Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
06/2005
06/07/2005US6903221 Reacting arylhalogenide with 1,3-diketone in carbon monoxide atmosphere; herbicides
06/07/2005US6903216 Antiarrhythmic agents for the treatment and prophylaxis of atrial arrhythmias, atrial fibrillation (AF) or atrial flutter; potassium channel modulators, beta-blocker
06/07/2005US6903215 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/07/2005US6903128 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
06/07/2005CA2281090C Sulfonamide compounds and salts for treatment of endothelin-mediated disorders
06/02/2005WO2005049623A1 PREPARATION OF 1-AZA-2-OXA-DIBENZO[e,h]AZULENES AND THEIR USE FOR THE MANUFACTURE OF PHARMACEUTICAL FORMULATIONS FOR THE TREATMENT AND PREVENTION OF CENTRAL NERVOUS SYSTEM DISEASES AND DISORDERS
06/02/2005WO2005049589A2 Heterocyclic compounds for the treatment of hyperlipidemia, diabetes, obesity and similar diseases
06/02/2005WO2005049064A1 Drug therapy for celiac sprue
06/02/2005WO2005048953A2 Amide derivatives as kinase modulators
06/02/2005WO2005048948A2 Urea derivatives as kinase modulators
06/02/2005US20050119332 Substituted thiophene compounds as modulators of protein tyrosine phosphatases (PTPases)
06/02/2005US20050119225 Phosphodiesterase 4 inhibitors, including N-substituted aniline and diphenylamine analogs
06/02/2005CA2546620A1 Preparation of 1-aza-2-oxa-dibenzo[e,h]azulenes and their use for the manufacture of pharmaceutical formulations for the treatment and prevention of central nervous system diseases and disorders
06/02/2005CA2545711A1 Urea derivatives as kinase modulators
06/01/2005EP1535912A1 Muscarinic agonists
06/01/2005EP1535909A2 Cyclic amine derivatives and their use as drugs
06/01/2005EP1534696A1 Therapeutic compounds for treating dyslipidemic conditions
06/01/2005EP1534693A2 1, 3-diamino-2-hydroxypropane prodrug derivatives
06/01/2005EP1534683A2 Cyclooxygenase-2 selective inhibitors, compositions and methods of use
06/01/2005EP1534666A1 Compounds for modulating the glycolosis enzyme complex and/or transaminase complex
06/01/2005EP1534273A2 Modulators of the glucocorticoid receptor and method
06/01/2005EP1351959B1 Novel pleuromutilin derivatives
06/01/2005EP1345902B1 Substituted heterocyclo-norbornylamine derivatives, method for producing the same, their use as medicament or diagnostic agent and medicament containing the same
06/01/2005EP0946499B1 N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
06/01/2005CN1621404A Drug and method for regulating cholesterol and triglyceride
06/01/2005CN1203852C Valdecoxib compositions
05/2005
05/31/2005US6900345 Antibiotics; mutilin 14-[N-(2-carbamoyloxyethoxycarbonyl)]carbamate; therapy for bacteria infections; chemical synthesis
05/31/2005US6900334 Antiallergens; autoimmune diseases
05/31/2005US6900333 Dissolving in aqueous solution containing alcohols; distillation; purification
05/26/2005WO2005047236A1 Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses
05/26/2005US20050113440 Compounds that modulate PPAR activity and methods for their preparation
05/26/2005US20050113424 E.g., 4-{3-[4-(3-{4-[amino(imino)methyl]phenoxy}propyl)-1-piperazinyl]propoxy}benzamidine; an antifungal agent with good pharmacokinetics and excellent antifungal action; side effect reduction such as nephrotoxicity; action to Mycomycetes
05/26/2005US20050113419 Therapeutic compounds for treating dyslipidemic conditions
