| Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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| 01/30/2001 | US6180087 Tunable indocyanine dyes for biomedical applications |
| 01/30/2001 | US6180085 Useful for optical tomographic, endoscopic, photoacoustic and sonofluoresence applications for detection and treatment of tumors and other abnormalities |
| 01/30/2001 | US6179883 2-imino-2,3-dihydro-1H-indole derivatives for dyeing keratin fibers |
| 01/25/2001 | WO2001005791A2 NEW PROCESS FOR THE PREPARATION OF N-(1,1-DIMETHYLETHYL)-4-[[5'-ETHOXY-4-cis-[2-(4-MORFOLINO)ETHOXY]-2'-OXOSPIRO[CYCLOHEXAN-1,3'-[H]INDOL]-1'(2'H)-yl]-SULFONYL]-3-METHOXYBENZAMIDE AND ITS SALTS |
| 01/25/2001 | WO2001005765A1 Cyclic amides and imides having selective antagonist activity at alpha-1d adrenergic receptor |
| 01/25/2001 | WO2001005761A1 sPLA2 INHIBITORS |
| 01/25/2001 | WO2001005760A2 New process for the preparation of spiro [(4-cyclohexanone)-[3h]indol]-2'[1'h]-one derivatives |
| 01/25/2001 | WO2001005759A2 Process for the preparation of spiro-[cis-4-(beta-hydroxyethyloxy)cyclohexane-(3h) indol)-2'(1'h)-one derivatives |
| 01/25/2001 | WO2001005758A2 Indoles and indazoles for the treatment of migraine |
| 01/25/2001 | DE19934433A1 New N-(indolyl-carbonyl)-N'-ethyl-piperazine derivatives, are 5-HT-2A receptor antagonists useful e.g. for treating schizophrenia, depression, Parkinson's disease, Alzheimer's disease or anorexia |
| 01/25/2001 | DE19934321A1 New N-phenyl-naphthalenesulfonamide derivatives are antiviral agents especially useful for treating cytomegalovirus infections |
| 01/25/2001 | DE19934283A1 Agent for coloring fibres, especially for temporary coloration of the hair, made by mixing prior to use of one component containing an enamine compound and another component containing at least one carbonyl compound |
| 01/25/2001 | CA2379208A1 Spla2 inhibitors |
| 01/25/2001 | CA2378047A1 Heterocyclic compounds for the treatment of migraine |
| 01/24/2001 | EP1070705A1 Indole derivatives |
| 01/24/2001 | EP1070703A1 Cyclobutene derivatives |
| 01/24/2001 | EP1070051A1 Process for the production of r-(+)-6- carboxamido- 3-n- methylamino- 1,2,3,4- tetrahydrocarbazole |
| 01/24/2001 | EP1070050A1 N-aryloxyethyl-indoly-alkylamines for the treatment of depression (5-ht1a receptor active agents) |
| 01/24/2001 | EP1070048A1 Calcilytic compounds |
| 01/24/2001 | EP1070046A1 Propanolamine derivatives |
| 01/24/2001 | EP0712389B1 Therapeutic compound - fatty acid conjugates |
| 01/24/2001 | EP0559687B1 2-aminocinnamic acid esters |
| 01/24/2001 | CN1281436A N-Benzyl-3-indenylacetamides derivatives for treating neoplasia |
| 01/24/2001 | CN1281429A Novel aryloxy-alkyl-dialkylamines |
| 01/24/2001 | CN1281334A Method for treating Alzheimer's disease |
| 01/24/2001 | CN1061069C Purification of indigo |
| 01/24/2001 | CN1061034C Tricyclic indole-2-carboxylic acid derivatives |
| 01/23/2001 | US6177570 Reaction of dicarboxylic anhydride with an amine in the presence of a tertiary amine. |
| 01/23/2001 | US6177466 Matrix metalloproteinase inhibitors |
| 01/23/2001 | US6177440 Substituted tricyclics |
| 01/23/2001 | US6177426 Morpholino-N-ethyl ester prodrugs of indole sPLA2 inhibitors |
| 01/23/2001 | US6177401 Use of organic compounds for the inhibition of Flk-1 mediated vasculogenesis and angiogenesis |
| 01/23/2001 | CA2197272C Pro-drugs of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)ethyl)-6- chloro-1,3-dihydro-2h-indol-2-one |
| 01/22/2001 | CA2312203A1 Cyclobutene derivatives, their preparation and their therapeutic uses |
