Patents
Patents for C07D 225 - Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom (1,649)
01/1996
01/09/1996US5482938 Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
11/1995
11/29/1995CN1112548A Polyiodinated compounds, process for preparing them and diagnostic compositions
10/1995
10/31/1995US5462934 Cholinesterase inhibitor; learning enhancement
10/24/1995CA1337401C Compositions comprising 1-oxo- or thiohydrocarbyl substituted azacycloalkanes
10/04/1995EP0675105A1 Polyiodinated compounds, process for their preparation and diagnostic composition
09/1995
09/23/1995CA2145035A1 Polyiodinated compounds, process for preparing them and diagnostic compositions
09/08/1995WO1995023788A1 Improved process for the acylation of lactams
08/1995
08/23/1995CN1107146A A process for preparing a composition containing benzoheterocycles
08/17/1995WO1995021614A1 New protein trafficking inhibitors
08/16/1995CN1106802A Tricyclic benzazepine vasopressin antagonists
08/15/1995CA1336711C Lactam derivatives, their preparation and their use as hypotensive agents
08/09/1995EP0659179A4 Benzo-fused lactams promote release of growth hormone.
08/02/1995EP0664702A1 Tumoricidal activity of benzoquinonoid ansamycins against prostate cancer and primitive neural malignancies
07/1995
07/18/1995US5434261 Benzo-fused lactams promote release of growth hormone
07/05/1995EP0660825A1 Anti-inflammatory macrolactam (cyclamenol)
07/04/1995US5430150 N-(1-(((1H-benzimidazol-2-ylmethyl)amino)carbonyl)-2-methyl -butyl)-3-(((1,1-dimethylethyl)amino)-carbonyl)decahydro-gamma-hydroxyalpha -(phenylmethyl)-2-isoquinolinepentanamide compounds; AIDS
06/1995
06/28/1995EP0659179A1 Benzo-fused lactams promote release of growth hormone
06/20/1995US5426103 Certain macrocyclic lactam derivatives
06/06/1995US5422371 Contacting a cell with a fatty acid or fatty alcohol to prevent reduction of testosterone to 5a-dihydrotestosterone
05/1995
05/17/1995EP0652749A1 METHODS AND COMPOSITIONS FOR INHIBITING 5$g(a)-REDUCTASE ACTIVITY
05/10/1995EP0651738A1 Natural amino acid derivatives as metalloproteinase inhibitors
05/09/1995US5413997 Triphenylmethane derivatives
04/1995
04/27/1995WO1995011231A1 Amidino derivatives useful as nitric oxide synthase inhibitors
04/27/1995CA2173468A1 Amidino derivatives useful as nitric oxide synthase inhibitors
04/19/1995EP0550635B1 Fused ring analogs of nitrogen containing nonaromatic heterocycles
03/1995
03/01/1995EP0640592A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists
02/1995
02/07/1995US5387590 Analgesics
02/02/1995WO1995003289A1 Benzo-fused lactams promote release of growth hormone
01/1995
01/12/1995WO1995001342A1 Ansamycin derivatives as antioncogene and anticancer agents
01/12/1995CA2166320A1 Ansamycin derivatives as antioncogene and anticancer agents
01/11/1995CN1097192A Retroviral protease inhibitors
12/1994
12/14/1994EP0628030A1 2,3,4,5-TETRAHYDRO-1H --3-BENZAZEPINES HAVING ANTI-PSYCHOTIC ACTIVITY, AND SYNTHESIS OF $g(a)-SUBSTITUTED-ARYLACETAMIDES
12/13/1994US5373008 Phenylamidine and phenylguanidine derivatives and their use as anti-diabetic agents
08/1994
08/23/1994US5340822 Substance P, neurokinin antagonists
08/03/1994EP0608336A1 Azabicyclo arylacetylene and arylenyne oximes as cholinergic agents and methods of treatment
07/1994
07/27/1994EP0607864A2 Tricyclic condensed heterocyclic compounds for the treatment of senile dementic
07/20/1994EP0325616B1 Penetration enhancers for transdermal delivery of systemic agents
06/1994
06/23/1994WO1994008578A3 Tumoricidal activity of benzoquinonoid ansamycins against prostate cancer and primitive neural malignancies
06/22/1994EP0602306A1 Retroviral protease inhibitors
06/17/1994CA2111454A1 Retroviral protease inhibitors
06/01/1994EP0599444A1 Dual action inhibitors
04/1994
04/28/1994WO1994008578A2 Tumoricidal activity of benzoquinonoid ansamycins against prostate cancer and primitive neural malignancies
04/28/1994CA2146668A1 Tumoricidal activity of benzoquinonoid ansamycins against prostate cancer and primitive neural malignancies
04/26/1994US5306718 Analgesics, cognition activators
04/06/1994CN1084849A Dual action inhibitors
03/1994
03/31/1994WO1994006774A1 Anti-inflammatory macrolactam (cyclamenol)
03/31/1994CA2144747A1 New natural substance cyclamenol and chemical derivatives
03/24/1994DE4231289A1 Neuer Naturstoff Cyclamenol und chemische Derivate New natural product cyclamenol and chemical derivatives
03/17/1994WO1994005634A1 Benzo-fused lactams promote release of growth hormone
