Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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04/02/2003 | EP1296931A2 Polyamine analogues as cytotoxic agents |
04/02/2003 | EP1296716A2 New formulation |
04/02/2003 | EP1296687A2 Treatment of male sexual dysfunction |
04/02/2003 | EP1296681A2 Use of microsomal triglyceride transfer protein (mtp) inhibitors for reducing the number of postprandial triglyceride-rich lipoprotein particles (pptrl) |
04/02/2003 | EP1296674A2 Use of substituted indole compounds for increasing nitric oxide synthase activity |
04/02/2003 | EP1121108B1 Novel therapeutic use of compounds with beta-3-agonist activity |
04/02/2003 | EP1019887B1 Fluorescent cyanine dyes |
04/02/2003 | EP1000027B1 Thermodynamically stable modification of 1-(4-carbazolyloxy)-3- 2-(2-methoxyphenoxy)ethylamino]-2-propanole, process for its preparation and pharmaceutical compositions containing it |
04/02/2003 | EP0894089B9 Novel heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them |
04/02/2003 | EP0882029B1 Heterocyclic derivatives as antidiabetic and antiobesity agents |
04/02/2003 | EP0587800B1 Immunomodulatory azaspiranes |
04/02/2003 | CN1407053A Blue light emitting compound and electroluminescert device with it as color display substance |
04/02/2003 | CN1406937A 1-[1-(hetero) aryl-1-perhydroxyalkylmethyl]-piperazine compound, preparation thereof and pharmaceutics containing it |
04/02/2003 | CN1104435C Process for the preparation of N-[(l-nButyl-4-piperidyl) methyl-3, 4-dihydro-2h-[1,3] oxazino [3,2-2] indole-10-carboxamide and salts and intermediates in the process |
04/01/2003 | US6541669 Multibinding amine compounds which are beta 2 adrenergic receptor agonists useful in treatment and prevention of respiratory diseases such as asthma, bronchitis |
04/01/2003 | US6541644 Adsorption by polymer; elution, desorption |
04/01/2003 | US6541643 Process for the preparation of spiro[cis-4-(β-hydroxyethyloxy)cyclohexane-[3h]indol]-2′[1′H]one derivatives |
04/01/2003 | US6541507 Notably 4,6-dimethoxyindole-2-carboxylic acid and derivatives thereof |
04/01/2003 | US6541506 Enediyne carboxylated on one end and having a pyrrole, furan or thiophene ring on the other; may be isolated from annarrhinum bellidofolium |
04/01/2003 | US6541505 Inhibiting the activity of Factor Xa; treating a disease state associated with a physiologically detrimental excess amount of thrombin. |
04/01/2003 | US6541503 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors |
04/01/2003 | US6541477 Inhibitors of p38-a kinase |
04/01/2003 | US6541474 Administering a pharmaceutically effective dose of the heterocycle-containing carboxylic acid derivative or salt to a patient suffering form acute promyelocytic leukemia |
04/01/2003 | US6541473 Resorcinol derivatives |
03/27/2003 | WO2003025017A1 Cytokine receptor |
03/27/2003 | WO2003024933A1 2-phenyl-3-heteroarylpropionic acid derivative or salt thereof and medicine containing the same |
03/27/2003 | WO2003024923A1 Sulfonamide compounds as protease inhibitors |
03/27/2003 | WO2003024899A2 CYCLIC HYDROXAMIC ACIDS AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-α CONVERTING ENZYME (TACE) |
03/27/2003 | WO2003024448A2 Inhibitors of histone deacetylase |
03/27/2003 | WO2002094263A3 Caspase inhibitors and uses thereof |
03/27/2003 | WO2002060859A3 Cyclic derivatives as modulators of chemokine receptor activity |
03/27/2003 | WO2002014261A3 4-substituted d-glutamic acid derivatives for use as antibiotic |
03/27/2003 | WO2001092218A3 Polyamine analogues as therapeutic and diagnostic agents |
03/27/2003 | US20030060635 Methods of using bis-indolylquinones |
03/27/2003 | US20030060498 5-arylsulfonyl indoles useful for treating disease |
03/27/2003 | US20030060497 Use of indole Mannich bases in the production of medicaments that are used to treat pain |
03/27/2003 | US20030060465 Such as 1-(p-chlorobenzoyl)-5-methoxy-2-methylindole-3-acetic acid morpholinocarbonyloxyethyl ester; for reducing gastrointestinal side effects |
03/27/2003 | US20030060461 Cyclic diamine compound with condensed-ring groups |
03/27/2003 | US20030060459 Diamines as modulators of chemokine receptor activity |
03/27/2003 | CA2465978A1 Inhibitors of histone deacetylase |
03/27/2003 | CA2460151A1 Cytokine receptor |
03/27/2003 | CA2460149A1 2-phenyl-3-heteroarylpropionic acid derivative or salt thereof and medicine containing the same |
03/26/2003 | EP1296142A2 Calcium receptor active molecules |
03/26/2003 | EP1295867A1 Biphenyl compound |
03/26/2003 | EP1294823A1 Double-spiro organic compounds and electroluminescent devices |
03/26/2003 | EP1294718A2 6,5-fused bicyclic heterocycles |
03/26/2003 | EP1294713A2 Compounds possessing antibacterial, antifungal or antitumor activity |
03/26/2003 | EP1294695A2 Substituted diamide derivatives useful as motilin antagonists |
03/26/2003 | EP1294691A1 Serine protease inhibitors |
