Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
09/1999
09/07/1999CA1340721C 1,4-dihydro-quinoline-and naphthyridine-3-carboxylic acid antibacterial agents
09/02/1999WO1999043672A1 Inhibitors of phospholipase a2
09/02/1999WO1999043670A1 Benzylpiperazinyl- and benzylpiperidinyl ethanone derivatives, their preparation and their use as dopamine d4 receptor antagonists
09/02/1999WO1999043655A1 Method for purifying (±)-2-azabicyclo(2.2.1)hept-5-en-3-one
09/02/1999WO1999043654A2 Inhibitors of phospholipase enzymes
09/02/1999WO1999043652A1 Indole derivatives and medicinal compositions containing the same
09/02/1999WO1999043651A2 Inhibitors of phospholipase enzymes
09/02/1999WO1999043650A2 Process(es) for the preparation of 6-trifluoromethyl-indoline derivatives
09/02/1999WO1999043649A1 Arylphenyl-substituted cyclic keto-enols
09/02/1999WO1999043644A1 N-sulphonyl and n-sulphinyl phenylglycinamide___________________
09/02/1999WO1999043643A2 Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes
09/02/1999WO1999024460A3 Dipeptide nitriles
09/02/1999WO1998034632A9 Compounds and compositions for delivering active agents
09/02/1999CA2322163A1 Inhibitors of phospholipase a2
09/02/1999CA2322162A1 Inhibitors of phospholipase enzymes
09/02/1999CA2322161A1 Inhibitors of phospholipase enzymes
09/02/1999CA2321830A1 Benzylpiperazinyl- and benzylpiperidinyl ethanone derivatives, their preparation and their use as dopamine d4 receptor antagonists
09/02/1999CA2320838A1 N-sulphonyl and n-sulphinyl phenylglycinamide___________________
09/01/1999EP0939078A2 Substituted phthalimido-cinnamic acid derivatives with herbicidal activity
09/01/1999EP0939077A2 3-Substituted 1-arylindole compounds as 5-HT2 antagonists
09/01/1999EP0938712A1 System and method for remotely grouping contents of an action history stack
09/01/1999EP0938491A1 Heterocyclic metallocenes and polymerization catalysts
09/01/1999EP0938474A2 Cyclopropylindole compounds and their use as prodrugs
09/01/1999EP0938466A1 Method for preparing cyclopropylamines
09/01/1999EP0938308A1 Antiparasitic agents
09/01/1999EP0724563B1 Intermediates for the preparation of a substituted 2,5-diamino-3-hydroxyhexane.
09/01/1999CN1227542A N-substituted indol-3-glyoxylamid with antiasthmatic, antiallergic and immunosuppressive/immunomodulating effect
09/01/1999CN1227540A Hydroxamic and carboxylic acid derivatives having MMP and TNF inhibitory activity
09/01/1999CN1227487A Pharmaceutical compositions containing mesembrine and related compounds
08/1999
08/31/1999US5945542 Isolation of natural L-β-3-indolylalanine and enrichment of natural aliphatic amino acid mixtures with natural L-β-3-indolylalanine
08/31/1999US5945443 Kappa agonist compounds and pharmaceutical formulations thereof
08/31/1999US5945317 Isolated from fermentation cultures of nodulisporum species; for insecticides, nematocides, miticides
08/31/1999CA2173328C Hiv protease inhibitors
08/31/1999CA2163216C Anxiolytic agent
08/31/1999CA2145835C Hydroxamic acid derivatives with tricyclic substitution
08/26/1999WO1999042457A2 Substituted alxoxycarbonyl compounds
08/26/1999WO1999042445A1 Phtalimido arylpiperazines as alpha 1a receptor antagonists useful in the treatment of benign prostatic hyperplasia
08/26/1999WO1999042444A1 Substituted isoindolones and their use as cyclic gmp modulators in medicaments
08/26/1999WO1999042443A1 Sulfonylamino derivatives which inhibit matrix-degrading metalloproteinases
08/26/1999WO1999042442A1 Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof
08/26/1999WO1999042436A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
08/26/1999WO1999042102A1 Indole-3-propionic acids, salts and esters thereof used as medicaments
08/26/1999DE19844192A1 New substituted alkoxycarbonyl compounds
08/26/1999DE19807423A1 New isoindolone derivatives useful as soluble guanylate cyclase activators for treating cardiovascular disorders, asthma, renal insufficiency, diabetes, cirrhosis or cognitive dysfunction
08/26/1999CA2321460A1 Substituted alxoxycarbonyl compounds
08/26/1999CA2320469A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
08/26/1999CA2316944A1 Aminoguanidinehydrazone derivative, production and use thereof
08/25/1999EP0937726A1 Intermediates for the preparation of duocarmycin sa and derivatives thereof, and process for the production of the intermediates
08/25/1999EP0937715A1 Tetrahydrobenzindole compounds
