Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
07/2003
07/01/2003US6586627 N-protected/N-substituted-beta-amino hydroxy sulfonates
07/01/2003US6586599 Catalyzed coupling reactions of aryl halides with silanes
07/01/2003US6586598 α, α-dibromo-α-chloro-acetophenones as synthons
07/01/2003US6586592 Bis-arylsulfones
07/01/2003US6586475 5-chloro-N-(2-N,N-diethylamino)ethyl)-2- methoxy-4-(1-naphthoylamino)benzamide and prodrugs, used for prevention of neurodegenarative diseases such as Alzheimer's disease
07/01/2003US6586466 Carbohydrazide-protease inhibitors
07/01/2003US6586454 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
07/01/2003US6586433 Anticholesterol agents; antilipemic agents; cardiovascular disorders
07/01/2003US6586432 Neurokinin-1 receptor antagonists
07/01/2003US6586418 Heteroaryl-phenyl substituted compounds that are inhibitors of trypsin-like serine protease enzymes; anticoagulant for treatment and prevention of thromboembolic disorders
07/01/2003US6586187 2-benzyloxycarbonylamino-3-(2-(4-(2-(3-benzylureido)-ethyl) -piperazin-1-yl)acetylamino)-propionic acid, for example; method of synthesis using Wang resins; various uses including anticancer, antiinflammatory and antiviral agents
06/2003
06/26/2003WO2003051855A1 N,n'-disubstituted piperazine compounds and the use of the same as analgesics
06/26/2003WO2003051842A2 Compositions decreasing activity of hormone-sensitive lipase
06/26/2003WO2003051841A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/26/2003WO2003051825A1 Human adam-10 inhibitors
06/26/2003WO2003051824A1 α-CYANOACRYLATES
06/26/2003WO2003051819A1 Substituted 1,5-diaminopentan-3-ol compounds
06/26/2003WO2003051369A1 Pharmaceutical containing n, n'-disubstituted piperazine compounds
06/26/2003WO2003051353A1 Substituted beta-aminoalcohols used as medicaments
06/26/2003WO2003051348A2 Composition, synthesis and therapeutic applications of polyamines
06/26/2003WO2003051276A2 Therapeutic heterocycles
06/26/2003WO2003002491A3 ENANTIOSELECTIVE TRANSFORMATION OF α, β-UNSATURATED ALDEHYDES USING CHIRAL ORGANIC CATALYSTS
06/26/2003US20030120115 Supported cobalt catalysts for nitrile hydrogenations
06/26/2003US20030120034 N-(2-hydroxyethyl)-2,4,6-triiodo-5-(2-(2,4,6-triiodo-3-(N-meth yl acetamido)-5-(methylcarbamyl)benzamidoacetamido)-isophthalmic acid, derivatives
06/26/2003US20030119902 Novel aminobenzoephenones
06/26/2003US20030119876 Compounds for the treatment of protozoal diseases
06/26/2003US20030119851 In the treatment or prevention of psychotic disorders such as schizophrenia psychotic depression, mania and other central nervous system diseases
06/26/2003US20030119833 Treating cardiovascular diseases
06/26/2003US20030119827 Peptidyl carbamates; treatments for osteoporosis and autoimmune diseases
06/26/2003US20030119819 Anticancer agents
06/26/2003US20030119803 In particular N-epsilon-amino acid substituted L-lysine derivatives possessing aspartyl protease inhibitory properties.
