Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
---|
11/15/2000 | EP0901453B1 Method for organic reactions |
11/15/2000 | EP0876342B1 Fluorinated melt additives for thermoplastic polymers |
11/15/2000 | EP0842227B1 Azothiophenes |
11/14/2000 | US6147254 Reacting chiral base in solution with enantiomeric mixture of n-protected-cis-4-amino-2-cyclopentene-1-carboxylic acids to produce, in diastereoselective manner by fractional crystallisation, substantially pure salt |
11/14/2000 | US6147253 N-protected/N-substituted-beta-amino-hydroxy sulfonates |
11/14/2000 | US6147106 Indolinone combinatorial libraries and related products and methods for the treatment of disease |
11/14/2000 | US6147105 Use in the treatment of estrogen-related diseases |
11/14/2000 | US6147082 Chalcones having antiproliferative activity |
11/14/2000 | US6147073 Substituted tetralymethylen-Oxindoles analogues as tyrosine kinase inhibitors |
11/14/2000 | CA2080221C An improved process for the preparation of substituted indolone derivatives |
11/09/2000 | WO2000066556A1 Indoline derivatives as progesterone antagonists |
11/09/2000 | WO2000066555A1 Thio-oxindole derivatives |
11/09/2000 | WO2000066554A1 3,3-substituted indoline derivatives |
11/09/2000 | WO2000066553A1 Substituted indole sulfonamides as antiviral agents |
11/09/2000 | WO2000066546A2 Monofluoroalkyl derivatives |
11/09/2000 | WO2000066528A2 Quinones for treatment of diseases |
11/09/2000 | WO2000066489A1 Synthesis of hydrogen peroxide |
11/09/2000 | WO2000066104A2 Ace-2 inhibiting compounds and methods of use thereof |
11/09/2000 | WO2000039087A3 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds as factor xa inhibitors |
11/09/2000 | WO2000035906A3 4- and 5-alkynyloxindoles and 4- and 5-alkenyloxindoles |
11/09/2000 | WO2000028981A3 Methods for treating, preventing, and reducing the risk of the onset of alzheimer's disease using an hmg coa reductase inhibitor |
11/09/2000 | DE19921424A1 Substituierte Benzoylketone Substituted benzoyl ketones |
11/09/2000 | DE19920791A1 Substituierte Benzoylisoxazole Substituted benzoylisoxazoles |
11/09/2000 | CA2372611A1 Quinones for treatment of diseases |
11/09/2000 | CA2372595A1 Contraceptive compositions containing indoline derivatives and progestational agents |
11/09/2000 | CA2372591A1 Contraceptive compositions containing 3,3-substituted indoline derivatives and uses thereof |
11/09/2000 | CA2372490A1 Monofluoroalkyl derivatives |
11/09/2000 | CA2372387A1 Ace-2 inhibiting compounds and methods of use thereof |
11/09/2000 | CA2371638A1 Indoline derivatives as progesterone antagonists |
11/09/2000 | CA2371633A1 Thio-oxindole derivatives |
11/09/2000 | CA2371629A1 3,3-substituted indoline derivatives |
11/09/2000 | CA2371621A1 Substituted indole sulfonamides as antiviral agents |
11/08/2000 | EP1050534A1 2,3-methano-amino acid derivatives, process for their preparation and pharmaceutical compositions containing them |
11/08/2000 | EP1049664A1 Inhibition of raf kinase using symmetrical and unsymmetrical substituted diphenyl ureas |
11/08/2000 | EP1049472A1 Antagonists of gonadotropin releasing hormone |
11/08/2000 | CN1272842A 2-acylaminopropanamines as tachykinin receptor antagonists |
11/08/2000 | CN1272841A Novel lactam metalloprotease inhibitors |
11/08/2000 | CN1058265C Quinazoline derivatives and its preparing method and compositions containing the same |
11/07/2000 | US6143902 Semi-synthesis of paclitaxel using a protected c-2 hydroxyl protected-n-acyl (2r,3s)-3-phenylisoserine activated esters |
11/07/2000 | US6143775 Physical form of zafirlukast; asthma |
11/07/2000 | US6143734 Nitroso esters of β-oxo-amides and aryl propionic acid derivatives of non-steroidal antiinflammatory drugs |
11/07/2000 | US6143180 By liquid chromatography with a separating agent, improved by passing said optical isomers through a polysaccharide derivative as the active component in the reverse phase condition using a basic mobile phase |
11/07/2000 | US6143153 DNA sequencing |
11/07/2000 | US6143151 DNA sequencing |
11/07/2000 | CA2156455C Glycinamide derivatives, processes for their preparation and medicines containing them |
11/02/2000 | WO2000064989A1 Cyanine dye |
11/02/2000 | WO2000064986A1 Novel carbopyronine fluorescence dyes |
11/02/2000 | WO2000064888A1 Di-aryl acid derivatives as ppar receptor ligands |
11/02/2000 | WO2000064872A1 INHIBITORS OF c-JUN N-TERMINAL KINASES (JNK) |
11/02/2000 | WO2000064866A1 Diphenylurea derivatives |
11/02/2000 | WO2000064864A1 N-protected amines and their use as prodrugs |
11/02/2000 | EP1048650A2 Process for producing 2-azabicyclo (2.2.1) hept-5-en-3-one |
11/02/2000 | EP1047692A1 Methods of synthesizing and screening inhibitors of bacterial nad synthetase enzyme, compounds thereof and methods of treating bacterial and microbial infections with these inhibitors |