08/25/1999EP0937714A1 Process for the preparation of an optically active indoline-2-carboxylic acid or derivative thereof
08/25/1999EP0937036A1 Substituted 4-biphenyl-4-hydroxybutyric acid derivatives as matrix metalloprotease inhibitors
08/25/1999CN1226911A Condensed azo compound and process for producing the same
08/25/1999CN1226594A Method for coal liquefaction
08/24/1999US5942536 Useful for treating migraine
08/24/1999US5942493 LH-RH antagonists having improved action
08/24/1999CA2212548C Use of carbazole compounds for the treatment of congestive heart failure
08/24/1999CA2193348C Substituted alkyldiamine derivatives and their use as tachykinin antagonists
08/19/1999WO1999041276A1 β-SHEET MIMETICS AND METHODS RELATING TO THE USE THEREOF
08/19/1999WO1999041239A1 B cell inhibitors
08/19/1999WO1999041224A1 Biaryl-acetic acid derivatives and their use as cox-2 inhibitors
08/19/1999WO1999040913A1 Chemical compounds
08/19/1999DE19808136C1 Extraction process for purification of aqueous racemic 2- azabicycloÝ2.2.1¨hept-5-en-3-one solution useful as starting material for antiviral and chemotherapeutic nucleoside analogues
08/19/1999CA2319766A1 .beta.-sheet mimetics and methods relating to the use thereof
08/19/1999CA2318966A1 Biaryl-acetic acid derivatives and their use as cox-2 inhibitors
08/19/1999CA2317456A1 Chemical compounds
08/18/1999EP0935918A1 Antibacterial compositions with activity against Ralstonia solanacearum
08/18/1999EP0935463A2 Anti-neurogenic inflammatory compounds and compositions and methods of use thereof
08/18/1999CN1226229A Glyoxalic acid derivative
08/17/1999US5939587 N-protected/N-substituted-beta-amino hydroxy sulfonates
08/17/1999US5939583 Antiarthritic agents; bone, cardiovascular, brain, nervous system disorders; antitumor and antimetastasis agents
08/17/1999US5939563 Fungicides
08/17/1999US5939462 NPY5 receptor antagonists and methods for using same
08/17/1999US5939451 Use of sulfonamides
08/17/1999US5939450 N,N-dimethyl-8,8-dipropyl-2-azaspiro 4.5!decane-2-propanamine dimaleate
08/17/1999US5939443 Selective β3 adrenergic agonists
08/17/1999US5939437 CCK and gastrin receptor ligands
08/17/1999US5939381 4-(4-(phenoxyacetyl)aminophenyl)butyric acid as a carrier for drug delivery
08/17/1999US5939268 Diels-alder reaction product of a diene and a dienophile; chemical intermediates for drugs, solid phase synthesis
08/12/1999WO1999040072A1 Five-membered, benzo-condensed heterocycles used as antithrombotic agents
08/12/1999WO1999040064A1 Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament
08/12/1999WO1999028304A3 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
08/12/1999CA2319555A1 Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament
08/12/1999CA2319494A1 5-membered heterocyclic condensed benzoderivatives, the preparation thereof and their use as pharmaceuticals
08/11/1999EP0934992A1 Light-emitting material for organo-electroluminescence device and organic electroluminescence device
08/11/1999EP0934931A2 3-Benzylidene-2-indolinones and their analogues as tyrosine kinase activity modulators
08/11/1999EP0934319A1 1H-PYRIDO[3,4-b]INDOLE-4-CARBOXAMIDE DERIVATIVES, PREPARATION AND APPLICATION THEREOF IN THERAPEUTICS
08/11/1999EP0934316A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
08/11/1999EP0934307A1 Substituted azabicylic compounds and their use as inhibitors of the production of tnf and cyclic amp phosphodiesterase
08/11/1999EP0934288A1 Oxadiazoles, processes for their preparation and their use as medicaments
08/11/1999EP0934269A1 Analogs of cc-1065 and the duocarmycins
08/11/1999EP0934268A1 Process for preparing 2-azadihydroxybicyclo 2.2.1]heptane compounds and the l-tartaric acid salt of the compound
08/11/1999EP0934267A1 $g(a)-AMINO SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE INHIBITORS
08/11/1999EP0934262A1 Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors
08/11/1999EP0934252A1 Amide derivatives and their use as pesticides
08/11/1999EP0934068A1 Compounds and methods
08/11/1999CN1225634A Synthesis of indolylmaleimides
08/11/1999CN1225630A Methanesulphonate salt of an arylpiperzine derived from tryptamine and its solvates for pharmaceutical use
08/11/1999CN1225623A Inhibition of matrix metalloproteases by acetylene contg. compounds
08/11/1999CN1225622A Substituted oxobutyric acids as matrix metalloprotease inhibitor
08/11/1999CN1225620A Substituted 4-arylbutyric acid derivatives as matrix metalloprotease inhibitors