Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
09/2000
09/05/2000US6114372 Matrix metalloproteinase (mmp); tumor necrosis factor(tnf); compounds such as n2-((2s)-acetylmercapto)acetyl-5-phthalimidopentanoyl)-n1-((4 -methoxybenzene)sulphonyl)-n1-(phenylmethyl)hydrazine
09/05/2000US6114371 3-(cyclohexanoheteroarylidenyl)-2-indolinone protein tyrosine kinase inhibitors
09/05/2000US6114360 Pyrrole compounds
09/05/2000US6114350 Cyanine dyes and synthesis methods thereof
09/05/2000US6114175 Amyloid-binding compounds which are non-azo derivatives of chrysamine g to determine degree of brain deposits quantitatively characterized by amyloidosis; down's syndrome; prevent cell degeneration; radioactive imaging
08/2000
08/31/2000WO2000050408A1 Pyridazin-3-one derivatives and medicines containing the same
08/31/2000WO2000050395A1 Sulfonamide-containing indole compounds
08/31/2000WO2000050389A1 Efficient carbamate synthesis
08/31/2000WO2000050377A1 Efficient synthesis of secondary amines by selective alkylation of primary amines
08/31/2000WO2000050376A2 Efficient synthesis of alkyl carbonates
08/31/2000DE19908699A1 Preparation of 2-aryl-1,3-ketoenol compounds, which may be useful as insecticides, by reaction of ketene compound with ketone, thioketone or imine
08/30/2000EP1031569A1 Processes for producing 7-isoindolinequinolonecarboxylic derivatives and intermediates therefor, salts of 7-isoindolinequinolonecarboxylic acids, hydrates thereof, and composition containing the same as active ingredient
08/30/2000EP1030844A1 Compounds which inhibit tryptase activity
08/30/2000EP1030843A1 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000EP1030838A1 Method of synthesis of pyrrole amides
08/30/2000EP1030661A1 N,N-DIETHYLGLYCOLAMIDO ESTER PRODRUGS OF INDOLE sPLA 2? INHIBITORS
08/30/2000EP0690843B1 Formyl- or cyano- substituted indole derivatives having dopaminergic activity
08/30/2000CN1265108A 4-oxo-3,5-dihydro-4H-pyridazino [4,5-b]-indole-1-acetamide derivatives, their prepn. and their application in therapy
08/30/2000CN1265096A Hydrazine derivatives
08/29/2000US6111116 Dibenzorhodamine dyes
08/29/2000US6110958 Pyrrole compounds having parasiticidal properties
08/29/2000US6110957 Antitumor agent treating cell proliferative disorders such as cancer, dyes, fungicides, bactericides
08/29/2000US6110956 N-aryloxyethylamine derivatives for the treatment of depression
08/29/2000US6110934 Substituted benzamide derivatives and their use as anticonvulsants
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/29/2000US6110917 Selective serotonin (5-ht) receptor agonist for treating migraines, vasospasms
08/29/2000US6110872 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides
08/24/2000WO2000049080A1 Photo curable liquid resin composition and photofabricated cured product
08/24/2000WO2000048993A1 Arylaminoalkylamides
08/24/2000WO2000048606A1 Compositions and methods for use in targeting vascular destruction
08/24/2000WO2000002887B1 Ligands for metals and metal-catalyzed processes
08/23/2000EP1029909A1 Organic electroluminescence device and phenylenediamine derivative
08/23/2000EP1029861A1 Benzisothiazol-piperazinyl derivative and its use as neuroleptic
08/23/2000EP1029541A1 Therapeutic or prophylactic agent for glomerulopathy
08/23/2000EP1029297A2 Method of virtual retrieval of analogs of lead compounds
08/23/2000EP1028942A2 Dipeptide nitriles
08/23/2000EP1028940A1 Process to produce oxazolidinones
08/23/2000EP1028725A1 Application of vasopressin antagonists for treating disturbances or illnesses of the inner ear
08/23/2000EP1028716A1 Method for treating and preventing heart failure and ventricular dilatation
08/23/2000EP0844873A4 Carotenoid-nicotinamide-zinc compositions and methods of treatment using same
08/23/2000EP0658159B1 Arylidene and heteroarylidene oxindole derivatives as tyrosine kinase inhibitors
08/23/2000CN1264366A Thermodynamically stable modification of 1-(4-carbazolyloxy)-3-[2-(2-methoxyphenoxy) ethylamino]-2-propanole, process for its preparation and pharmaceutical compositions containing it
08/23/2000CN1264365A 3-benzoylindole derivatives and drugs containing the same
08/23/2000CN1264300A Arylsubstituted piperazines useful in the threatement of bening prostatic hyperlasia
08/22/2000USRE36832 N-heteroaryl-N'-phenylurea derivatives, their production and use
08/22/2000US6107519 Amido-substituted secondary alcohol intermediates and preparation thereof
