Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
10/2000
10/19/2000CA2369670A1 Indigoid bisindole derivatives
10/19/2000CA2369103A1 Nitrogen-containing heterocyclic compounds and benamide compounds and drugs containing the same
10/19/2000CA2368840A1 3-bicycloaryl-2-aminomethyl bicycloalkanes as serotonine reuptake inhibitors
10/19/2000CA2368490A1 Short-chain peptide dye conjugates used as contrast agents for optical diagnostics
10/18/2000EP1044979A2 1-[(N-(un)substituted)amidoalkyl]spiroindolinonaphthoxazines, their preparation, compositions and (co)polymer matrices containing them
10/18/2000EP1044978A2 1-N-alkyl-5'-[(N'-(un)substituted)amido]spiroindolinonaphthoxazines, their preparation, compositions and (co)polymer matrices containing them
10/18/2000EP1044187A1 N-benzyl-3-indenylacetamides derivatives for treating neoplasia
10/18/2000EP1043991A1 Treatment for alzheimer's disease
10/18/2000EP0633886B1 Pharmaceutically active bicyclic-heterocyclic amines
10/18/2000EP0493606B1 Heterocycle-substituted benzene derivative, production thereof, and herbicide containing the same as active ingredient
10/18/2000CN1270518A Therapeutic or prophylactic agent for glomerulopathy
10/18/2000CN1270166A Derivatives of tricyclo-substituted isohydroxyloxime acid
10/17/2000US6133454 Method for preparing a substituted perhydroisoindole
10/17/2000US6133453 Reacting a substituted or unsubstituted 2,3-dihydrofuran with a salt of an aryl hydrazine
10/17/2000US6133305 Prevention and treatment of protein kinase related disorders such as cancer
10/17/2000US6133283 Mono- or polyenic carboxylic acid derivatives
10/17/2000US6133265 Treating physiological disorders associated with an excess of neuropeptide y, such as eating disorders, e.g., obesity, bulimia, and certain cardiovascular diseases, e.g., hypertension
10/17/2000US6133259 Diagnosis of alzheimer's disease
10/17/2000US6133252 Fungicides for the control of take-all disease of plants
10/12/2000WO2000059904A2 Compounds and methods to treat cardiac failure and other disorders
10/12/2000WO2000059888A1 N-benzimidazolylmethyl- and n-indolylmethyl-benzamides and their use as crf modulators
10/12/2000WO2000059885A1 Method for the preparation of tricyclic amino alcohol derivatives through azides
10/12/2000WO2000059883A2 Method for producing n-aryl-aza-heterocycles in the presence of cesium carbonate
10/12/2000WO2000059880A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
10/12/2000WO2000059875A2 Novel inhibitors of formation of advanced glycation endproducts (age's)
10/12/2000WO2000059868A1 Substituted aniline compounds
10/12/2000WO2000059504A1 Method for the treatment of neurological or neuropsychiatric disorders
10/12/2000WO1998025597A3 Method for treating and preventing heart failure and ventricular dilatation
10/12/2000WO1993012754A3 Tertiary and secondary amines as alpha-2 antagonists and serotonin uptake inhibitors
10/12/2000CA2369553A1 N-benzimidazolylmethyl and n-indolylmethyl-benzamides and their use as crf modulators
10/12/2000CA2369238A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
10/12/2000CA2368703A1 Substituted aniline compounds
10/12/2000CA2366850A1 Method for the treatment of neurological or neuropsychiatric disorders
10/12/2000CA2365503A1 Method for the preparation of tricyclic amino alcohol derivatives through azides
10/12/2000CA2360923A1 Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate
10/11/2000EP1043313A1 New acrylates and actinic radiation-curable compositions containing them
10/11/2000EP1043311A1 Biphenylamidine derivatives
10/11/2000EP1042329A1 Novel farnesyl transferase inhibitors, preparation, pharmaceutical, compositions containing them and use for preparing medicines
10/11/2000EP1042316A1 Indole derivatives useful a.o. for the treatment of osteoporosis
10/11/2000EP1042305A1 INHIBITION OF p38 KINASE USING SYMMETRICAL AND UNSYMMETRICAL DIPHENYL UREAS
10/11/2000EP1042289A1 Indole]naphthopyrans, preparation, compositions and (co)polymer matrices containing them, synthesis intermediates
10/11/2000EP1042288A1 Tripeptidyl peptidase inhibitors
10/11/2000EP1042287A1 Indole derivatives as inhibitors of factor xa
10/11/2000EP1042286A1 Gamma-glutamyl and beta-aspartyl containing immunomodulator compounds and methods therewith
10/11/2000EP1042285A1 iso-CBI AND iso-CI ANALOGS OF CC-1065 AND THE DUOCARMYCINS
10/11/2000EP1042279A1 Substituted beta-alanines
10/11/2000EP1042272A1 Derivatives of 2,2-dimethyl 3-(2-fluoro vinyl) cyclopropane carboxylic acid, their preparation process and their use as pesticides
10/11/2000CN1269775A Enantioselective reduction of ketones with silane agent/metal compound/chiral ligand system
10/10/2000US6130315 Substrates in which the scissile amide bond has been replaced by an activated electrophilic ketone moiety; antiinflammatory agents; antiproliferative/anticarcinogenic/antiarthritic agents; treatment of autoimmune diseases
10/10/2000US6130251 Use as agents for combating pests.
10/10/2000US6130241 Insect-repellent formulations
10/10/2000US6130240 Compound for treatment of cardiac arrhythmia, synthesis, and methods of use
10/10/2000US6130238 3-(cyclohexanoheteroarylidenyl)-2-indolinone protein tyrosine kinase inhibitors
10/10/2000US6130237 Condensed N-aclyindoles as antitumor agents
10/10/2000US6130235 Piperidine moieties coupled to indole, benzimidazole or benzotriazole.
