| Patents for C07D 225 - Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom (1,649) |
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| 03/10/2010 | EP1423376B1 Bicyclic compound, production and use thereof |
| 03/10/2010 | EP1023315B1 Methods and compositions for destruction of selected proteins |
| 03/02/2010 | US7671190 Transformed host cells that make the anticancer polyketides herbimycin and geldanamycin; biosynthesis |
| 02/24/2010 | CN100591673C Herbimycin derivant, preparation method and antineoplastic application thereof |
| 02/18/2010 | US20100041640 Beta-crystalline form of ivabradine hydrochloride, a process for its preparation and pharmaceutical compositions containing it |
| 02/17/2010 | CN101652348A C21-de0xy ansamycin derivatives as antitumor agents |
| 02/16/2010 | US7663301 for use as robust red organic phosphors |
| 02/16/2010 | US7662977 Such as 2-cationic amino-4-oxo-chromene derivatives; water solubility, pharmacokinetics; reduced side effects; anticancer agents |
| 02/16/2010 | CA2445329C 20-hydroxyeicosatetraenoic acid production inhibitors |
| 02/16/2010 | CA2287387C Methods and compositions for destruction of selected proteins |
| 02/04/2010 | WO2010012812A1 Benzazepines and benzazocines as sigma-receptor ligandes |
| 02/04/2010 | US20100029932 Process for production of amide or lactam |
| 02/04/2010 | DE102008035596A1 Derivate benzoannelierter Stickstoff-Heterocyclen Derivatives benzoannelierter nitrogen heterocycles |
| 01/26/2010 | US7652003 Macrocyclic β-secretase inhibitors |
| 01/19/2010 | US7648976 Potential as an anticancer agent; an inhibitor of heat shock protein-90; superior for the preparation of dispersion-based pharmaceutical formulations |
| 01/14/2010 | US20100009959 Pentacyclic Indole Derivatives as Antiviral Agents |
| 01/13/2010 | EP2142595A1 Oxime free anti-skinning combination |
| 01/12/2010 | US7645872 Compounds and methods for labeling oligonucleotides |
| 12/24/2009 | US20090318416 Beta d-crystalline form of ivabradine hydrochloride, a process for its preparation and pharmaceutical compositions containing it |
| 12/16/2009 | EP1904057B1 Hydroquinone ansamycins in the treatment of gastrointestinal stromal tumors |
| 12/15/2009 | CA2338000C Water-soluble 4-thio-maleimido derivatives and methods for their production |
| 12/10/2009 | US20090306368 Polynuclear complex |
| 12/10/2009 | US20090306367 Process for preparing amides from ketoximes |
| 12/09/2009 | EP2129662A2 C21-deoxy ansamycin derivatives as antitumor agents |
| 12/03/2009 | US20090298804 Novel Compounds and Methods for Their Production |
| 12/03/2009 | US20090297454 Perfluoroalkyl-Containing Complexes, Process For Their Production As Well As Their Use |
| 12/02/2009 | CN101595095A 18, 21-didesoxymacbecin derivatives for the treatment of cancer |
| 11/26/2009 | WO2009142206A1 Process for producing laurolactam |
| 11/25/2009 | EP2123635A1 Method for production of laurolactam |
| 11/25/2009 | EP2121957A1 Macrolactams by engineered biosynthesis |
| 11/25/2009 | CN101585809A Novel compound with antibacterial and antitumor activities |
| 11/19/2009 | WO2009138542A1 Use of hsp90 protein inhibiting compounds and pharmaceutical composition intended for anti-tumour therapy |
| 11/18/2009 | CN101580815A Omega-amino carboxylic acids, omega-amino carboxylic acid esters, or recombinant cells which produce lactams thereof |
| 11/11/2009 | EP2116529A1 Process for production of amide or lactam |
