Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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11/26/2002 | US6486173 Serotonin-7 (5-ht7); treatment of central nervous system disorders such as sleep disorders, depression and schizophrenia; for example 1,3-dihydro-2-((4-(4-fluorophenyl)-4-oxobutyl))isoindole |
11/26/2002 | US6486165 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
11/26/2002 | US6486153 Phenylindole derivatives as 5-HT2A receptor ligands |
11/26/2002 | CA2222312C Dye compositions for keratinic fibres containing n-subsituted 4-hydroxyindole derivatives, new derivatives, method for synthesis, their use in dyeing, and dyeing method |
11/21/2002 | WO2002092568A1 5-cyano-1h-indole derivatives as antagonists of the interleukine-8 receptors |
11/21/2002 | WO2002092567A1 Novel 5-phenyl-1h-indole derivatives as antagonists of interleukine-8 receptors |
11/21/2002 | WO2002092565A2 3-aminoalkyl-2-aryl-indole derivatives and their use as gnrh antagonists |
11/21/2002 | WO2002092564A2 Synthesis of cyclopentadiene derivatives |
11/21/2002 | WO2002092078A1 Oral controlled release pharmaceutical composition for one-a-day therapy for the treatment and prophylaxis of cardiac and circulatory diseases |
11/21/2002 | WO2002074309A3 Use of tryptophan derivatives for the specific cytostatic treatment of serotonin-producing tumors |
11/21/2002 | WO2002066426A3 Fluoro oxindole derivatives as modulators of kcnq potassium channels |
11/21/2002 | WO2002062290A3 Heterocyclic substituted 2-methyl-benzimidazole antiviral agents |
11/21/2002 | WO2002060340A9 Method for identifying maxi-k channel blockers |
11/21/2002 | US20020173659 Indole derivatives for the treatment of osteoporosis |
11/21/2002 | US20020173531 Central nervous system disorders; psychological disorders |
11/21/2002 | US20020173529 Fungicide active substance combinations |
11/21/2002 | US20020173527 Tumor necrosis factor antagonist; antiinflammatory agents |
11/21/2002 | US20020173518 Anticoagulant in mammls |
11/21/2002 | US20020173495 Selective androgen receptor modulators and methods of use thereof |
11/21/2002 | US20020173494 Ammonium salts of inositol hexaphosphate, and uses thereof |
11/21/2002 | US20020172885 For increasing sensitivity of photoresist useful for microfabrication of integrated circuits utilizing deep ultraviolet rays (from excimer lasers) and x-rays; resolution; profile |
11/21/2002 | CA2447305A1 Novel 5-phenyl-1h-indole derivatives as antagonists of interleukine-8 receptors |
11/21/2002 | CA2447184A1 5-cyano-1h-indole derivatives as antagonists of the interleukine-8 receptors |
11/21/2002 | CA2447005A1 Oral controlled release pharmaceutical composition for one-a-day therapy for the treatment and prophylaxis of cardiac and circulatory diseases |
11/20/2002 | EP1258252A1 Integrin expression inhibitors |
11/20/2002 | EP1257544A2 Piperazine and piperidine derivatives for treatment or prevention of neuronal damage |
11/20/2002 | EP1042285A4 iso-CBI AND iso-CI ANALOGS OF CC-1065 AND THE DUOCARMYCINS |
11/20/2002 | EP0925302B1 Palladium catalyzed indolization |
11/20/2002 | EP0892780B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS |
11/20/2002 | CN1380880A Process for producing substituted aromatic compound |
11/20/2002 | CN1380838A Method of separating imide compound |
11/20/2002 | CN1380287A 2-acryl-3-substituted indoacetamide derivative and its medical application |
11/19/2002 | US6482957 Useful as an intermediate of a carbocyclic nucleoside anti-viral agent; reacting 2-azabicyclo(2.2.1)hept-5-en-3-one with a sulfonyl halide or phosphoryl halide and then with a nucleic acid base |
11/19/2002 | US6482951 Isoindolin-1-one glucokinase activators |
11/19/2002 | US6482860 Pentafluorobenzenesulfonamides and analogs |
11/19/2002 | US6482849 Inhibitors of α4β1 mediated cell adhesion |
11/19/2002 | US6482846 Compositions and methods to prevent toxicity induced by nonsteroidal antiinflammatory drugs |
11/19/2002 | US6482835 Such as (r)-1-cyclopropyl-8-difluoromethoxy-7-(1-methyl-2,3-dihydro-1h-5-isoindolyl)-4-oxo-1,4-dihydro-3-quinolinecarboxyl ic acid methanesulfonate; chemical intermediates; bactericides; catalysis |
11/19/2002 | US6482832 Heterocyclically substituted amides, their production and their use |
11/19/2002 | CA2115143C Macromonomers having reactive end groups |
11/14/2002 | WO2002090347A1 Amide compounds |
11/14/2002 | WO2002090330A1 Substituted 2-pyridine-cyclohexane-1,4-diamine derivatives |
11/14/2002 | WO2002090327A1 Piperazinyl-isatins |
11/14/2002 | WO2002090319A1 Labelling reagents, method for synthesis of said reagents and methods for detecting biological molecules |
11/14/2002 | WO2002090317A1 Substituted cyclohexane-1,4-diamine derivatives |
11/14/2002 | WO2002090313A1 Aloe-emodin derivatives and their use in the treatment of neoplastic pathologies |
11/14/2002 | WO2002089783A1 Substituted cyclohexan-1,4-diamine derivatives with constipating and peripheral analgesic properties |
11/14/2002 | WO2002074764A3 Piperazine derivatives and their use as 5-ht1b ligands |
11/14/2002 | WO2002060339A3 Ophthalmic compositions for treating ocular hypertension |