| 01/18/2001 | WO2001004173A1 Process for the polymerisation of cycloolefins and polymerisable cycloolefins |
| 01/18/2001 | WO2001004092A1 Process for the preparation of tricyclic amino alcohol derivatives |
| 01/18/2001 | WO2001003684A2 Albumin-binding compounds that prevent nonenzymatic glycation and that may be used for treatment of glycation-related pathologies |
| 01/18/2001 | DE19933313A1 Agent for coloring fibres, especially for temporary coloration of the hair, made by mixing prior to use of one component containing an enamine compound and another component containing at least one carbonyl compound |
| 01/18/2001 | CA2377760A1 Process for the preparation of tricyclic amino alcohol derivatives |
| 01/17/2001 | EP1069125A2 Carbamate derivatives of 4-amino-3-isoxazolidinones, 3-amino-1-hydroxypyrrolidin-2-ones and 1-amino-1-cyclopropanecarboxylic acid analogs, a process for their preparation and their use as medicaments |
| 01/17/2001 | EP1069111A1 Indole derivatives with antiviral activity |
| 01/17/2001 | EP1069110A1 Sulfonamide derivatives |
| 01/17/2001 | EP1068865A1 Use of 4,6-dimethoxy-indole 2 carboxylic acid or derivatives thereof for seborrhea treatment |
| 01/17/2001 | EP1068858A1 Use of 4,6-dimethoxyindole-2-carboxylic acid for stimulating or inducing hair growth and/or arresting hair loss |
| 01/17/2001 | EP1068306A1 Pentaerythritol lipid derivatives |
| 01/17/2001 | EP1068199A2 N-aryloxyethyl-indoly-alkylamines for the treatment of depression |
| 01/17/2001 | EP1068193A1 Benzylpiperazinyl- and benzylpiperidinyl ethanone derivatives, their preparation and their use as dopamine d 4? receptor antagonists |
| 01/17/2001 | EP1068184A1 N-aryloxyethylamine derivatives for the treatment of depression |
| 01/17/2001 | EP1068178A1 NON-PEPTIDE GnRH AGENTS |
| 01/17/2001 | EP1067950A1 Neo-tryptophan |
| 01/17/2001 | EP1067925A1 Antidiabetic agents |
| 01/17/2001 | CN1280578A Bis-quaternary ammonium derivatives as neuromuscular relaxants |
| 01/17/2001 | CN1280566A Method of synthesis of pyrrole amides |
| 01/17/2001 | CN1280561A Amidocarboxylic acid derivatives |
| 01/17/2001 | CN1280560A Adamantane derivatives |
| 01/17/2001 | CN1060761C New aryl (alkyl) propylamides, process for preparing them and pharmaceutical compositions containing them |
| 01/16/2001 | US6175021 Human non-pancreatic secretory phospholipase a2 (spla2); inhibits release of arachidonic acid to treat septic shock; ((3-(2-amino-1,2-dioxoethyl)-2-methyl-1-(phenylmethyl)-1h-indol-4 -yl)oxylacetic acid, for example |
| 01/16/2001 | US6175020 2-(((alk)oxy or amino)carbonylmethyl),9-((protected)aminomethyl)-1-azaspiro(4.4)nonane compounds, useful as template for constructing synthetic receptors and as intermediates in the synthesis of enzyme inhibitors |
| 01/16/2001 | US6175015 Fused indolecarboxamides: dopamine receptor subtype specific ligands |
| 01/16/2001 | US6175014 Process for the preparation of lactam derivatives |
| 01/16/2001 | US6174924 Treating nerve cell death comprising administering to a subject exhibiting symptoms of nerve cell death or susceptible to nerve cell death a substituted guanidine compound |
| 01/16/2001 | US6174889 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors |
| 01/16/2001 | US6174883 3-substituted-2-oxindoles derivatives |
| 01/16/2001 | US6174839 As herbicide |
| 01/16/2001 | CA2314539A1 Use of 4,6-dimethoxy-indole 2-carboxylic acid or its derivatives for the treatment of seborrhoea |
