Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
12/2002
12/11/2002EP1263716A2 Amino acid derivatives as hiv aspartyl protease inhibitors
12/11/2002EP1263504A2 Compounds with 5-ht1a activity useful for treating disorders of the outer retina
12/11/2002EP1263434A1 Compounds with 5-ht 2 and 5-ht 1a agonist activity for treating glaucoma
12/11/2002EP1263414A1 Pharmaceutical compositions of glycogen phosphorylase inhibitors
12/11/2002EP1100805B1 Medicine nitrate salts
12/11/2002EP1061956B1 Manganese chelates with high relaxivity in serum
12/11/2002EP1058678B1 Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes
12/11/2002EP0966436B1 Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases
12/11/2002EP0805796B1 Cell adhesion inhibitors
12/11/2002EP0752813B1 Inhibitors of metazoan parasite proteases
12/11/2002EP0628030B1 2,3,4,5-TETRAHYDRO-1H --3-BENZAZEPINES HAVING ANTI-PSYCHOTIC ACTIVITY, AND SYNTHESIS OF $g(a)-SUBSTITUTED-ARYLACETAMIDES
12/11/2002CN1384821A Method for improving solubility of tricyclic amino alcohol derivatives
12/11/2002CN1384756A Pharmaceutical formulations and use thereof in prevention of stroke, diabetes and/or congestive heart failure
12/11/2002CN1384741A Selective COX-2 inhibitory novel esters from indolealkanols and novel amides from indolealkylamines
12/11/2002CN1095835C Tricyclo-substituted isohydroxyloxime acid derivative
12/10/2002US6492562 Invention also relates to novel intermediates and the resulting modified polyketides and antibiotics.
12/10/2002US6492555 Reaction of a carbamate with either a (s)-secondary alcohol or (s)-epoxide or (s)-ester; bactericides
12/10/2002US6492428 Macrophage migration inhibitory factor (mif); substituted iminoquinone or orthoquinone ring systems
12/10/2002US6492422 Tricyclic sulfonamides and their derivatives as inhibitors of matrix metalloproteinases
12/10/2002US6492412 Prevention of loss and restoration of bone mass by certain prostaglandin agonists
12/10/2002US6492394 Procollagen c-proteinase inhibitors; treating fibrotic diseases
12/10/2002US6492362 Compounds and compositions as cathepsin S inhibitors
12/10/2002US6492351 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
12/10/2002CA2057604C Process for producing an aryl-imido-peralkanoic acid
12/09/2002WO2002004403A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments
12/09/2002CA2412116A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments
12/05/2002WO2002096902A1 Carbazole derivatives and their use for the preparation of pharmaceutical compositions for the treatment of npy related diseases
12/05/2002WO2002096873A1 Isoindole and isoquinoline derivatives as inhibitors of factor xa
12/05/2002WO2002096867A2 Inhibitors of protein kinase for the treatment of disease
12/05/2002WO2002096864A1 Carboxamide-substituted phenylurea derivatives and method for production thereof as medicaments
12/05/2002WO2002096858A1 Cinnamide derivatives as kcnq potassium channel modulators
12/05/2002WO2002096424A1 Hetereocyclic beta-aminoacids and their use as anti-epileptogenic agents
12/05/2002WO2002078693A3 N-(2-arylethyl)benzylamines as antagonists of the 5-ht6 receptor
12/05/2002US20020183526 Catalytically reducing a nitrocarbazole, in presence of an iron compound
12/05/2002US20020183513 Tricyclic alkylhydroxamate derivatives
12/05/2002US20020183397 Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
12/05/2002US20020183377 Use of melatonin for treating androgenetic and diffuse alopecia
12/05/2002US20020183370 3-(cycloalkanoheteroarylidenyl)-2-indolinone protein tyrosine kinase inhibitors
12/05/2002US20020183369 For therapy of diabetes, insulin resistance, diabetic neuropathy, diabetic nephropathy, diabetic retinopathy, cataracts, hyperglycemia, hypercholesterolemia, hypertension, hyperinsulinemia, hyperlipidemia, atherosclerosis
12/05/2002US20020183364 Methods of modulating protein tyrosine kinase function with substituted indolinone compounds
12/05/2002US20020183349 For therapy and prophylaxis of disorders of the central nervous system; damage to the central nervous system; cardiovascular disorders; gastrointestinal disorders; diabetes, sleep apnea
12/05/2002US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm
12/05/2002US20020183321 Carbocyclic and heterocyclic substituted semicarbazones and thiosemicarbazones and the use thereof
12/05/2002DE10125567A1 New N-aroyl-N'-(carbamoyl-phenyl)-urea derivatives, are glycogen phosphorylase a inhibiting hypoglycemic agents, especially useful for treating type II diabetes
12/05/2002CA2448894A1 Cinnamide derivatives as kcnq potassium channel modulators
12/05/2002CA2448160A1 Heterocyclic beta-amino acids and their use as anti-epileptogenic agents
12/05/2002CA2448023A1 Carboxamide-substituted phenylurea derivatives and method for production thereof as medicaments
