Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
10/2002
10/10/2002WO2002057215A3 Sodium channel modulators
10/10/2002WO2002053516A3 N(phenylsulphonyl)glycine derivatives and their therapeutic use
10/10/2002WO2001072728A9 Novel piperazine derivatives
10/10/2002US20020147359 Neurokinin antagonist; antiinflammatory agents, antiallergens
10/10/2002US20020147342 Alkynyl containing hydroxamic acid compounds as matrix metalloproteinase and tace inhibitors
10/10/2002US20020147336 Glucocorticoid receptor modulators
10/10/2002US20020147193 Novel couplers for use in oxidative hair dyeing
10/10/2002US20020147187 Antiproliferative agents; anticancer agents
10/10/2002US20020147186 Side effect reduction
10/10/2002US20020144361 Novel couplers for use in oxidative hair dyeing
10/10/2002US20020144359 Derivatives of 2-aminophenol; providing good oxidative coloration of hair and for providing acceptable light fastness, selectivity, fastness to shampooing
10/10/2002US20020144358 2-substituted-4-amino-phenol derivative compounds providing good oxidative coloration of hair and acceptable light fastness, fastness to shampooing and permanent wave treatment
10/10/2002US20020144357 Benzene-1,4-diamine compounds having a weaker sensitization potential than p-phenylenediamine
10/10/2002DE10116768A1 Hypoglycemic medicaments useful for treating type II diabetes contain new or known N-aroyl-N'-phenyl-urea derivatives which are glycogen phosphorylase a inhibitors
10/10/2002DE10115994A1 (p-Amino-hydroxyphenyl)acrylamid-Derivate und diese Verbindungen enthaltende Färbemittel (P-amino-hydroxyphenyl) acrylamide derivatives and compositions containing these compounds colorant
10/10/2002CA2443304A1 (p-amino-hydroxyphenyl)-acrylamide derivatives and dyes containing said compounds
10/09/2002EP1246847A2 Dna encoding a human melanin concentrating hormone receptor (mch1) and uses thereof
10/09/2002EP1246819A1 A method for the preparation of substituted benzene derivatives
10/09/2002EP1246817A1 4-phenyl-1-piperazinyl, -piperidinyl and -tetrahydropyridyl derivatives
10/09/2002EP1246803A1 Piperidine and piperazine derivatives which function as 5-ht 2a? receptor antagonists
10/09/2002EP1246795A2 Antibacterial agents
10/09/2002EP1246790A1 Substituted 1 and 2 naphthol mannich bases
10/09/2002EP1246625A2 Methods and compositions for mitigating pain using nitrate esters
10/09/2002EP0882704B1 3,4-disubstituted phenylethanolaminotetralincarboxamide derivatives
10/09/2002EP0874836B1 Sulfonamide inhibitors of matrix metalloproteinases
10/09/2002CN1373765A Calcium complex of phosphorus contg. ethylenediamine derivs.
10/09/2002CN1373754A Antibacterial agents
10/09/2002CN1373750A 2'-substd. 1,1'-biphenyl-2-carbonamides, method for production thereof, use thereof as medicament and pharmaceutical preparation contg. said compounds
10/09/2002CN1373747A Process for making amine componds
10/08/2002US6462198 Used in the control or prevention of acute and/or chronic neurological disorders such as restricted brain function caused by bypass operations or transplants, poor blood supply to the brain, spinal cord injuries, head injuries, hypoxia,
10/08/2002US6462092 Such as 3-((3-fluorophenyl)-((3-(trifluoromethyl)phenyl)-methyl)amino)-1,1,1 -trifluoro-2-propanol; cardiovascular disease, i.e. atherosclerosis and other coronary artery diseases
10/08/2002US6462073 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
10/08/2002US6462064 Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents, especially for cervical cancers and dysplasias
10/08/2002US6462056 Oxazolidines as 5-HT2A-antagonists
10/08/2002US6462042 Tumor necrosis factor alpha converting enzyme inhibitors; inflammatory diseases, autoimmune diseases, cancer, cardio-vascular diseases, rheumatoid arthritis, osteoarthritis, osteoporosis, neurodegeneration, alzheimer's disease, stroke
10/08/2002CA2081766C Leukotriene b4 antagonists
10/03/2002WO2002077609A2 Identification of compounds for the treatment or prevention of proliferative diseases
10/03/2002WO2002076968A1 Malonates as inhibitors of the ice/ced-6 family of cysteine proteases
10/03/2002WO2002076965A1 Non peptide mimetics based on the active sequence s42fllr46 of the thrombin receptor for the treatment of thrombosis and cancer
10/03/2002WO2002076964A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
10/03/2002WO2002076947A1 Mch antagonists and their use in the treatment of obesity
10/03/2002WO2002076929A1 Aryl and biaryl compounds having mch modulatory activity
10/03/2002WO2002076926A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc chemokine receptor antagonists
10/03/2002WO2002076925A2 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
10/03/2002WO2002076924A1 Ionic liquid, electrolyte salt for storage device, electrolytic solution for storage device, electric double layer capacitor, and secondary battery
10/03/2002WO2002076923A1 1,3-diamino-4-(aminomethyl)-benzene derivatives and colorants containing said compounds
10/03/2002WO2002076918A1 NF-λB INHIBITOR CONTAINING SUBSTITUTED BENZOIC ACID DERIVATIVE AS ACTIVE INGREDIENT
10/03/2002WO2002076916A1 Self-reducing anthraquinone compounds
