Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
01/2003
01/15/2003CN1391473A VLA-4 inhibitor compounds
01/15/2003CN1391469A Npyy5拮抗剂 Npyy5 antagonist
01/15/2003CN1390834A Indenoindolone compounds, their preparation and medicinal compositions containing them
01/15/2003CN1098838C Substituted N-(indole-2-carbonyl)-beta-alanimamides and derivatives as antidiabetic agents
01/14/2003US6506876 LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use
01/14/2003US6506787 Aids therapy
01/14/2003US6506786 HIV protease inhibitors based on amino acid derivatives
01/14/2003US6506785 Establishing the status of the mammal as presently or prospectively being in early stages of degeneration of articular cartilage or subchondral bone in one or more joinsts, administering a xanthine chondroprotective compound
01/14/2003US6506763 3-(substituted)-2-indolinones compounds and use thereof as inhibitors of protein kinase activity
01/14/2003US6506758 Indole derivatives useful A.O. for the treatment of osteoporosis
01/09/2003WO2003003482A1 Organic light emitting diode devices using thermostable hole-injection and hole-transport compounds
01/09/2003WO2003002545A1 Peptoid compounds
01/09/2003WO2003002533A1 Triamide-substituted indoles, benzofuranes and benzothiophenes as inhibitors of microsomal triglyceride transfer protein (mtp) and/or apolipoprotein b (apo b) secretion
01/09/2003WO2003002532A1 Cyclic diamine compounds having fused-ring groups
01/09/2003WO2003002519A1 Phenol derivatives and their use in medicaments
01/09/2003WO2003002491A2 ENANTIOSELECTIVE TRANSFORMATION OF α, β-UNSATURATED ALDEHYDES USING CHIRAL ORGANIC CATALYSTS
01/09/2003WO2003002255A1 Hydroxylation of beta-dicarbonyls with zirconium catalysts
01/09/2003WO2002057231A3 Benz(g) indoles and their use as spla2 inhibitors
01/09/2003US20030009055 Process for the preparation of 1-aminomethyl-1- cyclohexaneacetic acid
01/09/2003US20030009036 To produce polymers; cancer therapy
01/09/2003US20030009033 Substituted condensation products of N-benzyl-3-indenylacent amides with heterocyclic aldehydes for neoplasia
01/09/2003US20030008915 Acylated 6,7,8,9-tetrahydro-5H-benzocycloheptenyl amines and their use as pharmaceutical agents
01/09/2003US20030008913 For controlling harmful insects, acarids and nematodes
01/09/2003US20030008911 Treating or preventing the early stages of degeneration of articular cartilage or subchondral bone in mammals using carprofen and derivatives
01/09/2003US20030008909 For therapy of uterine myometrial fibroids, endometriosis, benign prostatic hypertrophy; carcinomas and adenocarcinomas of endometrium, ovary, breast, colon, prostate, pituitary, meningioma and other hormone-dependent tumors
01/09/2003US20030008900 Compounds and compositions for delivering active agents
01/09/2003US20030008898 Indole derivatives and their use for the treatment of malignant and other diseases based on pathological proliferation
01/09/2003US20030008895 Prostaglandin agonists
01/09/2003US20030008884 Fungicidal phenyl (thio) urea and phenyl (thio) carbamate derivatives
01/09/2003US20030008360 Microorganisms for use in the generation of preferential cyclopentene
01/09/2003US20030008234 Optical data carrier comprising a cyanine dye as light-absorbent compound in the information layer
01/09/2003US20030005525 Composition for dyeing keratin fibers with a cationic direct dye and a thickening polymer
01/08/2003EP1273343A1 Method of separating imide compound
01/08/2003EP1273330A1 Sublimation purifying method and apparatus
01/08/2003EP1272900A2 High speed photothermographic materials containing tellurium compounds and methods of using same
01/08/2003EP1272468A1 Indolin-2-one derivatives, preparation and their use as ocytocin receptor ligands
01/08/2003EP1272467A1 Cathepsin cysteine protease inhibitors
01/08/2003EP1272456A1 Hydrazide and alkoxyamide angiogenesis inhibitors
01/08/2003EP1124819B1 Method of lithiating five-membered heterocycles
