Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
07/2008
07/30/2008CN101233112A Benzoquinazoline derivatives and their use in treating bone disorders
07/30/2008CN101230042A Uracil weeding compounds introducing amide structure
07/30/2008CN101230036A Method for preparing heterocyclic aryl-aryl biphenyl compounds
07/30/2008CN101230015A Substituted cinnamic acid derivatives containing amine substituent group and expression purification cytotoxicity thereof
07/30/2008CN101229165A Pyrimidine-2,4-dione derivatives as gonadotropin-releasing hormone receptor antagonists
07/30/2008CN100406453C 4-anilino-quinazoline derivatives as antiproliferative agents
07/29/2008US7405230 Phosphodiesterase 4 inhibitors, including N-substituted aniline and diphenylamine analogs
07/29/2008US7405221 2-(4-fluorobenzyloxy)-4-(2,4-dichlorophenyl)-5-(4-chlorophenyl)pyrimidine; antagonists or inverse agonists of the Cannabinoid-1 (CB1) receptor; antidepressant, neuroleptic, anxiolytic, antiinflammatory agent, cognition activator; psychosis, epilepsy, Parkinson's disease, and schizophrenia
07/29/2008US7405220 Pyrazolopyrimidines
07/29/2008US7405214 Antitumor agents; 2-fluoro-cyclopentenyl nucleosides such as 4-Amino-1-(2-fluoro-4-hydroxy-3-hydroxymethyl-cyclopent-2-enyl)-1H-pyrimidin-2-one; synthesis using 1-((4S,5S)-2,2-Dimethyl-5-vinyl-1,3-dioxolan-4-yl)-2-trityloxy-ethanone intermediates
07/29/2008CA2438813C Alkoxycarbonylamino heteroaryl carboxylic acid derivatives as ip antagonists
07/29/2008CA2178174C Process and intermediates for the manufacture of herbicidal 1-{[2-(cyclopropylcarbonyl)phenyl]sulfamoyl}-3-(4,6-dialkoxy-2-pyrimidinyl)urea compounds
07/29/2008CA2168192C 4-aminobenzoylguanidine derivatives
07/25/2008CA2617463A1 Linear dicationic terphenyls and their aza analogues as antiparasitic agents
07/24/2008WO2008089459A1 Inhibitors of mek
07/24/2008WO2008088727A2 Endothelin receptor antagonists
07/24/2008WO2008087021A1 Synthesis of 4-amino-pyrimidines
07/24/2008WO2008086931A1 Dithiolene metal complex colorless ir absorbers
07/24/2008WO2008086730A1 Tetrahydroquinazoline compounds and their use in preparing medicaments for treating and preventing virosis
07/24/2008WO2008055068A8 Inhibitors of histone deacetylase
07/24/2008WO2007120638A3 Methods and compositions for modulating glycosylation
07/24/2008US20080177069 Process for producing 4-aminoquinazoline compound
07/24/2008US20080177068 Quinazole derivatives
07/24/2008US20080177064 Dipeptidyl peptidase inhibitors
07/24/2008US20080176881 Compounds and compositions as protein kinase inhibitors
07/24/2008US20080176880 Activity against strains having acquired resistance nonnucleoside reverse transcriptase inhibitors; human alpha1 acid glycoprotein nonbinding; such as 4-[[(5-bromo-4,6-dichloro)-2-pyrimidinyl]amino]-benzonitrile
07/24/2008US20080176878 Crystalline rosuvastatin calcium
07/24/2008US20080176876 Substituted 2-Alkyl Quinazolinone Derivatives as Parp Inhibitors
07/24/2008US20080176875 Substituted quinazolines
07/24/2008US20080176869 e.g. N-(4-fluorobenzyl)-3-hydroxy-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine-2-carboxamide; viricide in combination with other HIV/AIDS antivirals, immunomodulators, antibiotics or vaccines; AIDS
07/24/2008US20080176867 e.g., N-[[5-(4-bromophenyl)-4-(2,4-dichlorophenyl)pyrimidin-2-yl]methyl]-3-(trifluoromethyl)benzenesulfonamide; cannabinoid receptor modulator; metabolic and gastrointenstinal disorders, antidiabetic, antiinflammatory, analgesic agent; neurodegenerative diseases
07/24/2008US20080176866 3-(5-Bromo-2-{4-[5-bromo-4-((1R,2R)-2-hydroxy-1-methyl propylamino)-pyrimidin-2-ylamino]phenylamino}pyrimidin-4-ylamino)butan-2-ol; cell cycle and tyrosine kinase receptor inhibitor; antiproliferative, anticarcinogenic agent