10/03/2002WO2002076450A1 Dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
10/03/2002WO2002076447A1 Hallogenated aminobenzophenones and aminobenzoylpyridines as inhibitors of il-1 and tnf
10/03/2002WO2002062784A8 Piperidinee derivatives as neurokinin 1 antagonists
10/03/2002WO2002062766A3 Melanocortin-4 receptor binding compounds and methods of use thereof
10/03/2002WO2002030880A3 N-substituted amino acid derivatives (factor xa inhibitors)
10/03/2002US20020143177 For inhibiting beta-secretase enzyme activity and A beta peptide production, inhibition of beta-secretase enzyme activity halts or reduces production of A beta from APP and reduces or eliminates the formation of beta-amyloid deposits
10/03/2002US20020143056 As inactivator of antigen- specific T cells is useful in the prophylaxis or therapy of autoimmune diseases, disorders involving an autoimmune component or neoplastic diseases
10/03/2002US20020143036 Pentafluorobenzenesulfonamides and analogs
10/03/2002US20020143020 Novel piperazine derivatives
10/03/2002US20020143003 As serotonin, norepinephrine and dopamine reuptake inhibitors, for therapy of central nervous system and other disorders
10/03/2002US20020142969 Using didepsipeptide for the control of endoparasites in medicine and veterinary medicine
10/03/2002US20020142947 By muta-synthesis using a mutated micro-organism to influence the biosynthesis of at least one of the precursors of group B streptogramines; mutant strain employed is preferably derived from the strain S. pristinaespiralis SP92
10/03/2002US20020138919 Novel couplers for use in oxidative hair dyeing
10/03/2002CA2443289A1 1,3-diamino-4-(aminomethyl)-benzene derivatives and colorants containing said compounds
10/03/2002CA2441092A1 Dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
10/03/2002CA2441080A1 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
10/03/2002CA2436351A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc chemokine receptor antagonists
10/03/2002CA2410816A1 Nf-.kappa.b inhibitor containing substituted benzoic acid derivative as active ingredient
10/02/2002EP1245568A1 Sulfonyl derivatives of amino acids and their use as inhibitors of dipeptidyl-peptidase IV (DPP IV)
10/02/2002EP1245561A1 N-substituted benzyl or phenyl aromatic sulfamides compounds and the use thereof
10/02/2002EP1245550A1 Novel selective deacetylating agents
10/02/2002EP1244643A1 Tryptase inhibitors
10/02/2002EP1244624A1 Anthracene derivatives as anti-cancer agents
10/02/2002EP1244617A1 Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
10/02/2002EP1244451A1 Substituted piperazine and piperidine calcium channel blockers
10/02/2002EP0871465B1 Use of ritonavir (abt-538) for improving the pharmacokinetics of drugs metabolized by cytochrome p450 in a method of treating aids
10/02/2002CN1372541A Sulfonyl carboxamide derivatives, method for their production and their use as medicaments
10/02/2002CN1372539A Quaternary bis-ammonium salt precursors and their uses as prodrugs having an antiparasitic activity
10/01/2002US6458957 α,α-dibromo-α-chloro-acetophenones as synthons
10/01/2002US6458953 Valency platform molecules comprising carbamate linkages
10/01/2002US6458852 Use of substituted N, N-bis-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
10/01/2002US6458849 Method of treating or preventing a ceip-mediated disorder in a subject by administering a therapeutically effective amount of a compound for strokes
10/01/2002US6458806 Aryl alkenamides derivatives as MCP-1 antagonists
10/01/2002US6458803 Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
10/01/2002US6458787 Novel pyrrolidine compounds that are potent and selective inhibitors of pde4, as well as methods of making the same, are disclosed. use of the compounds in the treatment of inflammatory diseases and other diseases involving elevated
10/01/2002US6458781 Blockers calcium channel antagonists for strokes, brain disorders
10/01/2002CA2203850C Novel n-phenyl-n-phenyliminonethylbenzamidines and their analogues as muscarinic receptor agonists
09/2002
09/26/2002WO2002074756A2 Urokinase inhibitors
09/26/2002WO2002074755A1 Method of producing n-substituted 2,6-dialkyl morpholines
09/26/2002WO2002074743A1 Aryl-substituted alicyclic compound and medical composition comprising the same
09/26/2002WO2002074740A1 Biguanide derivatives
09/26/2002WO2002074731A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
09/26/2002WO2002074296A1 Remedies for solid cancer containing hydroxamic acid derivatives as the active ingredient
09/26/2002WO2002034698A3 Phosgene-free process for preparing carbamates
09/26/2002WO2002028810A3 Retinoids for the treatment of emphysema
09/26/2002WO2002024636A3 N-acylsulfonamide apoptosis promoters
09/26/2002WO2002018334B1 Sodium channel modulators
09/26/2002WO1997019953A8 New lh-rh antagonists with improved effectiveness
09/26/2002US20020137974 Catalysis using phosphine oxide and sulfoxide compounds
09/26/2002US20020137939 Novel guanidinobenzamides
09/26/2002US20020137774 Carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
09/26/2002US20020137742 Benzenesulfonamide compounds