12/05/2002CA2447234A1 Carbazole derivatives and their use for the preparation of pharmaceutical compositions for the treatment of npy related diseases
12/04/2002EP1262536A2 Fluorescent group-containing carbodiimide compound and process for producing the compound
12/04/2002EP1262475A1 Indole derivatives, process for preparation of the same and use thereof
12/04/2002EP1261630A2 Bacterial genes and proteins that are essential for cell viability and their uses
12/04/2002EP1261601A1 Substituted indoles for modulating nfkb activity
12/04/2002EP1261586A2 Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase iv, processes for their preparation, and their use
12/04/2002EP1261585A1 Substituted indole mannich bases
12/04/2002EP1261583A1 INHIBITORS OF THE ICE/Ced-3 FAMILY OF CYSTEINE PROTEASES
12/04/2002EP1261579A1 Dehydroamino acids
12/04/2002EP1261362A2 Novel amino acid and peptide inhibitors of staphylococcus virulence
12/04/2002EP1001930B1 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
12/03/2002US6489489 Organic electroluminescent device
12/03/2002US6489488 Serotonin (5-ht) subtype 6 receptor (5-ht6); 3-(2-aminoethyl)indole derivatives; drug screening
12/03/2002US6489480 Coordination polymerization catalyst for alpha-olefins
12/03/2002US6489475 Method of producing heterocyclic derivatives
12/03/2002US6489353 Antiinflammatory agents; autoimmune diseases; central nervous system disorders
12/03/2002US6489352 Antiepileptic agents; nervous system disorders
12/03/2002US6489337 Treatment of alzheimer's disease, epilepsy, eating disorders, learning and memory disorders, migraine, sleep/wake disorders, allergic rhinitis, schizophrenia, mild cognitive impairment, and asthma
12/03/2002US6489046 Containing such as 8,15-diphenyl or a 8,15-bis(biphenyl)-benzo(a)pentacene; emits high purity reddish light; efficient, long life; planar light emitting member for televisions; back light for displays
11/2002
11/30/2002CA2386755A1 Fluorescent group-containing carbodiimide compound and process for producing the compound
11/28/2002WO2002094809A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives
11/28/2002WO2002094799A2 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
11/28/2002WO2002094770A2 Aminoalcohol derivatives
11/28/2002WO2002094263A2 Caspase inhibitors and uses thereof
11/28/2002WO2002094262A1 Heteroaryloxy 3-substituted propanamines s serotonin and norepinephrine reuptake inhibitors
11/28/2002WO2002094220A1 Liquid pharmaceutical composition
11/28/2002WO2002048106A3 Isoindolin-1-one glucokinase activators
11/28/2002US20020177720 Adsorption by polymer; elution, desorption
11/28/2002US20020177594 Inhibitors of histone deacetylase
11/28/2002CA2448080A1 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
11/28/2002CA2448076A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives
11/28/2002CA2445010A1 Heteroaryloxy 3-substituted propanamines s serotonin and norepinephrine reuptake inhibitors
11/27/2002EP1260511A1 Process for the preparation of 5-chloro-1-(4-fluorophenyl)-3-(1,2,3,6-tetrahydropyridin-4-yl)indole and method of manufacturing sertindole
11/27/2002EP1259505A2 Novel 1,3-dihydro-2h-indol-2-one, preparation method and pharmaceutical compositions containing same
11/27/2002EP1259492A1 Substituted piperazine derivatives as mtp inhibitors
11/27/2002EP1259488A1 Ortho-sulfonamido aryl hydroxamic acids, process for their preparation and their use as matrix metalloproteinase inhibitors
11/27/2002EP1259236A1 Tyrosine kinase inhibitors
11/27/2002EP1259231A2 Naphthoquinone derivatives as cd45 inhibitors
11/27/2002EP1019319B1 Synthesis method for solution with high grade chloramine
11/27/2002EP1001934B1 Indole compounds as cox-2 inhibitors
11/27/2002EP0971890B1 Substituted analogs of indole-3-carbinol and of diindolymethane as antiestrogens
11/27/2002EP0825982B1 Alkyl dihalogenated phenyl-substituted ketoenols useful as pesticides and herbicides
11/27/2002EP0585267B1 Herpesvirus particle preparation and vaccine
11/27/2002CN1382124A Bicycle androgen and progesterone receptor modulator compounds and methods
11/27/2002CN1382123A Process for preparation of indole derivatives or salts thereof
11/27/2002CN1381446A Process for preparing pineal hormone
11/27/2002CN1094927C Process for preparing 2-azadihydroxybicyclo [2,2,1] heptane compounds and L-tartaric acid salt of the compound
11/26/2002US6486343 Substituted phenyl keto enols as pesticides and herbicides
11/26/2002US6486342 Substituted chiral allosteric hemoglobin modifiers
11/26/2002US6486326 iso-CBI and iso-CI analogs of CC-1065 duocarmycins
11/26/2002US6486192 Indole compounds useful for treating bacterial infections
11/26/2002US6486185 3-heteroarylidene-2-indolinone protein kinase inhibitors
11/26/2002US6486178 Indane derivatives