Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
07/2003
07/23/2003CN1432001A 1-aryl-4-oxo-1,4-dihydro-3-quinolinecarboxamides as antiviral agents
07/23/2003CN1115330C N-(4-carbamimido-phenyl)-phenylglycinamid derivatives
07/22/2003US6596863 Matrix metalloproteinase inhibitor is useful as an anticancer agent, angiogenesis inhibitor, a tumor cell infiltration inhibitor or a tumor metastasis inhibitor; inflammatory diseases, osteoarthritis, rheumatoid arthritis
07/22/2003US6596773 Central nervous system disorders
07/22/2003US6596772 Relates to trifluoromethyl sulfonyl and trifluoromethyl sulfonamido compounds and the physiologically acceptable salts and the prodrugs thereof. These compounds are expected to modulate the activity of protein tyrosine enzymes which are
07/22/2003US6596752 Inhibitors of α4β1 mediated cell adhesion
07/22/2003US6596743 Carbamic acid derivatives
07/22/2003US6596716 2-propane-sulphonamide derivatives
07/22/2003US6596445 Initiators for photopolymerization of radically polymerizable compounds
07/17/2003WO2003057666A2 Inhibitors of dipeptidyl peptidase iv
07/17/2003WO2003057664A1 Carboxamidine derivatives and their use in the treatment of vascular diseases
07/17/2003WO2003057198A1 Pharmaceutical formulations with modified release
07/17/2003WO2003057169A2 4-dedimethylamino tetracycline compounds
07/17/2003WO2003057144A2 Change inhibitors of dipeptidyl peptidase iv
07/17/2003WO2002055496A8 Aryl piperidine and piperazine derivatives as inducers of ldl-receptor expression
07/17/2003US20030134874 Multicyclic compounds which inhibit leukocyte adhesion mediated by VLA-4
07/17/2003US20030134859 Substituted 2-chloro-5-nitrobenzamides; treating retrograde osteoporosis and diabetes mellitus
07/17/2003US20030134840 Novel compounds
07/17/2003US20030134802 Novel effectors of dipepetidyl peptidase IV
07/17/2003CA2471752A1 Carboxamidine derivatives and their use in the treatment of vascular diseases
07/17/2003CA2471204A1 Inhibitors of dipeptidyl peptidase iv
07/16/2003EP1327630A1 New derivatives of cyano-aryl (or cyanoheteroaryl)-carbonyl-piperazinyl-pyrimidines, their preparation and application as medication
07/16/2003EP1326840A2 Substituted heterocyclic compounds for treating multidrug resistance
07/16/2003EP1326834A2 2-substituted heterocyclic compounds
07/16/2003EP1326833A2 Substituted heterocyclic compounds for treating multidrug resistance
07/16/2003EP1326827A2 Insecticidal 1,8-naphthalenedicarboxamides
07/16/2003EP1326824A1 Pharmaceutical compounds
07/16/2003EP1210353B1 Calcium complex of phosphorus containing ethylenediamine derivatives
07/16/2003CN1430597A Novel MMP-2/MMP-9 inhibitors
07/16/2003CN1114596C Biphenyl derivatives
07/16/2003CN1114594C D4 receptor selectivity piperazine derivatives
07/16/2003CN1114591C Cyclic amide compounds
07/15/2003US6593474 Adrenergic blocking agents
07/15/2003US6593473 Evaporating form aqueous solution; solidification
07/15/2003US6593347 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use
07/15/2003US6593345 Naphthyl compounds, intermediates, compositions, and methods of use
07/15/2003US6593327 Compounds and compositions as protease inhibitors
07/15/2003US6593312 Cyclic α-amino-γ-hydroxyamide compounds
07/15/2003US6592884 Method of using alpha-keto enamine derivatives as ingredients and products incorporating same
07/15/2003CA2238465C Triaromatic compounds, compositions containing them and uses
07/10/2003WO2003055851A1 Hydroxamic acid derivative and mmp inhibitor containing the same as active ingredient
07/10/2003WO2003055850A1 β-AMYLOID PROTEIN PRODUCTION/SECRETION INHIBITORS
07/10/2003WO2003055848A2 Urea derivatives as vr1- antagonists
07/10/2003WO2003055847A1 Carboxylic acid derivative
07/10/2003WO2003055492A1 Use of oxindole derivatives in the treatment of dementia related diseases, alzheimer's disease and conditions associated with glycogen synthase kinase-3
07/10/2003WO2003055479A1 Compounds and their therapeutic use related to the phosphorylating activity of the enzyme gsk-3
07/10/2003WO2003055478A1 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders
07/10/2003US20030130509 Process to produce 3-carbon amino alcohol salts
07/10/2003US20030130349 Inhibitors of alpha 4beta1 mediated cell adhesion
07/10/2003US20030130339 Such as (E)-2-pyridineethenyl-4-fluorobenzyl sulfone; antitumor/anticancer agents
07/10/2003US20030130320 Alpha 4 integrin antagonists