| 11/11/2009 | CN101578268A Novel compounds and methods for their production |
| 11/11/2009 | CN101578267A 17-allylamino-17-demethoxygeldanamycin polymorphs and formulations |
| 11/05/2009 | WO2009134987A1 Difluoromethyl-containing macrocyclic compounds as hepatitis c virus inhibitors |
| 11/05/2009 | WO2009133801A1 Process for production of amide or lactam |
| 11/04/2009 | CN101573333A Inhibitors of histone deacetylase |
| 10/29/2009 | WO2009130706A1 A process for isolation and purification of geldanamycin |
| 10/27/2009 | US7608613 Soluble 17-amino-analogs of geldanamycin in acid addition salt form; water solubility; anticancer agents; storage stability |
| 10/27/2009 | US7608611 18,21-didehydro-18,21-dideoxo-18,21-dihydroxy-geldanamycin derivatives as anticarcinogenic agent; with a metal chelating agent |
| 10/22/2009 | US20090264397 Highly fluorinated oils and surfactants and methods of making and using same |
| 10/21/2009 | CN100551911C Polyphenols compound modified by azo-containing heterocyclic and use thereof |
| 10/21/2009 | CN100551910C Styryl compound modified by azo-containing heterocyclic and use thereof |
| 10/15/2009 | WO2009125720A1 Laurolactam production method |
| 10/13/2009 | US7601695 11-N-[4-(4-Pyridin-3-yl-imidazol-1-yl)-butyl]-6-O-methyl-5-O-(3-dimethylamino-2-hydroxy-propoxy)-3-oxo-erythronolide A, 11,12-carbamate; functionalized macrolides; antiviral, antiprotozoal, anticancer and antigastrointestinal |
| 10/08/2009 | US20090253667 18 ,21-Didesoxymacbecin Derivatives for the Treatment of Cancer |
| 10/08/2009 | US20090253653 Soluble 17-amino-analogs of geldanamycin in acid addition salt form; water solubility; anticancer agents; storage stability |
| 10/07/2009 | CN101550046A A method for synthesis of medium-ring compounds of 9 to 12 rings |
| 10/01/2009 | WO2009119167A1 Aniline derivative having anti-rna viral activity |
| 09/30/2009 | CN101547908A Heterocyclic derived metalloprotease inhibitors |
| 09/24/2009 | WO2009117594A1 Fluorinated macrocyclic compounds as hepatitis c virus inhibitors |
| 09/24/2009 | WO2009116537A1 Manufacturing method for laurolactam |
| 09/24/2009 | US20090240050 reacting macrocyclic metal-free cyanine compound dissolved in solvent and vanadium acetylacetonate; low cost |
| 09/11/2009 | WO2009110938A2 Novel macrocyclic polyene lactams |
| 09/09/2009 | EP2098512A1 Compounds and methods for treating dyslipidemia |
| 09/09/2009 | EP1670768B1 Compounds and methods for treating dyslipidemia |
| 09/09/2009 | CN101528705A Method of treating breast cancer using 17-aag or 17-ag or a prodrug of either in combination with a her2 inhibitor |
| 09/02/2009 | EP1794129A4 Synthesis by chiral diamine-mediated asymmetric alkylation |
| 09/01/2009 | US7582280 Conjugates of antioxidants with metal chelating ligands for use in diagnostic and therapeutic applications |
| 08/26/2009 | EP2091919A1 Derivatives of 18-amino substituted analogs of the geldamycin hydroquinon with cytotoxic activity for the treatment of cancer |
| 08/25/2009 | US7579463 Crown ether derivatives |
| 08/25/2009 | US7579462 Reacting allyl amine and geldanamycin in volatile aprotic solvent (tetrahydrofuran), concentrating by evaporation, adding volatile protic solvent (iisopropanol), removing protic solvent to purify, then filtering; making 17-allylamino-geldanamycin (Tanespimycin) |
| 08/25/2009 | US7579337 Analogs of benzoquinone-containing ansamycins and methods of use thereof |
