| Patents for C07D 225 - Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom (1,649) |
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| 05/07/2009 | US20090117127 Novel Compounds and Methods for Their Production |
| 04/30/2009 | WO2007053284A3 Method of treating breast cancer using 17-aag or 17-ag or a prodrug of either in combination with a her2 inhibitor |
| 04/30/2009 | US20090111869 Benzoquinone ansamycins |
| 04/30/2009 | US20090111816 Polycyclic aryl substituted triazoles and polycyclic heteroaryl substituted triazoles useful as axl inhibitors |
| 04/29/2009 | CN101421246A Layout of power semiconductor contacts on a cooling surface |
| 04/23/2009 | US20090105471 Macrocyclic compounds as inhibitors of viral replication |
| 04/16/2009 | US20090099080 Mitochondria-targeted anti-tumor agents |
| 04/16/2009 | US20090098047 Bioconjugates of metal complexes of nitrogen-containing macrocyclic ligands |
| 04/14/2009 | CA2409841C Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
| 04/14/2009 | CA2408934C Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
| 04/02/2009 | US20090088567 Purification of a crude lactam mixture by means of melt crystallization |
| 04/02/2009 | US20090088414 Soluble 17-amino-analogs of geldanamycin in acid addition salt form; water solubility; anticancer agents; storage stability |
| 04/02/2009 | US20090083912 Gas-Resistant Phtalocyanine Dyes |
| 03/19/2009 | US20090075975 Arylsulfonamides and uses related thereto |
| 03/18/2009 | EP2035380A2 Parp inhibitors |
| 03/17/2009 | US7504378 Viricides; induction immunology response; compounds according to invention specifically inhibit NS3 protease and do not show significant inhibitory activity against other serine proteases such as human leukocyte elastase, porcine pancreatic elastase, bovine pancreatic chymotrypsin, or cysteine proteases |
| 03/17/2009 | US7504088 Lipophilic derivatives of chelate monoamides |
| 03/12/2009 | US20090069281 Ansamycin formulations and methods of use thereof |
| 03/12/2009 | US20090069280 17-amino analogs of geldanamycin, used for treating and modulating disorders associated with hyperproliferation, such as cancer; antiproliferative and anticarcinogenic agents |
| 03/05/2009 | WO2008055068A3 Inhibitors of histone deacetylase |
| 03/05/2009 | US20090062528 Ansamycin formulations and methods of use thereof |
| 03/05/2009 | US20090062250 Soluble 17-amino-analogs of geldanamycin in acid addition salt form; water solubility; anticancer agents; storage stability |
| 02/26/2009 | US20090053137 Chelating Conjugates Having a Substituted Aromatic Moiety and Derivatives Thereof |
| 02/24/2009 | US7494986 central nervous system disorders like Depression, anxiety, cognition enhancer, antiinflammatory agents; 4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-phenylazocane |
| 02/19/2009 | WO2007075772A3 Compounds, screens, and methods of treatment |
| 02/19/2009 | US20090048253 Benzenoid ansamycin derivative |
| 02/12/2009 | US20090042847 17-allylamino-17-demethoxygeldanamycin polymorphs and formulations |
| 02/03/2009 | US7485631 macrolactone antibiotics; Phorboxazole mimetics; carcinogenic agent; cancer cell division inhibitor; pancreatic, breast, non-small lung, colon, and prostate cancers, leukemia |
| 02/03/2009 | US7485630 e.g. 2-{[(3'-Amino-1'-aza-2'-oxobicyclo[6.3.0]-undecyl)-11'-carbonyl]amino}-1,5-pentanedioic acid; tripeptide Gly-Pro-Glu (GPE) mimetic; enzymatic degradation, ischemic injury, hypoxic injury, reperfusion injury, and asphyxia |
| 01/29/2009 | WO2008116339A3 Organic compounds |
| 01/29/2009 | US20090030032 Bicyclic Compound, Production and Use Thereof |
| 01/29/2009 | US20090029960 Macrocyclic compounds useful as base inhibitors |
| 01/22/2009 | US20090023916 Tetrazine-based bio-orthogonal coupling reagents and methods |
| 01/22/2009 | US20090022704 Method for the treatment of gout or pseudogout |
| 01/21/2009 | EP0951466B1 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds |
| 01/14/2009 | CN101346354A 21-deoxymacbecin analogues useful as antitumor agents |
| 01/08/2009 | WO2009004146A2 Novel herbimycin a analogue derivatives, compositions containing same and use thereof |
| 12/30/2008 | US7470469 Medical device having surface modification with superoxide dismutase mimic |
| 12/30/2008 | CA2312098C A process for the preparation of ring-opened epothilone intermediates which are useful for the preparation of epothilone analogs |
| 12/25/2008 | US20080318338 Drug screening using a high affinity form of Heat Shock Protein-90 (HSP90) that has a 17-allylamino-geldanamycin (17-AAG) binding affinity |
| 12/23/2008 | US7468434 Administering lithium ion-chelated in a crown ether- or aza-crown ether-containing chromene or diazene derivative and a carrier; exposing eye to an external light soure to cause the aza-crown ether or crown ether of a chromene or a diazene compound to release lithium, glaucoma |
| 12/18/2008 | US20080312317 12 membered-ring macrolactam derivatives |
| 12/16/2008 | US7465718 Ansamycins having improved pharmacological and biological properties |
| 12/10/2008 | CN101318930A Herbimycin derivant, preparation method and antineoplastic application thereof |