11/02/2000 | EP1047672A1 Process for preparing sparingly soluble aromatic amines |
11/02/2000 | EP1047664A1 Novel tricyclic compounds, preparation method and pharmaceutical compositions containing same |
11/02/2000 | EP1047645A1 Compound for use as a mineral fibre binder and process for providing such |
11/02/2000 | EP1047411A1 Substituted diphenyl indanone, indane and indole compounds and analogues thereof useful for the treatment or prevention of diseases characterized by abnormal cell proliferation |
11/02/2000 | DE19919793A1 Neue Sulfonamide New sulfonamides |
11/02/2000 | DE19919119A1 Neue Carbopyronin-Fluoreszenz-Farbstoffe New carbopyronine fluorescent dyes |
11/02/2000 | CA2368205A1 N-protected amines and their use as prodrugs |
11/01/2000 | CN1272095A Synthesis method for solution with high grade chloramine |
10/31/2000 | US6140504 Substituted intermediate compounds for the preparation of n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides |
10/31/2000 | US6140372 Acyl derivatives of melatonin and of melatoninergic analogues and their use as medicinal products |
10/31/2000 | US6140358 Substituted phenyl keto enols as pesticides and herbicides |
10/31/2000 | US6140353 Used as medicaments for the treatment and/or prevention of thromboses, apoplexy, cardiac infarction, inflammation and arteriosclerosis or as antitumor agents |
10/31/2000 | US6140352 Carbazolyl-substituted ethanolamines as selective β-3 agonists |
10/31/2000 | US6140327 Morpholino-n-ethyl ester derivative of an indole sPLA2 inhibitor |
10/26/2000 | WO2000063296A2 Cyanine dyes and synthesis methods thereof |
10/26/2000 | WO2000063171A1 Tricyclic compounds |
10/26/2000 | WO2000063170A1 Cyclobutene-3,4-dione derivatives as inhibitors of phosphodiesterase 5 |
10/26/2000 | WO2000035886A3 (hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors |
10/26/2000 | WO2000021508A3 Novel therapeutic use of compounds with beta-3-agonist activity |
10/26/2000 | DE19918725A1 New heterocyclic-substituted N-cyano-sulfonanilide compounds, useful as total or selective pre- or post-emergence herbicides, showing desiccant, defoliant, germination inhibiting and especially weed-killing activities |
10/26/2000 | CA2335240A1 Cyanine dyes and synthesis methods thereof |
10/25/2000 | EP1046627A2 Enantiopure reagents and process for the separation of enantiomers |
10/25/2000 | EP1045833A1 2,3-substituted indole compounds as cox-2 inhibitors |
10/25/2000 | EP0720601B1 Gastrin and cck receptor ligands |
10/25/2000 | EP0714418B1 Cosmetic melanins |
10/25/2000 | CN1271343A Utilizing spirocyclic phenyl keto-enols as pesticides and herbicides |
10/24/2000 | US6137007 Enantiomer compositions of (1R,4S)-1-butyrylamino-4-(hydroxymethyl)-2-cyclopentene |
10/24/2000 | US6136949 Resins containing phenylethynl-terminated compounds |
10/24/2000 | US6136861 Bicyclo[2.2.1]heptanes and related compounds |
10/24/2000 | US6136843 Indole derivatives useful as endothelin receptor antagonists |
10/24/2000 | US6136842 Sulphur derivatives comprising an amide bond, method for preparing same, use thereof as drugs, and pharmaceutical compositions containing such derivatives |
10/24/2000 | US6136157 Method for organic reactions |
10/21/2000 | CA2305944A1 Process for separating enantiomers and enantiopur reagent |
10/19/2000 | WO2000061583A1 Xanthine derivatives and analogs as cell signaling inhibitors |
10/19/2000 | WO2000061556A1 Nitrogen-containing heterocyclic compounds and benamide compounds and drugs containing the same |
10/19/2000 | WO2000061555A1 Indigoid bisindole derivatives |
10/19/2000 | WO2000061554A1 1-amino ethylindole derivatives for the treatment of urinary incontinence |
10/19/2000 | WO2000061553A1 2-aminoethyl-indole derivatives, their preparation and therapeutic use |
10/19/2000 | WO2000061549A2 Pharmaceutical compounds |
10/19/2000 | WO2000061539A1 3-bicycloaryl-2-aminomethyl bicycloalkanes as serotonine reuptake inhibitors |
10/19/2000 | WO2000061537A2 Pharmaceutical compounds |
10/19/2000 | WO2000061194A2 Short-chain peptide dye conjugates used as contrast agents for optical diagnostics |
10/19/2000 | WO2000061124A2 Use off cell membrane penetrating indigoid bisindole derivatives |
10/19/2000 | DE19917713A1 Kurzkettige Peptid-Farbstoffkonjugate als Konstrastmittel für die optische Diagnostik Short-chain peptide-dye conjugates as contrast agents for optical diagnostics |
10/19/2000 | DE19917504A1 New hydroxy-indole derivatives, useful in treatment of degenerative joint disease, viral and parasitic infections, bronchial, dermatological, neurodegenerative and prostate disorders, etc. |
10/19/2000 | CA2370406A1 Pharmaceutical compounds |
10/19/2000 | CA2369981A1 Therapeutic compounds for inhibiting interleukin-12 signaling and methods for using same |