06/26/2003US20030119788 N-cyanomethyl carbonamides and sulfonamides which are cysteine protease, particularly cathepsin K, inhibitors
06/26/2003CA2510128A1 Composition, synthesis and therapeutic applications of polyamines
06/26/2003CA2473938A1 Human adam-10 inhibitors
06/26/2003CA2473877A1 Substituted beta-aminoalcohols as pharmaceutical preparations
06/26/2003CA2471500A1 Substituted 1,5-diaminopentan-3-ol compounds
06/26/2003CA2469944A1 Medicaments comprising n, n'-disubstituted piperazine compounds and their use
06/26/2003CA2469716A1 .alpha.-cyanoacrylates
06/26/2003CA2468978A1 Therapeutic heterocycles
06/26/2003CA2468413A1 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/25/2003EP1320520A1 Sulfonylguanidine
06/25/2003EP1025086B1 Benzamidine derivatives as factor xa inhibitors
06/25/2003CN1426412A Novel compounds
06/25/2003CN1426395A Inhibitors of dipeptidyl peptidase IV
06/25/2003CN1426394A Novel compounds
06/25/2003CN1426393A Novel compounds
06/25/2003CN1426392A Propenecarboxylic acid amidoxime derivatives, process for preparation thereof, and pharmaceutical compositions containing same
06/25/2003CN1112361C Process for preparing N-formyl morpholine
06/24/2003US6583286 Method for hydrogenating unsaturated heterocyclic compounds
06/24/2003US6583282 Formation of a urea by reacting an aromatic carbamate with a aromatic amine
06/24/2003US6583183 Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
06/24/2003US6583180 Glucocorticoid receptor modulators
06/24/2003US6583179 Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
06/24/2003US6583165 Anticarcinogenic, -inflammatory and -proliferative agents; viricides; bactericides; vascular restenosis, autoimmune diseases; psoriasis; anticolesterol and -lipemic agents
06/24/2003CA2288910C Pyrazolopyrimidinones for sexual dysfunction
06/24/2003CA2126337C 2-amino-1,3-propanediol compound and immunosuppressant
06/19/2003WO2003050099A1 Phenylalkynes
06/19/2003WO2003049690A2 Hiv integrase inhibitors
06/19/2003US20030114665 Such as 7-(((5-amino-1,2,4-thiadiazol-3-yl)-(Z)-(fluoro-methoxyimino)acetyl)amino)-3-(imino-1-piperazinylmethyl) methylhydrazono)methyl-3-cephem-4-carboxylic acid
06/19/2003US20030114521 Oxamic acids and derivatives as thyroid receptor ligands
06/19/2003US20030114508 Fused imidazolium derivatives
06/19/2003US20030114496 Treatment or prevention of Alzheimer's disease
06/19/2003US20030114490 New phenylalanine derivatives
06/19/2003US20030114454 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
06/19/2003US20030114442 Reducing concentration of blood lipoproteins
06/19/2003US20030114440 Compositions and methods of treatment for conditions responsive to testosterone elevation
06/19/2003US20030114427 Remedies and/or preventives for nervous system disorders
06/19/2003US20030114423 Arylamines as inhibitors of chemokine binding to US28
06/19/2003CA2469893A1 Phenylalkynes
06/18/2003EP1318980A2 Hydroxamate derivatives useful as deacetylase inhibitors
06/18/2003EP1318978A2 N-acylsulfonamide apoptosis promoters
06/18/2003EP1318977A1 Substituted phenylcyclohexane carboxylic acid amides and the use thereof
06/18/2003EP1318811A1 Cyclopentyl modulators of chemokine receptor activity
06/18/2003EP1183248B1 Non-linear optical devices and materials therefor
06/18/2003EP1140829A4 Contrast media for angiography
06/18/2003EP1082297B1 Substituted dithio-bis-nitrobenzenes and their applications
06/18/2003CN1425005A Cyclic quaternary ammonium compound
06/18/2003CN1424910A IL-8 receptor antagonists
06/18/2003CN1111520C Matrix metalloprotease inhibitors
06/17/2003US6579890 Matrix metalloprotease inhibitors
06/17/2003US6579881 Muscle relaxants, antiserotonine agent
06/17/2003US6579872 Bezamide derivatives for the treatment of diseases mediated by cytokines
06/17/2003US6579870 5-(1,4-diazepan-1-yl)-2-((3 -fluorophenyl)sulfonyl)phenylamine for example; treatment of diseases or disorders of the central nervous system; modulation of serotonin (5-HT) activity
06/17/2003US6579823 Group 8-10 metal complex comprising a bidentate or variable denticity ligand; polymerization of olefins
06/17/2003CA2059044C The use of n-(aminoalkyl) pyrrolidines as catalysts for the polyisocyanate polyaddition process
06/12/2003WO2003048158A1 Glycinamides as factor xa inhibitors
06/12/2003WO2003048121A1 Therapeutic benzamide derivatives
06/12/2003WO2003048118A1 5-ht7 receptor antagonists
06/12/2003WO2003048115A1 Bacterial enzyme inhibitors
06/12/2003WO2003048109A1 Novel glucagon antagonists
06/12/2003WO2003048108A2 Compounds for treatment of inflammation, diabetes and related disorders
06/12/2003WO2003048081A2 Glycinamides as factor xa inhibitors
06/12/2003WO2003047625A1 Neural transmission promoters
06/12/2003WO2003047575A1 Therapeutic benzamide derivatives
06/12/2003WO2003047568A1 N-aryl-n'-arylcycloalkyl-urea derivatives as mch antagonists for the treatment of obesity
06/12/2003WO2003047515A2 P2x7 receptor antagonists
06/12/2003WO2002047679A3 Nonpeptide agonists and antagonists of vasopressin receptors
06/12/2003WO2002017712A3 Disubstituted benzenes as insecticides
06/12/2003US20030109718 Enantioselective transformation of alpha, beta-unsaturated aldehydes using chiral organic catalysts
06/12/2003US20030109703 Antiinflammatory agents; autoimmune disease