Patents
Patents for C07D 225 - Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom (1,649)
10/2002
10/31/2002WO2002086078A2 Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
10/30/2002WO2001083444A1 Method for producing cyclic lactams
10/30/2002CA2407813A1 Method for producing cyclic lactams
10/22/2002US6468406 Anion-complexing compound, method of preparing the same, an ion-selective membrane and a sensor provided with such a compound or membrane
10/10/2002WO2002079167A1 Geldanamycin derivative and method of treating cancer using same
10/08/2002US6462092 Such as 3-((3-fluorophenyl)-((3-(trifluoromethyl)phenyl)-methyl)amino)-1,1,1 -trifluoro-2-propanol; cardiovascular disease, i.e. atherosclerosis and other coronary artery diseases
10/01/2002US6458852 Use of substituted N, N-bis-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
10/01/2002US6458849 Method of treating or preventing a ceip-mediated disorder in a subject by administering a therapeutically effective amount of a compound for strokes
10/01/2002US6458803 Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
09/2002
09/24/2002US6455519 Use of substituted N, N-disubstituted fused-heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
09/18/2002EP0804427B1 Lta4 hydrolase inhibitors
09/17/2002US6451830 Use of substituted N,N-disubstituted non-fused heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
09/17/2002US6451823 Use of substituted N-phenoxy-N-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
09/10/2002US6448295 Treating cardiovascular disease; atherosclerosis, dyslipidema hypercholesterolaemia; decreasing concentrations of low density lipoprotein and raising level of high density lipoprotein
09/10/2002US6448286 Imino pyrrolidine derivatives useful as nitric oxide synthase inhibitors
09/03/2002CA2140626C Hydroxamic acid derivatives as metalloproteinase inhibitors
08/2002
08/29/2002WO2002016369A3 Novel macrocycles and uses thereof
08/29/2002US20020120011 Substituted N, N-disubstituted diamino compounds useful for inhibiting cholesteryl ester transfer protein activity
08/01/2002WO2002058679A2 Antiangiogenic compounds and an assay for inhibitors of cell invasion
07/2002
07/25/2002WO2002057218A1 Alanine 2,6-dialkoxyphenyl ester derivatives as hypnotics
07/25/2002US20020099084 Pharmaceutically active compounds and methods of use
07/16/2002US6420395 Disorders or diseases involving the cholinergic system of the central nervous system, pain, inflammatory diseases, diseases caused by smooth muscle contractions and as assistance in the cessation of chemical substance abuse.
07/16/2002US6420363 Mono- or polyenic carboxylic acid derivatives
07/11/2002WO2002026750A3 Phosphino-aminophosphines, catalyst complexes and enantioselective hydrogenation
07/11/2002WO2002026705A3 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and their preparation
07/11/2002US20020091151 Novel macrocycles and uses thereof
07/10/2002EP1221441A2 LTA4 Hydrolase inhibitors
07/03/2002EP0563345B1 Novel 4-arylpiperazines and 4-arylpiperidines
06/2002
06/18/2002US6407087 UCF116 derivatives
05/2002
05/30/2002WO2002020526A3 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
05/30/2002US20020065417 Useful as ligands for metal catalysts for asymmetric reactions, in particular as rhodium complexes for asymmetric hydrogenation of enamide, itaconate, and alpha-ketoester compounds
05/10/2002WO2002036574A1 Geldanamycin derivatives useful for the treatment of cancer
04/2002
04/18/2002WO2002002488A3 Methods and compounds for modulating nuclear receptor coactivator binding
04/18/2002US20020045570 Methods and compositions for degradation and/or inhibition of her-family tyrosine kinases
04/11/2002US20020042508 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same
04/09/2002US6369110 Substituted guanidine derivatives and process for producing the same
04/04/2002WO2002026750A2 Phosphino-aminophosphines, catalyst complexes and enantioselective hydrogenation
04/04/2002WO2002026705A2 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and their preparation
03/2002
03/28/2002US20020037560 Bicyclic terpenes and synthesis thereof
03/19/2002US6358993 Pharmaceutically active nitrogen ring compounds and methods of use thereof
03/19/2002US6358942 Microbiocides and bactericides for treating grampositive, bacteroides, clostridium, mycobacterium, staphylococcus and streptococcus infections
03/14/2002WO2002020526A2 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
03/14/2002CA2421506A1 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
03/07/2002WO2002017712A2 Disubstituted benzenes as insecticides
02/2002
02/28/2002WO2002016369A2 Novel macrocycles and uses thereof
02/14/2002WO2002012185A1 Process for preparing 2,3-diaminopropanols and synthesis of other compounds using 2,3-diaminopropanols
02/12/2002CA2067877C Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions in which they are present
02/07/2002WO2002009696A1 Methods for treating cell proliferative disorders and viral infections
