| Patents for C07D 225 - Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom (1,649) |
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| 06/07/2006 | EP1373188B1 Alanine 2,6-dialkoxyphenyl ester derivatives as hypnotics |
| 06/07/2006 | EP1315732B1 Radicicol and monocillin and their analogues and uses thereof |
| 06/07/2006 | CN1781909A Process for preparing phencynonate optical isomer |
| 05/24/2006 | CN1775752A Optical pure diamide compound and its use |
| 05/17/2006 | EP1656359A2 Macrocyclic beta-secretase inhibitors for the treatment of alzheimer's disease |
| 05/11/2006 | US20060100164 11-N-[4-(4-Pyridin-3-yl-imidazol-1-yl)-butyl]-6-O-methyl-5-O-(3-dimethylamino-2-hydroxy-propoxy)-3-oxo-erythronolide A, 11,12-carbamate; functionalized macrolides; antiviral, antiprotozoal, anticancer and antigastrointestinal |
| 05/02/2006 | US7038042 Process for producing cyclic compound |
| 04/26/2006 | EP1648873A2 Neuroprotective macrocylic compounds and methods for their use |
| 04/26/2006 | EP1648858A1 Method for production of alpha, beta-unsaturated amide compounds |
| 04/20/2006 | US20060084657 Piperazine derivative |
| 04/13/2006 | US20060079505 Modulators of muscarinic receptors |
| 04/12/2006 | CN1250530C 12-(imino ether)-1, 15-pentadelactam, as well as preparation method and its application in bactericide |
| 04/11/2006 | US7026350 Water-soluble drugs and methods for their production |
| 04/06/2006 | CA2581375A1 Specific kinase inhibitors |
| 04/04/2006 | US7022690 Carboxylic acid substituted heterocycles, derivatives thereof and methods of use |
| 03/29/2006 | EP1638549A2 Novel antibacterial agents |
| 03/16/2006 | WO2005118666A8 N-acylurea compounds for preparing polyurethanes |
| 03/14/2006 | CA2289987C Arylsubstituted piperazines useful in the treatment of benign prostatic hyperplasia |
| 03/02/2006 | WO2005122891A8 Lipophilic derivatives of chelate monoamides |
| 02/22/2006 | CN1738799A Methods for preparing phenylalkyne derivatives |
| 02/02/2006 | WO2005084296A3 Fused tricyclic compounds as inhibitors of 17beta-hydroxysteroid dehydrogernase 3 |
| 01/31/2006 | CA2314154C Azepine or larger medium ring derivatives and their use as pharmaceuticals |
| 01/26/2006 | US20060019941 Prophylaxis or prevention of aberrations in a signal transduction pathway mediated by a cKit kinase by administering 17-ammonium hydroquinone ansamycin analogs with improved solubility and air stability; antiproliferative and anticarcinogenic agents |
| 01/26/2006 | US20060019939 Analogs of benzoquinone-containing ansamycins and methods of use thereof |
| 01/19/2006 | US20060014731 Analogs of benzoquinone-containing ansamycins and methods of use thereof |
| 01/12/2006 | US20060008417 Lipophilic derivatives of chelate monoamides |
| 01/11/2006 | EP1613603A2 Migrastatin analogs and uses thereof |
| 12/29/2005 | WO2005122891A1 Lipophilic derivatives of chelate monoamides |
| 12/29/2005 | US20050288269 Analogs of benzoquinone-containing ansamycins and methods of use thereof |
| 12/29/2005 | CA2569461A1 Lipophilic derivatives of chelate monoamides |
| 12/28/2005 | EP1608626A1 Migrastatin analog compositions and uses thereof |
| 12/20/2005 | US6977303 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same |
| 12/15/2005 | WO2005118666A1 N-acylurea compounds for preparing polyurethanes |
| 12/15/2005 | WO2005117588A2 Analogs of dictyostatin, intermediates therefor and methods of synthesis thereof |
