Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
05/2000
05/18/2000CA2347228A1 Process for preparing solid percarboxylic acid raw bleach material
05/17/2000EP1000930A2 Tachykinin antagonists
05/17/2000EP1000621A2 Use of 6-heterocyclic-4-amino-1,3,4,5-tetrahydrobenz (CD) indoles for treating motion sickness and vomiting
05/17/2000EP1000090A1 Novel photoinitiators and applications therefor
05/17/2000EP1000063A1 4-OXO-3,5-DIHYDRO-4H-PYRIDAZINO 4,5-$i(b)]-INDOLE-1-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY
05/17/2000EP1000047A1 1-(n-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of the phenyl ring
05/17/2000EP1000027A1 Thermodynamically stable modification of 1-(4-carbazolyloxy)-3- 2-(2-methoxyphenoxy)ethylamino]-2-propanole, process for its preparation and pharmaceutical compositions containing it
05/17/2000EP1000026A1 Special 3-azabicyclo 3.1.0]hexanes, method for producing and modifying the same, and their use
05/17/2000EP1000025A1 Substituted naphthopyrans
05/17/2000EP1000018A2 Urokinase inhibitors
05/17/2000EP0999834A1 Antithrombotic agents
05/17/2000CN1253555A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same
05/17/2000CN1253545A Aryl sulfonamides and analogues thereof and their use in treatment of neurodegenerative diseases
05/17/2000CN1253543A Process for producing ketoprofen and 5-benzoyl-3-methyl-2-indolinone
05/17/2000CN1253528A Optical recording media
05/17/2000CN1253507A Acid-labile and enzymatically divisible dye structure for diagnosis with near infrared light and for therapy
05/17/2000CN1253501A IL-8 receptor antagonists
05/17/2000CN1052482C Camptothecin derivatives, preparations thereof and antitumor agents
05/16/2000US6063807 Cyclo-oxygenase inhibitor and amidine derivatives salts, preparation method therefor, use thereof as drugs, and pharmaceutical compositions containing said salts
05/16/2000US6063806 Indolyl or indolinyl derivatives and medicinal use thereof as ACAT or lipid peroxidation inhibitors
05/16/2000US6063804 Pyrrole compounds
05/16/2000US6063785 Isomers of drugs for racemic mixtures
05/16/2000CA2126752C Benzopyran and related ltb4 antagonists
05/11/2000WO2000025778A1 5ht1 receptor agonists and metoclopramide for the treatment of migraine
05/11/2000WO2000025777A1 SUBSTITUTED PHENETHYLSULFONES AND METHOD OF REDUCING TNFαLEVELS
05/11/2000WO2000025776A1 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use
05/11/2000WO2000025770A1 Carbocyclic potassium channel inhibitors
05/11/2000WO2000009099A3 Treatment of vasodilatory headache
05/11/2000DE19851184A1 N-Arylsulfonyl-aminosäure-omega-amide N-arylsulfonyl-amino-omega-amides
05/11/2000CA2348543A1 5ht1 receptor agonists and metoclopramide for the treatment of migraine
05/10/2000EP0999220A2 Low molecular weight peptidomimetic growth hormone secretagogues
05/10/2000EP0999208A1 Nitrogenous heterocyclic compounds and hyperlipemia remedy containing the same
05/10/2000EP0998281A1 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
05/10/2000CN1252790A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
05/10/2000CN1252713A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
05/10/2000CN1252690A Fungicide active substance combinations
05/09/2000US6060609 Reacting a sulfonyl cyanide with cyclopentadiene in the presence of water and in a hydrocarbon solvent at a ph of 4 to 7
05/09/2000US6060608 Analogs of CC-1065 and the duocarmycins
05/09/2000US6060606 Optical recording medium having at least a recording layer and a reflective layer on a substrates; high density, compact disks
05/09/2000US6060586 Ureins derived from alpha, omega-diamono acids and process for their preparation
05/09/2000US6060513 Compounds and compositions for delivering active agents
05/09/2000US6060499 Concurrently administering mixture of long-acting non-steroidal antiinflammatory drug (la-nsaid) with 5ht agonist to reduce relapse
05/09/2000US6060498 N-(3-chloro-1h-indol-7-yl)-4-sulfamoylbenzenesulfonamide dissolved together with a base to form alkaline aqueous solution for parenteral injection
05/09/2000US6060492 Side effect reduction
05/09/2000US6060476 α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
05/09/2000US6060432 Synergistic mixture; crops, agriculture
05/04/2000WO2000024732A1 Method of lithiating five-membered heterocycles
05/04/2000WO2000024714A1 Intermediate for the synthesis of amlodipine, preparation process and corresponding utilization
05/04/2000WO2000006085A3 Compounds and methods
05/04/2000WO1999064038A9 Novel analgesic agents
05/04/2000WO1999064031A9 β2-ADRENERGIC RECEPTOR AGONISTS
05/04/2000WO1999043672A9 Inhibitors of phospholipase a2
