| Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619) |
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| 04/16/2008 | CN100381428C Quinazolone and quinazolone compound and application thereof |
| 04/16/2008 | CN100381427C Benzylamine compound, and its preparing method and use |
| 04/16/2008 | CN100381424C Biaryl sulfonamides and methods for using same |
| 04/15/2008 | US7358359 Antibacterial agents |
| 04/15/2008 | US7358262 Using transgenic tumor cells as models for antitumor agent efficacy; tissue targeted therapy and antiproliferative agents |
| 04/15/2008 | US7358257 sulfonylurea derivatives, sulfonylthiourea derivatives, sulfonylguanidine derivatives, sulfonylcyanoguanidine derivatives, thioacylsulfonamide derivatives, and acylsulfonamide derivatives; effective for prevention and treatment of cardiovascular diseases, antithrombotic agents |
| 04/15/2008 | US7358256 Antiproliferative agents; tyrosine kinase inhibitors; anticancer; diseases associated with signal transduction pathways operating through growth factor receptors; 4-amino-1-((4-(3-methoxyphenylamino) quinazolin-5-yl)methyl)-N-methylpiperidine-3-carboxamide |
| 04/15/2008 | US7358248 treatment of diabetes and/or cancer; useful in the treatment of syndrome X; capable of inhibiting Protein tyrosine phosphatases |
| 04/15/2008 | US7358239 Treating impaired fundic relaxation; [1(R),[A-(3 alpha ,4 alpha )]]-1-[1-[(3,4-dihydro-2H-1-benzopyran-2-yl)methyl]-3-methoxy-4-piperidinyl]-2(1H)-pyrimidinone |
| 04/15/2008 | CA2349325C Process for converting an alcohol to the corresponding fluoride |
| 04/15/2008 | CA2211981C Production of enantiomerically enriched ortho-substituted .alpha.,.alpha.-diaromatic methanols |
| 04/10/2008 | WO2008040652A1 Process for synthesis of phenoxy diaminopyrimidine derivatives |
| 04/10/2008 | WO2008003702A3 Fused bicyclic compounds interacting with the histamine h4 receptor |
| 04/10/2008 | WO2007110868A3 Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
| 04/10/2008 | WO2007065662A3 Trisubstituted quinazolinone derivatives as vanilloid antagonists |
| 04/10/2008 | US20080086004 To a cooled solution of ammonia was added the cooled sulfolane solution of 5-(2,4-diamino-pyrimidin-5-yloxy)-4-isopropyl-2-methoxy-benzenesulfonyl chloride to form -(2,4-diamino-pyrimidin-5-yloxy)-4-isopropyl-2-methoxy-benzenesulfonamide sulfolane solvate |
| 04/10/2008 | US20080085910 For inflammatory bowel disease; oral administration, bioavailability, pharmacokinetics; 2-(2,6-Dichlorobenzamido)-5-[4-(ethyl-pyrimidin-2-ylamino)phenyl]pent-4-enoic acid methyl ester for example |
| 04/10/2008 | US20080085907 Reverse transcriptase inhibitors; use against HIV with drug resistance to NNRTI's (Non Nucleoside Reverse Transcriptase Inhibitor drugs); Diaryl Pyrrolo(2,3-d)pyrimidines, diaryl purines, diaryl v-triazolo(4,5-d)pyrimidines |
| 04/10/2008 | US20080085900 Sulfonylguanidine compounds and pharmaceutical uses thereof |
| 04/10/2008 | US20080085890 Substituted isoquinoline-1,3(2H,4H)-diones, 1-thioxo-1,4-dihydro-2H-isoquinoline-3-ones and 1,4-dihydro-3 (2H)-isoquinolones and methods of use thereof |
| 04/10/2008 | CA2664305A1 Process for synthesis of phenoxy diaminopyrimidine derivatives |
| 04/09/2008 | EP1907368A1 2-cyano-pyrimidines and -triazines as cysteine protease inhibitors |
| 04/09/2008 | EP1907367A1 Design and synthesis of novel tubulin polymerization inhibitors: bonzoylphenyluria (bpu) sulfur analogs |
| 04/09/2008 | EP1309565B1 Heterocyclic mutilin esters and their use as antibacterials |
| 04/09/2008 | EP0964864B1 Pyrido 2,3-d pyrimidines and 4-aminopyrimidines as inhibitors of cellular proliferation |
| 04/09/2008 | EP0958287B2 Sulfamide-metalloprotease inhibitors |
| 04/09/2008 | CN101157657A Method for preparing azoxystrobin and its analogue |
| 04/09/2008 | CN100379730C Pyrimidine-sulfamides and their use as endothelian receptor antagonist |