07/10/2003US20030130287 Psychological disorders; central nervous system disorders; antidepressants; Parkinson's disease; Alzheimer's disease;cardiovascular disorders
07/10/2003US20030130272 Topoisomerase inhibitor; viricides
07/10/2003US20030130236 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
07/10/2003US20030130165 Method for treating neurodegenerative disorders
07/10/2003US20030129591 Linker arms for nanocrystals and compounds thereof
07/10/2003US20030129590 Linker arms for nanocrystals and compounds thereof
07/10/2003CA2482392A1 Carboxylic acid derivative
07/10/2003CA2469967A1 Urea derivatives as vr1- antagonists
07/09/2003EP1325912A1 2,2-diphenylbutanamide derivatives and medicines containing the same
07/09/2003EP1325903A1 2,3-diphenylpropionic acid derivatives or their salts, medicines or cell adhesion inhibitors containing the same, and their usage
07/09/2003EP1324970A2 Retinoids for the treatment of emphysema
07/09/2003CN1429229A Hydroxylamine esters as polymerization initiators
07/09/2003CN1429216A A new process for synthesis of morpholinylbenzenes
07/09/2003CN1429210A Substituted thioacetamides
07/09/2003CN1429199A Insecticidal 1,8-naphthalenedicarboxamides
07/09/2003CN1429133A Dosing form for reagents, use of said dosing form in organic chemical synthesis and production of said dosing form
07/09/2003CN1429107A Compositions cotaining benzamide disulfide derivative for treating allergic diseases
07/09/2003CN1113876C Preparation of N-formyl morpholine, N-formyl piperazine and their homologues
07/09/2003CN1113866C Process for preparation of piperidines
07/09/2003CN1113855C Preparation of alkylamines
07/08/2003CA2290501C Anti-inflammatory piperazinyl-benzyl-tetrazole derivatives and intermediates thereof
07/03/2003WO2003053942A1 Aryloxyphenyl and arylsulfanylphenyl derivatives
07/03/2003WO2003053927A1 Piperazine derivative
07/03/2003WO2003053919A1 Substituted cyclohexane derivatives
07/03/2003WO2003053918A2 Method for producing perfluoroalkane sulfonic acid esters and the salts thereof
07/03/2003WO2003053915A2 Compounds for the treatment of inflammatory disorders
07/03/2003WO2003053912A1 α-(N-SULPHONAMIDO)ACETAMIDE DERIVATIVES AS β-AMYLOID INHIBITORS
07/03/2003WO2003053885A1 Method for forming a carbon-carbon or carbon-heteroatom linkage
07/03/2003US20030125558 5-bromosalicylaldehyde is reacted in a one-pot reaction firstly with haloaceticalkyl or benzylester and then with formamide to give 5-L-benzofuran-2-carboxamide, then transition metal-catalyzed ammination with piperazines
07/03/2003US20030125557 1-[1-(hetero) aryl-1-perhydroxyalkylmethyl]-piperazine compounds, process for their preparation and pharmaceutical compositions containing them
07/03/2003US20030125549 Process for the catalytic asymmetric disubstitution of carboxamides using 2 different Grignard reagents
07/03/2003US20030125354 Aromatic compounds containing urea or thiourea groups are useful for terating cytokine mediated diseases
07/03/2003US20030125348 Minocycline compound substitued at 9-position by a group selected from nitro, alkyl, alkenyl, alkynyl, aryl, alkoxy, alkylthio, alkylsufinyl, alkylsulfonyl, amino, thionitroso, arylalkynyl or carbamate, urea, and sulfonamide
07/03/2003US20030125329 Treating atherosclerosis and other coronary artery diseases
07/03/2003US20030125328 Treating atherosclerosis and other coronary artery diseases
07/03/2003US20030125324 Alpha 4 beta 1 integrin and CD49d/ CD29 (vla-4); antiinflammatory agents
07/03/2003CA2471038A1 Process for the preparation of perfluoroalkanesulfonic acid esters and salts thereof
07/03/2003CA2470808A1 Piperazine derivative
07/03/2003CA2470141A1 Method for forming a carbon-carbon or carbon-heteroatom linkage
07/03/2003CA2467118A1 Aryloxyphenyl and arylsulfanylphenyl derivatives
07/02/2003EP1322610A2 PIPERAZINE BASED INHIBITORS OF FACTOR Xa
07/02/2003EP1322602A1 Substituted cinnamic acid guanidides, method for the production thereof, their use as a medicament, and to a medicament containing these compounds
07/02/2003EP1322590A1 5-amino-1-pentene-3-ol substituted derivatives
07/02/2003EP1322331A2 Fatty acid synthase inhibitors
07/02/2003EP0973780B1 Antibacterial substituted 7-acylamino -3-(methylhydrazono) methyl-cephalosporins and intermediates
07/02/2003EP0944582B1 Ketobenzamides as calpain inhibitors
07/02/2003CN1427829A Substituted phenylacetamides and their use as glucokinase activators
07/02/2003CN1427816A Process for forming amide bond
07/02/2003CN1427809A Nitroaromatic solubilizer for nitroxyls in aromatic solvents