Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
11/1999
11/17/1999EP0572537B1 Cytokine inhibitors
11/17/1999CN1235280A Photographic element containing yellow dye-forming photographic coupler
11/17/1999CN1046510C Preparation of N-tert-butylamides
11/16/1999US5986106 Multistage reaction of halogenation, hydrolysis, decarboxylation, alkylation, amination, oxidation and oxidation, reaction of oxalyl chloride and ammonia
11/16/1999US5986105 Quinolone- and naphthyridonecarboxylic acid derivatives
11/16/1999US5985911 C-terminal ketone inhibitors of matrix metalloproteinases and TNFα secretion
11/16/1999US5985910 Estrogen agonists/antagonists useful for the treatment of diseases associated with estrogen deficiency
11/16/1999US5985909 Anticancer drugs used as prodrugs for antibody-directed enzyme-prodrug therapy (adept) and gene-directed enzyme-prodrug therapy (gdept) for cancer
11/16/1999US5985908 MCBI analogs of CC-1065 and the duocarmycins
11/16/1999US5985887 Aza-anthracyclinone derivatives
11/11/1999WO1999057117A2 Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
11/11/1999WO1999057100A1 Spla2 inhibitor compounds for treatment of disease
11/11/1999WO1999057098A2 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
11/11/1999WO1999056765A1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME
11/11/1999WO1999056752A1 sPLA2 INHIBITOR ESTER
11/11/1999WO1999056745A1 New use
11/11/1999WO1999042457A3 Substituted alxoxycarbonyl compounds
11/11/1999DE19838506A1 Indolderivate und deren Verwendung zur Behandlung von malignen und anderen, auf pathologischen Zellproliferationen beruhenden Erkrankungen The indole derivatives and their use for the treatment of malignant and other diseases based on pathological cell proliferations
11/11/1999CA2496859A1 Indole derivatives and their use for the treatment of malignant and other diseases based on pathological cell proliferation
11/11/1999CA2331070A1 New use
11/11/1999CA2331036A1 Spla2 inhibitor ester
11/11/1999CA2330856A1 Spla2 inhibitor compounds for treatment of disease
11/11/1999CA2329704A1 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
11/11/1999CA2327507A1 Succinamide inhibitors of interleukin-1.beta. converting enzyme
11/10/1999EP0863873B1 Indole carbamates as leukotriene antagonists
11/10/1999CN1234792A Nitric ester derivatives and use in treatment of urinary incontinence and other diseases
11/10/1999CN1046283C Process for preparation of 9-amino camptothecin
11/10/1999CN1046269C HIV protease inhibitors
11/10/1999CN1046268C Dihydro-indolin-2-one derivative
11/09/1999US5981762 Substituted indole-2-carboxylic acids as glucosyl transferase inhibitors
11/09/1999US5981755 Tachykinin antagonists
11/09/1999US5981752 Tricyclic compounds having fungicidal activity, their preparation and their use
11/09/1999US5981584 Useful in the manufacture of a medicament for inhibiting the aggregation of blood platelets, inhibiting angiogenesis, inhibiting osteoclast mediated bone resorption, preventing platelet thrombosis
11/09/1999US5981580 Fatty acid analogs and prodrugs
11/09/1999US5981569 Substituted phenylacrylonitrile compounds and compositions thereof for the treatment of disease
11/09/1999US5981538 Skin disorders
11/09/1999US5981525 Indole derivatives useful in the treatment of osteoporosis
11/09/1999US5981513 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
11/09/1999US5981467 Containing quatenary nitrogen unit
11/09/1999US5981435 Methods for controlling algae
11/09/1999CA2177780C New arylalkyl(thio)carboxamide compounds, their preparation processes and the pharmaceutical compositions that contain them
11/09/1999CA2106452C Amidinophenol derivatives
11/04/1999WO1999055696A1 New hydroxyindoles, their use as phosphodiesterase 4 inhibitors and method for producing same
11/04/1999WO1999055694A1 Indolyl derivatives as serotonergic agents
11/04/1999WO1999055688A1 Substituted diarylalkyl amides as calcium channel antagonists
11/04/1999WO1999055673A1 Arylphenyl-substituted cyclic keto enols
11/04/1999WO1999055672A2 Antipsychotic indolyl derivatives
11/04/1999WO1999055330A1 Ccr-3 receptor antagonists
11/04/1999DE19818964A1 New hydroxy-indole derivatives useful in treatment of degenerative joint disease, viral and parasitic infections, bronchial, dermatological, neurodegenerative and prostate disorders, etc.