| 01/11/2001 | WO2001002403A1 METHOD FOR PREPARING SUBSTITUTED [1,4]DIAZEPINO[6,7,1-hi]INDOL-4-ONES |
| 01/11/2001 | WO2001002388A1 Indole derivatives and their use for the treatment of osteoporosis amongst other applications |
| 01/11/2001 | WO2001002369A2 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use |
| 01/11/2001 | WO2001002368A1 N-heterocyclic derivatives with neuronal activity |
| 01/11/2001 | WO2001002355A2 Indole synthesis |
| 01/11/2001 | WO2000059904A3 Compounds and methods to treat cardiac failure and other disorders |
| 01/11/2001 | CA2376707A1 Process for the preparation of substituted ¬1,4|diazepino¬6,7,1-hi|indol-4-ones |
| 01/11/2001 | CA2376657A1 Indole derivatives and their use for the treatment of osteoporosis amongst other applications |
| 01/10/2001 | EP1066290A1 PYRROLO[1,2-a]PYRAZINE sPLA 2 INHIBITOR |
| 01/10/2001 | EP1066283A2 Substituted indolealkanoic acids |
| 01/10/2001 | EP1066258A1 Aryl phenyl substituted cyclic ketoenols |
| 01/10/2001 | EP1066257A2 Heterocylic classes of compounds for the modulating tyrosine protein kinase |
| 01/10/2001 | CN1279617A Combination of an aldose reductase inhibitor and a glycogen phosphorglase inhibitor |
| 01/10/2001 | CN1060472C Hydroxamic acid derivatives with tricylic substitution, their preparing methods, medicines containing them and uses thereof |
| 01/09/2001 | US6172261 Biosynthesis using chain extension |
| 01/09/2001 | US6172255 Alkoxy-alkyl-substituted 1-H-3-aryl-pyrrolidine-2,4-diones used as herbicides and pesticides |
| 01/09/2001 | US6172113 Bicyclic amino derivatives and PGD2 antagonist containing the same |
| 01/09/2001 | US6172108 Hydrazide compounds |
| 01/09/2001 | US6172100 Administering aminated 1-benzyl-2-phenylindole derivatives; benzylation |
| 01/09/2001 | US6172099 Tricyclic compounds having saturated rings and medicinal compositions containing the same |
| 01/09/2001 | US6172084 Quinoline-indole antimicrobial agents, uses and compositions related thereto |
| 01/09/2001 | US6172082 α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors |
| 01/09/2001 | US6172073 Benzimidazolyloxy alkanamines as serotonin reuptake inhibitors; nicotine and tobacco withdrawal; psychological, eating, brain, gastrointestinal, sleep, and sexual disorders |
| 01/09/2001 | US6172072 Heterocyclically substituted benzamides and their use in fighting diseases |
| 01/09/2001 | US6172057 Antiinflammatory agents; antiarthritic agents; antitumor agents |
| 01/04/2001 | WO2001000658A1 C-terminal modified (n-substituted)-2-indolylcarbonyldipeptides as inhibitors of the ice/ced-3 family of cysteine proteases |
| 01/04/2001 | WO2001000576A1 Indole and indazole urea-peptoids as thrombin receptor antagonists |
| 01/04/2001 | WO2001000206A1 Vla-4 inhibitor compounds |
| 01/04/2001 | WO2001000197A2 Methods of treating fungal infections with inhibitors of nad synthetase enzyme |
| 01/04/2001 | CA2376892A1 Methods of treating fungal infections with inhibitors of nad synthetase enzyme |
| 01/04/2001 | CA2369308A1 Vla-4 inhibitor compounds |
| 01/04/2001 | CA2365341A1 C-terminal modified (n-substituted)-2-indolylcarbonyldipeptides as inhibitors of the ice/ced-3 family of cysteine proteases |
| 01/03/2001 | EP1065204A1 Bicycliccarbonyl indole compounds as anti-inflammatory/analgesic agents and as COX-2 inhibitors |
| 01/03/2001 | EP1065203A2 Heterocyclic compounds as retinoic acid receptor antagonists |
| 01/03/2001 | EP1064941A1 Use of melatoninergic ligands for obtaining pharmaceutical compositions for the prevention or the treatment of gastrointestinal pathologies |