arylalkanoic acid derivative and use thereof
02/24/2005WO2005016346A1 Quinazoline analogs as receptor tyrosine kinase inhibitors
02/24/2005WO2005016344A1 Piperazine derivatives for the treatment of hiv infections
02/24/2005WO2005016326A2 Analogs of thalidomide as potential angiogenesis inhibitors
02/24/2005WO2005016000A1 Derivatives of cyclic quinone and uses thereof
02/24/2005WO2005005393A3 Cck-1 receptor modulators
02/24/2005WO2004093789A3 Use of galr3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods
02/24/2005WO2004087056A3 BI-CYCLIC PYRIMIDINE INHIBITORS OF TGFβ
02/24/2005WO2004046103A3 Arylpyridine compounds
02/24/2005WO2004031175A3 N-substituted-2-oxodihydropyridine derivatives as npy antagonists
02/24/2005US20050043552 Process for the synthesis of amine ethers from secondary amino oxides
02/24/2005US20050043543 Benzotriazole/HALS molecular combinations and compositions stabilized therewith
02/24/2005US20050043535 4-(Piperidyl-and pyrrolidyl-alkyl-ureido)-quinolines as urotensin II receptor antagonists
02/24/2005US20050043390 Viricides against herpes virus
02/24/2005US20050043388 Therapy, prevention of metabolism disorders; insulin resistance; antidiabetic agents; hypoglycemic agents; anticholesterol agents; obesity; polycystic ovarian syndrome
02/24/2005US20050043381 Aminopyrazole compounds
02/24/2005US20050043379 Leukotriene hydrolase inhibitors; antiinflammatory agents; antihistamines; chronic onstructive pulmonary disorders; atherosclerosis; multiple sclerosis; inflammatory bowel disorders; antiarthritic agents ;psoriasis
02/24/2005US20050043378 LTA4H modulators
02/24/2005US20050043368 Osteoporosis therapy; bone disorders
02/24/2005US20050043366 Antiinflamamtory agents; immunology disorders; autoimmune diseases; antiallergens; aids viricides; antiarthritic agents; muscular disorders; Parkinson's disease; Alzheimer's disease; kidney damage
02/24/2005US20050043364 Novel pyrrole-based HMG-CoA reductase inhibitors
02/24/2005US20050043363 Efficient microbial preparation of capravirine metabolites M4 and M5
02/24/2005US20050043357 Mitotic kinesin inhibitors
02/24/2005US20050043354 Substance P antagonist
02/24/2005US20050043352 human YAK family of serine/threonine protein kinases (hyak); use treating diseases of the hematopoietic systems, including anemias, polycythemia, myelodysplastic syndrome, myelosuppression, cytopenia, male contraceptives; 2-(3-Chloro-phenylamino)-7-methoxy-quinoline-3-carboxylic acid for example
02/24/2005US20050043348 Phenyl-substituted imidazopyridines
02/24/2005US20050043338 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
02/24/2005US20050043337 Selective beta3 adrenergic agonists
02/24/2005US20050043336 Quinazoline derivatives as antitumor agents
02/24/2005US20050043335 Heterocyclic derivatives of glycinamide and their medical use
02/24/2005US20050043334 Such as N6-(4,5-dihydrooxazol-2-yl)-N4-[3-methyl-4-(6-methylpyridin-3-yloxy)-phenyl]-quinazoline-4,6-diamine; for treatment of hyperproliferative disorders such as cancer
02/24/2005US20050043333 Quinazolinone derivative
02/24/2005US20050043331 Substituted 3-(2,5-disubstituted)pyridyl-4-aryl pyrroles for treating inflammatory diseases
02/24/2005US20050043330 Antiinflammation agents
02/24/2005US20050043316 Piperidine derivatives, process for preparation thereof, and pharmaceutical composition for alzheimer's disease containing the same
02/24/2005US20050043315 Aminopyrimidine compounds, processes for their preparation and pharmaceutical compositions containing them
02/24/2005US20050043314 Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same
02/24/2005US20050043313 1-(phenylaminocarbonylmethyl)-3-alkylamino-5,6-disubstituted-2-pyazinones; serine protease inhibitors; anticoagulants; coronary artery and cerebrovascular diseases
02/24/2005US20050043310 Such as (R)-4-bromo-N-[1-(2,4-dichlorophenyl)-ethyl]-2-(quinoxaline-5-quinoxaline-sulfonylamino)-benzamide via sulfonylation; cholecystokinin receptor modulators
02/24/2005US20050043307 Novel heterocycle as agonist or antagonist for nervous systems which can contain double or triple bonds with nitrogen, oxygen or sulfur with carbon or azo groups and or salts and as modulators or receptors with carriers
