Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
10/1999
10/05/1999US5962658 (3-oxoisoindolin-1-ylidine)propandinitrile derivatives and method for preparing the same
10/05/1999US5962502 Polyamidic acid derivatives with antigastrin activity, a method for their preparation, and their pharmaceutical use
10/05/1999US5962501 Headaches
10/05/1999US5962498 Protein kinase C modulators. C. indolactam structural-types with anti-inflammatory activity
10/05/1999US5962473 Methods of treating or ameliorating the symptoms of common cold or allergic rhinitis with serotonin 5-HT1F
10/05/1999US5962470 Heterocyclic compounds having anti-diabetic activity and their use
10/05/1999US5962469 Cyclic nitrones
10/05/1999US5962465 Brain disorders; psychological disorders
10/05/1999CA2175204C Certain fused pyrrolecarboxanilides; a new class of gaba brain receptor ligands
09/1999
09/30/1999WO1999048869A1 Aryl phenyl substituted cyclic ketoenols
09/30/1999WO1999048868A2 Heterocyclic classes of compounds for the modulating tyrosine protein kinase
09/30/1999WO1999048522A1 Pharmaceutical composition containing a cysteine protease inhibitor for prophylaxis and therapy of brain tissue impairment
09/30/1999WO1999006340A3 Sulfonylamino substituted hydroxamic acid derivatives as metalloprotease inhibitors
09/30/1999DE19813354A1 Arylphenylsubstituierte cyclische Ketoenole Arylphenylsubstituierte cyclic ketoenols
09/30/1999CA2325935A1 Heterocyclic families of compounds for the modulation of tyrosine protein kinase
09/30/1999CA2324566A1 Pharmaceutical composition containing a cysteine protease inhibitor for prophylaxis and therapy of brain tissue impairment
09/30/1999CA2236827A1 Methods of identifying antagonists of glycosaminoglycan-protein interactions
09/29/1999EP0944601A1 Guanidinylamino heterocycle compounds useful as alpha-2 adrenoceptor agonists
09/29/1999EP0944597A1 Metalloproteinase inhibitors
09/29/1999EP0944596A1 Seco precursors of cyclopropylindolines and their use as prodrugs
09/29/1999EP0944595A1 5-cyclo indole compounds as 5-ht1d receptor ligands
09/29/1999EP0944590A2 Aminoguanidines and alkoxyguanidines as protease inhibitors
09/29/1999EP0944584A1 Benzamidoaldehydes and their use as cysteine protease inhibitors
09/29/1999EP0944583A1 Novel compounds useful as therapeutic agents and assay reagents
09/29/1999EP0944581A1 Process of preparing substituted acrylamides
09/29/1999EP0944580A2 N-(aryl/heteroaryl) amino acid esters, pharmaceutical compositions, and methods for inhibiting beta-amyloid peptide release and/or its synthesis
09/29/1999EP0553107B1 Protein kinase c modulators with anti-inflammatory and antiviral activity
09/29/1999CN1230187A Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
09/29/1999CN1230110A Cell adhesion inhibitors
09/29/1999CN1045294C Method for prepn. of indole derivatives
09/28/1999US5959146 Tricyclic compounds
09/28/1999US5958965 4-aminoethoxy indoles
09/28/1999US5958839 Herbicidal compounds
09/28/1999US5958838 Controlling weeds in crops.
09/28/1999US5958683 Screening method using the RZR receptor family
09/28/1999CA2181351C Process and intermediates for preparing naphthyridonecarboxylic acid salts
09/23/1999WO1999047525A1 Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
09/23/1999WO1999047508A1 Benzenesulfonamide-derivatives and their use as medicaments
09/23/1999WO1999047497A2 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
09/23/1999WO1999047490A1 Bicyclo[2.2.1]heptanes and related compounds
09/23/1999CA2323783A1 Benzenesulfonamide-derivatives and their use as medicaments
09/23/1999CA2322742A1 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
09/22/1999EP0942902A2 Novel immunotherapeutic imides/amides
09/22/1999EP0942756A2 Optical diagnostic agents for diagnosis of neurodegenerative diseases by means of near infra-red radiation (nir radiation)
09/22/1999EP0942728A1 Use of nk-1 receptor antagonists for treating sexual dysfunction
09/22/1999CN1229082A Amine compound and its acid addition salt
09/21/1999US5955501 Derived from phorboids of the diterpene- and benzolactam-classes.