02/1994
02/03/1994WO1994002447A1 Hydroxamic acid derivatives as metalloproteinase inhibitors
02/03/1994WO1994002446A1 Natural amino acid derivatives as metalloproteinase inhibitors
02/01/1994US5283241 Animal growth regulators
01/1994
01/20/1994WO1994001100A1 METHODS AND COMPOSITIONS FOR INHIBITING 5α-REDUCTASE ACTIVITY
01/04/1994US5276165 Preparation of N-substituted lactams
12/1993
12/01/1993CN1078969A Condensed heterocyclic ketone derivatives, their production and use
11/1993
11/16/1993US5262547 Vapor phase reaction of a hydrocarbon with oxygen
10/1993
10/19/1993US5254682 Cyclic renin inhibitors containing 3(S)-amino-4-cyclohexyl-2(R)-hydroxy-butanoic acid or 4-cyclo-hexyl-(2R, 3S)-dihydroxybutanoic acid or related analogs
10/06/1993EP0563345A1 Novel 4-arylpiperazines and 4-arylpiperidines
10/05/1993CA1322795C Process for extracting organic composites and solutions and aqueous suspensions thereof
09/1993
09/29/1993EP0562049A1 Novel 4-arylpiperazines and 4-arylpiperidines
09/21/1993US5246940 Substituted n-biphenylyl lactams
09/21/1993CA1322368C Fused heteroalkylene quinolinamines, a process and intermediates for their preparation and their use as medicaments
09/15/1993EP0560235A1 Condensed heterocyclic ketone derivatives, their production and use
09/14/1993US5244889 Treatment of cardiovascular disorders
09/10/1993CA2091216A1 Condensed heterocyclic ketone derivatives, their production and use
09/07/1993US5242912 Cyclic anthranilic acid derivatives and process of preparing the same
09/02/1993WO1993016997A1 2,3,4,5-TETRAHYDRO-1H^_-3-BENZAZEPINES HAVING ANTI-PSYCHOTIC ACTIVITY, AND SYNTHESIS OF α-SUBSTITUTED-ARYLACETAMIDES
08/1993
08/31/1993US5241065 Selectively antagonize dopamine D-1 receptors
08/04/1993CN1074937A 4,5-dihydro geldanamycin, preparation of its hydroquinone, and applications
08/03/1993CA1320956C Catalytic preparation of cyanoalkyl lactams
07/1993
07/22/1993WO1993014215A1 Process and uses for 4,5-dihydrogeldanamycin and its hydroquinone
07/22/1993CA2127457A1 Process and uses for 4,5-dihydrogeldanamycin and its hydroquinone
06/1993
06/29/1993US5223498 Phenylamidine and phenylguanidine derivatives and their use as antidiabetic agents
06/29/1993CA1319613C Penetration enhancers for transdermal delivery of systemic agents
06/09/1993EP0545150A1 Process for the preparation of N-substituted lactams by reductive amination of dicarboxylic acid derivatives with mixtures of primary, secondary and tertiary amines
06/02/1993EP0544620A1 Macrocyclic lactams as inhibitors of atrial natriuretic factors (ANF)-degrading neutral endopeptidase (NEP)
05/1993
05/27/1993CA2083622A1 Certain macrocyclic lactam derivatives
05/19/1993EP0542554A1 Substituted N-biphenylyl lactams
05/14/1993CA2082787A1 Substituted n-biphenylyl lactams
04/1993
04/29/1993WO1993008192A1 Azabicyclo arylacetylene and arylenyne oximes as cholinergic agents and methods of treatment
04/27/1993US5206751 Process for the production of an impact-resistant liquid crystal switching and display device
03/1993
03/18/1993WO1993004682A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/18/1993CA2095847A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/16/1993CA1314655C Hydroxylamine derivatives
03/12/1993WO1993004684A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/12/1993CA2095826A1 4-arylpiperazines and 4-arylpiperidines
03/02/1993US5190937 Lactam derivatives
02/1993
02/02/1993CA1313371C Fused azepinone and azocinone derivatives, processes for their preparation, agents containing them and their use, and intermediates in their preparation
01/1993
01/26/1993US5182288 Substituted n-biphenylyl lactams
12/1992
12/23/1992EP0518943A1 Mercaptoacyl aminolactam endopeptidase inhibitors
12/16/1992EP0518672A2 Cyclic renin inhibitors
12/12/1992CA2070972A1 Cyclic renin inhibitors
11/1992
11/11/1992EP0512901A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them
10/1992
10/20/1992US5156837 Cosmetic compositions containing quaternized nitrogen compounds
10/15/1992WO1992012133A3 Arthropodicidal carboxanilides
10/14/1992EP0368933B1 Compositions comprising 1-oxo- or thiohydrocarbyl substituted azacycloalkanes
07/1992
07/23/1992WO1992012133A2 Arthropodicidal carboxanilides
06/1992
06/24/1992CN1062134A Production of hydrocarbon derivatives
06/23/1992US5124322 Antiarthritic agents
06/17/1992EP0257063B1 Compositions comprising 1-substituted azacycloalkanes and their uses
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