Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
07/2008
07/15/2008US7399760 1-(4-Methylsulfanyl-phenyl)-6-phenyl-pyrimidin-2,4-(1H)-dione;cyclooxygenase and prostaglandin inhibitor; tumor necrosis factor and interleukins 1, 6, 8, 12 antagonist;
07/15/2008US7399537 Organic electroluminescence device and phenylenediamine derivative
07/15/2008US7399505 Nematic or cholesteric or chiral-smectic; high absolute values of dielectric anisotropy combined with a favorable ratio of viscosity to clearing point; light- and UV-stable, and also thermally stable; high voltage holding ratio
07/15/2008CA2275400C Process for the preparation of substituted pyrimidine desrivatives
07/15/2008CA2144473C Pna synthesis using a base-labile amino protecting group
07/14/2008CA2675265A1 Process for the preparation of ethyl-n-(2, 3-dichloro-6-nitrobenzyl) glycine hydrochloride
07/10/2008WO2008083280A1 Compounds and methods of treating insulin resistance and cardiomyopathy
07/10/2008WO2008083101A1 Phosphoramidate alkylator prodrugs for the treatment of cancer
07/10/2008WO2008080965A2 Hiv inhibiting 5,6-substituted pyrimidines
07/10/2008WO2008080964A1 Hiv inhibiting 6-substituted pyrimidines
07/10/2008US20080167464 Processes for the preparation of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile
07/10/2008US20080167330 Anticancer agents
07/10/2008US20080167329 3,4-Dihydroquinazolin-2(1H)-ones, e.g., 4-Ethyl-6-chloro-4-phenyl-3-(2,2,2-trifluoroethyl)-3,4-dihydroquinazolin-2(1H)-one; treatment of epilepsy, pain, movement disorders, cognitive disorders, psychological disorders, sleep disorders, hot flashes, fibromyalgia, and drug withdrawl
07/10/2008US20080167328 Antitumor agents
07/10/2008US20080167327 Crystalline, formed by crystallizing from an aqueous solution without agitation; treating cancer
07/10/2008US20080167310 Syndrome X, antidiabetic agents; hypoglycemic agents;antilipemic agents; artherosclerosis; cardiovascular disorders
07/10/2008US20080167308 Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors
07/10/2008US20080167307 Carboxylic Acid Derivative Containing Thiazole Ring and Pharmaceutical Use Thereof
07/10/2008US20080167301 Novel Hydroxy-6-Heteroarylphenanthridines and Their Use as Pde4 Inhibitors
07/10/2008US20080167287 Imidazotriazines and imidazopyrimidines as kinase inhibitors
07/10/2008US20080166358 Quinazoline derivatives and methods of treatment
07/10/2008CA2674185A1 Hiv inhibiting 5,6-substituted pyrimidines
07/10/2008CA2674178A1 Hiv inhibiting 6-substituted pyrimidines
07/09/2008EP1942105A1 Aminodihydrothiazine derivative
07/09/2008EP1940827A1 Carbamate compounds which inhibit leukocyte adhesion mediated by vla-4
07/09/2008EP1940826A1 Pyrimidinyl amide compounds which inhibit leukocyte adhesion mediated by vla-4
07/09/2008EP1940814A1 Piperazine derivatives as antimalarial agents
07/09/2008EP1940804A2 Novel pyrimidine-2,4-diamine derivatives and their use as modulators of small-conductance calcium-activated potassium channels
07/09/2008EP1940407A2 N-(4-oxo-3,4-dihydroquinazolin-2-yl)butanamides as androgen receptor modulators
07/09/2008EP1768978B1 2,4,6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer
07/09/2008CN101218211A Quinoxaline derivatives as antitumor agents
07/09/2008CN101218210A Processes for the manufacture of rosuvastatin and intermediates
07/09/2008CN101215264A Method for synthesizing pyrimidinamine
