Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
06/2008
06/26/2008WO2007074391A3 Preparation of a key intermediate in the synthesis of rosuvastatin
06/26/2008US20080153869 2-hydroxy-1H-indol derivatives enzyme inhibitors for preventing or treating inflammation, inflammatory bowel disease, psoriasis, dementia related diseases Alzheimer's Disease, Cognitive Impairment, arthritis, neurodegenerative diseases, amyotrophic lateral sclerosis, Down syndrome, Huntington's Disease
06/26/2008US20080153859 5-{[6-Fluoro-2,5-dihydroxy-4,4,7-dimethyl-2-(trifluoromethyl)-1,2,3,4-tetrahydronaphthalen-1-yl]amino}-isoquinolin-1(2H)-one; anti-allergic, immunosuppressive and antiproliferative action
06/26/2008US20080153852 Tryptophan hydroxylase inhibitors; anticarcinogenic agents; gastrointestinal, cardiovascular, and respiratory system disorders
06/26/2008US20080153837 4-(Benzimidazol-2-yl)fluorene and 4-(azabenzimidazol-2-yl)fluorene derivatives; treating disorders related to Hsp90 protein; anticarcinogenic, antimetastasis, antitumor, anticoagulant, antiproliferative, antihistamine, and antidiabetic agents; metabolic, muscular, rheumatic and nervous system disorders
06/26/2008US20080153836 1H-Quinazoline-2,4-Diones
06/26/2008US20080153835 Therapeutic agents useful for treating pain
06/26/2008US20080153815 Pinane-substituted pyrimidinediamine derivatives useful as axl inhibitors
06/26/2008US20080153809 Novel amides useful for treating pain
06/26/2008US20080152950 Anthracene derivative and organic electroluminescent device using the same
06/26/2008US20080152702 Improved blood circulation lifetime of drug-carrying liposomes having a surface coating of releasable hydrophilic polymer covalently and reversibly linked to an phospholipid or polypeptide through a dithiobenzyl linkage
06/26/2008DE102007023102A1 Bisoxime als Fungizide Bisoximes as fungicides
06/26/2008CA2695613A1 Sulfonamide derivatives with therapeutic indications
06/26/2008CA2672668A1 4-amino-1h-pyrimidin-2-one-based compounds, compositions comprising them and methods of their use
06/26/2008CA2671414A1 Process for the preparation of substituted cyanophenoxy-pyrimidinyloxy-phenyl acrylate derivatives
06/25/2008EP1935887A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands
06/25/2008EP1935885A2 Melanin concentrating hormone receptor ligands : substituted 1-benzyl-4-aryl piperazine analogues.
06/25/2008EP1935869A1 Retinoids for the treatment of emphysema
06/25/2008EP1934233A1 Sulfonamide derivatives as glycokinase activators useful in the treatment of type 2 diabetes
06/25/2008EP1492534B1 Carbamic acid compounds comprising a piperazine linkage as hdac inhibitors
06/25/2008CN101208310A New crystal forms of 4-[6-methoxy-7-(3-piperidin-1-yl-propoxy)quinazolin-4-yl]piperazine-1-carboxylic acid(4-isopropoxyphenyl)-amide
06/25/2008CN101208309A Chloro-substituted guanidines
06/25/2008CN101208308A 8-alk0xy-4-methyl-3, 4-dihydr0-quinaz0lin-2-yl amines and their use as 5-ht5a receptor ligands
06/25/2008CN101208307A Process for preparing amorphous rosuvastatin calcium free of impurities
06/25/2008CN101205215A Method for preparing cidofovir key intermediate
06/25/2008CN100396785C Resoldution method for racemic compound of nucleoside enantiomorph
06/25/2008CN100396679C Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase
06/25/2008CN100396668C Non-imidazole aryloxypiperidines
06/24/2008US7390908 Such as 2-[3,5-Di(2-chlorobenzyloxy)benzoyl)amino]-thiazole; for treatment of diabetes
06/24/2008US7390835 Aralkyl amines as cannabinoid receptor modulators
