Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
02/2003
02/25/2003US6525042 Sulfonyl derivatives
02/25/2003US6525036 Compounds and compositions as protease inhibitors
02/25/2003US6525020 For drug delivery
02/20/2003WO2003014111A1 Arylpiperazines and arylpiperidines and their use as metalloproteinase inhibiting agents
02/20/2003WO2003014098A1 Arylpiperazines and arylpiperidines and their use as metalloproteinase inhibiting agents
02/20/2003WO2003014097A1 Arylsulfonyl derivatives with 5-ht6 receptor affinity
02/20/2003WO2003014064A1 Naphthylurea and naphthylacetamide derivatives as vanilloid receptor 1 (vr1) antagonists
02/20/2003WO2002085871A3 Serotonergic agents with long-acting in vivo effects
02/20/2003WO2002068399B1 Aryl carbamate derivatives, preparation and use thereof
02/20/2003WO2002048097B1 Compounds, compositions and methods for treatment of parasitic infections
02/20/2003WO2002024635A3 Aminoalcohol derivatives
02/20/2003US20030036558 Useful in the treatment of chronic complications arising from diabetes, such as neuropathy; may also contain an angiotensin converting enzyme inhibitor.
02/20/2003US20030035784 Hair condition
02/20/2003DE20217957U1 Oxidative dyeing agent for keratin fibers uses 2-aminomethylene-substituted resorcinols as couplers, some of which are novel compounds
02/20/2003CA2456250A1 Arylsulfonyl derivatives with 5-ht6 receptor affinity
02/20/2003CA2455754A1 Amine derivatives
02/19/2003EP1284262A1 Process for the preparation of cis-2,6-dimethylpiperazine
02/19/2003EP1284140A2 Use of ritonavir (ABT-538) for improving the pharmacokinetics of drugs metabolized by cytochrome P450 in a method of treating aids
02/19/2003EP1283825A1 N-substituted peptidyl nitriles as cysteine cathepsin inhibitors
02/19/2003EP1283823A1 Novel mmp-2/mmp-9 inhibitors
02/19/2003CN1398260A 二肽腈组织蛋白酶k抑制剂 Dipeptide nitrile cathepsin inhibitors k
02/19/2003CN1398247A Colchinol derivatives as vascular damaging agents
02/19/2003CN1397554A Novel N-benzyl diethylenediamine compound, its prepn. process and medicinal compsns. contg. them
02/19/2003CN1397547A Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them
02/19/2003CN1101807C 异羟肟酸衍生物 Hydroxamic acid derivatives
02/18/2003US6521755 Process for preparing 10,11-methanobenzosuberane derivatives
02/18/2003US6521707 (poly)ether amine ester isocyanate derivatives that can be reacted with hydroxy and amino compounds to form urethanes or ureas used in the isolation of nucleic acids
02/18/2003US6521666 Inhibitors of α4 mediated cell adhesion
02/18/2003US6521619 Bind to the interaction-domain of integrin lfa-1 interrupting enothelial cell-leukocyte adhesion
02/14/2003WO2002018326A1 Novel propenohydroxamic acid derivatives
02/14/2003CA2423733A1 Novel propenohydroxamic acid derivatives
02/13/2003WO2003011851A2 Aromatic hydroxamic acid derivatives useful as hdac inhibitors
02/13/2003WO2003011844A2 Reagent and method for perfluoroalkylation
02/13/2003WO2003011817A1 1, 3, 5-tricyano-2, 4, 6-tris(vinyl)benzene derivatives and method for preparing the same
02/13/2003WO2003011296A1 Pharmaceutical preparations containing aminobenzene- sulfonic acid derivatives as the active ingredient
02/13/2003WO2003011282A1 Pharmaceutical compositions, kits and methods comprising combinations of estrogen agonists/antagonists, estrogens and progestins
02/13/2003WO2002096855A3 Anticholinergic compounds and methods of use
02/13/2003US20030032803 Novel amide derivatives as inhibitors of matrix metalloproteinases, TNF-alpha, and aggrecanase
02/13/2003US20030032644 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
02/13/2003US20030032641 Certain salts of discodermolide acid, pharmaceutical compositions containing them and their use in treating tumors
02/13/2003CA2455858A1 Pharmaceutical preparations containing aminobenzene- sulfonic acid derivatives as the active ingredient
02/13/2003CA2449804A1 Aromatic hydroxamic acid derivatives useful as hdac inhibitors
02/13/2003CA2448235A1 Pharmaceutical compositions, kits and methods comprising combinations of estrogen agonists/antagonists, estrogens and progestins
02/12/2003EP1283039A1 -secretase inhibitors
02/12/2003EP1282630A1 Hydroxylamine esters as polymerization initiators
02/12/2003EP1282611A1 Substituted phenylacetamides and their use as glucokinase activators
02/12/2003EP1282600A1 Inhibitors of dipeptidyl peptidase iv
02/12/2003EP1282597A1 Method for the production of $g(v)-aminoalkylsulphonic acids
02/12/2003EP0988292B1 Piperazine derivatives and their use as anti-inflammatory agents
02/12/2003CN1396916A Process for preparation of quetiapine and intermediates therefor
