Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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12/10/2002 | US6492424 Glucocorticoid and thyroid hormone receptor ligands for the treatment of metabolic disorders |
12/10/2002 | US6492423 Hepatitis c and b viricides |
12/10/2002 | US6492418 Administering benzamide-disulfide derivative for therapy and prophylaxis of allergic disease of the eye, nose, skin, ear, gastrointestinal tract or lung and manifestations of systemic mastocytosis |
12/10/2002 | US6492396 Substituted thioacetamides |
12/10/2002 | US6492393 Compounds useful as anti-inflammatory agents |
12/10/2002 | US6492375 Administering a piperidine compound |
12/10/2002 | US6492372 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 |
12/10/2002 | US6492370 Urea derivatives and pharmaceutical compositions thereof |
12/10/2002 | US6492369 Drug abruse |
12/10/2002 | US6492368 Benzamidine derivatives as factor XA inhibitors |
12/10/2002 | US6492367 Sulfamato hydroxamic acid metalloprotease inhibitor |
12/10/2002 | US6492365 Microsomal triglyceride transfer protein |
12/10/2002 | US6492363 2-(4-bromo or 4-iodo phenylamino) benzoic acid derivatives |
12/10/2002 | US6492362 Compounds and compositions as cathepsin S inhibitors |
12/10/2002 | US6492355 Adamantane derivatives |
12/10/2002 | US6492351 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
12/10/2002 | CA2230445C Fibrinogen receptor antagonists and medicinal preparations containing the same as the active ingredient |
12/09/2002 | WO2002004403A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments |
12/09/2002 | CA2412116A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments |
12/05/2002 | WO2002097050A2 Novel estrogen receptor ligand binding domain variants and novel ligands and pharmaceutical compositions |
12/05/2002 | WO2002096897A1 PHOSPHINYLMETHYL AND PHOSPHORYLMETHYL SUCCINIC AND GLUTARIC ACID ANALOGS AS β-SECRETASE INHIBITORS |
12/05/2002 | WO2002096884A2 Substituted benzoylketones as herbicidal agents for use as plant treatment agent |
12/05/2002 | WO2002096876A1 Carbamate and oxamide compounds as inhibitors of cytokine production |
12/05/2002 | WO2002096874A2 Method for producing biperiden iv |
12/05/2002 | WO2002096869A2 Piperazine mono(dithio)carbamate ester compounds and analogs thereof |
12/05/2002 | WO2002096864A1 Carboxamide-substituted phenylurea derivatives and method for production thereof as medicaments |
12/05/2002 | WO2002096858A1 Cinnamide derivatives as kcnq potassium channel modulators |
12/05/2002 | WO2002096855A2 Anticholinergic compounds and methods of use |
12/05/2002 | WO2002096854A1 N-benzyl-m-phenylenediamine derivatives and dyes containing said compounds |
12/05/2002 | US20020183518 Use for treatment of human and animal disorders, for purification of proteins or glycoproteins, and in diagnosis |
12/05/2002 | US20020183517 Reacting dihydric alcohol characterized by four to six carbons, preferably 1,5-pentanediol, with excess ammonia in presence of ZSM-5 catalyst modified with nickel, copper or cobalt |
12/05/2002 | US20020183512 Compounds for use in treatment of cancer |
12/05/2002 | US20020183397 Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity |
12/05/2002 | US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm |
12/05/2002 | US20020183334 For therapy of sleepiness, promotion of wakefulness, treatment of Parkinson's disease, cerebral ischemia, stroke, sleep apneas, eating disorders, stimulation of appetite and weight gain, treatment of attention deficit hyperactivity disorder |
12/05/2002 | US20020183316 Amidoalkyl-piperidine and amidoalkyl-piperazine derivatives useful for the treatment of nervous system disorders |
12/05/2002 | DE10126929A1 Production of compounds with perfluoroalkanesulfonic acid residues, used e.g. in electrolytes and batteries, involves reacting perfluoroalkanesulfonic anhydride with dialkyl carbonate in presence of perfluoroalkanesulfonic acid |
12/05/2002 | DE10125567A1 New N-aroyl-N'-(carbamoyl-phenyl)-urea derivatives, are glycogen phosphorylase a inhibiting hypoglycemic agents, especially useful for treating type II diabetes |
12/05/2002 | CA2448894A1 Cinnamide derivatives as kcnq potassium channel modulators |
12/05/2002 | CA2448626A1 Carbamate and oxamide compounds as inhibitors of cytokine production |
12/05/2002 | CA2448023A1 Carboxamide-substituted phenylurea derivatives and method for production thereof as medicaments |
12/05/2002 | CA2443346A1 Anticholinergic compounds and methods of use |
12/05/2002 | CA2442212A1 N-benzyl-m-phenylenediamine derivatives and dyes containing said compounds |
12/05/2002 | CA2411082A1 Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament |
12/04/2002 | EP1261595A1 Arylpiperazines and arylpiperidines and their use as metalloproteinase inhibiting agents |
12/04/2002 | EP1261594A1 5,10-dihydroacridines as calcium channel blockers |
12/04/2002 | EP1261590A1 Piperidine- and piperazine substituted n-hydroxyformamides as inhibitors of metalloproteinases |
12/04/2002 | EP1261329A2 Il-8 receptor antagonists |
12/04/2002 | EP1261321A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof |
12/04/2002 | CN1382440A Method and medicine case for treating depression or preventing degeneration of cognitive function |
12/03/2002 | US6489480 Coordination polymerization catalyst for alpha-olefins |