05/26/2005US20050113373 medicine to inhibit proliferative conditions, such as cancer and psoriasis; detecting or identifying a histone deactylase (HDAC) in a biological sample
05/26/2005US20050113357 Cholinergic agents such as 3-[3-(4-methoxypiperidine)-1-yl-propyl]-1H-indole; for therapy of cognitive dysfunction, forgetfulness, confusion, memory loss, attention deficits, deficits in visual perception, depression, pain, sleep disorders, and psychosis
05/26/2005US20050113356 Inhibitors of cathepsin S
05/26/2005US20050112197 Celecoxib dissolving in polyethylene glycol; antiinflammatory agents, osteoporosis, respiratory system disorders, antitumor agents, analgesics
05/25/2005EP1533292A1 Dibenzylamine compound and medicinal use thereof
05/25/2005EP1531812A1 Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthristis
05/19/2005WO2005044808A1 A process for the manufacture of zonisamide
05/19/2005WO2005012220A9 Cycloalkylidene compounds as modulators of estrogen receptor
05/19/2005US20050107444 E.g., 2-(3-{3-[(2-chloro-3-(trifluoromethyl)-benzyl)-(2,2-diphenylethyl)-amino]-propoxy}phenyl)-1-morpholin-4-yl-ethanone; agonists of the nuclear receptors, LXR alpha and LXR beta used to increase ABCA1, ABCG1, and apolipoprotein E expression and inhibiting cholesterol absorption
05/19/2005US20050107435 antibiotics such as (5S,5S')-N-(3-{4'-[5-(Acetylamino-methyl)-2-oxo-oxazolidin-3-yl]-2,2'-difluoro-biphenyl-4-yl}-2-oxo-oxazolidin-5-ylmethyl)-acetamide, used for treating a bacterial infections in mammals
05/19/2005DE10348023A1 Neue Alanyl-Aminopeptidasen-Inhibitoren zur funktionellen Beeinflussung unterschiedlicher Zellen und zur Behandlung immunologischer, entzündlicher, neuronaler und anderer Erkrankungen New alanyl aminopeptidase inhibitors for functional interference of different cells and for the treatment of immunological, inflammatory, neuronal and other diseases
05/19/2005CA2545119A1 A process for the manufacture of zonisamide
05/18/2005CN1617852A Alpha-(n-sulphonamido)acetamide derivatives as beta-amyloid inhibitors
05/18/2005CN1617850A Dibenzylamine compound and medicinal use thereof
05/17/2005US6893650 Fungicides; locus infestation; such as N,N-dimethyl-N'-(4-(3-trifluoromethylbenzylthio)-2,5-xylyl)formamidine
05/12/2005WO2005042513A1 Phenyl carboxamide and sulfonamide derivatives for use as 11-beta-hydroxysteroid dehydrogenase
05/12/2005WO2005041959A1 Phenoxyacetic acids derivatives useful as peroxisome proliferator-activated receptor (ppar) dual agonists
05/12/2005WO2005007635A8 Combretastatin derivatives with cytotoxic action
05/12/2005WO2003006454A8 Heterocyclic carboxamides and their use as fungicides
05/12/2005CA2544317A1 Phenoxyacetic acids derivatives useful as peroxisome proliferator-activated receptor (ppar) dual agonists
05/12/2005CA2540843A1 Phenyl carboxamide and sulfonamide derivatives for use as 11-beta-hydroxysteroid dehydrogenase
05/11/2005EP1529530A1 Compounds affecting glucokinase
05/11/2005EP1056341A4 Method and apparatus for the preparation of ketones
05/11/2005EP0951464B1 N-(aryl/heteroarylacetyl) amino acid esters, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
05/11/2005CN1615305A Coumarin derivatives, process for their production and use thereof
05/11/2005CN1613853A PDF enzyme inhibitor-hydroxamic acid serial compounds synthetic method and use thereof
05/10/2005US6890956 Cyclohexyl sulphones as gamma-secretase inhibitors
05/10/2005US6890942 Acyl sulfonamides as inhibitors of HIV integrase