02/24/2005US20050043304 Lower alkyl molecular weight amine as enzyme inhibitors for use in the treatment of tryptase enzyme inhibitors inhibitorsfor respiratory system disorders, antiinflammatory agents, inflammatory bowel disease, hyperprolific skin disorders, vascular edema and rheumatoid arthritis
02/24/2005US20050043302 New indole derivatives as factor Xa inhibitors
02/24/2005US20050043301 Substituted heterocyclic compounds and methods of use
02/24/2005US20050043300 Piperazine derivatives
02/24/2005US20050043299 Inhibitors of dipeptidyl peptidase iv
02/24/2005US20050043292 eg S)-[5-amino-6-oxo-6-(3,3,4,4-tetrafluoro-pyrrolidin-1-yl)-hexyl-carbamic acid benzylester; Type 2 diabetes, metabolic syndrome (syndrome X or insulin resistance syndrome), hyperglycemia, impaired glucose tolerance, glucosuria, metabolic acidosis, arthritis, cataracts, diabetic neuropathy
02/24/2005US20050043291 Heterocyclic substituted aminoazacycles useful as central nervous system agents
02/24/2005US20050043290 for treating neurodegenerative disease such as Alzheimer's disease
02/24/2005US20050043277 Production of imidazole derivatives and novel intermediates of the derivatives
02/24/2005US20050042771 Identifying non-drug targets; use in drug design for improving knowledge of drug-target and drug-non-target interactions, so that drug adverse reactions can be reduced or eliminated in drugs such as troglitazone, rosiglitazone, pioglitazone, methotrexate, atorvastatin, celecoxib, rofecoxib, cerivastatin
02/24/2005US20050042614 Point mutations; dipeptidyl-peptidase inhibitors; kits
02/24/2005US20050042304 Novel substituted benzimidazole dosage forms and method of using same
02/24/2005DE10331500A1 Neue Acridin-Derivate und deren Verwendung als Arzneimittel New acridine derivatives and their use as medicaments
02/24/2005DE102004010545A1 Pyrazoline Pyrazolines
02/24/2005CA2743534A1 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor
02/24/2005CA2535665A1 Substituted arylalkanoic acid derivative and use thereof
02/24/2005CA2535619A1 4-pyrimidone derivatives and their use as peptidyl peptidase inhibitors
02/24/2005CA2535406A1 Gabanergic modulators
02/24/2005CA2535020A1 Substituted quinolines serving as antimicrobial agents
02/24/2005CA2534950A1 Cyclic amine bace-1 inhibitors having a benzamide substituent
02/24/2005CA2534887A1 Process for the preparation of 2- (quinoxalin-5-ylsulfonylamino) -benzamide compounds
02/24/2005CA2534866A1 Piperazine derivatives for the treatment of hiv infections
02/24/2005CA2532104A1 Process for preparing isomerically pure prodrugs of proton pump inhibitors
02/24/2005CA2518774A1 Heterocyclic n-aryl carboxamides as cytokine inhibitors
02/23/2005EP1508569A2 Process for the preparation of tetrasubstituted imidazole derivatives and novel crystalline structures thereof
02/23/2005EP1507826A2 Amelioration of the development of cataracts and other opthalmic diseases
02/23/2005EP1507775A1 Heterocyclic compounds which inhibit leukocyte adhesion mediated by alpha4 integrins
02/23/2005EP1507774A1 Processes for preparation of polymorphic forms of desloratadine
02/23/2005EP1507773A1 Macrocyclic compounds useful as pharmaceuticals
02/23/2005EP1507768A1 Aryl-alkyne compounds as herbicides
02/23/2005EP1507767A1 4-substituted imidazole-2-thiones and imidazol-2-ones as agonists of the alpha-2b and alpha-2c adrenergic receptors
02/23/2005EP1507764A1 Novel enantiomers of tetrahydroisoquinoline derivatives and their pharmaceutically acceptable salts, their preparations and pharmaceutical compositions
02/23/2005EP1507761A1 Pyridine carboxamide derivatives and their use as pesticides
02/23/2005EP1507760A1 Cyanoguanidine prodrugs
02/23/2005EP1507759A1 Cyanoguanidine produgs
02/23/2005EP1507535A1 Pyrimidine-2,4,6-trione metallo-proteinase inhibitors
02/23/2005EP1507534A2 Compounds, compositions and methods
02/23/2005EP1507531A2 Stable pharmaceutical compositions of desloratadine
02/23/2005EP1507529A1 Combination of organic compounds