Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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09/03/2003 | CN1440396A Colchinol derivatives as angiogenesis inhibitors |
09/03/2003 | CN1440395A COLCHINOL derivatives as vascular damaging agents |
09/03/2003 | CN1440390A Substituted diamide derivatives useful as motilin antagonists |
09/03/2003 | CN1440383A PPARγ调制剂 PPARγ modulators |
09/02/2003 | US6613944 Process to produce 3-carbon amino alcohol salts |
09/02/2003 | US6613942 Glucagon antagonists/inverse agonists |
09/02/2003 | US6613805 For therapy and prophylaxis of neurodegenerative diseases such as Alzheimer's disease, Down's syndrome, Parkinson's disease, Creutzfeldt-Jacob disease, amyotrophic sclerosis on lateral fasciculus, multiple sclerosis, and neurological disorders |
09/02/2003 | US6613796 Use of estrogen antagonists and estrogen agonists in inhibiting pathological conditions |
09/02/2003 | US6613769 Tryptase inhibitors |
09/02/2003 | US6613764 Aspartic protease inhibitors |
09/02/2003 | US6613729 Comprising organic counterion of sunflower seed-amidopropyl morpholine |
09/02/2003 | US6613572 Agent for expression of long-term potentiation of synaptic transmission comprising compound having brain somatostatin activation property |
09/02/2003 | US6613458 Benzo(a)perylene derivative dopant |
08/28/2003 | WO2003070713A1 Substituted aryl alkenoic acid heterocyclic amides possessing pungent taste |
08/28/2003 | WO2003070690A2 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative |
08/28/2003 | WO2003070675A2 Substituted 10-aryl-11h-benzo[b]fluorenes and 7-aryl-5,6-dihydro-benzo[a]anthracenes for selective effects on estrogen receptors |
08/28/2003 | WO2003070220A1 Ph-sensitive cationic lipids, and liposomes and nanocapsules containing the same |
08/28/2003 | WO2003017998B1 Platinum complexes and their use in cancer treatment |
08/28/2003 | US20030162830 3,4-diphenyl-bicyclo(4.3.0)nonyl derivatives |
08/28/2003 | US20030162820 Heterocyclic amides used as dipeptidyl aminopeptidase (DPIV) inhibitors, for prophylaxis of arthritis, obesity, allograft surgery, cancer, autoimmune, nervous system and skin disorders |
08/28/2003 | US20030162817 Pentafluorobenzenesulfonamides and analogs |
08/28/2003 | US20030162799 Squaric acid derivatives |
08/28/2003 | US20030162793 Methods for preventing or treating cardiac arrhythmia |
08/28/2003 | US20030162778 Carbocyclic side chain containing metalloprotease inhibitors |
08/28/2003 | US20030161860 Novel substituted aryl alkenoic acid heterocyclic amides |
08/28/2003 | CA2474785A1 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative |
08/27/2003 | EP1337519A1 Process for the preparation of 1,5-disubstituated-3-amino-1,2,4-triazoles and substituted aminoguanidines as intermediate compounds |
08/27/2003 | EP0901469B1 Arylalkylpiperazine compounds as antioxidants |
08/27/2003 | EP0874809B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials |
08/27/2003 | CN1438999A Serine protease inhibitors |
08/27/2003 | CN1438897A Remedial agent for anxiety neurosis or depression and piperazine derivative |
08/27/2003 | CN1438883A Beta Secretase inhibitors |
08/27/2003 | CN1119338C Alpha-(1-piperazinyl) ocetamido arenecarboxylic aicd derivatives as antidiabetic agents |
08/27/2003 | CN1119336C Novel compounds with analgesic effect |
08/27/2003 | CN1119149C 10,11 methanodibenzosuberane derivatives used as chemo sensitizing agents |
08/26/2003 | US6610882 Affinity for bradykinin receptors; antithrombotics |