02/07/2002CA2417495A1 Methods for treating cell proliferative disorders and viral infections
01/2002
01/16/2002CN1077886C Amidino derivatives useful as nitric oxide synthase inhibitors
01/10/2002WO2002002488A2 Methods and compounds for modulating nuclear receptor coactivator binding
01/10/2002US20020004501 Therapy for muscular disorders, urogenital disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002US20020004494 Muscular disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002CA2415103A1 Methods and compounds for modulating nuclear receptor coactivator binding
01/09/2002EP1169319A1 Methods and compositions for degradation and/or inhibition of her-family tyrosine kinases
01/02/2002EP1165532A1 Antibacterial agents
12/2001
12/20/2001WO2001096342A1 Bicyclic terpenes and synthesis thereof
11/2001
11/29/2001WO2001090082A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
11/29/2001WO2001090081A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
11/28/2001EP0850234B1 Novel heterocyclic compounds for the treatment of pain and use thereof
11/22/2001US20010044532 By reacting phosgene and lactam in the presence of a non-nucleophilic aliphatic tertiary amine, such as N,N-diisopropylethylamine; high purity, good yields
11/21/2001EP0659179B1 Benzo-fused lactams promote release of growth hormone
11/21/2001CN1322718A Process for producing N.N'-carbonyl dilactan
11/08/2001DE10021193A1 Verfahren zur Herstellung cyclischer Lactame A process for preparing cyclic lactams
11/07/2001EP1151996A2 Process for the preparation of N,N'-carbonyl-bis-lactames
11/06/2001US6313307 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/2001
10/28/2001CA2345846A1 Preparation process for n,n'-carbonylbis-lactams
10/24/2001EP0856002B1 Phenyloxazolidinones having a c-c bond to 4-8 membered heterocyclic rings
10/10/2001EP1140897A1 Protease inhibitors
10/10/2001EP0840731B1 Polycyclic alcaloid-derivatives as nmda-receptor antagonists
10/03/2001CN1072222C Phenyloxazolidinones having C-C bond to 4-8 membered heterocyclic rings
10/02/2001CA2037541C Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
09/2001
09/19/2001CN1313281A Autolytic mycin
09/18/2001US6291508 Potent ability to bind to retinoic acid receptors thus useful in treating psoriasis and rheumatoid arthritis.
09/12/2001CN1070859C 6-methoxy-1H-benzotriazole-5-carboxamide derivatives, process for producing same, and medicinal composition containing same
08/2001
08/28/2001US6281354 Analogs of duocarmycin and cc-1065
08/23/2001WO2001060768A1 Process for producing cyclic compound
08/23/2001CA2400979A1 Process for producing cyclic compound
08/21/2001US6277839 Antiinflammatory agents, antipyretics, analgesics; side effect reduction
08/01/2001EP1119555A1 Biphenylene lactams as prostaglandin receptor ligands
08/01/2001CN1305993A Cyclic guanyl preparation used as nitrogen oxide synthetic enzyme inhibitor
07/2001
07/18/2001EP1115695A1 (r)-chiral halogenated 1-substitutedamino-(n+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity
07/18/2001EP1115693A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL $i(TERTIARY)-HETEROALKYLAMINES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY
07/18/2001CN1304309A Semi-synthetic ecteinascidins
07/05/2001WO2001047558A1 Nerve protective drugs
07/05/2001CA2395996A1 Neuroprotective drug
06/2001
06/26/2001US6251885 Treating microorganism infection, lung cancer, breast cancer or leukemia in mammal
05/2001
05/30/2001EP0794184B1 6-methoxy-1h-benzotriazole-5-carboxamide derivatives, process for producing the same, and medicinal composition containing the same
05/22/2001CA2200892C Process for preparing lauryllactam through photonitrosation of cyclododecane in the presence of trichloronitrosomethane
05/16/2001EP1098666A2 Water-soluble drugs and methods for their production
05/10/2001WO1999002514A3 Epothilone derivatives
05/02/2001CN1293669A Benzylpiperazingl-and benzylipeeridinyl ethanone derivatives, their preparation method and their use as dopamine D receptor antagonists
04/2001
04/11/2001CN1064354C Trilcyclic benzazepine vasopressin antagnonists
03/2001
03/27/2001US6207824 Using macroporous cation exchange resin
03/14/2001EP1083166A1 Novel substituted guanidine derivatives and process for producing the same
03/14/2001CN1063171C Process for producing lauryllactam by photonitrosation of cyclododecane in presence of trichloronitrosomethane
02/2001
02/07/2001EP1073629A1 Anion-complexing compound, method of preparing the same, an ion-selective membrane and a sensor provided with such a compound or membrane
01/2001
01/17/2001EP1068193A1 Benzylpiperazinyl- and benzylpiperidinyl ethanone derivatives, their preparation and their use as dopamine d 4? receptor antagonists
01/17/2001EP1067933A1 Semi-synthetic ecteinascidins
01/09/2001US6172234 Optically active cyclic amino acid ester derivatives and processes for producing the same
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