11/04/1999CA2330452A1 Antipsychotic indolyl derivatives
11/04/1999CA2330436A1 Indolyl derivatives as serotonergic agents
11/04/1999CA2329821A1 Ccr-3 receptor antagonists
11/03/1999EP0953871A1 Photographic element containing yellow dye-forming photographic coupler
11/03/1999EP0953567A2 Bicyclic substituted piperazine-, piperidine- and tetrahydropyridine derivatives, their preparation and their use as agents with central dopaminergic (dopamine D4 receptor) activity
11/03/1999EP0952978A1 Metallocenes and catalysts for olefin-polymerisation
11/03/1999EP0834074B1 Detection of transmembrane potentials by optical methods
11/03/1999EP0650599B1 Method of colorimetric analysis of malonic dialdehyde and 4-hydroxy-2-enaldehydes as indexes of lipid peroxidation, kits for carrying out said method, substituted indoles for use in said method and their preparation
11/03/1999CN1234024A 4-aminoethoxy indolone derivatives
11/03/1999CN1234023A 4-aminoethoxy indoes as dopamin D2 agonists and as 5HT1A ligands
11/03/1999CN1234020A Amide derivatives and their use as pesticides
11/02/1999US5977379 Process for the preparation of flame-resistant halogenated imide compounds
11/02/1999US5977365 Heterocyclic compound having anti-diabetic activity
11/02/1999US5977361 Transition metal-catalyzed process for preparing N-aryl compounds
11/02/1999US5977359 Substituted heterocyclic compounds, method of preparing them and pharmaceutical compositions in which they are present
11/02/1999US5977154 Obesity, diabetes
11/02/1999US5977137 Sulfonamide inhibitors of aspartyl protease
11/02/1999US5977130 Intimal hypertrophy inhibitors
11/02/1999US5977125 Mono-or polyenic carboxylic acid derivatives
11/02/1999US5977108 Leukemia
10/1999
10/28/1999WO1999054303A1 Optically active tetrahydrobenzindole derivatives
10/28/1999WO1999054302A1 Process for the production of r-(+)-6- carboxamido- 3-n- methylamino- 1,2,3,4- tetrahydrocarbazole
10/28/1999WO1999054301A1 Substituted 2-oxo-alkanoic acid-[2-(indol-3-yl)-ethyl] amides
10/28/1999WO1999054300A1 Process for preparing 4-substituted-1h-indole-3-glyoxamides
10/28/1999WO1999054295A1 Process for preparing 4-hydroxy indole, indazole and carbazole compounds
10/28/1999WO1999047497A3 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
10/28/1999WO1999043654A3 Inhibitors of phospholipase enzymes
10/28/1999WO1999024460B1 Dipeptide nitriles
10/28/1999DE19818732A1 New aryl substituted cyclic ketoenol compounds useful for control of insects and as herbicides
10/28/1999DE19808261A1 Arylphenylsubstituierte cyclische Ketoenole Arylphenylsubstituierte cyclic ketoenols
10/28/1999CA2329319A1 Optically active tetrahydrobenzindole derivatives
10/28/1999CA2328875A1 Substituted 2-oxo-alkanoic acid-[2-(indol-3-yl)-ethyl] amides
10/28/1999CA2326515A1 Process for preparing 4-substituted-1h-indole-3-glyoxamides
10/28/1999CA2326505A1 Process for preparing 4-hydroxy indole, indazole and carbazole compounds
10/27/1999EP0952154A2 N-acyl and N-aroyl aralkyl amides
10/27/1999EP0952149A2 Substituted carbazoles, process for their preparation and their use as sPLA2 inhibitiors
10/27/1999EP0951842A2 Infant formula
10/27/1999EP0584088B1 Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
10/27/1999CN1233250A Process for the preparation of N-[cl-nButyl-4-piperidyl) methyl-3,4-dihydro-2h-[1,3] oxazino [3,2-a] indole-10-carboxamide and salts and intermediates in the process
10/27/1999CN1233248A 1H-pyrido [3,4-b] indole-4-carboxamide derivatives, preparation and application thereof in therapeutics
10/27/1999CN1233245A Oxadiazoles, processes for their preparation and their use as medicaments
10/27/1999CN1233239A Process for preparing 2-azadihydroxybicyclo [2,2,1] heptane compounds and the L-tartaric acid salt of the compound
10/27/1999CN1233238A Acylaminoalkenylene-amide derivatives as NK1 and NK2 antagonists
10/27/1999CN1233180A Treatment of the common cold or allergic rhinitis
10/27/1999CN1233176A Substituted tricyclics
10/27/1999CN1233150A Method for inhibiting the expression of FAS
10/26/1999USRE36359 Long chain carboxylic acid imide ester
10/26/1999US5973165 Process for preparing 2-oxindole
10/26/1999US5973075 Methods for preparing rigid-rod macromonomers with reactive end groups
10/26/1999US5972982 Containing 5-to 9-membered heteroaryl mono- or bicyclic ring system having no more than 1 carbonyl carbon in the ring system; viricides, bactericides
10/26/1999US5972964 Aminomethylindans, -benzofurans and -benzothiophenes