08/26/2003 | US6610850 Contrast media for angiography |
08/26/2003 | US6610715 Cathecol hydrazone derivatives, process for preparing the same and pharmaceutical composition containing the same |
08/26/2003 | US6610710 Inflammatory bowel diseases, diabetes, tumor proliferation and tumor metastasis. |
08/26/2003 | US6610705 Process for the preparation of diaryl naphthyl methanes |
08/26/2003 | US6610704 Antithrombotic amides |
08/26/2003 | US6610702 Ammonium salts of inositol hexaphosphate, and uses thereof |
08/26/2003 | US6610689 Viricides |
08/26/2003 | US6610660 O2-arylated or O2-glycosylated 1-substituted diazen-1-ium-1,2-diolates and O2-substituted 1-[(2-carboxylato) pyrrolidin-1-yl] diazen-1-ium-1,2-diolates |
08/21/2003 | WO2003068759A1 Piperazine derivatives as anti-inflammatory agents |
08/21/2003 | WO2003068217A1 Biphenil derivatives and their use as antiandrogenic agents |
08/21/2003 | WO2003018549A3 Bicyclic compounds as inhibitors of chemokine binding to us28 |
08/21/2003 | WO2003007930A3 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors |
08/21/2003 | WO2002002512A3 Compounds to treat alzheimer's disease |
08/21/2003 | US20030158406 Enzyme inhibitor treating autoimmune diseases, Alzheimer's disease, atherosclerosis |
08/21/2003 | US20030158252 Especially trypsin-like serine proteases, such as chymotrypsin, trypsin, thrombin, plasmin and factor Xa. |
08/21/2003 | US20030158236 Treating, e.g., an HIV infection. |
08/21/2003 | US20030158231 Sulfonamide compounds as protease inhibitors |
08/21/2003 | US20030158225 Novel compounds |
08/21/2003 | US20030158209 Amidomethylcarbonyl-substituted piperazine derivatives containing additional amine groups, useful in treating eating, sexual and skin disorders |
08/21/2003 | US20030158208 Dopamine D4 ligands for the treatment of novelty-seeking disorders |
08/21/2003 | US20030158207 N-benzylpiperazine compounds |
08/21/2003 | US20030158205 N-benzyl-substituted, e.g., (2S)-1-(p-chlorophenoxy)methyl)-carbonyl-2-methyl-4-(p -fluorobenzyl)piperazine; inhibit the activity of the chemokines, MIP-1 alpha and RANTES |
08/21/2003 | US20030158202 Substituted fused ring sulfonamides containing, e.g., naphthalene, isoquinoline, quinoline, benzofuran or benzothiophene rings; treatment of conditions relating to obesity, type II diabetes and CNS disorders |
08/21/2003 | US20030158186 Compositions and methods for treating heart failure |
08/21/2003 | US20030158185 Novel use of phenylheteroakylamine derivatives |
08/21/2003 | US20030158180 Antidepressants; treating anxiety, stress, eating disorders, bipolar disorder, drug abuse and drug dependence, schizophrenic disorders, psychotic disorders, cognitive activators, obesity, emesis, rheumatoid arthritis, cancer |
08/21/2003 | US20030158176 Quaternary ammonium compounds |
08/21/2003 | CA2474171A1 Biphenil derivatives and their use as antiandrogenic agents |
08/20/2003 | EP1336608A1 Dibenzosberanyl piperazine derivatives and drug-resistance overcoming agents containing the derivatives |
08/20/2003 | EP1204592B1 Zeolite ssz-52 |
08/20/2003 | EP1194415B1 Novel piperazinylalkylthiopyrimidine derivatives, pharmaceutical compositions containing the same, and a process for their preparation |
08/20/2003 | EP1150944B1 N2-phenylamidine derivatives |
08/20/2003 | CN1437589A Process for the preparation of pyrazolopyrimidin ones |
08/20/2003 | CN1437578A (P-amino-hyaroxyphenyl)-acrylamide derivatives and dyes containing said compounds |