12/03/2002 | US6489374 Organonitrogen compounds that yield amines, imines or amidines when exposed to visible or ultraviolet radiation; polymerization catalysts used in one-pot systems having storage stability |
12/03/2002 | US6489327 Tryptase inhibitors |
11/28/2002 | WO2002095393A2 Drug evolution: drug design at hot spots |
11/28/2002 | WO2002094801A1 Method for producing biperiden i |
11/28/2002 | WO2002094800A1 Method for the production of biperidin |
11/28/2002 | WO2002094799A2 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues |
11/28/2002 | WO2002094794A1 4 (phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain anxiety or gastrointestinal disorders |
11/28/2002 | WO2002094781A1 Method for the production of biperiden ii |
11/28/2002 | WO2002094208A1 Novel couplers for use in oxidative hair dyeing |
11/28/2002 | WO2002062777A3 Amino ceramide-like compounds and therapeutic methods of use |
11/28/2002 | US20020177598 Inhibit activity of chemokines, macrophage inflammatory protein-1 (MIP-1 alpha) and RANTES; 1-((4-chlorophenoxy)methyl)-carbonyl-2-methyl-4-(4-fluorobenzyl)piperazine for example |
11/28/2002 | US20020177594 Inhibitors of histone deacetylase |
11/28/2002 | DE10125451A1 New N-benzyl-m-phenylenediamine derivatives and physiologically-compatible, water-soluble salts are used in oxidative colorant for keratin fibers, especially human hair |
11/28/2002 | DE10125432A1 New benzoyl-substituted aliphatic ketones or aldehydes, useful as herbicides or fungicides, especially as pre- and post-emergence selective herbicides against a broad spectrum of weeds |
11/28/2002 | DE10124867A1 New substituted (hetero)aryl-alkenes or -alkynes, used as thrombin inhibitors, serine protease inhibitors, antithrombotic agents and intermediates |
11/28/2002 | CA2448080A1 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues |
11/28/2002 | CA2434036A1 Novel couplers for use in oxidative hair dyeing |
11/27/2002 | EP1260504A1 Process for the preparation of antihistaminic 4-diphenylmethyl piperidine derivatives |
11/27/2002 | EP1259493A2 Substituted piperazine compounds |
11/27/2002 | EP1259492A1 Substituted piperazine derivatives as mtp inhibitors |
11/27/2002 | EP1259484A1 Carboxamides useful as inhibitors of microsomal triglyceride transfer protein and of apolipoprotein b secretion |
11/27/2002 | EP1259478A1 Covalent derivatives of alkanolamides of monocarboxylic and dicarboxylic acids functionally active on the cb2 cannabinoid receptor |
11/27/2002 | EP1259475A1 Transition metal-catalyzed process for addition of amines to carbon-carbon double bonds |
11/27/2002 | EP1259470A2 A group of anti-cancer compounds with specific structure and their production method |
11/27/2002 | EP1114024B1 Urokinase inhibitors |
11/27/2002 | EP1109557B1 Use of cetirizine for preventing the onset of asthma |
11/27/2002 | EP1000048B1 Substituted 1,2,3,4-tetrahydronaphthalene derivatives |
11/27/2002 | CN1382135A Amine and amide derivatives as ligands for neuropeptide YY5 receptor usefu in treatment of obesity and other disorders |
11/27/2002 | CN1381454A Method for preparing oxazolidone amine |
11/27/2002 | CN1381449A Aralkylone pipeazine derivative and its application |
11/27/2002 | CN1381448A Aralkylformylalkyl piperazine derivative and its application as brain nerve protector |
11/26/2002 | US6486324 Forming libraries of bactericides; immobilization; side effect reduction |
11/26/2002 | US6486178 Indane derivatives |
11/26/2002 | US6486165 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
11/26/2002 | CA2231364C Novel n-aminoalkylfluorenecarboxamides; a new class of dopamine receptor subtype specific ligands |
11/24/2002 | CA2354921A1 Drug evolution: drug design at hot spots |
11/22/2002 | WO2003101942A1 Amidine substituted aryl and heteroaryl derivatives with an antithrombotic and factor xa inhibiting action |
11/22/2002 | CA2445571A1 Substituted aryl and heteroaryl derivatives, the preparation thereof and the use thereof as pharmaceutical compositions |
11/21/2002 | WO2002092585A1 Novel, arylsusfonamide compounds for the treatment of obesity, type ii diabetes and cns-disorders |
11/21/2002 | WO2002092574A1 Substituted benzoylcyclohexenones and their use as herbicidal agents |
11/21/2002 | WO2002092068A1 Carboxylic acid derivatives and drugs containing the same as the active ingredient |
11/21/2002 | WO2002091993A2 Estrogen receptor modulators |
11/21/2002 | WO2002072084A3 Glycyrrhetinic acid derivatives, progesterone and progesterone derivatives and their use for the manufacture of a medicament to inhibit 11beta-hydroxysteroid dehydrogenase activity |
11/21/2002 | US20020173665 Use treating pain, urinary incontinence and bladder overactivity |
11/21/2002 | US20020173664 An 3-acyl-4-substituted-oxazolidin-2,5-dione that readily reacts with nucleophilic reagents such as free amino acids; use in peptide synthesis for example |
11/21/2002 | US20020173645 Acylating a 2-aryl-6-alkoxy-benzo(b)thiophene with a p-(tertiaryaminoethoxy)benzoic acid hydrohalide salt or the corresponding benzoyl halide in presence of a boron trihalide |
11/21/2002 | US20020173508 Enzyme inhibitors; antiinflammatory agents, antiarthritic agents |
11/21/2002 | US20020173494 Ammonium salts of inositol hexaphosphate, and uses thereof |
11/21/2002 | US20020173488 Boronic Ester and acid compounds, synthesis and uses |