06/24/2008US7390833 osteoarthritis; compounds inhibit Aggrecanase Activity of a disintegrin and metalloprotease with thrombosondin type I motifs; biaryl sulfonamid derivatives; N-({4'-[2-4-methylisoquinolin-3-yl)ethyl]-1,1 '-biphenyl-4-yl}sulfonyl)-D-valine
06/24/2008US7390818 3-(2,4-dimethoxyphenyl)-1,9-dimethyl-2-oxo-2,9-dihydro-1H-pyrido[2,3-b]indole-6-carboxylic acid; gamma-aminobutyric acid modulator; anticarcinogenic, antitumor, antiproliferative agent
06/24/2008US7390815 Pyrazole compounds useful as protein kinase inhibitors
06/24/2008US7390814 Substituted hexahydropyrazino [1,2-a] pyrimidine-4,7-dione derivatives, process for their preparation and their use as medicaments
06/24/2008US7390806 Antibiotics containing borinic acid complexes and methods of use
06/19/2008WO2008073928A1 Composition for treating a pulmonary hypertension
06/19/2008WO2008073687A2 Compounds and compositions as protein kinase inhibitors
06/19/2008WO2008073370A1 Aspartyl protease inhibitors containing a tricyclic ring system
06/19/2008WO2008073365A1 Aspartyl protease inhibitors
06/19/2008WO2008073125A1 Moxonidine analogs, preparation processes and uses therefor
06/19/2008WO2008072078A1 An improved process for preparing rosuvastatin caclium
06/19/2008WO2008049123A3 2,4-pyrimidinediamine derivatives as inhibitors of jak kinases for the treatment of autoimmune diseases
06/19/2008US20080146620 Dibenzylamine Compounds and Pharmaceutical Use Thereof
06/19/2008US20080146600 potent proline transporter inhibitors such as (S)-2-(4-((3'-chlorobiphenyl-4-yl)(hydroxy)methyl)piperidin-1-yl)pyrimidin-5-ol, used as cognition activators or for treatment of brain disorders
06/19/2008US20080146599 receptor tyrosine kinase inhibitors such as 2-chloro-N-{3-[(4,6-diaminopyrimidin-5-yl)ethynyl]phenyl}benzenesulfonamide, used as angiogenesis inhibitors in mammals
06/19/2008US20080146597 Therapeutic Tetrahydroisoquinoline-Based Compositions for Cancer Therapy
06/19/2008US20080146594 Thrombopoietin activity modulating compounds and methods
06/19/2008US20080146574 Heterocycle Substituted Carboxylic Acids
06/19/2008US20080146571 potent deoxycytidine kinase inhibitors; O-linked pyrimidin-4-amine-based compounds
06/19/2008US20080146570 Chemical Compounds
06/19/2008US20080146569 Nicotinamide Derivatives
06/19/2008US20080146562 Halogenated quinazolinyl nitrofurans as antibacterial agents
06/19/2008US20080145453 4-(piperimidine-2thione)phenyl derivatives; kinesin Eg5 inhibitor; anticarcinogenic agent; the aldehyde, the ketone and the thiourea are reacted together in the solid phase, grafted onto resin by esterification, and detached by hydrolysis
06/19/2008US20080142759 For irradiation with blue/red laser; write only read many (WORM); digital versatile discs
06/19/2008CA2672295A1 Aspartyl protease inhibitors containing a tricyclic ring system
06/19/2008CA2672293A1 Aspartyl protease inhibitors
06/19/2008CA2669536A1 Composition for treating a pulmonary hypertension
06/18/2008EP1931643A1 2-substituted hydroxylaminopyrimidine, method for the production and the use thereof in the form of pesticides
06/18/2008EP1931642A2 Novel pyrimidine carboxamides
06/18/2008EP1931627A1 Amino-alkyl-amide derivatives as ccr3 receptor ligands
06/18/2008EP1585521B1 Derivatives of aryl-quinazoline/aryl-2amino-phenyl methanone which promote the release of parathyroid hormone
06/18/2008CN101203522A Antineoplastic compounds and pharmaceutical compositions thereof
06/18/2008CN101203496A Process for preparing pure amorphous rosuvastatin calcium
06/18/2008CN101200451A Method for preparing hydrochloride urapidil
06/18/2008CN100395293C Water-soluble fiber-reactive dyes, method for the production and use thereof