08/19/2003 | US6608212 Palladium catalyzed coupling of a vinylphosphate and aryl-metal halide; preparation of such as 1-(4-(2-(pyrrolidin-n-yl)-ethoxy)phenyl)-6-methoxy-3,4-dihydronaphthalene |
08/19/2003 | US6608196 Structurally diverse; parallel approach |
08/19/2003 | US6608195 Process for the preparation of 2-(4-alkyl-1-piperazinyl)-benzaldehyde and -benzylidenyl compounds |
08/19/2003 | US6608100 HIV protease inhibitors based on amino acid derivatives |
08/19/2003 | US6608066 Tissue factor antagonists and methods of use thereof |
08/19/2003 | US6608057 Compounds useful as reversible inhibitors of cathepsin S |
08/19/2003 | US6607868 Photoresist monomers, polymers thereof, and photoresist compositions containing the same |
08/14/2003 | WO2003066889A2 Assay for acytyltransferase or deacetylase activity |
08/14/2003 | WO2003066613A1 N-phenyl-2-pyrimidine-amine derivatives |
08/14/2003 | WO2003066604A2 Novel aryl- and heteroarylpiperazines |
08/14/2003 | WO2003066579A2 Novel bicyclic hydroxamates as inhibitors of histone deacetylase |
08/14/2003 | WO2003066570A1 Transition-metal-catalyzed carbon-nitrogen bond-forming methods using carbene ligands |
08/14/2003 | WO2003066056A1 Method of promoting neuronal growth |
08/14/2003 | WO2003066035A2 Compounds for inhibiting insulin secretion and methods related thereto |
08/14/2003 | WO2003065989A2 (oxime)carbamoyl fatty acid amide hydrolase inhibitors |
08/14/2003 | WO2003031408A3 Tricyclic compounds useful for modulating lxr |
08/14/2003 | WO2003024945A3 Method for producing polyphosphates of organic bases |
08/14/2003 | US20030153788 Oxidizing an amino alcohol (obtained by ring opening the epoxy, aziding, reducing and reacting it with a carboxylic acid); stereoselectivity; protease inhibitors: antiallergens; anticarcinogenic and hypotensive agents |
08/14/2003 | US20030153781 Increased enantioselectivity of asymmetric addition of organic zinc and aldehyde by providing ligands to perform as superior catalysts to form a predominance of secondary alcohol; efficiency |
08/14/2003 | US20030153780 Water-soluble specialty surfactants to lower the surface tension of water to <20 dynes/cm.; reacting amines with allyl glycidyl ether, followed by reaction with a perfluoroalkyl iodide; oily surfaces; coatings for addition polymers |
08/14/2003 | US20030153768 Efficient synthesis of ceramide-like compounds by reacting an aldehyde and an amidomethylisonitrile to form a 4-amido-2-oxazoline; suppress biosynthesis of glycosphingolipids; antitumor agents; Tays-Sach, Gaucher's |
08/14/2003 | US20030153596 Novel thiourea derivatives and the pharmaceutical compositions containing the same |
08/14/2003 | US20030153577 Cyclic amine derivatives-CCR-3 receptor antagonists |
08/14/2003 | US20030153568 Serine/threonine and tyrosine kinases inhibitors |
08/14/2003 | US20030153564 New oxabispidine compounds useful in the treatment of cardiac arrhythmias |
08/14/2003 | US20030153559 Treatment of an oxygen and/or energy deficit; a poly(adenosine diphosphate ribose)-polymerase inhibitor; treating autoimmune, neurodegenerative and diseases caused by a toxic effect; viricides |
08/14/2003 | US20030153537 Reducing tetracycline resistance in living cells |
08/14/2003 | US20030153510 Novel compounds inhibiting factor xa activity |
08/14/2003 | US20030153507 HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis |
08/14/2003 | CA2737565A1 N-phenyl-2-pyrimidine-amine derivatives |