Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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08/07/2002 | EP0829473B1 Processes for preparing cyclic compounds |
08/07/2002 | CN1362960A Method for preparing substituted [1,4] diazepino (6,7,1-hi) indol-4-ones |
08/07/2002 | CN1362947A N-cyanomethylamides as protease inhibitors |
08/07/2002 | CN1362640A Silver-halides photo-sensitive emulsion layer with reinforced photographic photosensibility |
08/07/2002 | CN1362397A Dialkoyl-halogen phenyl substituted keto-enol |
08/07/2002 | CN1088709C Amine compound and its acid addition salt |
08/07/2002 | CN1088702C Disubstituted bicyclic heterocycles, their production and use as medicaments |
08/07/2002 | CN1088585C Compound active at novel site on receptor-operated calcium channels use full for treatment of neurological disorders and diseases |
08/06/2002 | US6429317 Indane derivatives for antipsychotic compositions |
08/06/2002 | US6429221 Inhibitors of tumor necrosis factor; used to treat cachexia, endotoxic shock, and retrovirus replication |
08/06/2002 | US6429212 Aminopeptidase n inhibitor used to treat cancer, tumors, and retinopathy; few side effects; angiogenesis inhibitor |
08/06/2002 | US6429207 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases |
08/06/2002 | CA2231812C Cyclic nitrones and pharmaceutical compositions containing them |
08/06/2002 | CA1341380C Process for the preparation of n-alkylated amino acids and their esters, use in the synthesis of carboxyalkyl dipeptides |
08/01/2002 | WO2002059165A2 Polymerization of olefinic compounds |
08/01/2002 | WO2002059124A2 Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists |
08/01/2002 | WO2002059122A1 ANTI-CANCER 2,3-DIHYDRO-1H-PYRROLO[3,2-f]QUINOLINE COMPLEXES OF COBALT AND CHROMIUM |
08/01/2002 | WO2002059117A1 Piperazine- and piperidine-derivatives as melanocortin receptor agonists |
08/01/2002 | WO2002059108A1 Melanocortin receptor agonists |
08/01/2002 | WO2002059107A1 Substituted piperidines/piperazines as melanocortin receptor agonists |
08/01/2002 | WO2002059095A1 Melanocortin receptor agonists |
08/01/2002 | WO2002059092A1 Process for the preparation of (3-cyano-1h-indol-7-yl)(4-(4-fluorophenethyl)piperazin-1-yl)-methanone and salts thereof |
08/01/2002 | WO2002059089A2 Process for the preparation of heterocyclic indene analogs |
08/01/2002 | WO2002059088A1 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands |
08/01/2002 | WO2002059082A2 Aryl and aminoaryl substituted serotonin receptor agonist and antagonist ligands |
08/01/2002 | WO2002059080A2 Trisubstituted carbocyclic cyclophilin binding compounds and their use |
08/01/2002 | WO2002058690A2 Methods for the treatment of diseases using malonyl-coa decarbox ylase inhibitors |
08/01/2002 | WO2002058679A2 Antiangiogenic compounds and an assay for inhibitors of cell invasion |
08/01/2002 | WO2002032285A3 Hydrophilic light absorbing compositions for determination of physiological function in critically ill patients |
08/01/2002 | WO2001078697A3 Method and compositions for the treatment of allergic conditions using pgd2 receptor antagonists |
08/01/2002 | WO2001078654A3 Halogentated 2-amino-3, 4 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
08/01/2002 | US20020103383 Selective 5-HT6 receptor ligands |
08/01/2002 | US20020103382 Serotonin (5-HT) subtype 6 receptor (5-HT6); 3-(2-aminoethyl)indole derivatives; drug screening |
08/01/2002 | US20020103248 Indole derivatives which are agonists of the progesterone receptor and useful for treatment of carcinoma and adenocarcinomas of uterine leiomyomata, endometriosis or polycystic ovary syndorme in a mammal |
08/01/2002 | US20020103247 Indole and dihydroindole derivatives |
08/01/2002 | US20020103234 Heterocycl-containing carboxylic acid derivative and drug containing the same |
08/01/2002 | US20020103217 Triphenylpropanamide compounds; useful in treating inflammations but which do not demonstrate side effects associated with other anti-inflammatory treatments such as glucocorticoids |
08/01/2002 | US20020103197 For use in protecting human and animal hair and skin against damaging action of UV radiation |
08/01/2002 | US20020103192 Perfluoroalkylketones, ketooxazoles, ketoamides, ketoesters, and diketones, and their dihydroxy derivatives, such as 7-((1,1'-biphenyl)-3-yloxy)-1-(1,3-oxazol-2-yl)-1-heptanone |
08/01/2002 | US20020103188 Peroxisome Proliferator-Activated Receptors (PPAR); diabetes and obesity; 3-(4-(2-(10,1-Dihydro-dibenzo(b,f)azepin-5-yl)ethoxy)-pheny)-2-ethoxy -propionic acid, for example |
08/01/2002 | US20020103164 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
08/01/2002 | US20020102608 Library of indolinone compounds for use in the treatment of cancer |
08/01/2002 | CA2435829A1 Trisubstituted carbocyclic cyclophilin binding compounds and their use |
08/01/2002 | CA2435653A1 Anti-cancer 2,3-dihydro-1h-pyrrolo[3,2-f]quinoline complexes of cobalt and chromium |
08/01/2002 | CA2435633A1 Antiangiogenic compounds and an assay for inhibitors of cell invasion |
08/01/2002 | CA2435566A1 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands |
08/01/2002 | CA2433025A1 Substituted piperidines/piperazines as melanocortin receptor agonists |
08/01/2002 | CA2432988A1 Melanocortin receptor agonists |
08/01/2002 | CA2432985A1 Piperazine- and piperidine-derivatives as melanocortin receptor agonists |
08/01/2002 | CA2432122A1 Aryl and aminoaryl substituted serotonin receptor agonist and antagonist ligands |
08/01/2002 | CA2431996A1 Melanocortin receptor agonists |
07/31/2002 | EP1227095A2 A process for the purification of (S)-4-((3-(dimethylamino)ethyl)-1H-indol-5yl)-methyl)-2-oxazolidinone |
07/31/2002 | EP1226138A1 Fab i inhibitors |
07/31/2002 | EP1226121A1 Method of inhibiting neurotrophin-receptor binding |
07/31/2002 | EP1226120A2 Benz[f]indoles for use in the treatment of 5ht receptor related disorders |
07/31/2002 | EP1226116A1 Processes for the preparation of sumatriptan and related compounds |
07/31/2002 | EP1225955A1 Aryl olefinic azacyclic, and aryl acetylenic azacyclic compounds, pharmaceutical compositions containing them and their use as inhibitors of nicotinic cholinergic receptors |
07/31/2002 | EP1225895A1 Fab i inhibitors |
07/31/2002 | EP1225894A1 Fab i inhibitors |
07/31/2002 | EP1225886A2 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits |
07/31/2002 | EP1225882A1 Selective cox-2 inhibitory novel esters from indolealkanols and novel amides from indolealkylamines |
07/31/2002 | EP0764152B1 Substituted indolylmethylene-oxindole analogues as tyrosine kinase inhibitors |
07/31/2002 | EP0719267B1 Second messenger cell signaling inhibitors |
07/31/2002 | CN1361768A Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases |
07/31/2002 | CN1361716A Preparation and use of ionic liquids in microwave-assisted chemical transformation |
07/31/2002 | CN1361100A New heterocyclic derivative and its medical use |
07/30/2002 | US6426349 Substituted condensation products of N-benzyl-3-indenylacetamides with heterocyclic aldehydes for neoplasia |
07/30/2002 | US6426344 Aryl and heteroaryl substituted indolealkanoic acids |
07/30/2002 | CA2344707C N-substituted cycloalkyl and polycycloalkyl alpha-substituted trp-phe- and phenethylamine derivatives |
07/30/2002 | CA2093353C Hydrolytically and oxidatively stable polyimides |
07/30/2002 | CA2078039C Process for the production of lactams |
07/25/2002 | WO2002057231A2 Benz(g) indoles and their use as spla2 inhibitors |
07/25/2002 | WO2002057216A1 Terphenyl compounds bearing substituted amino groups |
07/25/2002 | WO2002038545A3 Crystalline ethanolate solvate form of zafirlukast, process for manufacture and pharmaceutical compositions thereof |
07/25/2002 | WO2002032901A3 Bridged piperazine derivatives |
07/25/2002 | WO2002030867A3 Drugs for diabetes |
07/25/2002 | WO2001070222A3 Compounds with 5-ht1a activity useful for treating disorders of the outer retina |
07/25/2002 | WO2001040188A9 Curcumin analogues for treating cancer |
07/25/2002 | US20020099224 Hydrolysis of [R (R*, R*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid esters with calcium hydroxide |
07/25/2002 | US20020099223 Cyclocarbonylating acetic acid (or benzoic acid)-1-(1-benzenesulfonyl-1H-indol-2-yl)-allyl ester to obtain 9-benzenesulfonyl-9H-carbazol-4-yl ester; saponifying |
07/25/2002 | US20020099208 Heterocyclic substituted 2-methyl-benzimidazole antiviral agents |
07/25/2002 | US20020099096 Useful for oral testosterone replacement therapy, male contraception, maintaining sexual desire in women, treating prostate cancer and imaging prostate cancer |
07/25/2002 | US20020099084 Pharmaceutically active compounds and methods of use |
07/25/2002 | US20020099080 Indole derivatives useful A.O. for the treatment of osteoporosis |
07/25/2002 | US20020099071 Protein tyrosine kinase and protein serin/threonine kinase inhibitory activity; anticancer agents; treating chemotherapy induced alopecia |
07/25/2002 | US20020099054 2-phenyl benzimidazole derivatives as MCP-1 antagonists |
07/25/2002 | DE10130830A1 Indol-Derivate Indole derivatives |
07/25/2002 | DE10102944A1 Production of 3-cyano-1H-indol-7-yl)-(4-(4-fluorophenethyl)piperazin-1-yl)-methanone useful as a selective 5-HT2A antagonist comprises use of an indolecarboxylic acid ester as the starting material |
07/25/2002 | CA2431506A1 Benz(g) indoles and their use as spla2 inhibitors |
07/24/2002 | EP1225169A1 Radiation-activated cytotoxin therapy |
07/24/2002 | EP1224170A1 6-position substituted indoline, production and use thereof as a medicament |
07/24/2002 | EP1224169A2 Production of 5-substituted indolinones and use thereof as medicaments |
07/24/2002 | EP1224168A1 Antifungal enediynes |
07/24/2002 | EP1224165A1 Novel compounds |
07/24/2002 | EP1223929A1 Cannabimimetic indole derivatives |
07/24/2002 | EP0885230B1 Camptothecin derivatives and the use thereof as antitumor agents |
07/24/2002 | EP0859759B1 Sulphonic acids and their use as u/v absorbers |
07/24/2002 | CN1360580A Substd. benzoyl ketones, methods for producing them and their use as herbicides |
07/24/2002 | CN1360576A Process for preparation of spiro [(4-cyclohexanone)-[3H] indol]-2'[iH]-one derivs. |
07/24/2002 | CN1360575A Process for preparation of spiro-[cis-4-(beta-hydroxyethyloxy) cyclohexane-(3H) indol]-2'[1'H]-one derivs. |