07/24/2008US20080176860 8-[4-{4-[5-(Acetylamino-methyl)-2-oxo-oxazolidin-3-yl]-2-fluoro-phenoxymethyl}-4-(3,4,5,6-tetrahydroxy-tetrahydro-pyran-2-carbonyloxy)-piperidin-1-yl]-1-cyclopropyl-7-fluoro-9-methyl; microbioside; multi-drug resistant bacteria; bacterial topoisomerases and protein synthesis inhibitor
07/24/2008US20080176833 Dihydropyridine derivatives as useful as protein kinase inhibitors
07/24/2008US20080176830 Compounds, Compositions, and Methods
07/24/2008US20080176813 Carbocyclic nucleosides and process for obtaining such
07/24/2008US20080176744 Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them
07/24/2008US20080175814 Quinoline derivatives for modulating dna methylation
07/24/2008CA2712073A1 Nucleoside and nucleotide analogues with quaternary carbon centers and methods of use
07/24/2008CA2675358A1 Inhibitors of mek
07/23/2008EP1947103A1 Aryloxypropanolamines, methods of preparation thereof and use of aryloxypropanolamines as medicaments
07/23/2008EP1947092A1 Nucleic acid base having perfluoroalkyl group and method for producing the same
07/23/2008EP1947091A1 Pyrimidyl nitrile derivatives as cysteine protease inhibitors
07/23/2008EP1947086A1 Benzene derivative or salt thereof
07/23/2008EP1945627A1 Pyrimidine derivatives for the treatment of cancer
07/23/2008EP1945213A2 3-piperidin-4-yl-indole orl-1 receptor modulators
07/23/2008EP1368413B1 Two-layer imageable element comprising thermally reversible polymers
07/23/2008EP1325745B1 Preventives and remedies for complications of diabetes
07/23/2008EP1315715B1 Quinazoline derivatives as kinase inhibitors
07/23/2008EP1080092B1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation
07/23/2008EP1073638B1 Heterocyclically substituted amides, their production and their use
07/23/2008CN101228136A 2-cyano-pyrimidines and -triazines as cysteine protease inhibitors
07/23/2008CN101228129A Fluorinated pyridine N-oxide thrombin modulators and process for N-oxidation of nitrogen containing heteroaryls
07/23/2008CN101225083A Tetrahydro quinazoline ketone compound and use thereof in preparation of medicine treating and preventing virus diseases
07/23/2008CN101223883A Weedicide compound of water dissolved saline of novel structure sulfonylurea compound
07/23/2008CN100404537C Quinazolin allkaloids compound, preparation method and use thereof
07/23/2008CN100404517C Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
07/23/2008CN100404032C Novel crystalline forms of the anti-cancer compound ZD1839
07/22/2008US7402589 such as 1-(4-Fluorophenyl)-1-{2-[(1S)-2-hydroxy-1,2-dimethyl-propylamino]-pyrimidin-4-yl}-3-o-tolyl-urea; Interleukin-1, Cycloxygenase-2, Tumor Necrosis Factor- alpha antagonist; antiinflammatory agent; rheumatoid arthritis or osteoarthritis
07/22/2008US7402586 3-Benzylsulfonylamino-6-methyl-1-[(3-guanidinooxypropyl)aminocarbonylmethyl]-2-pyridinone trifluoroacetate; anticoagulants either embedded in or physically linked to materials used in the manufacture of devices used in blood collection, blood circulation, and blood storage
07/22/2008US7402585 For example, 2-(3-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]amino}-1H-pyrazol-5-yl)-N-phenylacetamide; use in the treatment of certain diseases, in particular to proliferative disease such as cancer
07/22/2008US7402557 Reducing epithelial toxicity such as a skin rash or diarrhea during cancer therapy, by coadministering KGF with erlotinib (N-(3-ethynylphenylamino)-6,7-bis(2-methoxyethoxy)-4-quinazoline amine)
07/17/2008WO2008086462A2 AMINO-SUBSTITUTED QUINAZOLINE DERIVATIVES AS INHIBITORS OF β-CANTENIN/TCF-4 PATHWAY AND CANCER TREATMENT AGENTS
07/17/2008WO2008084872A1 Hydrazone derivative
