Patents
Sitemap › C07 - Organic chemistry › C07D - Heterocyclic compounds › C07D 225 - Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom
Patents for C07D 225 - Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom (1,649)
01/2001
01/04/2001WO2001000583A1 Ucf116 derivatives as antitumor agents
01/03/2001EP1065203A2 Heterocyclic compounds as retinoic acid receptor antagonists
12/2000
12/26/2000US6166056 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
12/21/2000DE19927912A1 Catalytic preparation of cyclic and/or polymer compounds by educt metathesis is performed in the presence of one or more heterogeneous catalysts and ionic liquids
12/06/2000CN1275912A Novel amide derivatives
10/2000
10/19/2000WO2000061578A1 Methods and compositions for degradation and/or inhibition of her-family tyrosine kinases
10/19/2000CA2370007A1 Methods and compositions for degradation and/or inhibition of her-family tyrosine kinases
10/18/2000CN1270589A Epothilone derivatives
10/17/2000US6133283 Mono- or polyenic carboxylic acid derivatives
10/05/2000WO2000058294A1 Antibacterial agents
10/04/2000EP1040099A1 Azepine or larger medium ring derivatives and their use as pharmaceuticals
09/2000
09/27/2000EP1038867A1 Process for the purification of N-substituted lactames, with acidic macroporous cation exchange resins
09/26/2000US6124293 Semi-synthetic ecteinascidins
09/14/2000DE19910504A1 Verfahren zur Reinigung von N-substituierten Lactamen A process for purifying N-substituted lactams
09/13/2000EP1035093A2 Metathesis in the presence of ionic liquids
09/13/2000EP0983248A4 Analogs of duocarmycin and cc-1065
09/07/2000DE19909600A1 Catalytic preparation of cyclic and/or polymer compounds by educt metathesis is performed in the presence of one or more heterogeneous catalysts and ionic liquids
09/06/2000EP1032556A1 Pharmaceutically active compounds and methods of use
09/05/2000US6114381 To control brain damage associated with anoxia or ischemia which typically follows stroke, cardiac arrest or perinatal asphyxia; compound is an antagonist to inhibit excitotoxic actions at excitatory amino acid receptor sites
08/2000
08/23/2000CN1264300A Arylsubstituted piperazines useful in the threatement of bening prostatic hyperlasia
08/22/2000US6107291 Antiinflammatory agent
08/02/2000EP1023315A1 Methods and compositions for destruction of selected proteins
07/2000
07/26/2000EP1021423A1 MACROCYCLIC INHIBITORS OF MATRIX METALLOPROTEINASES AND TNF$g(a) SECRETION
07/26/2000EP1021190A1 Novel amide derivatives
07/19/2000EP1019389A2 Epothilone derivatives
07/13/2000WO2000003737A9 Water-soluble drugs and methods for their production
07/06/2000WO2000039115A1 Protease inhibitors
06/2000
06/21/2000CN1257485A Azacyclooctane and heptane derivatives, their preparation and usein therapy
06/06/2000US6071915 Arylsubstituted piperazines useful in the treatment of benign prostatic hyperplasia
06/06/2000US6071906 Inhibits or modulates the inducible isoform of nitric oxide synthase over the the constitutive isoforms; antiarthritic, -diabetic, ischemic, thrombosis agents; cardiovascular disorders; toxic shock syndrome; autoimmune diseases
05/2000
05/02/2000US6057311 Benzodiazonine derivatives binding to cholecystokinin or gastrin receptors
04/2000
04/25/2000US6054579 Reacting a difunctional component containing an activated carbon, an amine capable of forming an imine with the activated carbon, and an isocyanide in a nucleophilic polar protic solvent
04/25/2000US6054474 Activating opioid receptors
04/20/2000WO2000003737A3 Water-soluble drugs and methods for their production
04/18/2000US6051716 Antimicrobial agents
04/13/2000WO2000020398A1 Biphenylene lactams as prostaglandin receptor ligands
04/13/2000CA2346445A1 Biphenylene lactams as prostaglandin receptor ligands
04/06/2000WO2000018724A1 (R)-CHIRAL HALOGENATED 1-SUBSTITUTEDAMINO-(n+1)-ALKANOLS USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY
04/06/2000WO2000018721A1 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
04/04/2000US6046211 Amidino derivatives useful as nitric oxide synthase inhibitors
03/2000
03/28/2000US6043266 Microbiocides treating gram-positive bacteria infections and persons with aids
03/28/2000US6043261 Pyrrolodino imidines useful as nitric oxide synthase inhibitors
03/15/2000EP0984943A1 Azacyclooctane and heptane derivatives, their preparation and usein therapy
03/15/2000EP0984777A1 Arylsubstituted piperazines useful in the treatement of benign prostatic hyperlasia
03/08/2000EP0983248A1 Analogs of duocarmycin and cc-1065
03/01/2000EP0782573B1 Brefeldin a and analogs to improved synaptic transmission
02/2000
02/29/2000US6030964 Binds to retinoic acid receptors and useful for treating psoriasis, autoimmune diseases, tumors, rheumatoid arthritis and for inducing immunosuppression in organ transplantation
02/15/2000US6025355 Substituted indolinyl and derivatives thereof, neurological injury and neurodegenerative disorders.
