Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
09/2002
09/26/2002US20020137687 Novel compounds that inhibit tryptase activity
09/26/2002DE10114084A1 New 1,3-diamino-4-aminomethyl-benzene derivatives, useful as coupler substances in oxidative hair dye formulations based on a developer-coupler combination
09/26/2002CA2445754A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
09/25/2002EP1243577A1 Novel phenylalanine derivatives
09/25/2002EP1242427A1 Novel piperidine and piperazine derivatives
09/25/2002EP1242400A1 Pyrrolidine derivatives as cyclic amp-specific phosphodiesterase inhibitors
09/25/2002EP1242399A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS
09/25/2002EP1242398A2 Partially saturated calcium channel blockers
09/25/2002EP1242379A1 Curcumin analogues for treating cancer
09/25/2002EP0994710B1 Pharmaceutical compositions for oral administration, comprising a benzhydrylpiperazine and a cyclodextrin
09/25/2002EP0912534B1 Muscarinic antagonists
09/25/2002CN1091438C 0-acyl-4-phenyl-cyclohexanols, their salts, medicaments containing such compounds and their use, as well as method of preparing them
09/24/2002US6455737 Cationic dyes and oxidation bases having intense shades or colors and colorfastness used on human keratin fibers such as hair; multicompartment kits
09/24/2002US6455735 Reacting a tertiary or secondary amine with hydrogen peroxide in presence of a recyclable heterogeneous layered double hydroxide exchanged with one of the anions of transition metal oxides as a catalyst in a solvent
09/24/2002US6455700 Process for preparing guanidine and amidine derivatives
09/24/2002US6455581 Inhibitors of hiv protease.
09/24/2002US6455572 Estrogen agonist/antagonist metabolites
09/24/2002US6455550 N-alkanoylphenylalanine derivatives
09/24/2002US6455533 Substituted benzhydrylpiperazines such as cetirizine, hydroxyzine, efletirizine, meclizine and buclizine, the optically active isomers thereof and the pharmaceutically acceptable salts thereof.
09/24/2002US6455531 Metalloproteinase inhibitors
09/24/2002US6455528 Tumor necrosis factor antagonist and/or interleukin promoter; antiallergens, antiinflammatory agents; autoimmune disease treatment
09/24/2002US6455519 Use of substituted N, N-disubstituted fused-heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
09/24/2002US6455502 Compounds and compositions as protease inhibitors
09/19/2002WO2002072563A1 Extraction of metal salts from aqueous solution
09/19/2002WO2002072545A2 9-aminoacyl tetracycline compounds and methods of use thereof
09/19/2002WO2002072524A2 Method for producing vinyl, aryl and heteroaryl acetic acids and derivatives thereof
09/19/2002WO2002072097A1 Remedies and/or preventives for diabetic ischemic heart diseases
09/19/2002WO2002072084A2 Glycyrrhetinic acid derivatives, progesterone and progesterone derivatives and their use for the manufacture of a medicament to inhibit 11beta-hydroxysteroid dehydrogenase activity
09/19/2002WO2002062308A3 Primary intermediates for oxidative coloration of hair
09/19/2002WO2002055519A3 Novel process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2r, 4r)-4-hydroxy -6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide
09/19/2002WO2001007020A3 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof
09/19/2002US20020133026 Novel process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2r,4r)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide
09/19/2002US20020133012 Therapy for neurokinin sensitive disease
09/19/2002US20020132853 Diaryl piperazines and related compounds useful in the treatment of a chronic and acute pain conditions, itch and urinary incontinence.
09/19/2002US20020132852 Symmetrically disubstituted aromatic compounds and pharmaceutical compositions for inhibiting poly (ADP-ribose) glycohydrolase, and methods for their use
09/19/2002US20020132816 Estrogen agonists/antagonists for preventing breast cancer
09/19/2002US20020131951 Biodegradable poly(beta-amino esters) and uses thereof
09/19/2002US20020131932 Radiopharmaceuticals for diagnosing alzheimer's disease
09/19/2002DE10113027A1 3-Diaminophenyl-acrylamide derivatives or their physiologically acceptable, water-soluble salts, used as developers in combination with couplers in oxidative dye formulations, especially for dyeing hair are new
09/19/2002DE10109204A1 Use of new and known diphenylurea compounds for the preparation of a medicament for the inhibition of intracellular protein-degradation pathway
09/19/2002DE10058461A1 Substituierte Cyclohexanderivate und ihre Verwendung Substituted cyclohexane derivatives and their use
09/19/2002CA2440670A1 Agent for therapeutic and/or prophylactic treatment of diabetic ischemic heart disease
09/19/2002CA2440295A1 Method for producing vinyl, aryl and heteroaryl acetic acids and derivatives thereof
09/18/2002EP1241174A1 Chiral ligands for asymmetric synthesis
09/18/2002EP1241160A1 Tetracycline derivatives and their use as antibiotic agents
09/18/2002EP1241159A1 Aromatic diamide derivatives, chemicals for agricultural or horticultural use and usage thereof
09/18/2002EP1240154A1 Serine protease inhibitors
09/18/2002EP1240143A1 New modulators of dopamine neurotransmission