05/06/2005WO2005040161A1 Biaryl linked hydroxamates: preparation and pharmaceutical applications
05/06/2005WO2005040142A1 Novel keto-oxadiazole derivatives as cathepsin inhibitors
05/06/2005WO2005040138A1 Substituted benzylaminoalkylene heterocycles
05/06/2005WO2005040121A2 Amides that inhibit vanilloid receptor subtype 1 (vr1) receptor
05/06/2005WO2005040100A1 Tetrahydro-naphthalene and urea derivatives
05/06/2005CA2542695A1 Substituted benzylaminoalkylene heterocycles
05/06/2005CA2542494A1 Tetrahydro-naphthalene and urea derivatives
05/06/2005CA2539967A1 Amides that inhibit vanilloid receptor subtype 1 (vr1) receptor
05/05/2005US20050096362 4-((Phenoxyalkyl)thio)-phenoxyacetic acids and analogs
05/05/2005US20050096357 Antibiotics; therapy for infections which is caused by drug-resistant Streptococcus, or bacteria infections
05/04/2005EP1528059A2 Substituted isoxazoles for the treatment of inflammation
05/04/2005EP1528058A1 Polymorphic crystalline forms of celecoxib
05/04/2005EP1528055A2 Sulphonamide Derivatives
05/04/2005EP1526895A2 Methods for treating carbonic anhydrase mediated disorders
05/04/2005EP1526869A1 Compositions of a cyclooxygenase-2 selective inhibitor and a carbonic anhydrase inhibitor for the treatment of neoplasia
05/04/2005EP1373229A4 Process for the preparation of 1,2-benzisoxazole-3-acetic acid
05/03/2005US6887905 Treatment of depression or generalized anxiety disorder
05/03/2005US6887877 Viricide for hepatitis virus
05/03/2005US6887871 Use of phenylheteroakylamine derivatives
05/03/2005US6887863 Such as (2RS,3R)-3-amino-4-cyclohexyl-2-hydroxy-N-phenoxybutanamide; methionine aminopeptidase type 2 inhibitors
05/03/2005CA2133337C Compounds useful for treating allergic or inflammatory diseases
04/2005
04/28/2005WO2005037271A2 Large conductance calcium-activated k channel opener
04/28/2005WO2005037257A2 Novel alanyl-amino peptidase inhibitors for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/28/2005WO2004014844A3 Aryl and heteroaryl compounds and methods to modulate coagulation
04/28/2005CA2542723A1 Novel alanyl-amino peptidase inhibitors for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/27/2005EP1525883A1 Ciclooxygenase-2 inhibitor compositions having rapid onset of therapeutic effect
04/27/2005EP1525191A2 Novel method for preparing styryl pyrazole, isoxazole and isothiazole derivatives
04/27/2005EP1524974A2 Transcription factor modulating compounds and methods of use thereof
04/27/2005EP1011651B1 Method of treating diabetes and related disease states
04/27/2005CN1610659A Carboxylic acid derivative
04/27/2005CN1198838C Antipicornaviral compounds, their prepn. and use
04/26/2005US6884821 Alkyloxypropanoic acid derivative containing sulfonamide or amide group are useful as insulin resistance agent
04/26/2005US6884814 Phenyl benzisoxazoles as estrogenic agents
04/26/2005CA2213124C Benzoyl derivatives
04/21/2005WO2005035514A2 Modulators of atp-binding cassette transporters containing cycloalkyl or pyranyl groups
04/21/2005WO2005035510A1 Derivatives of 4-phenylthiazoles and 4-phenylimidazoles and the use thereof as medicaments for treating neurodegenerative diseases, pain and epilepsy
04/21/2005WO2005034848A2 Inhibitors of cathepsin s
04/21/2005WO2004111019A3 Protective groups cleavable by serumal albumins
04/21/2005US20050085667 N-biphenylmethyl aminocycloalkanecarboxamide derivatives
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