Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
04/2005
04/21/2005CA2541667A1 Substituted pyrazinone compounds for the treatment of inflammation
04/21/2005CA2541582A1 Indoles and azaindoles as antiviral agents
04/21/2005CA2541162A1 Fused lactam compounds
04/21/2005CA2540868A1 Pyrrolidinyl urea derivatives as angiogenesis inhibitors
04/21/2005CA2540867A1 Process for the preparation of n-amino substituted heterocyclic compounds
04/21/2005CA2539882A1 Substituted isoquinolinones
04/21/2005CA2526017A1 5-h-benzo[d]naphth[2,1-b]azepine derivative as selective d1/d5 receptor antagonists for the treatment of obesity and cns disorders
04/20/2005EP1524272A1 Growth hormone secretagogues
04/20/2005EP1524265A1 Prolinamide derivatives as sodium and/or calcium channel blockers or selective MAO-B inhibitors
04/20/2005EP1523481A1 3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them
04/20/2005EP1523480A2 Derivatives of 3-guanidinocarbonyl-1-heteroaryl-pyrrole, process for their preparation and their pharmaceutical use
04/20/2005EP1523473A1 Indoline derivatives substituted in position 6, production and use thereof as medicaments
04/20/2005EP1523313A1 Crystalline 2,5-dione-3-(1-methyl-1h-indol-3-yl)-4- 1-(pyridin-2-ylmethyl)piperidin-4-yl]-1h-indol-3-yl]-1h-pyrrole mono-hydrochloride
04/20/2005EP1448547B1 Pyridine derivatives as nmda receptor ligands
04/20/2005EP1443934B1 Benzotriazepines as gastrin and cholecystokinin receptor ligands
04/20/2005EP1373249B1 Imidazolidine derivatives, their preparation, and their use as antiinflamatory agent
04/20/2005EP1349847B1 Oxybenzamides derivatives as factor xa inhibitors
04/20/2005EP1254133B1 Indol-3-yl derivatives and their use as integrin inhibitors
04/20/2005EP1252158B1 Nicotinamide benzofused-heterocyclyl derivatives useful as selective inhibitors of pde4 isozymes
04/20/2005EP1200414B1 Process for the preparation of substituted pyrimidines
04/20/2005EP1177185B1 4, 5, 6, 7-tetrahydroindazole derivatives as antitumor agents
04/20/2005EP1140904B1 Farnesyl protein transferase inhibitors
04/20/2005EP1042287B1 Indole derivatives as inhibitors of factor xa
04/20/2005EP1029851B1 Piperazine compounds and medicinal use thereof
04/20/2005EP1015431B1 2-aminopyridines as inhibitors of cyclooxygenase-2
04/20/2005EP0766669B1 Tri-substituted phenyl derivatives useful as pde iv inhibitors
04/20/2005EP0721455B9 Tetrahydropyridine-(or 4-hydroxypiperidine)alkylazoles having an affinity for sigma and/or 5ht1a receptors
04/20/2005CN1608063A Indolinone derivatives
04/20/2005CN1608062A Salt forms of e-2-methoxy-n-(3-{4-[3 methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide and method of production
04/20/2005CN1608061A Therapeutic isoquinoline compounds
04/20/2005CN1608060A Diaryl 1, 2, 4-triazole derivatives as a highly selective cyclooxygenase-2 inhibitor
04/20/2005CN1608059A Bipyridyl derivatives as a highly selective cyclooxygenase-2 inhibitor
04/20/2005CN1608054A Therapeutic quinolone compounds with 5-HT-antagonistic properties
04/20/2005CN1608053A Heterocyclic derivatives of glycinamide and its pharmaceutical uses
04/20/2005CN1607951A Quinoline derivatives as neuropeptide y antagonists
04/20/2005CN1197861C Method for preparing solid optical pure neutral S- (-) - and (R) - (+) -Omeprazole
04/20/2005CN1197860C FAB I inhibitors
04/20/2005CN1197859C Febrifugine and isofebrifugine and processes for the preparation of both
04/20/2005CN1197849C 2, 3, 4, 5-tetrahydro-1H-[1, 4] benzodiazepine-3-hydroxamic acid as matrix metalloproteinase inhibitors
04/20/2005CN1197574C Method for stabilizing benzimidazole compounds
04/19/2005US6881848 Process for preparing 4-trifluoromethylsulfinylpyrazole derivative
04/19/2005US6881844 Indole-3-carboxamides as glucokinase activators
04/19/2005US6881815 Comprises polymerization catalysts; aromatization; elminates need for nitration
04/19/2005US6881753 Potassium channel inhibitors and method
04/19/2005US6881747 Small molecules for inhibition of function and drug delivery to leukocytes
04/19/2005US6881743 Pyridine matrix metalloproteinase inhibitors
04/19/2005US6881740 Pharmaceutical agents
04/19/2005US6881738 Analogs of choline for neuroprotection and cognitive enhancement in neurodegenerative disorders
04/19/2005US6881737 Substituted triazinyl acrylamide derivatives and methods of use
04/19/2005US6881735 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
04/19/2005US6881536 Particle based electrochemiluminescent assays
04/19/2005CA2315189C Integrin receptor antagonists
04/19/2005CA2273894C Novel n-benzenesulphonyl-l-proline derivatives, method for preparing and therapeutic use
04/19/2005CA2172162C Optically active imidazolidinone derivative and process for producing the same
04/19/2005CA2116631C Process for the preparation of aqueous nicotinaldehyde
04/14/2005WO2005033108A1 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones
04/14/2005WO2005033106A1 Azolidinecarbonitriles and their use as dpp-iv inhibitors