07/17/2008WO2008084493A2 A novel process for the preparation of 2-halo-4-aminoquinazolines
07/17/2008WO2008067440A3 Rosuvastatin dehydroabietylamine salt
07/17/2008WO2008067219A3 Quinazolinone modulators of tgr5
07/17/2008US20080171878 Dealkoxycarbonylating a 4-oxo-1,6-dihydro-pyrimidinyl carboxylic acid ester; one-pot procedure, without isolation of intermediate
07/17/2008US20080171877 N-(4-Heptadecyl-6-oxo-1,6-dihydropyrimidin-2-yl)-N'-phenylguanidine; low viscosity values at the jetting temperature of a hot melt ink jet printer
07/17/2008US20080171876 3-[2-[4-(6-fluorobenzo[d]isoxazol-3-yl)-1-piperidyl]ethyl]-7-hydroxy-4-methyl-1,5-diazabicyclo[4.4.0]deca-3,5-dien-2-one, with less than 0.2% of the impurity 3-[2-[4-(6-fluorobenzo[d]isoxazol-3-yl)-1-oxypiperidin-1-yl]ethyl]-7-hydroxy-4-methyl-1,5-diazabicyclo[4.4.0]deca-3,5-dien-2-one
07/17/2008US20080171875 Process for the synthesis of 9-hydroxy risperidone (paliperidone)
07/17/2008US20080171874 Method for the regioselective preparation of substituted benzo[g]quinoline-3-carbonitriles and benzo[g]quinazolines
07/17/2008US20080171756 e.g. N-{[4-hydroxy-6-oxo-2-phenyl-1-(phenylmethyl)-1,6-dihydro-5-pyrimidinyl]carbonyl}glycine; anemia caused by increasing the production of erythropoietin (Epo), ischemia, stroke, and cytoprotection
07/17/2008US20080171742 e.g. 6-methyl-2-{2-[3-(pyrid-2-yl)isoxazol-5-yl]pyrrolidin-1-yl}-4-(pyrid-2-ylamino)pyrimidine; insulin-like growth factor 1 receptor (somatomedin) antagonist; antiproliferative, antitumor, anticarcinogenic agent;
07/17/2008US20080171692 Substituted amides
07/16/2008EP1944298A1 Quinazoline derivative and pharmaceutical
07/16/2008EP1944289A1 Compounds which potentiate glutamate receptor and uses thereof in medicine
07/16/2008EP1943240A2 Chemical process
07/16/2008EP1943233A2 Compounds and compositions for protein kinase inhbitors
07/16/2008EP1943232A1 Squaric acid derivatives as inhibitors of histone deacetylase
07/16/2008EP1943213A2 Ppar modulating biaromatic compounds
07/16/2008EP1942905A2 Niacin receptor agonists, compositions containing such compounds and methods of treatment
07/16/2008EP1660445A4 Lactams of alkylated acyclic diamine derivatives as modulators of chemokine receptor activity
07/16/2008EP1392655B1 Potassium channel openers
07/16/2008EP1054004B1 Novel pyrimidine-5-carboxamide derivatives
07/16/2008CN101223147A Pyrimidindione derivatives as prokineticin 2 receptor antagonists
07/16/2008CN101223146A Modulators of ATP-binding cassette transporters
07/16/2008CN101219999A N- (3-ethynylphenyl) -6, 7-bis (2-methoxyethoxy) -4-quinazolinamine mesylate anhydrate and monohydrate
07/16/2008CN101219998A Acyclic pyrimidine nucleoside derivant and method for producing the same
07/16/2008CN101219997A Synthesis of 2-chlorine-5- amido pyrimidine
07/16/2008CN101219987A New nitrogen-containing heterocyclic derivative and organic electroluminescent element using the same
07/16/2008CN100402627C C-nitrosoaniline compounds and their blends as polymerization inhibitors
07/16/2008CN100402515C Substituted phthalides as anti-convulsive drugs
07/16/2008CN100402506C Ozagrel lysine, preparing method and usage
07/16/2008CN100402495C Aminoalkylamide substituted cyclohexyl derivatives
07/15/2008US7399884 Substituted benzamides; anticarcinogenic agents, antiinflammatory agents, antiarthritic agents, transplant rejection; controlled release formulations
07/15/2008US7399856 Processes for the preparation of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-2pyrimidinyl]amino]benzonitrile
07/15/2008US7399775 β-amyloid protein production/secretion inhibitor
07/15/2008US7399767 Heterocyclic benzo[c]chromene derivatives useful as modulators of the estrogen receptors
07/15/2008US7399765 Substituted diazabicycloalkane derivatives