Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
09/2008
09/17/2008EP1392639B1 Pyruvate derivatives
09/17/2008CN101268059A 2-substituted hydroxylaminopyrimidine, method for the production and the use thereof in the form of pesticides
09/17/2008CN101268058A 4-phenyl-6-substituted-pyrimidine-2-carbonitrile derivatives
09/17/2008CN101268043A Amino-alkyl-amide derivatives as CCR3 receptor ligands
09/17/2008CN101265235A Method for preparing herbicide bispyribac-sodium
09/17/2008CN101265234A Method for synthesizing aditoprim
09/17/2008CN100418954C 3h-quinazolin-4-one derivatives
09/17/2008CN100418952C Biphenyl derivatives and their use as fungicides
09/17/2008CN100418951C Cycloamine derivative and its use as medicine
09/16/2008US7425631 Compounds and methods of use
09/16/2008US7425629 Stereoselective synthesis of certain trifluoromethyl-substituted alcohols
09/16/2008US7425564 Quinoline derivative and quinazoline derivative inhibiting self-phosphorylation of hepatocytus prolifertor receptor and medicinal composition containing the same
09/16/2008US7425559 Medicine containing pyrimidine derivative
09/16/2008US7425557 Inhibitors of glycogen synthase kinase 3
09/16/2008CA2515338C Inhibitors of histone deacetylase
09/16/2008CA2427221C Process and intermediates for preparing anti-cancer compounds
09/16/2008CA2182228C Codrugs as a method of controlled drug delivery
09/12/2008WO2008109697A2 Ppar active compounds
09/12/2008WO2008109417A1 Mgmt inhibitor combinations for the treatment of neoplastic disorders
09/12/2008WO2008109178A1 Metalloprotease inhibitors containing a squaramide moiety
09/12/2008WO2008109027A2 Tri-aryl/heteroaroaromatic cannabinoids and use thereof
09/12/2008WO2008107436A1 Bicyclic organic compounds suitable for the treatment of inflammatory or allergic conditions
09/12/2008WO2008107211A2 Novel p2y12 receptor antagonists
09/12/2008WO2008107096A1 Diaminopyrimidines as fungicides
09/12/2008WO2008089933A3 Benzoquinazole derivatives
09/12/2008WO2007117399A3 Benzoimidazol-2-yl pyrimidines and pyrazines as modulators of the histamine h4 receptor
09/12/2008CA2680177A1 Metalloprotease inhibitors containing a heterocyclic moiety
09/12/2008CA2679844A1 Ppar active compounds
09/12/2008CA2679488A1 Diaminopyrimidines as fungicides
09/12/2008CA2678492A1 Bicyclic organic compounds suitable for the treatment of inflammatory or allergic conditions
09/11/2008US20080221325 And sulfonated poly(aryl ether ketone) monomers; crosslinked with barbituric acid; fuel cells, seawater desalination, heavy water and sewage treatment and biomass-energy resources; improved water holding capacity, chemical resistance, electrochemical stability and heat resistance
09/11/2008US20080221324 Iclaprim; protecting the phenol group of 5-[(2-hydroxy-3,4-dimethoxy-benzaldehyde)methyl]-2,4-dilkylamidopyrimidine, reacting with cyclopropyl methyl ketone, reducing the ketone, acid catalyzed cyclization, deprotecting; dihydrofolate reductase inhibitors; fewer crystalline intermediates, improved yield
09/11/2008US20080221323 Production of Rosuvastatin Calcium Salt
09/11/2008US20080221132 Multi-Functional Small Molecules as Anti-Proliferative Agents
09/11/2008US20080221127 Ppar active compounds
09/11/2008US20080221103 4-(3-Methyl-2,5-dioxo-2,5-dihydro-1H-pyrrol-1-ylamino)-6-(methylthio)-2-phenylpyrimidine-5-carbonitrile; having significant in vitro TNF- alpha inhibitory activity useful for the treatment of various inflammatory diseases such as arthritis, inflammatory bowel disease, psoriasis, asthma, COPD, cancer etc.