08/22/2000US6107329 Hypotensive agents; cardiovascular disorders
08/22/2000US6107292 Indenoindoles and benzocarbazoles as estrogenic agents
08/22/2000US6107066 Coumarin derivative-n-linked lipid used as a fluorophore capable of undergoing energy transfer
08/17/2000WO2000047212A1 Quinazoline derivatives as angiogenesis inhibitors
08/17/2000WO2000027819A3 Antrhranilic acid amides and the use thereof as medicaments
08/16/2000EP1027332A1 Novel lactam metalloprotease inhibitors
08/16/2000EP1027056A1 Alpha-ketoamide multicatalytic protease inhibitors
08/16/2000EP1027046A1 Antagonists of gonadotropin releasing hormone
08/16/2000CN1263092A Carboxylic compound and its preparation method and application
08/15/2000US6103937 Producing unsaturated nitrogen containing compounds such as enamides, enamines and aryl amineslamides using as catalyst nickel and an organophosphine or carbene ligand
08/15/2000US6103905 Quinoline-indole antimicrobial agents, uses and compositions related thereto
08/15/2000US6103761 Agents acting at cholecystokinin receptors
08/15/2000US6103752 Therapeutic heterocyclic compounds
08/10/2000WO2000046199A2 Indole derivatives as anti-inflammation agents
08/10/2000WO2000046198A1 Anti-inflammatory indole derivatives
08/10/2000WO2000046197A1 Indole derivatives and their use as mcp-1 receptor antagonists
08/10/2000WO2000046196A1 Indole derivatives and their use as mcp-1 antagonists
08/10/2000WO2000046195A1 Anti-inflammatory indole derivatives
08/10/2000WO2000046184A1 N2-phenylamidine derivatives
08/10/2000WO2000015206A3 Tryptophanyl ester and their n-acyl derivatives for the prevention and treatment of diseases caused or exacerbated by oxidation processes
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/10/2000CA2357013A1 Anti-inflammatory indole derivatives
08/10/2000CA2356898A1 Indole derivatives and their use as mcp-1 antagonists
08/10/2000CA2355734A1 Indole derivatives as anti-inflammation agents
08/09/2000EP1026149A1 Amidocarboxylic acid derivatives
08/09/2000EP1025099A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants
08/09/2000EP1025077A1 Novel aryloxy-alkyl-dialkylamines
08/09/2000EP1024697A1 Method for treating alzheimer's disease
08/09/2000EP0734384B1 3-substituted 1-arylindole compounds
08/09/2000CN1262272A HIV proteinase inhibitor
08/08/2000US6100420 Heterocyclylbenzonitriles
08/08/2000US6100404 Erythromycin compounds
08/08/2000US6100398 Transition metal-catalyzed process for preparing N-aryl amine compounds
08/08/2000US6100397 Process for the preparation of N-[(1-n butyl-4-piperidyl)methyl]-3,4-dihydro-2H-[1,3]oxazino[3,2-a] indole-10-carboxamide and salts and intermediates in the process
08/08/2000CA2177743C New alkoxy-aryl compounds, process for preparing the same and pharmaceutical compositions containing them
08/03/2000WO2000044731A1 Novel hydroxyamidino carboxylate derivatives useful as nitric oxide synthase inhibitors
08/03/2000WO2000044722A1 Chondrongenesis promotors and indolin-2-one derivatives
08/03/2000WO2000044721A1 3,7-disubstituted indole derivatives and medicinal compositions containing the same
08/03/2000WO2000044717A2 Synthesis of oligoketides
08/03/2000WO2000044713A1 Alkynyl containing hydroxamic acid compounds as tace inhibitors
08/03/2000WO2000044709A2 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
08/03/2000WO2000044705A1 Synthesis method of nitroxymethylphenyl esters of aspirin derivatives
08/03/2000WO2000044373A1 Antibacterial hydroxamic acid derivatives
08/03/2000WO2000003975A3 Aryl vinyl ether derivatives and their use as herbicides
08/03/2000DE19903126A1 New sulphur substituted sulphonylaminocarboxylic acid N-arylamide derivatives used for treating e.g. cardiovascular diseases and atherosclerosis
08/03/2000CA2361454A1 Synthesis method of nitroxymethylphenyl esters of aspirin derivatives
08/03/2000CA2361040A1 Synthesis of oligoketides
08/03/2000CA2356346A1 Alkynyl containing hydroxamic acid compounds as tace inhibitors
08/03/2000CA2356299A1 Acetylenic .alpha.-amino acid-based sulfonamide hydroxamic acid tace inhibitors
08/02/2000EP1024134A1 Aminobutanoic acid derivatives
08/02/2000EP1023898A1 Cyano-indoles as serotonine reuptake inhibitors and as 5-HT2c receptor ligands
08/02/2000EP1023295A1 Fibrinogen receptor antagonist prodrugs
08/02/2000CN1261906A Alkyl, alkenyl and alkynyl chrysamine G derivatives for the antemortem diagnosis of alzheimer's disease and in vivo imaging and prevention of amyloid deposition