10/10/2000US6130227 7-Substituted camptothecin derivatives and methods for inhibiting the growth of tumor cells therewith
10/05/2000WO2000058405A2 Squaraine dyes
10/05/2000WO2000058288A1 Pyridine-2,3-dicarboxylic acid diamides
10/05/2000WO2000058287A1 Novel method for manufacturing tricyclic amino alcohol derivatives
10/05/2000WO2000058286A2 Method of producing heterocyclic carbamates from aza-heterocyclic compounds and carbon dioxide
10/05/2000CA2368451A1 Pyridine-2,3-dicarboxylic acid diamides
10/05/2000CA2368448A1 Novel method for manufacturing tricyclic amino alcohol derivatives
10/05/2000CA2366263A1 Squaraine dyes
10/05/2000CA2361019A1 Process for the preparation of heterocyclic carbamates from aza-heterocycles and carbon dioxide
10/04/2000EP1040096A1 Neuroprotective agents
10/04/2000EP1039911A1 MORPHOLINO-N-ETHYL ESTER PRODRUGS OF INDOLE sPLA 2 INHIBITORS
10/04/2000CN1268509A Substituted phenyl heterocyclic compound weedicide
10/04/2000CN1268352A Method for preparing medicinal prepns. contg. 6-heterocycle-4-amino-1,3,4,5-tetrabenzo [cd] indole
10/04/2000CN1057085C Heterocyclically substituted phenyl-cyclohexane carboxylcic acid derivatives
10/04/2000CN1057083C Tricyclic 1-aminoethylpyrrol derivative
10/03/2000US6127544 1-substituted-3-ureido-indolin-2-ones which exhibit selective antagonism against gastrin receptors without causing side effects attributed to cck-a receptor antagonism; such as for treatment of peptic ulcers, gastritis
10/03/2000US6127542 Chemical intermediates to specified pyrazino(2',1':6,1)pyrido(3,4b)indole-1,4-diones which are selective inhibitors of cyclic guanosine 3',5'-monophosphate specific phosphodiesterase; to treat cardiovascular disorders
10/03/2000US6127539 N-phosphorylation or sulfonylation of 2-azabicyclo(2.2.1) hept-5-en-3-one in the presence of an organolithium compound and at a subzero temperature, then reacting with a purine base to yield the cyclopentenyl nucleoside
10/03/2000US6127404 Tissue selective compounds in the treatment of endometrial proliferation
10/03/2000US6127403 An enzyme inhibitor for treating arteriosclerotic lesions of arteriosclerosis, hyperlipemia and diabetes, as well as ischemic diseases of brain, heart
10/03/2000US6127373 Method of treating tourette's syndrome and obsessive compulsive disorder
10/03/2000US6127364 Anthelminthics, insecticides, acaricides, and nematicides.
10/03/2000US6126932 Insoluble polymer bearing pendant side chains, said side chains each terminating with the 1-(3-(1-pyrrolidinyl)-propyl)-3-ethylcarbodiimide moiety.
10/03/2000CA2177773C New aryl(alkyl)propylamides, process for preparing the same and pharmaceutical compositions containing them
09/2000
09/28/2000WO2000056711A1 Tricyclic indole-2-carboxylic acid compound used as nmda receptor antagonist
09/28/2000WO2000056710A1 3-(anilinomethylene) oxindoles as protein tyrosine kinase and protein serine/threonine kinase inhibitors
09/28/2000WO2000056709A1 Indolinone compounds as kinase inhibitors
09/28/2000WO2000056335A1 Methods for treating neurodegenerative disorders using aspartyl protease inhibitors
09/28/2000DE19913483A1 Verfahren zur Herstellung von Heterocyclischen Carbamaten aus Aza-Heterocyclen und Kohlendioxid Process for the preparation of heterocyclic carbamates from carbon dioxide and aza heterocycles
09/28/2000CA2368041A1 Indolinone compounds as kinase inhibitors
09/28/2000CA2367112A1 Methods for treating neurodegenerative disorders using aspartyl protease inhibitors
09/28/2000CA2362700A1 Tricyclic indole-2-carboxylic acid compound used as nmda receptor antagonist
09/27/2000EP1038873A2 Benzo(3,4)cyclobuta(1,2-c)pyrrole derivatives as inhibitors of serotonine reuptake
09/27/2000EP1038868A2 Sulfonamides as antiviral agents
09/27/2000EP1038863A2 Substituted dimeric compounds, process for their preparation and pharmaceutical compositions thereof
09/27/2000EP1037865A1 Synthesis of cc-1065/duocarmycin analogs
09/27/2000EP1037637A1 Use of 5ht1a receptor antagonists for preventing and/or treating temporal lobe epilepsy
09/27/2000EP1037630A2 Method for the treatment of disorders associated with apoptosis using n-heterocyclic glyoxylamide compounds
09/27/2000EP1037626A1 Multicatalytic protease inhibitors for use as anti-tumor agents
09/27/2000CN1268134A Bis-indole derivatives having antimetastatic activity, A process for their preparation and pharmaceutical compositions containing them
09/27/2000CN1268119A Process for preparing 4-substituted-1H-indole-3-glyoxamides
09/27/2000CN1056842C Amino acid derivative having anti CCK activity
09/27/2000CN1056828C Preparation process for esters of 2,2-dimethyl-3-[(2)-1-propenyl] cyclopropane carboxylic acid and intermediates thereof
09/26/2000US6124465 Farnesyl transferase inhibitors, their preparation, the pharmaceutical compositions which contain them and their use in the preparation of medicaments
09/26/2000US6124340 Polymorphic compounds