09/11/2008US20080221096 Pyrido[3' ,2':4,5]Furo[3,2-d]Pyrimidine Derivatives
09/11/2008US20080221095 increased potency and selectivity in relation to currently known MMP-13, MMP-8 and MMP-3 inhibitors; treating rheumatoid arthritis, osteoarthritis or inflammation; squaramide or benzoxazinone moiety
09/11/2008US20080221089 Compositions and methods for inhibition of the jak pathway
09/11/2008US20080221083 Heterobicyclic metalloprotease inhibitors
09/11/2008US20080221078 Use of a CB1 Antagonist for Treating Side Effects and Negative Symptoms of Schizophrenia
09/11/2008US20080220454 Using erastin as therapeutic agent in treatment of cell proliferative disorders associated with mutation in ras gene
09/11/2008US20080216606 Grinding to uniform particle size; heating; pressurization;; extraction from ores, concentrates
09/10/2008EP1967513A1 Novel P2Y12 receptor antagonists
09/10/2008EP1966189A1 Bicyclic heterocycles, medicaments containing said compounds, use thereof, and method for the production thereof
09/10/2008EP1966163A1 Pyrimidine derivatives useful as inhibitors of pkc-theta
09/10/2008EP1966162A2 Pyrimidine derivatives
09/10/2008EP1966161A1 Carboxamides for controlling undesired micro-organisms in plant protection
09/10/2008EP1966160A1 SUBSTITUTED 2-AMINOPYRIMIDINE-4-ONES, THEIR PHARMACEUTICAL COMPOSITIONS AND THEIR USE IN THE TREATMENT AND/OR PREVENTION OF Aß-RELATED PATHOLOGIES
09/10/2008EP1966159A2 Chemical compounds
09/10/2008EP1966144A1 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors
09/10/2008EP1966141A1 Six-membered heterocycles useful as serine protease inhibitors
09/10/2008EP1965805A1 Urea derivatives useful as calcium receptor modulators
09/10/2008EP1965644A1 Novel herbicides
09/10/2008EP1646389B1 Pyrimidine-2,4-dione derivatives as gonadotropin-releasing hormone receptor antagonists
09/10/2008EP1597240B1 Bicyclic heterocycles, medicaments containing said compounds, use thereof, and method for the production thereof
09/10/2008EP1438053B1 Pyrimidine derivatives, pharmaceutical agent containing said compounds, use and method for making same
09/10/2008CN101263125A Quinazoline derivatives useful in cancer treatment
09/10/2008CN101263124A Quinazoline derivatives useful in cancer treatment
09/10/2008CN101263123A Pesticide pyrimidinyloxy substituted phenylamidine derivatives
09/10/2008CN101260107A Diheterocycle compound containing 4-thiazolidinone and pyrimidine, synthetic method and application thereof
09/10/2008CN101260082A Method for preparing 3,4-dihydropyrimidin-2(1-H)-ones compounds
09/09/2008US7423148 Small molecule PI 3-kinase inhibitors and methods of their use
09/09/2008US7423044 A cyclopenta[d]pyrimidine, or 5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine derivatives; treating metabolic disorders, type II diabetes, controlling glucose levels
09/09/2008US7422013 Dry powder dispersing apparatus and methods for their use
09/09/2008CA2225756C Substituted cyanophenyl uracils
09/09/2008CA2211646C Substituted phenyl compounds as endothelin antagonists
09/04/2008WO2008106692A1 Pim kinase inhibitors and methods of their use
09/04/2008WO2008106635A1 Pyrimidine-2,4-diamine derivatives and their use as jak2 kinase inhibitors
09/04/2008WO2008105968A1 Novel seh inhibitors and their use
09/04/2008WO2008105515A1 Novel hydroxamic acid derivative
09/04/2008WO2008105386A1 Rexinoid compound having alkoxy group
09/04/2008WO2008104994A2 2,2,2-tri-substituted acetamide derivatives as glucokinase activators, their process and pharmaceutical application