| 04/09/2008 | CN100379729C Nitro compounds and their application in preparation of pemetrexed |
| 04/08/2008 | US7355044 Self-assembling dyes |
| 04/08/2008 | US7354946 Biarylurea derivatives |
| 04/03/2008 | WO2008039520A2 Fused ring compounds for inflammation and immune-related uses |
| 04/03/2008 | WO2008038955A1 Benzophenone derivatives useful for inhibiting formation of microtubule |
| 04/03/2008 | WO2008038132A1 Crystalline diamine salts of rosuvastatin |
| 04/03/2008 | WO2008015563A3 Salts of rosuvastatin and processes for their preparation |
| 04/03/2008 | WO2007125547A3 Novel process for statins and its pharmaceutically acceptable salts thereof |
| 04/03/2008 | US20080081811 5-[2-(cyclohexyloxy)-6-methyl-4-pyrimidinyl]-2-[5-(4-methyl-1-piperazinyl)methyl-2-pyrazinyl]amino-1,3-thiazole; anticarcinogenic agent; G1 phase in cell cycle; great selectivity |
| 04/02/2008 | EP1905765A1 6-arylamino-5-cyano-4-pyrimidinone as PDE9A-inhibitors |
| 04/02/2008 | EP1905441A2 Non-sedating barbiturate compounds as neuroprotective agents |
| 04/02/2008 | EP1904459A1 New crystal forms of 4-[6-methoxy-7-(3-piperidin-1-yl-propoxy)quinazolin-4-yl]piperazine-1-carboxylic acid(4-isopropoxyphenyl)-amide |
| 04/02/2008 | EP1904458A1 Method for the production of quinazolinone derivatives |
| 04/02/2008 | EP1904457A2 Compositions and methods for inhibition of the jak pathway |
| 04/02/2008 | EP1904456A1 Processes for the manufacture of rosuvastatin and intermediates |
| 04/02/2008 | EP1575949B1 Fungicides |
| 04/02/2008 | EP1201648B1 Carbamate derivatives and agricultural/horticultural bactericides |
| 04/02/2008 | CN101155789A 1h-quinaz0line-2,4-diones and their use as ampa-receptor ligands |
| 04/02/2008 | CN101155788A Crystal of 4(3h)-quinazolinone derivative |
| 04/02/2008 | CN101155787A (3,4-dihydro-quinazolin-2-yl)-indan-1-yl-amines |
| 04/02/2008 | CN101155786A N-phenyl-2-pyrimidine-amine derivatives and process for the preparation thereof |
| 04/02/2008 | CN101155785A Novel adenosine a3 receptor modulators |
| 04/02/2008 | CN100378101C 1.3.4-triaza-phenalene and 1,3,4,6-tetraazaphenalene derivatives |
| 04/02/2008 | CN100378100C Pyrazolo(4,3-d)pyrimidine derivatives |
| 04/02/2008 | CN100378082C Pyrimidine compounds and pests controlling composition containing the same |
| 04/02/2008 | CN100378081C Process for the manufacture of organic compounds |
| 04/02/2008 | CN100378072C Heterocyclic methyl sulfone derivative |
| 04/01/2008 | US7351829 Compounds on the basis of 2- and 4-chromenylidene-merocyanines respectively, and their use |
| 04/01/2008 | US7351826 Aryl acid pyrimidinyl methyl amides, pyridazinyl methyl amides and related compounds |
| 04/01/2008 | US7351825 4-[5-((1S,2R)-1-Carboxy-2-phenyl-cyclopropylsulfamoyl)-thiophen-2-yl]-3,6-dihydro-2H-pyridine-1-carboxylic acid tert-butyl ester; aggrecanase and matrix metalloproteinase (with zinc in the catalytic active center) (MMP) inhibitor; antiarthritic agent: osteoarthritis, rheumatoid arthritis |
| 04/01/2008 | US7351733 Tetrahydrocarbazole derivatives and their pharmaceutical use |
| 04/01/2008 | US7351700 4-(2-Hexylsulfanyl-6-methyl-pyrimidin-4-ylmethyl)-morpholine; antidepressant, anxiolytic agent, cognition activator; epilepsy, schizophrenia, spasticity and skeletal muscle rigidity, spinal cord injury, multiple sclerosis, amyotrophic lateral sclerosis, neuropathic pain |
| 03/27/2008 | WO2008036843A2 Nitrogen containing substituted heterocycles as platelet adp receptor inhibitors |
| 03/27/2008 | WO2008036286A1 Crystalline rosuvastatin calcium |
| 03/27/2008 | WO2008035359A2 Oximinophenoxyalkanoic acid and phenylalkanoic acid derivatives |
| 03/27/2008 | WO2008002671A3 Metalloprotease inhibitors |
| 03/27/2008 | WO2007056163A3 Aminopyrimidines useful as kinase inhibitors |
| 03/27/2008 | WO2007020411A8 Amide derivatives |
| 03/27/2008 | US20080076914 Method of Deprotection |