05/03/2000EP0997458A1 Novel tricyclic compounds having saturated rings and medicinal compositions containing the same
05/03/2000EP0997457A1 3-benzoylindole derivatives and drugs containing the same
05/03/2000EP0861233B1 N-protected/n-substituted-beta-amino hydroxy sulfonates
05/03/2000CN1052003C Prodrugs of antiinflammatory 3-acyl-2-oxidole-1-carboxamides
05/02/2000US6057455 Preparation of intermediates useful in the synthesis of quinoline antibiotics
05/02/2000US6057449 Direct preparation of pyrrolo[3,4-c]pyrroles
05/02/2000US6057371 Sigma receptor ligands and the use thereof
05/02/2000US6057369 Use in the treatment of disease states associated with proteins that mediate cellular activity which are capable of being modulated by inhibiting a matrix metalloproteinase (mmp), tumor necrosis factor (tnf) or cyclic amp
05/02/2000US6057349 2-imidazoline, 2-oxazoline, 2-thiazoline, and 4-imidazole derivatives of methylphenyl, methoxphenyl, and aminophenyl alkylsulfonamides and ureas and their use
05/02/2000US6057347 Comprising nonsteroidal antiinflammatory drug and compound that donates, transfers, or releases nitric oxide, elevates endogenous synthesis levels of nitric oxide, or is substrate for nitric oxide synthase
05/02/2000US6057336 Lactam metalloprotease inhibitors
05/02/2000US6057323 Kappa agonist compounds pharmaceutical formulations and method of prevention and treatment of pruritus therewith
05/02/2000CA2136411C Immediate release tablet cores of insoluble drugs having sustained release coating
04/2000
04/27/2000WO2000023425A1 New compounds, their preparation and use
04/27/2000WO2000023424A1 Epibatidine analogues as acetylcholine receptor antagonists
04/27/2000WO2000023423A1 Method for producing (+)-exo-6-phenyl-3-azabicyclo-[3.2.0]heptanes
04/27/2000WO2000023421A1 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES
04/27/2000WO2000023420A1 Aromatic amine derivatives, process for the preparation thereof and agents containing the same
04/27/2000WO1999063933A9 Multivalent agonists, partial agonists and antagonists of the gaba receptors
04/27/2000DE19848521A1 Preparation of (+)-exo-6-phenyl-3-azabicyclo(3.2.0)heptane derivatives comprises photocyclization of bisallyl ammonium salts, isomer resolution using (-)-ditoluoyltartaric acid and crystallization
04/27/2000CA2348159A1 Aromatic amine derivatives, their production and use
04/27/2000CA2347792A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
04/26/2000EP0994862A2 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
04/26/2000EP0994854A1 Method for preparing a substituted perhydroisoindole
04/26/2000EP0994848A1 Glucagon antagonists/inverse agonists
04/26/2000EP0994712A1 Inhibitors of neutrophil mediated oxidant production
04/26/2000EP0973737A4 Efficient synthesis of a chiral mediator
04/26/2000EP0680469B1 Aminoacid derivates, medicaments containing these compounds and process for preparing the same
04/26/2000EP0554247B1 Neuroprotective indolone and related derivatives
04/25/2000US6054482 Hydrolysis of gabapentin or the lactam to form acid addition salt, conversion to pure compound by ion exchanging; antiepileptic agents
04/25/2000US6054457 Benzamide derivatives and their use as vasopressin antagonists
04/25/2000US6054445 Kappa opioid agonist activity; analgesics and anti-pruritic agents
04/25/2000CA2010827C Use of derivates of n-phenyl-3,4,5,6-tetrahydrophthalimide for the desiccation and abscission of plant organs
04/20/2000WO2000021950A1 2,3-dihydro-1h-isoindole derivatives useful as modulators of dopamine d3 receptors (antipsychotic agents)
04/20/2000WO2000021929A1 Process for preparing 4-substituted-1h-indole-3-glyoxamides
04/20/2000WO2000021923A1 Process for preparing toluenesulfinates
04/20/2000WO2000021563A1 Remedies or preventives for ischemic reflow failure
04/20/2000WO2000021508A2 Novel therapeutic use of compounds with beta-3-agonist activity
04/20/2000WO1999064000A9 Novel therapeutic agents that modulate neurokinin receptors
04/20/2000WO1999048868A9 Heterocyclic classes of compounds for the modulating tyrosine protein kinase
04/20/2000CA2347718A1 Process for preparing 4-substituted-1h-indole-3-glyoxamides
04/20/2000CA2346699A1 Process for preparing toluenesulfinates
04/20/2000CA2346334A1 Composition for treating or preventing ischemia reperfusion injury
04/19/2000EP0994104A1 Aryl (sulfide, sulfoxide and sulfone) derivatives and drugs containing the same as the active ingredient
04/19/2000EP0993831A2 Compounds and compositions for delivering active agents
04/19/2000EP0993458A1 3-benzylpiperidine
04/19/2000EP0993442A1 Hydrazine derivatives
04/19/2000EP0993441A1 INHIBITORS OF p38