09/04/2008WO2008104754A1 Novel pyrimidine derivatives 698
09/04/2008WO2008104474A1 Diaminopyrimidines
09/04/2008WO2008104472A1 2, 4 -diaminopyrimidine derivatives and their use as p2x antagonists or as prodrugs thereof
09/04/2008WO2008086462A3 AMINO-SUBSTITUTED QUINAZOLINE DERIVATIVES AS INHIBITORS OF β-CANTENIN/TCF-4 PATHWAY AND CANCER TREATMENT AGENTS
09/04/2008WO2008080965A3 Hiv inhibiting 5,6-substituted pyrimidines
09/04/2008WO2007126988A3 Selective androgen receptor modulators and methods of use thereof
09/04/2008US20080214812 Trisubstituted triazolopyrimidines for use in platelet aggregation inhibition
09/04/2008US20080214810 Dye-forming coupler, silver halide photographic light-sensitive material, and azomethine dye compound
09/04/2008US20080214809 Using 3-(2-chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrrido[1,2-a]-pyrimidin-4-one (CMHTP) as chemical intermediate for paliperidone (9-hydroxyrisperidone); catalytic hydrogenation
09/04/2008US20080214808 Preparation of Aseptic 3-[2-[4-((6-Fluoro-1,2-Benzisoxazol-3-Yl)-1-Piperidinyl]-6,7,8,9-Tetrahydro-9-Hydroxy-2-Methyl-4H-Pyrido[1,2-a]Pyrimidin-4-One Palmitate Ester
09/04/2008US20080214628 Administering a compound (2S)-(4E)-N-methyl-5-(5-isopropoxy-3-pyridyl-4-penten-2-amine; attention deficit disorder
09/04/2008US20080214588 replication inhibitors; show improved ability to inhibit the replication of mutant strains, in particular strains which show double or multiple mutations in the viral genome encoding for reverse transcriptase
09/04/2008US20080214587 Coupling of methyl (E)-2-{2-[6-chloropyrimidin-4-yloxy]phenyl}-3-methoxyacrylate with 2-cyanophenyl in DMF with 2 mol % DABCO; significantly smaller amounts of this relatively expensive catalyst may be used without compromising the yield
09/04/2008US20080214586 2-Amino-4-Phenylquinazoline Derivatives and the Use Thereof as Hsp90 Modulators
09/04/2008US20080214560 (4-{[5-Fluoro-4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)pyrimidin-2-yl]amino}phenyl)(phenyl)methanone hydrochloride; glycogen synthase kinase-3 inhibitors
09/04/2008US20080214558 2-[(2-(4-methylpyrazin-1-yl)-3-fluoro-5-pyridinyl)amino]-4-[(3-chloro-4-fluoro) or (3-cyanomethyl)phenylamino]pyrimidine; 2-[(4-(4-methylpyrazin-1-yl)-phenyl)amino]-4-[(3-chloro-4-fluoro) or (3-cyanomethyl)phenylamino]pyrimidine; colon, breast, stomach, urogenital, pancreatic cancers, leukemia lymphoma
09/04/2008US20080214548 2-Cyano-Pyrimidines and-Triazines as Cysteine Protease Inhibitors
09/04/2008US20080214543 Antiandrogen; prostate cancer; excellent oral pharmacokinetics
09/04/2008US20080214538 Pyridoindolone Derivatives Substituted in the 3-Position by a Phenyl, Their Preparation and Their Application in Therapeutics
09/04/2008DE102007010801A1 Use of new or known 2,4-diaminopyrimidine derivatives as fungicides
09/04/2008CA2679659A1 Pim kinase inhibitors and methods of their use
09/04/2008CA2679489A1 Pyrimidine-2,4-diamine derivatives and their use as jak2 kinase inhibitors
09/04/2008CA2679185A1 2,2,2-tri-substituted acetamide derivatives as glucokinase activators, their process and pharmaceutical application
09/03/2008EP1964839A2 Quinazoline derivatives as kinase inhibitors
09/03/2008EP1964575A1 Pharmaceutical comprising ppar agonist
09/03/2008EP1963284A1 Novel quinazoline-2,4-diamine derivatives and their use as modulators of small-conductance calcium-activated potassium channels
09/03/2008EP1963283A2 Trisubstituted quinazolinone derivatives as vanilloid antagonists