Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619) |
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09/17/2008 | EP1392639B1 Pyruvate derivatives |
09/17/2008 | CN101268059A 2-substituted hydroxylaminopyrimidine, method for the production and the use thereof in the form of pesticides |
09/17/2008 | CN101268058A 4-phenyl-6-substituted-pyrimidine-2-carbonitrile derivatives |
09/17/2008 | CN101268043A Amino-alkyl-amide derivatives as CCR3 receptor ligands |
09/17/2008 | CN101265235A Method for preparing herbicide bispyribac-sodium |
09/17/2008 | CN101265234A Method for synthesizing aditoprim |
09/17/2008 | CN100418954C 3h-quinazolin-4-one derivatives |
09/17/2008 | CN100418952C Biphenyl derivatives and their use as fungicides |
09/17/2008 | CN100418951C Cycloamine derivative and its use as medicine |
09/16/2008 | US7425631 Compounds and methods of use |
09/16/2008 | US7425629 Stereoselective synthesis of certain trifluoromethyl-substituted alcohols |
09/16/2008 | US7425564 Quinoline derivative and quinazoline derivative inhibiting self-phosphorylation of hepatocytus prolifertor receptor and medicinal composition containing the same |
09/16/2008 | US7425559 Medicine containing pyrimidine derivative |
09/16/2008 | US7425557 Inhibitors of glycogen synthase kinase 3 |
09/16/2008 | CA2515338C Inhibitors of histone deacetylase |
09/16/2008 | CA2427221C Process and intermediates for preparing anti-cancer compounds |
09/16/2008 | CA2182228C Codrugs as a method of controlled drug delivery |
09/12/2008 | WO2008109697A2 Ppar active compounds |
09/12/2008 | WO2008109417A1 Mgmt inhibitor combinations for the treatment of neoplastic disorders |
09/12/2008 | WO2008109178A1 Metalloprotease inhibitors containing a squaramide moiety |
09/12/2008 | WO2008109027A2 Tri-aryl/heteroaroaromatic cannabinoids and use thereof |
09/12/2008 | WO2008107436A1 Bicyclic organic compounds suitable for the treatment of inflammatory or allergic conditions |
09/12/2008 | WO2008107211A2 Novel p2y12 receptor antagonists |
09/12/2008 | WO2008107096A1 Diaminopyrimidines as fungicides |
09/12/2008 | WO2008089933A3 Benzoquinazole derivatives |
09/12/2008 | WO2007117399A3 Benzoimidazol-2-yl pyrimidines and pyrazines as modulators of the histamine h4 receptor |
09/12/2008 | CA2680177A1 Metalloprotease inhibitors containing a heterocyclic moiety |
09/12/2008 | CA2679844A1 Ppar active compounds |
09/12/2008 | CA2679488A1 Diaminopyrimidines as fungicides |
09/12/2008 | CA2678492A1 Bicyclic organic compounds suitable for the treatment of inflammatory or allergic conditions |
09/11/2008 | US20080221325 And sulfonated poly(aryl ether ketone) monomers; crosslinked with barbituric acid; fuel cells, seawater desalination, heavy water and sewage treatment and biomass-energy resources; improved water holding capacity, chemical resistance, electrochemical stability and heat resistance |
09/11/2008 | US20080221324 Iclaprim; protecting the phenol group of 5-[(2-hydroxy-3,4-dimethoxy-benzaldehyde)methyl]-2,4-dilkylamidopyrimidine, reacting with cyclopropyl methyl ketone, reducing the ketone, acid catalyzed cyclization, deprotecting; dihydrofolate reductase inhibitors; fewer crystalline intermediates, improved yield |
09/11/2008 | US20080221323 Production of Rosuvastatin Calcium Salt |
09/11/2008 | US20080221132 Multi-Functional Small Molecules as Anti-Proliferative Agents |
09/11/2008 | US20080221127 Ppar active compounds |
09/11/2008 | US20080221103 4-(3-Methyl-2,5-dioxo-2,5-dihydro-1H-pyrrol-1-ylamino)-6-(methylthio)-2-phenylpyrimidine-5-carbonitrile; having significant in vitro TNF- alpha inhibitory activity useful for the treatment of various inflammatory diseases such as arthritis, inflammatory bowel disease, psoriasis, asthma, COPD, cancer etc. |