09/18/2002EP1240142A1 New modulators of dopamine neurotransmission
09/18/2002EP1240141A1 New modulators of dopamine neurotransmission
09/18/2002EP1036059B1 Adamantane derivatives
09/18/2002EP0929516B1 Benzamidine derivatives and the use thereof as medicaments with ltb4-antagonistic effect
09/18/2002EP0804427B1 Lta4 hydrolase inhibitors
09/18/2002CN1091104C Prepn. of N-formyl piperidine
09/17/2002US6452012 3-phenyl-2,6-dioxopiperidin-3-ylpropionamide derivatives and method for preparing same
09/17/2002US6451973 Human immunodeficiency virus (hiv) protease inhibitors
09/17/2002US6451830 Use of substituted N,N-disubstituted non-fused heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
09/17/2002US6451824 Sulfonylaminocarboxylic acids
09/17/2002US6451823 Use of substituted N-phenoxy-N-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
09/17/2002US6451817 Alpha-substituted-1-benzyl-napthyls
09/17/2002US6451803 N-acyl and n-aroyl aralkyl amides useful in treating seritonergic disorders
09/17/2002US6451801 Compounds and methods for treatment of asthma, allergy and inflammatory disorders
09/17/2002US6451798 Substituted alkyl piperazine derivatives
09/17/2002US6451792 Matrix metalloprotease inhibitors
09/17/2002US6451791 Amidoaromatic ring sulfonamide hydroxamic acid compounds
09/17/2002US6451068 Oxidative color dyes for hair
09/17/2002CA2182241C Methods for the manufacture of nefazodone
09/12/2002WO2002070541A2 Peptide deformylase inhibitors
09/12/2002WO2002070496A1 Nitric oxide donors based on metallic centres
09/12/2002WO2002070492A1 New asymmetric process for the preparation of diarylmethylpiperazines derivatives and novel asymmetric diarylmetylamines as intermediates
09/12/2002WO2002070470A2 Benzophenones as inhibitors of reverse transcriptase
09/12/2002WO2002070467A1 Derivatives of diphenylurea, diphenyloxalic acid diamide and diphenylsulfuric acid diamide and their use as medicaments
09/12/2002WO2002070456A1 Benzene-1 2-diol mannich bases ligands polymers and method of selective metal ions removal
09/12/2002WO2002069937A1 Compounds and compositions for delivering active agents
09/12/2002WO2002069901A2 Cathepsin cysteine protease inhibitors
09/12/2002WO2002048122A3 Benzamidine derivatives
09/12/2002WO2002044113A3 Use of(-) (3-halomethylphenoxy) (4-halophenyl) acetic acid derivatives for treatment of insulin resistance, type 2 diabetes, hyperlipidemia and hyperuricemia
09/12/2002WO2002012213A3 (meth)acrylic acid derivatives and their polymers suitable for use in the manufacture of paper
09/12/2002US20020128499 Alkylthio-substituted benzoquinones by oxidizing with an alkali periodate in the presense of a phase transfer catalyst; Protective agents for rubber vulcanizates; aging and ozone resistance; fatigue; stabilizers
09/12/2002US20020128495 Carboxylic acid amides, pharmaceutical compositions containing these compounds, their use and the preparation thereof
09/12/2002US20020128434 Alpha-(1,3-dicarbonylenol ether) methyl ketones as cysteine protease inhibitors
09/12/2002US20020128308 Useful as medicines having an osteogenesis promoting effect and chondrogensis promoting effect.
09/12/2002US20020128275 Intermediates for the production of antiallergic pharmaceuticals
09/12/2002US20020128269 Piperazine derivatives
09/12/2002US20020128255 Substituted hydroxyl amine derivatives; inhibitors of beta-secretase, inhibit beta-secretase-mediated cleavage, inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques
09/12/2002US20020128247 Phenyl sulfamide derivatives as dietetics, antidiabetics, and hypotensive agents
09/12/2002US20020128231 Aryl-indane compounds
09/12/2002US20020128208 Such as 4-benzoylamino-(2-(2-hydroxyethyl)-piperazin-1-yl-methyl)-phenyl)-benzene -sulfonamide; for treatment of hypertension; treatment of kidney disorders
09/12/2002US20020127582 Generating adenovirus-associated vector; obtain cells, transform with expression vector, propagate, recover transformed cells, propagate and recover vectors
09/12/2002US20020127202 Compounds and compositions for delivering active agents
09/12/2002DE10111262A1 Verfahren zur Herstellung von Vinyl- Aryl- und Heteroarylessigsäuren und ihrer Devivate Process for the preparation of vinyl aryl and heteroaryl and its Devivate
09/12/2002CA2440104A1 New asymmetric process for the preparation of diarylmethylpiperazines derivatives and novel asymmetric diarylmetylamines as intermediates
09/12/2002CA2439827A1 Peptide deformylase inhibitors
09/12/2002CA2439820A1 Benzophenones as inhibitors of reverse transcriptase
09/12/2002CA2439634A1 Benzene-1 2-diol mannich bases ligands polymers and method of selective metal ions removal
09/12/2002CA2438849A1 Compounds and compositions for delivering active agents
09/11/2002EP1238966A2 Hair cosmetic, aminocarboxylic acid amide and method for producing the same
09/11/2002EP1237868A1 Hydroxamic acid derivatives as matrix metalloproteinase (mmp) inhibitors
09/11/2002EP1237867A1 Hydroxamic acid derivatives as matrix metalloproteinase (mmp) inhibitors
09/11/2002EP1237859A2 Use of bis-sulfonamides for producing medicaments used for preventing or treating hyperlipidaemia