04/14/2005WO2005033105A2 Vanilloid receptor ligands and their use in treatments
04/14/2005WO2005033097A1 P-glycoprotein inhibitor, method for preparing the same and pharmaceutical composition comprising the same
04/14/2005WO2005033096A1 Quinoline derivatives and quinazoline derivatives, medicaments containing said compounds, use thereof, and method for the production thereof
04/14/2005WO2005033095A1 Fungicidal 4-(2-aminopyridin-4-yl)-n-phenyl-1,3,5-triazin-2-amine derivatives
04/14/2005WO2005033081A1 4-piridinylmethylsulphonamide derivatives as fungicidal plant protection agents
04/14/2005WO2005033073A2 Spirocyclic heterocyclic derivatives and methods of their use
04/14/2005WO2005033048A2 Wnt pathway antagonists
04/14/2005WO2005032548A1 Substituted benzazoles and use thereof as inhibitors of raf kinase
04/14/2005WO2005032547A1 Bicyclo`3.1.1!heptane substituted benzimidazolone and quinazolinone derivatives as agonists on human orl1 receptors
04/14/2005WO2005032493A2 Amide compounds as ion channel ligands and uses thereof
04/14/2005WO2005032490A2 Cyclic diamines and derivatives as factor xa inhibitors
04/14/2005WO2005032484A2 Alkoxy substituted imidazoquinolines
04/14/2005WO2005032472A2 Pyrrolidine and piperidine derivatives as factor xa inhibitors
04/14/2005WO2005016883A3 Acrylamide derivatives as vla-1 integrin antagonists and uses thereof
04/14/2005WO2005014723A8 Cyanin-type compounds having an alkynyl linker arm
04/14/2005WO2005007111A3 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
04/14/2005WO2005002503A3 Asymmetric benzimidazoles and related compounds as potassium channel modulators
04/14/2005WO2005000281A3 Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
04/14/2005WO2004099154A3 Pyrazole-amides and sulfonamides as sodium channel modulators
04/14/2005WO2004092124A3 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors
04/14/2005WO2004091542A3 Nitrogen containing integrin targeting compounds
04/14/2005US20050080272 Halogenated nitrobutadienes for controlling animal pests
04/14/2005US20050080271 Peptidomimetic ligands for cellular receptors and ion channels
04/14/2005US20050080265 Sleep disorders; side effect reduction
04/14/2005US20050080258 Kinase inhibitors; autoimmune disease; antiinflammatory agents
04/14/2005US20050080129 Derivatives of andrimide and moiramide b having antibacterial properties
04/14/2005US20050080121 for example, 4S-[(naphthalene-2-carbonyl)-amino]-5-(2-oxo-pyrrolidin-3S-yl)-pent-2-enoic acid ethyl ester; treatment of viral infections caused by human rhinoviruses, human polioviruses, human coxsackieviruses, human echoviruses, among others
04/14/2005US20050080119 Diaminopropionic acid derivatives
04/14/2005US20050080111 Antagonists of liver X receptors; control of cholesterol, triglyceride, or bile acid levels; 6-(1-Benzyl-1H-pyrazol-4-yl)-1-(2,4-difluoro-benzyl)-2-oxo-4-trifluoromethyl-1,2-dihydro-pyridine-3-carbonitrile
04/14/2005US20050080108 such as (S)-1-ethyl-5-[(4'-trifluoromethyl-biphenyl-2-carbonyl)-amino]-1H-indole-2-carboxylic acid-[2-[benzyl(methyl)amino]-2-oxo-1-phenylethyl]amide; for treatment of obesity and lipid disorders; diabetes
04/14/2005US20050080106 Such as 2-[3,5-Di(2-chlorobenzyloxy)benzoyl)amino]-thiazole; for treatment of diabetes
04/14/2005US20050080101 N-[4-(pyrazolyl)-pyrimidin-2-yl]-N-phenyl-amine derivatives
04/14/2005US20050080096 Condensed heterocyclic compounds
04/14/2005US20050080095 Novel amides useful for treating pain
04/14/2005US20050080090 Such as 7-(Imidazolo[4,5-b]pyridin-1-yl)-1-(1-methylpyrrolidin-3-yl)naphthalene; for treating depression, anxiety, eating disorders, drug abuse, cluster headache, migraine, pain, and other disorders arising from deficient serotonergic neurotransmission
04/14/2005US20050080087 For treatment of metabolic disorders, eating disorders, appetitive disorders, psychiatric disorders, memory impairment, Parkinson's disease, Alzheimer's disease, substance abuse, leukocyte activation-associated disorders, and inflammatory diseases
04/14/2005US20050080082 Potassium channel modulators
04/14/2005US20050080078 Such as [1-(4-chloro-phenyl)-cyclobutyl]-(3-hydroxymethyl piperidin-1-yl)-methadone for treating cocaine and/or methamphetamine addiction
04/14/2005US20050079176 Treating stress response with chemokine receptor ccr5 modulators
04/14/2005DE19842833B4 2-Arylalkylthio-imidazole, 2-Arylalkenylthio-imidazole und 2-Arylalkinylthio-imidazole als Entzündungs-Hemmstoffe und Hemmstoffe der Cytokin-Freisetzung 2-arylalkylthio-imidazole, 2-Arylalkenylthio-imidazole and 2-Arylalkinylthio-imidazoles as inflammatory inhibitors and inhibitors of cytokine release
04/14/2005DE10343098A1 Tetrahydrochinoxaline und ihre Verwendung Tetrahydroquinoxalines and their use
04/14/2005DE10342503A1 Benzyl-Benzimidazolylderivate Benzyl-Benzimidazolylderivate
04/14/2005CA2541299A1 Amide compounds as ion channel ligands and uses thereof