09/11/2008 | US20080221096 Pyrido[3' ,2':4,5]Furo[3,2-d]Pyrimidine Derivatives |
09/11/2008 | US20080221095 increased potency and selectivity in relation to currently known MMP-13, MMP-8 and MMP-3 inhibitors; treating rheumatoid arthritis, osteoarthritis or inflammation; squaramide or benzoxazinone moiety |
09/11/2008 | US20080221089 Compositions and methods for inhibition of the jak pathway |
09/11/2008 | US20080221083 Heterobicyclic metalloprotease inhibitors |
09/11/2008 | US20080221078 Use of a CB1 Antagonist for Treating Side Effects and Negative Symptoms of Schizophrenia |
09/11/2008 | US20080220454 Using erastin as therapeutic agent in treatment of cell proliferative disorders associated with mutation in ras gene |
09/11/2008 | US20080216606 Grinding to uniform particle size; heating; pressurization;; extraction from ores, concentrates |
09/10/2008 | EP1967513A1 Novel P2Y12 receptor antagonists |
09/10/2008 | EP1966189A1 Bicyclic heterocycles, medicaments containing said compounds, use thereof, and method for the production thereof |
09/10/2008 | EP1966163A1 Pyrimidine derivatives useful as inhibitors of pkc-theta |
09/10/2008 | EP1966162A2 Pyrimidine derivatives |
09/10/2008 | EP1966161A1 Carboxamides for controlling undesired micro-organisms in plant protection |
09/10/2008 | EP1966160A1 SUBSTITUTED 2-AMINOPYRIMIDINE-4-ONES, THEIR PHARMACEUTICAL COMPOSITIONS AND THEIR USE IN THE TREATMENT AND/OR PREVENTION OF Aß-RELATED PATHOLOGIES |
09/10/2008 | EP1966159A2 Chemical compounds |
09/10/2008 | EP1966144A1 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors |
09/10/2008 | EP1966141A1 Six-membered heterocycles useful as serine protease inhibitors |
09/10/2008 | EP1965805A1 Urea derivatives useful as calcium receptor modulators |
09/10/2008 | EP1965644A1 Novel herbicides |
09/10/2008 | EP1646389B1 Pyrimidine-2,4-dione derivatives as gonadotropin-releasing hormone receptor antagonists |
09/10/2008 | EP1597240B1 Bicyclic heterocycles, medicaments containing said compounds, use thereof, and method for the production thereof |
09/10/2008 | EP1438053B1 Pyrimidine derivatives, pharmaceutical agent containing said compounds, use and method for making same |
09/10/2008 | CN101263125A Quinazoline derivatives useful in cancer treatment |
09/10/2008 | CN101263124A Quinazoline derivatives useful in cancer treatment |
09/10/2008 | CN101263123A Pesticide pyrimidinyloxy substituted phenylamidine derivatives |
09/10/2008 | CN101260107A Diheterocycle compound containing 4-thiazolidinone and pyrimidine, synthetic method and application thereof |
09/10/2008 | CN101260082A Method for preparing 3,4-dihydropyrimidin-2(1-H)-ones compounds |
09/09/2008 | US7423148 Small molecule PI 3-kinase inhibitors and methods of their use |
09/09/2008 | US7423044 A cyclopenta[d]pyrimidine, or 5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine derivatives; treating metabolic disorders, type II diabetes, controlling glucose levels |
09/09/2008 | US7422013 Dry powder dispersing apparatus and methods for their use |
09/09/2008 | CA2225756C Substituted cyanophenyl uracils |
09/09/2008 | CA2211646C Substituted phenyl compounds as endothelin antagonists |
09/04/2008 | WO2008106692A1 Pim kinase inhibitors and methods of their use |
09/04/2008 | WO2008106635A1 Pyrimidine-2,4-diamine derivatives and their use as jak2 kinase inhibitors |
09/04/2008 | WO2008105968A1 Novel seh inhibitors and their use |
09/04/2008 | WO2008105515A1 Novel hydroxamic acid derivative |
09/04/2008 | WO2008105386A1 Rexinoid compound having alkoxy group |
09/04/2008 | WO2008104994A2 2,2,2-tri-substituted acetamide derivatives as glucokinase activators, their process and pharmaceutical application |