06/18/2008CN100395246C Method for producing folic acid antagonist and its intermediate
06/17/2008US7388014 Quinazoline derivatives and therapeutic use thereof
06/17/2008CA2384188C Antiviral compositions
06/17/2008CA2356380C Immunosuppressive effects of pteridine derivatives
06/17/2008CA2331737C Agents for relieving side effects caused by use of an anti-tumour agent
06/17/2008CA2286772C Fungicide active substance combinations
06/17/2008CA2272291C Crf antagonistic quino- and quinazolines
06/17/2008CA2249446C Irreversible inhibitors of tyrosine kinases
06/12/2008WO2008069609A1 Pyrimidinone derivatives or pyridazinone derivatives for inhibition of factor viia activity
06/12/2008WO2008068470A1 Antibacterial polycyclic urea compounds
06/12/2008WO2008031556A3 2 amino-pyrimidine derivatives as h4 receptor antagonists, processes for preparing them and their use in pharmaceutical compositions
06/12/2008WO2008015517A3 Ep2 agonists
06/12/2008WO2007148208A3 Carbonylated (aza) cyclohexanes as dopamine d3 receptor ligands
06/12/2008US20080139811 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection
06/12/2008US20080139809 Compounds Capable of Activating Cholinergic Receptors
06/12/2008US20080139598 e.g. N-(3'-chloro-3-methylbiphenyl-4-yl)-1-(pyrimidin-2-yl)piperidin-4-amine; proline transporter inhibitor; cognition activator; Alzheimer's disease, Attention-Deficit/Hyperactivity Disorder, autism, Down syndrome, Fragile X syndrome, Huntington's disease, Parkinson's disease, schizophrenia, dementia
06/12/2008US20080139590 Quinazoline based egfr inhibitors containing a zinc binding moiety
06/12/2008US20080139589 2-Methyl-3-{4-[3-(1-pyrrolidinyl)propoxy]phenyl}-5-trifluoromethyl-4(3H)-quinazolinone; sleep, psychological, nervous system, and attention deficit disorders; drug abuse, alcoholism; antidiabetic agents, cognition activators; Alzheimer's and Parkinson's disease; histamine H3 receptor antagonists
06/12/2008US20080139547 N-Hydroxyalkynylbenzamide (or hydroxamate) derivatives; anticarcinogenic and antiproliferative agents
06/12/2008US20080139505 Potentiators Of Glutamate Receptors
06/12/2008US20080139455 (2S,3S,E)-2-amino-14,14-difluoro-3-hydroxytetradec-6-enoic acid; serine palmitoyl transferase ; insulin resistance, pancreatic beta cell apoptosis, obesity, pro-thrombotic conditions, myocardial infarction, hypertension, dyslipidemia
06/12/2008CA2670870A1 Antibacterial polycyclic urea compounds
06/11/2008EP1928862A1 2-aminopyrimidine derivatives as modulators of the histamine h4 receptor activity
06/11/2008EP1928857A1 Method for preparing (3-chloro-4-fluorophenyl)-(4-fluoro-4-{[(5methyl-pyrimidin-2-ylmethyl)-amino]-methyl}-piperidin-1-yl)-methanone and novel intermediate pyrimidine derivatives
06/11/2008EP1928844A2 Bis-aryl amide compounds and methods of use
06/11/2008EP1928843A1 Bis-aryl urea compounds for the treatment of protein kinase-mediated diseaes
06/11/2008EP1928842A1 4-phenyl-6-substituted-pyrimidine-2-carbonitrile derivatives
06/11/2008EP1928461A1 Pyrimidine compounds as serotonin receptor modulators
06/11/2008EP1928242A2 A use of sulfonanilides as herbicide
06/11/2008EP1485348B1 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
06/11/2008EP1313713B1 4-pyrimidinamine derivatives, pharmaceutical compositions and related methods
06/11/2008EP1255739B1 3-aminoquinazolin-2,4-dione antibacterial agents
06/11/2008CN101198596A 2-amino-quinaz0lin-5-ones as HSP90 inhibitors useful in treating proliferation diseases
06/11/2008CN101198595A Aspartyl protease inhibitors
06/11/2008CN101198590A Novel pyridine derivative and pyrimidine derivative (3)