| 12/04/2008 | WO2008145525A2 Process for the preparation of dibenzo [b,d]azepin-6-one derivative |
| 12/04/2008 | WO2007098229A3 Geldanamycin derivatives and method of use thereof |
| 12/04/2008 | CA2686645A1 Process for the preparation of dibenzo [b,d]azepin-6-one derivative |
| 11/27/2008 | WO2005025498A3 Substituted acetanilides and benzamides for the treatment of asthma and pulmonary inflammation |
| 11/27/2008 | US20080293731 Organic Compounds |
| 11/20/2008 | US20080283122 Beta-Substituted Porphyrins |
| 11/18/2008 | US7452992 Heterocyclic compounds as CCR5 antagonists |
| 11/13/2008 | US20080279781 Glycosylated Carboranylporphyrins and Uses Thereof |
| 11/12/2008 | CN101302199A Guidemycin and use thereof in tumor treatment |
| 11/11/2008 | US7449573 acid generators which generates a sulfonic acid having one or more SO3H groups and one or more SO2 bonds upon irradiation with an actinic ray or a radiation |
| 11/06/2008 | US20080275039 Geldanamycin Derivatives and the Method for Biosynthesis Thereof |
| 11/06/2008 | US20080275018 Antibacterial amide-macrocycles v |
| 10/30/2008 | WO2008104812A3 C21-de0xy ansamycin derivatives as antitumor agents |
| 10/23/2008 | WO2008128058A1 New gallium bisaminothiolate complexes for myocardial imaging |
| 10/23/2008 | WO2008127739A1 Oxime free anti-skinning combination |
| 10/21/2008 | CA2296012C Epothilone derivatives |
| 10/02/2008 | WO2008118327A1 Conformationally restrained epothilone analogues as anti-leukemic agents |
| 10/01/2008 | EP1975155A1 Process for production of lactam |
| 10/01/2008 | EP1973883A2 Novel compounds and methods for their production |
| 09/25/2008 | US20080234246 Benzoquinone imine-containing ansamycins and its acylation or alkylation derivatives; cellular proliferation, hyperproliferation; increase the bioavailability and reduce the toxicity associated with the natural product |
| 09/25/2008 | DE102007013765A1 Lejimalid Analoga und Verwendung davon Lejimalid analogues and use thereof |
| 09/24/2008 | EP1971578A1 21-deoxymacbecin analogues useful as antitumor agents |
| 09/17/2008 | EP1968583A2 Compounds, screens, and methods of treatment |
| 09/17/2008 | CN101267816A Methods of treatment using hydroquinone ansamycins |
| 09/11/2008 | US20080221077 Ansamycin formulations and methods of use thereof |
| 09/04/2008 | WO2008104812A2 C21-de0xy ansamycin derivatives as antitumor agents |
| 09/04/2008 | CA2679224A1 Novel compounds |
| 08/28/2008 | US20080206788 Reagents and methods for the detection and quantification of vancomycin in biological fluids |
| 08/27/2008 | CN101253154A Novel ansamycin derivatives |
| 08/26/2008 | US7417040 hormone sensitive diseases such as prostate hypertrophia, benign prostatic hyperplasia, adenomas and neoplasies of the prostate, prostate cancer, hirsutism, and polycystic ovary syndrome; dibenz[b,f]azocine, dibenzo[b,f][1,4]thiazocine, dibenz[b,f][1,5]oxazocine derivatives; anticancer, antitumor agents |
| 08/14/2008 | WO2008096873A1 Method for production of laurolactam |
| 08/13/2008 | CN101239948A Novel derivative Gdm-CT-1-1 of geldanamycin and preparation method thereof |
| 08/07/2008 | WO2008093912A1 Novel ansamycin derivatives and the method for mutational biosynthesis thereof |
| 08/07/2008 | US20080188651 Analogs of dictyostatin, intermediates therefor and methods of systhesis thereof |
| 08/07/2008 | US20080188450 Macrolactams by engineered biosynthesis |
| 08/06/2008 | EP1951223A2 17-allylamino-17-demethoxygeldanamycin polymorphs and formulations |
| 08/06/2008 | EP1951222A2 Method of treating breast cancer using 17-aag or 17-ag or a prodrug of either in combination with a her2 inhibitor |
| 07/31/2008 | WO2008056188A3 Novel compounds and methods for their production |
| 07/30/2008 | CN101230040A Process for preparing 17-allyl amino geldanamycin (17-AAG) and other ansamycins |
| 07/29/2008 | US7405208 Benzoquinone ansamycins |
| 07/24/2008 | WO2008055068A8 Inhibitors of histone deacetylase |
| 07/23/2008 | CN101227901A Anti-inflammatory agents |
| 07/22/2008 | US7402670 Synthesis by chiral diamine-mediated asymmetric alkylation |
| 07/17/2008 | WO2008083543A1 Nitrogen-containing heterocyclic modified compounds and uses thereof |
| 07/10/2008 | WO2008081726A1 Process for production of amide or lactam |
| 07/09/2008 | EP1940798A1 17-oxymacbecin derivatives and their use in the treatment of cancer and/or b-cell malignancies |
| 07/09/2008 | CN101217958A Inhibitors of AKT activity |
| 07/03/2008 | WO2008078642A1 Method for producing lactam compound |
| 07/03/2008 | US20080161287 Bicyclic compound, production and use thereof |
| 07/02/2008 | EP1937677A1 Cb-1 modulating compounds and their use |
| 07/02/2008 | EP1937644A1 Novel ansamycin derivatives |
| 07/02/2008 | EP1648858B1 Method for production of alpha, beta-unsaturated amide compounds |
| 07/02/2008 | CN101213178A Benzenoid ansamycin derivative |
| 06/24/2008 | US7390797 Fused indazole compounds |
| 06/11/2008 | EP1928837A2 18,21-didesoxymacbecin derivatives for the treatment of cancer |
| 06/11/2008 | EP1414794B1 Allylmercaptocaptopril compounds and uses thereof |