09/21/1999US5955492 Carboxylic acid indole inhibitors of chemokines
09/21/1999US5955491 Method for treating osteoporosis
09/21/1999US5955487 Treating high blood pressure, cardiac insufficiency, glaucoma
09/21/1999US5955462 Antiinflammatory agents for neurogenic inflammation and administering bisindole or compounds
09/21/1999US5955435 Peptidyl compounds having MMP and TNF inhibitory activity
09/21/1999US5955421 Peptides containing D-2-alkyl-Tryptophan
09/16/1999WO1999046268A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
09/16/1999WO1999046267A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999046244A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999046237A1 Modulators of protein tyrosine phosphatases
09/16/1999WO1999046236A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999045968A1 Manganese chelates with high relaxivity in serum
09/16/1999WO1999045967A1 Manganese chelates with high relaxivity in serum
09/16/1999WO1999028304A9 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
09/16/1999CA2323493A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999CA2323472A1 Modulators of protein tyrosine phosphatases
09/15/1999EP0941215A1 Glyoxylic acid amides and their use as pesticides
09/15/1999EP0759899B1 Nitro compounds and their compositions having anti-inflammatory, analgesic and anti-thrombotic acitivities
09/15/1999CN1228779A Spirocyclic metalloprotease inhibitors
09/15/1999CN1228768A Insect-repellent formulation
09/15/1999CN1228423A Process for preparation of optically active indoline-2-carboxylic acid or derivative thereof
09/15/1999CN1228422A Process for preparing naphthyridones and intermediates
09/15/1999CN1045101C Anilines as markers for mineral oils
09/14/1999US5952527 A complex of transitional metal compound, cyclooctadiene or cyclopentadiene and 2,2-bis/diphenylphosphinoamino/-5,5',6,6'7,7',8,8'-octahydro-1 ,1'-binaphthyl compound; used as hydrogenation catalyst
09/14/1999US5952511 Indolin-2-one derivatives
09/14/1999US5952497 N.sup.α -Bpoc amino acid pentafluorophenyl (Pfp) esters and 3,4-dihydro-4-oxo-1,2,3-benzotriazin-3-yl (ODhbt) esters
09/14/1999US5952386 Excellent insecticidal activity for the control of noxious insects
09/14/1999US5952377 Fatty acid analogs and prodrugs
09/14/1999US5952365 2- 2-(Dimethylamino)ethyl!-8,8-dipropyl-2-azaspiro 4.5!decane dimaleate
09/14/1999US5952362 2-imidazoline, 2-oxazoline, 2-thiazoline, and 4-imidazole derivatives of methylphenyl, methoxyphenyl, and aminophenyl alkylsulfonamides and ureas and their use
09/14/1999US5952355 Propenone derivatives
09/14/1999US5952343 HIV protease inhibitors
09/14/1999US5952322 Method of reducing tissue damage associated with non-cardiac ischemia using glycogen phosphorylase inhibitors
09/14/1999CA2006356C Arylpiperazinylbutyl-dihydroindoles and related compounds
09/14/1999CA1340734C Substituted bridged-diazabicycloalkyl quinolone carboxylic acids
09/10/1999WO1999044989A1 Matrix metalloproteinase inhibitors
09/10/1999WO1999044987A1 NON-PEPTIDE GnRH AGENTS
09/10/1999WO1999044624A2 Pharmaceutical composition for prophylaxis and therapy of diseases associated with ocular fundus tissue cytopathy
09/10/1999WO1999044613A1 Pharmaceutical compositions containing in combination two antagonists selective of arginine-vassopressin v receptors, even of v1a and v2 receptors
09/10/1999WO1999044608A1 New use
09/10/1999CA2322854A1 Pharmaceutical composition for prophylaxis and therapy of diseases associated with ocular fundus tissue cytopathy
09/10/1999CA2322444A1 Non-peptide gnrh agents
09/10/1999CA2320757A1 New use
09/10/1999CA2317502A1 Matrix metalloproteinase inhibitors
09/08/1999EP0940139A2 Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
09/08/1999EP0939627A1 Pentafluorobenzenesulfonamides and analogs
09/08/1999CN1228094A Palladium catalyzed indolization
09/07/1999US5948816 Non-tolerance-inducing antiviral agents
09/07/1999US5948808 Indole-3-carbinol, diindolylmethane and substituted analogs as antiestrogens
09/07/1999US5948807 Spiroindanamines and Spiroindanimides
09/07/1999US5948780 Administering a metalloproteinase inhibitor
09/07/1999US5948600 Method and material for the formation of a heat mode image
09/07/1999US5948593 Optical recording medium