| 03/27/2008 | US20080076785 Phytopathogenic |
| 03/27/2008 | US20080076784 Bicyclic, Nitrogen-Containing Heterocycles and Aromatase Inhibitors |
| 03/27/2008 | US20080076783 Cycloalkyl Keto Piperidine Tachykinin Receptor Antagonists |
| 03/27/2008 | US20080076667 Substituted fluoroalkoxyphenylsulfonylureas |
| 03/27/2008 | US20080076188 Luminescent compounds |
| 03/27/2008 | DE112005003498T5 Herstellungsverfahren für Chinazolinderivate und Anwendung zur Herstellung zur Behandlung von Tumorerkrankungen A method for manufacturing and application for the production of quinazoline derivatives for the treatment of tumor diseases |
| 03/27/2008 | DE102006021874B4 4,5-Diphenyl-pyrimidinyl-amino substituierte Carbonsäuren, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel 4,5-diphenyl-pyrimidinyl-amino substituted carboxylic acids, process for their preparation and their use as medicaments |
| 03/27/2008 | CA2664411A1 Platelet adp receptor inhibitors |
| 03/26/2008 | EP1903030A1 Method for catalytic manufacture of aromatic or heteroaromatic nitriles |
| 03/26/2008 | EP1902037A1 2,4-diamino-pyrimidines used as aurora inhibitors |
| 03/26/2008 | EP1902036A2 Process for the preparation of rosuvastatin |
| 03/26/2008 | EP1509218A4 Peptide deformylase inhibitors |
| 03/26/2008 | EP1455790B1 Use of pyridine-2,4-dicarboxylic acid diamides and of pyrimidine-4,6-dicarboxylic acid diamides for selective collagenase inhibition |
| 03/26/2008 | CN101151261A Pyrimidine compounds having tie2 (TEK) inhibitory activity |
| 03/26/2008 | CN101151258A Pyrimidine derivatives for treatment of hyperproliferative disorders |
| 03/26/2008 | CN101151255A 5-phenyl-pentanoic acid derivatives as matrix metalloproteinase inhibitors for the treatment of asthma and other diseases |
| 03/26/2008 | CN101151254A Diketo acids with nucleobase scaffolds: anti-HIV replication inhibitors targeted at HIV integrase |
| 03/26/2008 | CN101151253A Substituted n-[pyrimidin-2-ylmethyl]carboxamides and their use as herbicides and plant growth regulators |
| 03/26/2008 | CN101151252A Multimers of pyrimidinone derivatives and their use as human neutrophil elastase inhibitors |
| 03/26/2008 | CN101148439A Preparing method for gefitinib |
| 03/26/2008 | CN100376580C Pyrazolopyrimidines as cyclin-dependent kinase inhibitors |
| 03/26/2008 | CN100376571C 6-substituted pyrido-pyrimidines |
| 03/26/2008 | CN100376246C Pyrimidine-2,4-dione derivatives as gonadotropin-releasing hormone receptor antagonists |
| 03/25/2008 | US7348335 Compositions useful as inhibitors of JAK and other protein kinases |
| 03/25/2008 | US7348334 Monocyclic derivatives of aryl alkanoic acids and their use in medicine: process for their preparation and pharmaceutical compositions containing them |
| 03/25/2008 | US7348333 Treating bone disorder caused by osteoclasts, tumor growth and tumor metastasis, prophylaxis of cardiovascular disorders, nephropathies or retinopathies |
| 03/25/2008 | US7348332 (3,4-dihydro-quinazolin-2-yl)-(R)-indan-1-yl-amine; serotonin (5-HT5A) receptor antagonist/agonist; anxiolitic, antidepressant, sleep disorders and schizophrenia; amination thioquinazolin with 1-aminoindane |
| 03/25/2008 | US7348148 Polynucleotide analog with polyether, polythioether, polyether sulfone, and/or and polyether sulfoxide linkages; antisense drug therapy |
| 03/20/2008 | WO2008033834A1 Pyrimidines derivatives and their use as kinase inhibitors |
| 03/20/2008 | WO2008031888A2 Condensed pyrimidinones active on glutamatergic receptors |
| 03/20/2008 | WO2008031556A2 2 amino-pyrimidine derivatives as h4 receptor antagonists, processes for preparing them and their use in pharmaceutical compositions |
| 03/20/2008 | WO2008031509A1 ISOSERINE DERIVATIVES FOR USE AS COAGULATION FACTOR IXa INHIBITORS |
| 03/20/2008 | WO2007144769A3 Aryl- and heteroaryl-ethyl-acylguanidine derivatives, their preparation and their application in therapeutics |