03/26/2003 | EP1294689A1 Novel $g(b crystalline form of perindopril tert-butylamine salt, preparation method, and pharmaceutical compositions containing same |
03/26/2003 | EP1294688A2 Indolinone derivatives as protein kinase/phosphatase inhibitors |
03/26/2003 | EP1294687A2 1,2,4-trisubstituted benzenes as inhibitors of 15-lipoxygenase |
03/26/2003 | EP1294686A2 Indole derivatives and their use as 15-lipoxygenase inhibitors |
03/26/2003 | EP1294366A1 Pharmaceutical compounds for treating copd |
03/26/2003 | EP1294364A1 Stable gabapentin having ph within a controlled range |
03/26/2003 | EP1159269B1 Anti-imflammatory indole derivatives |
03/26/2003 | EP0885186B1 Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them |
03/26/2003 | EP0763026B1 Gastrin and cck antagonists |
03/26/2003 | CN1406223A Protease inhibitor and their pharmaceutical uses |
03/26/2003 | CN1103756C Estrogenic agents |
03/25/2003 | WO2003000254A1 Fused cyclic compounds and medicinal use thereof |
03/25/2003 | US6538038 A method of treating a warm-blooded animal having a vascular proliferative disorder, comprising administering, to the animal, an amount of a prodrug of a tubulin binding agent, other than combretastatin A4 disodium phosphate to achieve |
03/25/2003 | US6538003 Pyridopyranoazepine derivatives, their preparation and their therapeutic application |
03/25/2003 | US6537330 Colorants |
03/25/2003 | CA2423800A1 Fused cyclic compounds and medicinal use thereof |
03/21/2003 | WO2002022555A1 Substituted biphenyl derivatives, method for preparing same and pharmaceutical compositions containing same |
03/20/2003 | WO2003022816A1 Process for the preparation of base-free carbazolide anions |
03/20/2003 | WO2003022815A1 3-(4,5,6,7-tetrahydroindol-2-ylmethylidiene)-2-indolinone derivatives as kinase inhibitors |
03/20/2003 | WO2003022814A1 Indole derivatives |
03/20/2003 | WO2003022813A1 Indole derivatives, process for producing the same and drugs containing the same as the active ingredient |
03/20/2003 | WO2003022810A1 3-amino carbonyl-substituted benzoylcyclohexanediones that can be used as herbicides |
03/20/2003 | WO2003022806A2 Cbi analogues of cc-1065 and the duocarmycins |
03/20/2003 | WO2003022280A2 3-glyoxlylamideindoles for treating cancer |
03/20/2003 | WO2003022277A1 Arylsulfonamide derivatives for use as ccr3 antagonists in the treatment of inflammatory and immunological disorders |
03/20/2003 | WO2003022272A1 Appetite-stimulating agents and remedies for anorexia |
03/20/2003 | WO2003004466A3 Dye-sulfenates for dual phototherapy |
03/20/2003 | WO2002100845A8 Hv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis |
03/20/2003 | WO2002067865A3 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof |
03/20/2003 | US20030055109 Stability |
03/20/2003 | US20030055093 For therapy of cardiovascular diseases, stable or unstable angina pectoris, coronary heart disease, stable or unstable angina pectoris, coronary heart disease, Prinzmetal angina, acute coronary syndrome, heart failure, myocardial infarction |
03/20/2003 | US20030055086 Amino acid derivatives and use thereof as nep, ace and ece inhibitors |
03/20/2003 | US20030055077 Method and compositions for the treatment of allergic conditions using pgd2 receptor antagonists |
03/20/2003 | US20030055076 Novel compounds, their preparation and use |
03/20/2003 | US20030055037 Benzimidazole and indole derivatives as CRF receptor modulators |
03/20/2003 | CA2460347A1 3-glyoxlylamideindoles for treating cancer |
03/20/2003 | CA2459879A1 3-(4,5,6,7-tetrahydroindol-2-ylmethylidiene)-2-indolinone derivatives as kinase inhibitors |
03/20/2003 | CA2459515A1 Indole derivatives |
03/20/2003 | CA2459308A1 Cbi analogues of cc-1065 and the duocarmycins |
03/19/2003 | EP1293506A1 New 1-(1-(Hetero)aryl-1-perhydroxyalkylmethyl)-Piperazine derivatives, process for their preparation and pharmaceutical compositions containing the same |
03/19/2003 | EP1292574A1 3-azabicyclo[3.1.0]hexane derivatives having opioid receptor affinity |
03/19/2003 | EP1292564A2 Aminoalcohol derivatives |
03/19/2003 | EP1037637B1 Use of 5ht1a receptor antagonists for preventing and/or treating temporal lobe epilepsy |
03/19/2003 | EP1012131B1 Enantioselective reduction of ketones with a silane agent/metal compound/chiral ligand system |
03/19/2003 | CN1404479A Novel 1,3-dihydro-2H-indol-2-one derivatives their preparing method and the pharmceutical composition containing the same |
03/19/2003 | CN1404477A 哌嗪和哌啶衍生物 Piperazine and piperidine derivatives |
03/19/2003 | CN1403455A Synthesis of 2-oxazolidone derivate by one still process |
03/18/2003 | US6534660 CC-1065 analog synthesis |
03/18/2003 | US6534651 Substituted isoindolinone derivatives |
03/18/2003 | US6534650 Benzisoxazole and 4-amidino-3-hydroxyphenyl chemical intermediates |
03/18/2003 | US6534627 Synthesis and use of amino acid fluorides as peptide coupling reagents |