Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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09/11/2002 | EP1237852A1 N-phenylcarbamates having a microbicide, insecticide and acaricide effect |
09/11/2002 | EP1237849A1 Activators of soluble guanylate cyclase |
09/11/2002 | EP1177199B1 Ionic liquids and production and use thereof |
09/11/2002 | EP0958287B1 Sulfamide-metalloprotease inhibitors |
09/11/2002 | EP0813529B1 Arginine analogues having nitric oxide synthase inhibitor activity |
09/11/2002 | EP0799206B1 Aryl- and hetaryl-sulfonamide derivatives, their preparation and their use as endothelin antagonists |
09/11/2002 | EP0736009B1 N-oxides of 4-arylpiperazines and 4-arylpiperidines as antipsychotic drugs |
09/11/2002 | CN1368958A Arylsulfonamido-substituted hydroxamic acid derivatives |
09/11/2002 | CN1368956A Carbamate derivatives and agricultural/horticultural bactericides |
09/11/2002 | CN1368498A Preparation method of o-chloromethyl phenyl glyoxalic acid derivative |
09/11/2002 | CN1368497A Preparation method of o-chloromethyl phenyl glyoxalic acid derivative |
09/11/2002 | CN1090480C Phenoxy piperazine derivatives for treating disorders of dopamine system |
09/10/2002 | US6448445 Method for catalytically disubstituting carboxylic acid amides with at least one grignard reagent |
09/10/2002 | US6448373 Inhibitors of enzymes such as phospholipase a2; treatment of inflammatory diseases including atopic dermatitis and inflammatory bowel disease |
09/10/2002 | US6448295 Treating cardiovascular disease; atherosclerosis, dyslipidema hypercholesterolaemia; decreasing concentrations of low density lipoprotein and raising level of high density lipoprotein |
09/10/2002 | US6448293 Treatment or prevention of a disorder in which the regulation of monoamine transporter function is implicated, such as premature ejaculation. |
09/10/2002 | US6448250 Sulfamato hydroxamic acid metalloprotease inhibitor |
09/10/2002 | US6448244 Broad-spectrum antifungals, against which there is no existing resistance and which can be administered intravenously or transungually |
09/10/2002 | US6448243 Serotonin antagonist for treating, ameliorating and preventing spastic paralysis or central muscle relaxants for ameliorating myotonia |
09/10/2002 | US6448242 Cyclic amide compounds |
09/10/2002 | US6447748 Benzamide compounds for cancer imaging and therapy |
09/10/2002 | CA2239159C Acylated enol derivatives of .alpha.-ketoesters and .alpha.-ketoamides |
09/10/2002 | CA2198562C Method of treating conditions with estrogen agonists |
09/06/2002 | WO2002068399A1 Aryl carbamate derivatives, preparation and use thereof |
09/06/2002 | WO2002068390A1 Diamides which inhibit tryptase and factor xa activity |
09/06/2002 | WO2002068381A2 Aryl-n-cyanoguanidines and methods related thereto |
09/06/2002 | WO2002068377A1 Omega-aminoalkylamides of r-2-aryl-propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells |
09/06/2002 | WO2002068367A1 A method to inhibit ethylene responses in plants |
09/06/2002 | WO2002067919A1 Il-8 receptor antagonists |
09/06/2002 | WO2002043648A8 Compounds active at the glucocorticoid receptor ii |
09/06/2002 | WO2002032868A3 2-substituted heterocyclic compounds and their use in treating multidrug resistance |
09/06/2002 | WO2002022577A3 Hydroxamate derivatives useful as deacetylase inhibitors |
09/06/2002 | WO2001018011A9 Calcium complex of phosphorus containing ethylenediamine derivatives |
09/06/2002 | CA2475454A1 Aryl-n-cyanoguanidines and methods related thereto |
09/06/2002 | CA2438828A1 Aryl carbamate derivatives, preparation and use thereof |
09/06/2002 | CA2437114A1 Diamides which inhibit tryptase and factor xa activity |
09/05/2002 | US20020123637 Pharmaceutically active compounds and methods of use thereof |
09/05/2002 | US20020123498 For inhibiting transport protein; therapy |
09/05/2002 | US20020123489 Benzamidine derivatives |
09/04/2002 | EP1236723A1 Sulfamide derivatives useful as beta3 agonists and pharmaceutical uses thereof |
09/04/2002 | EP1236722A1 Optically active 4-(tert-butoxycarbonyl) piperazine compound, and method for producing the same |
09/04/2002 | EP1235831A2 New oxabispidine compounds useful in the treatment of cardiac arrhythmias |
09/04/2002 | EP1235807A1 B-amino acid-, aspartic acid- and diaminopropionic-based inhibitors of factor xa |
09/04/2002 | EP1235793A2 Vla-4 integrin antagonists |
09/04/2002 | EP1235776A1 Triphenylalkene derivatives and their use as selective estrogen receptor modulators |
09/04/2002 | EP1235764A1 Catalysis using phosphine oxide compounds |
09/04/2002 | EP1235575A2 Agent for expression of long-term potentiation of synaptic transmission comprising compound having brain somatostatin activation property |
09/04/2002 | EP0635008B1 Piperazides of substituted phenylalanine derivates as thrombin inhibitors |
09/04/2002 | CN1367783A Antipsychotic cyclic N-aralkyl amines |
09/03/2002 | US6444819 Benzylpiperazinyl and piperidinyl ethanone derivatives: dopamine receptor subtype specific ligands |