02/02/2000EP0976729A1 Optically active cyclic amino acid ester derivatives and processes for producing the same
01/2000
01/27/2000WO2000003737A2 Water-soluble drugs and methods for their production
01/27/2000WO1999051238A9 Semi-synthetic ecteinascidins
01/19/2000CN1048484C A process for preparing a composition containing benzoheterocycles
01/18/2000US6015659 Inducement of thermotolerance with benzoquinonoid ansamycins
01/04/2000US6011028 Cyclic amidino agents useful as nitric oxide synthase inhibitors
12/1999
12/21/1999CA2006577C Hypoglycaemic phenylamidines and phenylguanidines
12/02/1999WO1999061414A1 Novel substituted guanidine derivatives and process for producing the same
12/02/1999CA2331509A1 Novel substituted guanidine derivatives and process for producing the same
11/1999
11/23/1999US5990104 Inhibiting nmda receptor activation by administering derivatives of given formula, such as 5,6,7,8,9,11,12-heptahydro-3-hydroxy-5-methyl-10-thia-5,11 -methanobenzocyclodecen-13-amine (sulphazocine)
11/16/1999US5985869 Benzoheterocyclic compounds
11/02/1999US5977125 Mono-or polyenic carboxylic acid derivatives
10/1999
10/19/1999US5968962 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/19/1999US5968924 Benzo-fused lactams promote release of growth hormone
10/14/1999WO1999051570A1 Anion-complexing compound, method of preparing the same, an ion-selective membrane and a sensor provided with such a compound or membrane
10/14/1999WO1999051238A1 Semi-synthetic ecteinascidins
10/14/1999CA2326844A1 Anion-complexing compound, method of preparing the same, an ion-selective membrane and a sensor provided with such a compound or membrane
09/1999
09/29/1999EP0945436A1 Cytotrienins, process for preparing the same, and antitumor agent
09/07/1999US5948770 Controlling mammal and plant fungi
09/02/1999WO1999043670A1 Benzylpiperazinyl- and benzylpiperidinyl ethanone derivatives, their preparation and their use as dopamine d4 receptor antagonists
09/02/1999CA2321830A1 Benzylpiperazinyl- and benzylpiperidinyl ethanone derivatives, their preparation and their use as dopamine d4 receptor antagonists
08/1999
08/10/1999US5936100 Synthesis of functionalized macrocycles by ring closing metathesis
08/03/1999US5932568 6-methoxy-1H-benzotriazole-5-carboxamide derivatives and pharmaceutical compositions containing them
08/03/1999US5932566 Ansamycin derivatives as antioncogene and anticancer agents
07/1999
07/22/1999WO1999036403A1 Novel dopamine re-uptake inhibitors and methods of synthesizing and using the same
07/01/1999WO1999032451A1 Azepine or larger medium ring derivatives and their use as pharmaceuticals
06/1999
06/30/1999EP0925300A1 Pharmaceutically active compounds and methods of use
06/15/1999US5912360 Dioxolane intermediates
04/1999
04/29/1999WO1999020599A1 Pharmaceutically active compounds and methods of use
04/29/1999CA2307597A1 Pharmaceutically active compounds and methods of use
03/1999
03/16/1999US5883251 Enzyme inhibitors
03/04/1999WO1999009991A1 Novel amide derivatives
03/04/1999CA2301566A1 N-acylated lipophilic amino acid derivatives
03/03/1999EP0724570B1 Amidino derivatives useful as nitric oxide synthase inhibitors
02/1999
02/24/1999EP0897912A1 Amidino derivatives useful as nitric oxide synthase inhibitors
02/09/1999US5869483 Tricyclic benzazepine vasopressin antagonists
01/1999
01/21/1999WO1999002514A2 Epothilone derivatives
01/12/1999US5859239 Mercaptoalkanoylamino and acylmercaptoalkanoylamino benzoxazepines and benzothiazepines
01/07/1999WO1999000362A1 Synthesis of aminocarbonyl substituted lactams
01/05/1999US5856477 Hypotensive agents; congestive heart failure
01/05/1999US5856476 Processes for preparing azepiones useful as intermediates in the preparation of inhibitors of angiotensin converting enzyme and neutral endopeptidase
12/1998
12/29/1998US5854236 Tricyclic benzazepine vasopressin antagonists
12/29/1998US5854234 Amidino dervatives useful as nitric oxide synthase inhibitors
12/03/1998WO1998054152A1 Azacyclooctane and heptane derivatives, their preparation and usein therapy
12/03/1998CA2289576A1 Azacyclooctane and heptane derivatives, their preparation and use in therapy
12/01/1998US5843952 Tricyclic benzazepine vasopressin antagonists
11/1998
11/26/1998WO1998052925A1 Analogs of duocarmycin and cc-1065
11/26/1998CA2290789A1 Analogs of duocarmycin and cc-1065
11/19/1998WO1998051702A1 Methods and compositions for destruction of selected proteins
11/19/1998WO1998051298A1 Arylsubstituted piperazines useful in the treatement of benign prostatic hyperlasia
10/1998
10/28/1998CN1197457A Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/14/1998CN1196053A Novel heterocyclic compounds for treatment of pain and use thereof
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