| 12/15/2005 | CA2568221A1 Analogs of dictyostatin, intermediates therefor and methods of synthesis thereof |
| 12/08/2005 | WO2005115988A1 Method for producing decane-1,10-dicarboxylic imide |
| 12/01/2005 | US20050267122 Ansamycins having improved pharmacological and biological properties |
| 11/24/2005 | US20050261263 Benzoquinone ansamycins |
| 11/16/2005 | EP1483395A4 Process to prepare and isolate geldanamycin |
| 11/16/2005 | EP1330464B1 Phosphino-aminophosphines, catalyst complexes and enantioselective hydrogenation |
| 11/10/2005 | US20050250753 hormone sensitive diseases such as prostate hypertrophia, benign prostatic hyperplasia, adenomas and neoplasies of the prostate, prostate cancer, hirsutism, and polycystic ovary syndrome; dibenz[b,f]azocine, dibenzo[b,f][1,4]thiazocine, dibenz[b,f][1,5]oxazocine derivatives; anticancer, antitumor agents |
| 11/09/2005 | EP1019389B1 Epothilone derivatives |
| 10/26/2005 | EP1589000A2 (R)-Chiral halogenated 1-substitutedamino-(N+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity |
| 10/26/2005 | EP1289965B1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
| 10/20/2005 | WO2005097765A1 Anaplastic lymphoma kinase modulators and methods of use |
| 10/20/2005 | CA2559866A1 Anaplastic lymphoma kinase modulators and methods of use |
| 10/13/2005 | WO2005095347A1 Geldanamycin and derivatives inhibit cancer invasion and identify novel targets |
| 10/13/2005 | US20050227955 Reduction of the benzoquinone moiety to form a hydroquinone, and salt formation, producing 17-ammonium hydroquinone ansamycin analogs with improved solubility and air stability; antiproliferative and anticarcinogenic agents |
| 10/13/2005 | CA2560822A1 Geldanamycin and derivatives inhibit cancer invasion and identify novel targets |
| 10/06/2005 | US20050222126 Antiangiogenic compounds and an assay for inhibitors of cell invasion |
| 10/05/2005 | EP1581261A1 Cytotoxins and diagnostic imaging agents comprising hsp90 ligands |
| 09/20/2005 | US6946456 Administering compounds which inhibit heat shock protein 90 proteins; methods block Rb negative or deficient cells in the G2/M phase of the cell cycle and rapidly causes their destruction |
| 09/15/2005 | WO2005084296A2 Fused tricyclic compounds as inhibitors of 17beta-hydroxysteroid dehydrogernase 3 |
| 09/14/2005 | EP1258250B1 Nerve protective drugs |
| 09/09/2005 | WO2004093796A3 Lactam derivatives and methods of their use |
| 08/31/2005 | EP1567494A1 Methods for preparing phenylalkyne derivatives |
| 08/11/2005 | US20050176695 Process for preparing 17-allyl amino geldanamycin (17-aag) and other ansamycins |
| 08/04/2005 | US20050171082 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same |
| 08/03/2005 | CN1649847A Method for producing optically active sulfoxide derivative |
| 08/03/2005 | CN1213036C Novel amide derivatives |
| 07/28/2005 | WO2005068431A1 Composition for dyeing keratin fibres, comprising at least one para-phenylenediamine derivative |
| 07/14/2005 | WO2005063714A1 Analogs of benzoquinone-containing ansamycins for the treatment of cancer |
| 07/14/2005 | WO2005063388A1 Method for preparing solid acid catalyst and method for producing lactam compound using such catalyst |
| 07/07/2005 | WO2005061461A1 INHIBITORS AGAINST MEMBERS OF THE HEAT SHOCK PROTEIN 90 (hsp90) FAMILY |
| 07/07/2005 | WO2005037779A3 Novel dipeptidyl peptidase iv inhibitors used for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases |
| 06/30/2005 | WO2004084809A3 Neuroprotective macrocylic compounds and methods for their use |
| 06/23/2005 | WO2005056531A1 11-o-methylgeldanamycin compounds |
| 06/23/2005 | WO2005023792A3 Macrocyclic compounds useful as pharmaceuticals |
| 06/23/2005 | CA2545457A1 11-o-methylgeldanamycin compounds |
| 06/02/2005 | US20050119416 Ring-opening or closing metathesis reaction of olefin; reduction of carbonyl compound, catalysis, complexing; cyclization, reduction |
| 06/01/2005 | EP1115695B1 (r)-chiral halogenated 1-substitutedamino-(n+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity |
| 05/25/2005 | DE10348022A1 Neue Dipeptidylpeptidase IV-Inhibitoren zur funktionellen Beeinflussung unterschiedlicher Zellen und zur Behandlung immunologischer, entzündlicher, neuronaler und anderer Erkrankungen New dipeptidyl peptidase IV inhibitors for the functional influence of different cells and for the treatment of immunological, inflammatory, neuronal and other diseases |
| 05/24/2005 | US6897323 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same |
| 05/19/2005 | WO2005018545A3 Macrocyclic beta-secretase inhibitors for the treatment of alzheimer's disease |
| 05/19/2005 | US20050107606 Process for producing optically active sulfoxide derivative |
| 05/18/2005 | EP1531153A1 Epothilone derivatives |
| 05/12/2005 | US20050101656 As anti-proliferative agents |
| 05/10/2005 | US6890917 Particularly significant oral in vivo activity |
| 05/05/2005 | US20050096475 Cyclization in presence of solvent; 1-benzyl-8-bromo-1,2,3,4-tetrahydro-1-benzazocin -5-carboxylic acid methyl ester |
| 05/04/2005 | CN1612887A Phosphino-aminophosphines |
| 05/04/2005 | CN1199945C Method for producing cyclic lactams |
| 05/03/2005 | US6887993 11-O-methylgeldanamycin compounds |
| 04/28/2005 | WO2005037796A1 Compounds and methods for treating dyslipidemia |
| 04/28/2005 | WO2005037779A2 Novel dipeptidyl peptidase iv inhibitors used for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases |
| 04/28/2005 | CA2542807A1 Novel dipeptidyl peptidase iv inhibitors used for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases |
| 04/27/2005 | EP1526133A1 Epothilone derivatives |
| 04/20/2005 | CN1608050A Piperazine derivative |
| 04/13/2005 | CN1196684C Process for producing N.N'-carbonyl dilactan |
| 04/07/2005 | US20050074457 Simplified, high throughput screening for identification of heat shock protein 90 ligands selective for high affinity form |
| 04/06/2005 | EP1519735A2 Assays and implements for determining and modulating hsp90 binding activity |
| 04/05/2005 | US6875863 Anticancer agents |
| 03/29/2005 | US6872715 Anticancer agents; antiproliferative agent; 17-(N,N-bis(hydroxyethyl)aminoethylamino)-or 17-(cyclopropylmethylamino)-geldanamycin derivatives |
| 03/22/2005 | US6870049 Antibiotics such as 11-O-methyl-17-(2-dimethylaminoethyl)amino -17-demethoxy-geldanamycin) useful as antiproliferative agents |
| 03/17/2005 | WO2005023792A2 Macrocyclic compounds useful as pharmaceuticals |
| 03/17/2005 | US20050059699 N-acylated lipophilic amino acid derivatives |
| 03/10/2005 | WO2004087673B1 Migrastatin analogs and uses thereof |
| 03/10/2005 | US20050054683 Microbiocides; bacteriocides; oxazolidinone compound |
| 03/09/2005 | EP1511704A1 Polymerisation inhibitor |
| 03/09/2005 | EP1511476A2 Scorpionate-like pendant macrocyclic ligands, complexes and compositions thereof, and methods of using same |
| 03/08/2005 | US6864367 Process for producing cyclic compound |