| 08/20/2009 | WO2009004146A3 Novel herbimycin a analogue derivatives, compositions containing same and use thereof |
| 08/20/2009 | US20090209593 Novel antibacterial agents |
| 08/20/2009 | US20090209549 Analogs of Benzoquinone-Containing Ansamycins and Methods of Use Thereof |
| 08/20/2009 | US20090209507 15-O-Desmethylmacbecin Derivatives and Their Use in the Treatment of Cancer or B-Cell Malignancies |
| 08/20/2009 | US20090209494 21-deoxymacbecin analogues useful as antitumor agents |
| 08/20/2009 | US20090208590 Analogs of Benzoquinone-Containing Ansamycins and Methods of Use Thereof |
| 08/19/2009 | EP2089365A1 Heterocyclic derived metalloprotease inhibitors |
| 08/13/2009 | WO2009099134A1 Production method and beckmann rearrangement catalyst for producing a cyclic lactam compound |
| 08/13/2009 | WO2008145525A3 Process for the preparation of dibenzo [b,d]azepin-6-one derivative |
| 08/13/2009 | US20090203739 Anti-Inflammatory Agents |
| 08/13/2009 | US20090202521 Bifunctional Polyazamacrocyclic Chelating Agents |
| 08/06/2009 | US20090198050 Macrocyclic Modulators of the Ghrelin Receptor |
| 08/05/2009 | CN101500997A PARP inhibitors |
| 07/30/2009 | WO2009094443A1 Difluorinated tripeptides as hcv serine protease inhibitors |
| 07/30/2009 | WO2009092295A1 A set of geldanamycin derivatives and their preparation methods |
| 07/30/2009 | CA2713005A1 Difluorinated tripeptides as hcv serine protease inhibitors |
| 07/29/2009 | CN100519536C Group of geldanamycin derivative with nucleoside base |
| 07/28/2009 | US7566706 Drug delivery methods of 17-ammonium hydroquinone ansamycin analogs with improved solubility and air stability; antiproliferative and anticarcinogenic agents |
| 07/23/2009 | US20090186905 Anaplastic lymphoma kinase modulators and methods of use |
| 07/23/2009 | CA2755876A1 Synthesis of resorcylic acid lactones useful as therapeutic agents |
| 07/22/2009 | EP2079700A1 18, 21-didesoxymacbecin derivatives for the treatment of cancer |
| 07/16/2009 | US20090180984 Macrocyclic oximyl hepatitis c serine protease inhibitors |
| 07/16/2009 | US20090180983 Bicyclic, c5-substituted proline derivatives as inhibitors of the hepatitis c virus ns3 protease |
| 07/15/2009 | EP1765073A4 Analogs of dictyostatin, intermediates therefor and methods of synthesis thereof |
| 07/08/2009 | EP1278726B1 Method for producing cyclic lactams |
| 07/02/2009 | US20090170878 Macrocyclic compounds useful as bace inhibitors |
| 06/18/2009 | US20090155829 Heme choline esters and uses thereof |
| 06/17/2009 | EP1472230B1 Ansamycins having improved pharmacological and biological properties |
| 06/17/2009 | CN101460465A 18,21-didesoxymacbecin derivatives for the treatment of cancer |
| 06/16/2009 | US7547705 Ethyl-1'-[(2S)-2-hydroxy-2-phenylethyl]-6'-oxo-8'-(pyridin-4-yl)-1',3',4',6'-tetrahydro-1H-spiro[piperidine-4,2'-pyrimido[1,2-a]pyrimidine]-1-carbox; glycogen synthase kinase-3 beta, amyloid precursor protein, tau protein hyperphosphorylation inhibitor; neurodegenerative disease, type II diabetes |
| 06/11/2009 | US20090149395 Novel macrocyclic polyene lactams |
| 06/04/2009 | WO2009069522A1 Method for production of laurolactam |
| 06/04/2009 | WO2007061878A3 17-allylamino-17-demethoxygeldanamycin polymorphs and formulations |
| 05/20/2009 | CN101437802A 17-oxymacbecin derivatives and their use in the treatment of cancer and/or B-cell malignancies |
| 05/12/2009 | US7531543 Phenylpiperazine cycloalkanol derivatives and methods of their use |