11/14/2002 | WO2001097787A3 Use of microsomal triglyceride transfer protein (mtp) inhibitors for reducing the number of postprandial triglyceride-rich lipoprotein particles (pptrl) |
11/14/2002 | WO2001020995A9 Compounds directed against pilus biogenesis and activity in pathogenic bacteria; methods and compositions for synthesis thereof |
11/14/2002 | US20020169331 Method of separating imide compound |
11/14/2002 | US20020169326 Fatty acid derivatives |
11/14/2002 | US20020169322 Use of N-alkylamino-heterocylic compounds for the treatment of migraine |
11/14/2002 | US20020169200 Antitumor, antiinflammatory and antiarthritic agents, treating metastasis, restenosis, osteoporosis, inflammation, macular degeneration, and diabetic retinopathy |
11/14/2002 | US20020169198 Agonists of the progesterone receptor; contraceptives, hormone replacement therapy and treating menopause symptoms |
11/14/2002 | US20020169164 Tricyclic sulfonamides and their derivatives as inhibitors of matrix metalloproteinases |
11/14/2002 | US20020169157 An aromatic or heteroaromatic amino acid derivative, used for treating disorders related to overexpression of protein tyrosine phosphatase-1B |
11/14/2002 | US20020166180 For oxidative coloring agent for keratin fibers |
11/14/2002 | CA2446735A1 Substituted cyclohexane-1,4-diamine derivatives with an anti-diarrhoea and peripheral analgesic action |
11/13/2002 | EP1256576A1 Fused imidazolium derivatives |
11/13/2002 | EP1256574A1 Nitrogen-containing compounds having kinase inhibitory activity and drugs containing the same |
11/13/2002 | EP1255757A1 Amino acid derivatives and use thereof as nep, ace and ece inhibitors |
11/13/2002 | EP1255752A2 Pyrrole substituted 2-indolinone protein kinase inhibitors |
11/13/2002 | EP1255751A2 1,3-dihydro-2h-indol-2-one derivatives and their use as ligands for v1b or v1b and v1a arginine-vasopressin receptors |
11/13/2002 | EP1255734A1 Isatine derivatives with neurotrophic activity |
11/13/2002 | EP1255726A2 (r)-2-aryl-propionamides, useful in the inhibition of il-8 induced chemiotaxis of neutrophils |
11/13/2002 | EP1255542A1 Substituted amino acids as neutral sphingomyelinase inhibitors |
11/13/2002 | EP1255536A2 Indolinone derivatives for modulation of c-kit tyrosine protein kinase |
11/13/2002 | EP1112272B1 Muscarinic agonists and antagonists |
11/13/2002 | EP1068199B1 N-aryloxyethyl-indoly-alkylamines for the treatment of depression |
11/13/2002 | EP0843672B1 One pot synthesis of 2-oxazolidinone derivatives |
11/13/2002 | EP0760658B1 Compounds for inhibiting osteoclast-mediated bone resorption |
11/13/2002 | CN1379774A Compounds |
11/13/2002 | CN1379772A Substituted indoles for modulating NFKB activity |
11/13/2002 | CN1379761A Condensed indoline derivatives and their use as 5HT, in particular 5HT2C receptor ligands |
11/13/2002 | CN1379755A Substituted 2-dialkylamino alkylbiphenyl derivatives |
11/13/2002 | CN1379024A Process for preparing 5-phenylformyl-3-methyl-2-indolone |
11/12/2002 | US6479552 Use of substituted N, N-disubstituted diamino compounds for inhibiting cholesteryl ester transfer protein activity |
11/12/2002 | US6479534 Indoline derivatives and method of treating obesity |
11/12/2002 | US6479528 Methods for inhibiting or reversing tau filament formation polymerization |
11/12/2002 | US6479524 To prolong the thrombin time |
11/12/2002 | US6479503 Cycloalkano-indole and -azaindole derivatives |
11/12/2002 | US6479480 1h-indole derivatives bearing an optionally substituted phenyl moiety at the 2-position of the indole ring system and a methylene-linked heterocyclic moiety at the 3-position of the indole ring system; schizophrenia treatment |
11/12/2002 | US6479123 Dipyrromethene-metal chelate compound and optical recording medium using thereof |
11/12/2002 | CA2324959C Phthalimido compounds as intermediates for producing substance p receptor antagonists |
11/07/2002 | WO2002088274A1 Double-spiro organic compounds and electroluminescent devices |
11/07/2002 | WO2002088114A2 Heteroaryl ofefinic azacyclic and heteroaryl acetylenic azacyclic compounds for the treatment of cns disorders |
11/07/2002 | WO2002088094A1 2-iminoimidazole derivatives (1) |
11/07/2002 | WO2002088092A1 2-iminoimidazole derivative (2) |
11/07/2002 | WO2002088083A1 Process for producing tetrahydrocarbazole derivative |
11/07/2002 | WO2002088073A1 Anthranilic acid amides, method for the production thereof, their use as antiarrhythmia agents, and pharmaceutical preparations thereof |
11/07/2002 | WO2002064546A3 Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical |
11/07/2002 | WO2001085687A1 Substituted indoles as parp inhibitors |
11/07/2002 | US20020165412 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof |
11/07/2002 | US20020165402 Quarternary ammonium compounds |
11/07/2002 | US20020165398 Amino-thiophene-amido derivatives |
11/07/2002 | US20020165394 Inhibition of RAF kinase using quinolyl, isoquinolyl or pyridyl ureas |
11/07/2002 | US20020165343 Growth hormone secretagogues |
11/07/2002 | US20020165275 Trisubstituted carbocyclic cyclophilin binding compounds and their use |