09/03/2002 | US6444704 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors |
09/03/2002 | US6444701 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase |
09/03/2002 | US6444678 α- and β-amino acid hydroxyethylamino sulfamic acid derivatives useful as retroviral protease inhibitors |
09/03/2002 | US6444190 Slurry of a sodium aluminum hydride, lithium or titanium containing additive and a lewis base in solvent; non-pyrophoric; thermal stability |
09/03/2002 | CA2140626C Hydroxamic acid derivatives as metalloproteinase inhibitors |
09/01/2002 | CA2373578A1 .beta.3, agonists and uses thereof |
09/01/2002 | CA2356201A1 Compounds and compositions for delivering active agents |
08/29/2002 | WO2002066469A2 Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands |
08/29/2002 | WO2002066451A2 1,2-diphenyl-1-naphthyl ethene derivatives, analogs and use thereof |
08/29/2002 | WO2002066446A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands |
08/29/2002 | WO2002066432A1 Substituted propane-1,3-diamine derivatives and the pharmaceutical use thereof |
08/29/2002 | WO2002066428A2 Non-steroidal estrogen receptor ligands |
08/29/2002 | WO2002066422A1 Phenethanolamine derivatives for treatment of respiratory diseases |
08/29/2002 | WO2002066415A2 Non-steroidal modulators of estrogen receptors |
08/29/2002 | WO2002040466A3 Amidoalkyl-piperidine and amidoalkyl-piperazine derivatives for treating of nervous systems disorders |
08/29/2002 | WO2002002520A3 Compounds to treat alzheimer's disease |
08/29/2002 | WO2002002506A3 Compounds to treat alzheimer's disease |
08/29/2002 | WO2001012584A3 Pharmaceutical compounds |
08/29/2002 | WO1999064055A9 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht4 receptors |
08/29/2002 | US20020120148 Benzocycloheptenylamino derivatives; treatment of pollakiuria or urinary incontinence |
08/29/2002 | US20020120140 Phosgene-free process for preparing carbamates |
08/29/2002 | US20020120011 Substituted N, N-disubstituted diamino compounds useful for inhibiting cholesteryl ester transfer protein activity |
08/29/2002 | US20020120007 Benzamide inhibitors of factor Xa |
08/29/2002 | US20020119988 Modulators of TNF-alpha signaling |
08/29/2002 | US20020119979 Cancer therapy |
08/29/2002 | US20020119960 Drug resistance therapy |
08/29/2002 | US20020119953 Sickle cell anemia |
08/29/2002 | US20020119910 Drug delivery |
08/29/2002 | DE19941540C2 Sulfonylcarboxamide zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Hyperlipidämie Sulfonylcarboxamide for the preparation of medicaments for the prophylaxis or treatment of hyperlipidemia |
08/29/2002 | DE10108307A1 Substituierte Propan-1,3-diamin-Derivate Substituted propane-1,3-diamine derivatives |
08/29/2002 | CA2438318A1 Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands |
08/29/2002 | CA2438264A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands |
08/29/2002 | CA2437977A1 Phenethanolamine derivatives for treatment of respiratory diseases |
08/28/2002 | EP1233961A2 Method for producing 5-(1-piperazinyl)-benzofuran-2-carboxamide by transition metal-catalyzed amination |
08/28/2002 | EP1233955A1 Process for preparing piperazine-substituted aliphatic carboxylates |
08/28/2002 | EP1233954A1 A process for the preparation of 2- 4-(alpha-phenyl-p-chlorobenzyl)piperazin-1-yl]ethoxy acetic acid and novel intermediates therefor |
08/28/2002 | EP0868202B1 Cascade polymer complexes, process for producing the same and pharmaceuticals containing the same |
08/28/2002 | CN1366518A Biphenyl butyric acid derivative as matrix metalloproteinase inhibitor |
08/27/2002 | US6441237 Drugs; antiarrhthymia agents, antiischemic agents |
08/27/2002 | US6441193 Intermediates such as 1-(2-(4-(6-methoxy-3,4-dihydronaphtha-len-1-yl)phenoxy)ethyl)pyrrolidine and compounds such as cis-6-phenyl-5-(4-(2-pyrrolidin-1-ylethoxy)phenyl)-5,6,7,8 -tetrahydronaphthalen-2-ol, hydrobromide salt |
08/27/2002 | US6441179 Intermediates useful for the preparation of antihistaminic piperidine derivatives |
08/27/2002 | US6441049 Administering compound effective to inhibit binding of an amyloid beta peptide with alpha-7 nicotinic acetylcholine receptors |
08/27/2002 | US6441042 Hydroxamic acid derivatives as antibacterials |
08/27/2002 | US6441023 For therapy of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone disease, diabetes (insulin resistance) and hiv infection |
08/27/2002 | CA2224738C Use of ritonavir (abt-538) for improving the pharmacokinetics of drugs metabolized by cytochrome p450 in a method of treating aids |
08/22/2002 | WO2002064576A1 Heteroaryl alkyl piperazine derivatives as fatty acid oxidation inhibitors |
08/22/2002 | WO2002064551A1 Hiv protease inhibitors based on amino acid derivatives |
08/22/2002 | WO2002064550A1 Glucocorticoid receptor modulators |
08/22/2002 | WO2002064546A2 Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical |
08/22/2002 | WO2002064545A1 Acylated indanyl amines and their use as pharmaceuticals |