02/12/2003CN1101397C Preparation of beta-methyl carbepenem intermediate
02/11/2003US6518458 (Aminoiminomethyl) amino) alkane-carboxamides and their applications in therapy
02/11/2003US6518314 Pharmaceutical agents that impede the initiation and progression of primary and secondary DMS disruptions
02/11/2003US6518310 Non-peptidic; inhibits trypsin-like protease, thrombin and embolus formation; anticoagulant
02/11/2003US6518286 Compounds
02/11/2003US6518283 Squaric acid derivatives
02/11/2003US6518272 HT3 receptor agonists and antagonists; treatment of anxiety, depression, cognitive deficits, and prostate cancer
02/11/2003US6518267 Protease inhibitors
02/11/2003US6517811 Compounds for cancer imaging and therapy
02/06/2003WO2003010128A2 Perfluoroalkyl-substituted amines, acids, amino acids and thioether acids
02/06/2003WO2003009897A1 Medicament inhibiting sodium/calcium exchange system
02/06/2003WO2003009849A1 Process for the preparation of 2-(2-(4-(bis(4-fluorophenyl)methyl)-piperazin-1-yl)ethoxy)acetic acid derivatives or corresponding salt forms thereof and intermediates therefor
02/06/2003WO2003009807A2 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods
02/06/2003WO2002032871A3 Compounds and methods for treating multidrug resistance
02/06/2003US20030028026 Nitrate salts of Salbutamol, Cetirizine, Loratadine, Terfenadine, Emedastine, Ketotifen, Nedocromil, Ambroxol, Dextromethorphan, Dextorphan, Isoniazide, Erythromycin, and Pyrazinamide; respiratory system pathology treatment
02/06/2003US20030027862 Amino-and amido-diphenyl ethers
02/06/2003US20030027840 Estrogen receptor modulators
02/06/2003US20030027832 4-Phenyl-1-piperazinyl, -piperidinyl and -tetrahydropyridyl derivatives
02/06/2003US20030027831 Arylpiperzine derivatives are useful for treatment of anxiety, depression, hypertension, cognitive disorders, sexual dysfunction, brain trauma, memory loss, eating disorders, obesity, substance abuse, and obsessive-compulsive diseases
02/06/2003US20030027822 Sodium channel modulators
02/06/2003US20030026521 Optical interleaver
02/06/2003CA2454903A1 Substituted piperazines as modulators of the melanocortin receptor
02/06/2003CA2454681A1 Medicament inhibiting sodium/calcium exchange system
02/06/2003CA2454564A1 Process for the preparation of 2-(2-(4-(bis(4-fluorophenyl)methyl)-piperazin-1-yl)ethoxy)acetic acid derivatives or corresponding salt forms thereof and intermediates therefor
02/06/2003CA2452159A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods
02/05/2003EP1281702A2 Calcium receptor active molecules
02/05/2003EP1280785A1 Phenylsulphonylpiperazinyl derivatives as 5-ht receptor ligands
02/05/2003EP1280764A2 Inhibitors of histone deacetylase
02/05/2003EP1086078B1 Neuropeptide y5 receptor antagonists
02/05/2003EP1082121A4 Hiv integrase inhibitors
02/05/2003CN1395562A Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
02/05/2003CN1395467A Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
02/05/2003CN1394846A Alpha-substituted benzene acetic acid its preparation and farm pesticide containing said compound
02/05/2003CN1100774C Compounds having both potent calcium antagonist and antioxidant activity and use thereof as cytoprotective agents
02/05/2003CN1100767C Macrocyclic metal complex carboxylic acids, use and method for production thereof
02/05/2003CN1100748C Inhibition of matrix metalloproteases by 2-substituted-4-(4-substituted phenyl)-4-oxobutyric acids
02/04/2003US6515180 Method for the catalytic, symmetric disubstitution of carboxylic acid amides with grignard reagents
02/04/2003US6515028 Glucamine compounds for treating hepatitis virus infections
02/04/2003US6515027 Substituted benzanilides as CCR5 receptors ligands, antiinflammatory agents and antiviral agents
02/04/2003US6515024 Succinoylamino hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors
02/04/2003US6514976 Arylpiperazines having activity at the serotonin 1A receptor
02/04/2003US6514975 Anti-inflammatory piperazinyl-benzyl-tetrazole derivatives and intermediates thereof
02/04/2003US6514934 For treating sexual dysfunctions in males and females
02/04/2003CA2272927C Dimesylate salts of neuropeptide y ligands
02/03/2003WO2002016312A2 Novel compounds inhibiting factor xa activity
02/03/2003CA2418283A1 Novel compounds inhibiting factor xa activity
01/2003
01/31/2003WO2002012169A1 Amino diphenyl ethers and amido diphenyl ethers
01/31/2003CA2417880A1 Amino diphenyl ethers and amido diphenyl ethers
01/30/2003WO2003008559A2 Novel analogs of choline for neuroprotection and cognitive enhancement in neurodegenerative disorders
01/30/2003WO2003008399A1 Synthesis of udp-glucose: n-acylsphingosine glucosyltransferase inhibitors