07/09/2008CN100400523C Substituted piperazines,(1,4) diaszepines, and 2,5-diazabicyclo (2.2.1)iieptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists
07/09/2008CN100400487C Glucocorticoid receptor modulators
07/09/2008CN100400107C Drugs for diagnosis of tissue-reproductive activity or treatment of proliferative disease
07/08/2008US7396927 Process for preparation of rosuvastatin calcium
07/08/2008US7396844 3-(4-amidinobenzoylamino)-4-[5-amidino-2-(2-carboxy-2-oxoethyl)phenoxy]butanoic acid; anticoagulant; blood coagulation factor X and thrombin inhibitor; cerebral infarction, thrombosis, embolism, transient ischemic attack (TIA) and subarachnoidal hemorrhage (vasospasm); ischemic heart diseases
07/08/2008US7396836 Pyrimidine compound and medicinal composition thereof
07/08/2008US7396831 Vanilloid receptor ligands and their use in treatments
07/03/2008WO2008079907A1 Compositions and methods for inhibition of the jak pathway
07/03/2008WO2008079719A1 Pyrimidine kinase inhibitors
07/03/2008WO2008078674A1 Glucokinase-activating substance
07/03/2008WO2008077885A2 2- [(phenylamino) -pyrimidin-4ylamin0] -cyclopentane carboxamide derivatives and related compounds as inhibitors of kinases of the cell cycle for the treatment of cancer
07/03/2008WO2008077548A1 Pyrimidyl derivatives as protein kinase inhibitors
07/03/2008WO2008077507A1 Heteroaryl-substituted carboxamides and use thereof for the stimulation of the expression of no synthase
07/03/2008WO2008077453A1 5-fluorouracil derivatives and their use for the treatment of cancer
07/03/2008WO2008077188A1 Bicyclic pyrimidinones and uses thereof
07/03/2008WO2008061208A3 Arylsulfonamide compounds
07/03/2008WO2008061208A2 Arylsulfonamide compounds
07/03/2008WO2008053334A3 An improved process for preparing rosuvastatin calcium
07/03/2008WO2008043835A3 Crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2h)-pyrimidinyl]-4-fluoro-n-[[methyl-(1-methyl-ethyl)amino]sulphonyl]benzamide
07/03/2008WO2007039112A8 Novel phloroglucinol derivatives having selectin ligand activity
07/03/2008US20080161562 2-(6-Chloro-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethyl)-benzonitrile
07/03/2008US20080161561 Reacting N-[4-(2,2-Dimethyl-propionylamino)-5-(3,4,5-trimethoxy-benzyl)-pyrimidin-2-yl]-2,2-dimethyl-propionamide with an indole to produce 3-[4-(2,4-Bis-isobutyrylamino-pyrimidin-5-ylmethyl)-6,7-dimethoxy-benzofuran-2-carbonyl]-5-chloro-1-(toluene-4-sulfonyl)-1H-indole-2-carboxylicacid-dimethylamide
07/03/2008US20080161560 Reacting N-[4-(4-flurophenyl)-5-formyl-6-isopropylpyrimidin-2-yl]-N-methylmethylsulfonamide with (carbethoxymethylene)triphenylphosphorane producing the correct absolute stereochemistry at C-5 (S) of Rosuvastatin side chain followed by regioselective chain extension
07/03/2008US20080161322 e.g. 1-[2-tert-Butyl-6-(trifluoromethyl)pyrimidin-4-yl]-4-[3-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)propyl]piperazin-4-ium chloride3,4-Dihydroquinolin-2(1H)-one; dopamine D3 receptor antagonists or agonists; antidepressant, schizophrenia, Parkinson's disease
07/03/2008US20080161310 (2S)-4,4-difluoro-1-(2-{[1-(2-pyrazinyl)piperidin-4-yl]amino}acetyl)-2-pyrrolidine carbonitrile; enzyme inhibitors; diabetes
07/03/2008US20080161297 Rho kinase inhibitors
07/03/2008CA2673466A1 Substituted tetracycline compounds
07/03/2008CA2673184A1 New compounds
07/03/2008CA2673183A1 Bicyclic pyrimidinones and uses thereof
07/03/2008CA2673003A1 Quinazolines for pdk1 inhibition