09/04/2008 | WO2008104754A1 Novel pyrimidine derivatives 698 |
09/04/2008 | WO2008104474A1 Diaminopyrimidines |
09/04/2008 | WO2008104472A1 2, 4 -diaminopyrimidine derivatives and their use as p2x antagonists or as prodrugs thereof |
09/04/2008 | WO2008086462A3 AMINO-SUBSTITUTED QUINAZOLINE DERIVATIVES AS INHIBITORS OF β-CANTENIN/TCF-4 PATHWAY AND CANCER TREATMENT AGENTS |
09/04/2008 | WO2008080965A3 Hiv inhibiting 5,6-substituted pyrimidines |
09/04/2008 | WO2007126988A3 Selective androgen receptor modulators and methods of use thereof |
09/04/2008 | US20080214812 Trisubstituted triazolopyrimidines for use in platelet aggregation inhibition |
09/04/2008 | US20080214810 Dye-forming coupler, silver halide photographic light-sensitive material, and azomethine dye compound |
09/04/2008 | US20080214809 Using 3-(2-chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrrido[1,2-a]-pyrimidin-4-one (CMHTP) as chemical intermediate for paliperidone (9-hydroxyrisperidone); catalytic hydrogenation |
09/04/2008 | US20080214808 Preparation of Aseptic 3-[2-[4-((6-Fluoro-1,2-Benzisoxazol-3-Yl)-1-Piperidinyl]-6,7,8,9-Tetrahydro-9-Hydroxy-2-Methyl-4H-Pyrido[1,2-a]Pyrimidin-4-One Palmitate Ester |
09/04/2008 | US20080214628 Administering a compound (2S)-(4E)-N-methyl-5-(5-isopropoxy-3-pyridyl-4-penten-2-amine; attention deficit disorder |
09/04/2008 | US20080214588 replication inhibitors; show improved ability to inhibit the replication of mutant strains, in particular strains which show double or multiple mutations in the viral genome encoding for reverse transcriptase |
09/04/2008 | US20080214587 Coupling of methyl (E)-2-{2-[6-chloropyrimidin-4-yloxy]phenyl}-3-methoxyacrylate with 2-cyanophenyl in DMF with 2 mol % DABCO; significantly smaller amounts of this relatively expensive catalyst may be used without compromising the yield |
09/04/2008 | US20080214586 2-Amino-4-Phenylquinazoline Derivatives and the Use Thereof as Hsp90 Modulators |
09/04/2008 | US20080214560 (4-{[5-Fluoro-4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)pyrimidin-2-yl]amino}phenyl)(phenyl)methanone hydrochloride; glycogen synthase kinase-3 inhibitors |
09/04/2008 | US20080214558 2-[(2-(4-methylpyrazin-1-yl)-3-fluoro-5-pyridinyl)amino]-4-[(3-chloro-4-fluoro) or (3-cyanomethyl)phenylamino]pyrimidine; 2-[(4-(4-methylpyrazin-1-yl)-phenyl)amino]-4-[(3-chloro-4-fluoro) or (3-cyanomethyl)phenylamino]pyrimidine; colon, breast, stomach, urogenital, pancreatic cancers, leukemia lymphoma |
09/04/2008 | US20080214548 2-Cyano-Pyrimidines and-Triazines as Cysteine Protease Inhibitors |
09/04/2008 | US20080214543 Antiandrogen; prostate cancer; excellent oral pharmacokinetics |
09/04/2008 | US20080214538 Pyridoindolone Derivatives Substituted in the 3-Position by a Phenyl, Their Preparation and Their Application in Therapeutics |
09/04/2008 | DE102007010801A1 Use of new or known 2,4-diaminopyrimidine derivatives as fungicides |
09/04/2008 | CA2679659A1 Pim kinase inhibitors and methods of their use |
09/04/2008 | CA2679489A1 Pyrimidine-2,4-diamine derivatives and their use as jak2 kinase inhibitors |
09/04/2008 | CA2679185A1 2,2,2-tri-substituted acetamide derivatives as glucokinase activators, their process and pharmaceutical application |
09/03/2008 | EP1964839A2 Quinazoline derivatives as kinase inhibitors |
09/03/2008 | EP1964575A1 Pharmaceutical comprising ppar agonist |
09/03/2008 | EP1963284A1 Novel quinazoline-2,4-diamine derivatives and their use as modulators of small-conductance calcium-activated potassium channels |
09/03/2008 | EP1963283A2 Trisubstituted quinazolinone derivatives as vanilloid antagonists |