07/03/2008CA2672718A1 Pyrimidyl derivatives as protein kinase inhibitors
07/03/2008CA2672564A1 Substituted heteroaryl pyridopyrimidone derivatives
07/03/2008CA2672088A1 Glucokinase activator
07/03/2008CA2670645A1 Pyrimidine kinase inhibitors
07/03/2008CA2664118A1 Protease inhibitors
07/02/2008EP1939203A2 Inhibitors of human phosphatidyl-inositol 3-kinase delta isoform
07/02/2008EP1939187A1 Substituted heteroaryl pyridopyrimidone derivatives
07/02/2008EP1939186A1 5-Fluorouracil derivatives and their use for the treatment of cancer
07/02/2008EP1939185A1 New types of hetaryl-phenylendiamin-pyrimidines as protein kinase inhibitors for the treatment of cancer
07/02/2008EP1939181A1 Heteroaryl-substituted carboxamides and use thereof for the stimulation of the expression of NO synthase
07/02/2008EP1937672A1 N-[(4,5-diphenylpyrimidin-2-yl)methyl]amine derivatives, the preparation thereof and their therapeutic use
07/02/2008EP1937653A1 Pyrimidine derivatives and their use as kcnq potassium channels openers
07/02/2008EP1937652A1 Pyrimidine amide compounds as pgds inhibitors
07/02/2008EP1937237A1 Novel phloroglucinol derivatives having selectin ligand activity
07/02/2008EP1730117A4 Thiourea compositions and uses thereof
07/02/2008EP1496838A4 Substituted amides
07/02/2008CN101213180A Method for producing dihydroquinazolines
07/02/2008CN101213179A 2,4-diamino-pyrimidines used as Aurora inhibitors
07/02/2008CN101212969A Azinone and diazinone V3 inhibitors for depression and stress disorders
07/02/2008CN101212903A Polycyclic carbamoylpyridone derivative having HIV integrase inhibitory activity
07/02/2008CN101209997A Pyrimidine-4-formic acid esters and synthetic method thereof
07/02/2008CN100398543C Method of preparing fugutoxin water extract
07/02/2008CN100398524C Tetrahydroquinazolines and dihydrocyclopentapyrimidines as CFR antagonists
07/02/2008CN100398523C 2,4-dichlor phenoxyacetic amide pyrimidine derivative and its preparation method and agricultural composition
07/02/2008CN100398518C Process for the preparation of pyridinyl and pyrimidinyl mono-fluorinated beta keto-esters
07/02/2008CN100398206C Catalyst for producing ethyoxyl quinoline
07/01/2008US7393873 Arylsulfonamide derivatives
07/01/2008US7393855 Treating human herpes virus, human immunodeficiency virus, and hepatitis B virus; optionally administered with other antiviral agents; (E)-9-{[2,2-bis-(hydroxymethyl)cyclopropylidene]methyl}adenine
07/01/2008US7393367 Containing a 3-allyl-4-hydroxybenzaldehyde; quaternary (thi)oxopyrmidinium salt; hetero(carbonyl)acetonitrile (2-cyanomethylbenzimidazole); excellent brilliance and depth of color; wide range of color nuances; improved fastness
06/2008
06/26/2008WO2008076949A2 Quinazoline derivatives and methods of treatment
06/26/2008WO2008076778A1 4-amino-1h-pyrimidin-2-one based compounds, compositions comprising them, and methods of their use
06/26/2008WO2008075353A1 Sulfonamide derivatives with therapeutic indications
06/26/2008WO2008075341A1 Process for the preparation of substituted cynophenoxy-pyrimidinyloxy-phenyl acrylate derivatives
06/26/2008WO2008074578A2 Agent for dyeing fibers comprising keratin
06/26/2008WO2008074515A1 Novel hetaryl-phenylene-diamine pyrimidine as protein kinase inhibitors
06/26/2008WO2008074445A1 Novel tricyclic and heterotricyclic derivatives, processes for preparing them, pharmaceutical compositions thereof
06/26/2008WO2008074068A1 Substituted quinoline derivatives as antiamyloidogeneic agents