01/08/2003EP0863878B1 Cyclic nitrones and pharmaceutical compositions containing them
01/08/2003CN1390214A New phenylpiperazines
01/08/2003CN1390213A Aryloxy propanolamines for improving livestock production
01/07/2003US6504036 2- and 2.5-substituted phenylketoenols
01/07/2003US6503998 Nonlinear Optical (nlo) materials, sulfon-diol-ether derivatives
01/07/2003US6503949 Glucagon antagonists/inverse agonists
01/07/2003US6503939 Combination regimens using 3,3-substituted indoline derivatives
01/07/2003US6503938 Treatment of estrogen related disease or tumor, including prostatic hyperplasia, breast cancer, endometrial carcinoma, anovulatory infertility, melanoma or osteoporosis
01/07/2003US6503907 Indole and dihydroindole derivatives
01/07/2003US6503900 [1,4]diazepino [6,7,1-jk ]carbazoles and derivatives
01/07/2003CA2143208C Sulfonamide inhibitors of hiv-aspartyl protease
01/03/2003WO2003000688A1 Azaindoles
01/03/2003WO2003000684A1 Substituted naphthyl indole derivatives as inhibitors of plasminogen activator inhibitor type-1 (pai-1)
01/03/2003WO2003000680A1 Diamine derivatives
01/03/2003WO2003000657A1 Diamine derivatives
01/03/2003WO2003000649A1 6-(aryl-amido or aryl-amidomethyl)-naphthalen-2-yloxy-acidic derivatives as inhibitors of plasminogen activator inhibitor type-1 (pai-1)
01/03/2003WO2003000289A1 Composition comprising a pde-4 inhibitor and h1-receptor antagonist and the use thereof for the manufacture of a medicament for the treatment of respiratory diseases
01/03/2003WO2003000253A1 Substituted indole acid derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1)
01/03/2003WO2003000252A1 5-halo-tryptamine derivatives used as ligands of the 5-ht6 and/or 5-ht7 serotonin receptors
01/03/2003WO2003000251A1 Novel idolinones and uses thereof
01/03/2003WO2003000247A1 Carbamates of 2-heterocyclic-1,2-ethanediols
01/03/2003WO2003000181A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003WO2002008187A9 Novel peptides as ns3-serine protease inhibitors of hepatitis c virus
01/03/2003WO2002001653A3 Organic light emitting diode devices using aromatic amine compounds with high and tunable glass transition temperatures
01/03/2003CA2450758A1 Composition comprising a pde-4 inhibitor and h1-receptor antagonist and the use thereof for the manufacture of a medicament for the treatment of respiratory diseases
01/03/2003CA2450475A1 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003CA2450174A1 6-(aryl-amido or aryl-amidomethyl)-naphthalen-2-yloxy-acidic derivatives as inhibitors of plasminogen activator inhibitor type-1 (pai-1)
01/02/2003WO2002002529A1 Bicyclic lactams and sulfonamides with 5-ht1a-affinity and use thereof for preventing and treating cerebral ischaemia
01/02/2003US20030004351 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
01/02/2003US20030004181 Disubstituted bicyclic heterocycles, the preparation thereof, and their use as pharmaceutical compositions
01/02/2003US20030004162 Antidiabetic agents; dietetics
01/02/2003US20030004156 Anticholesterol agents; cardiovascular disorders; antidiabetic agents; antiproliferative agents
01/02/2003US20030004151 Cyclic derivatives as modulators of chemokine receptor activity
01/02/2003US20030004149 Antiangiogenic compounds and an assay for inhibitors of cell invasion
01/02/2003US20030004138 Hypoglycemic agents; antidiabetic agents; dietetics
01/02/2003US20030003396 Reflection, protective or covering layers which can be written on or read by blue, red or infrared light
01/02/2003EP1270565A1 4-Substituted furan-2-sulfonamide and its use in the preparation of sulfonyl urea derivatives
01/02/2003EP1270562A2 Cyclic alpha-amino-gamma-hydroxy-amides, process for their preparation and pharmaceutical compositions thereof
01/02/2003EP1270557A1 Ethylenediamine derivatives
01/02/2003EP1270554A1 Sulfonyl urea derivatives and their use in the control of interleukin-1 activity
01/02/2003EP1268479A1 Phenyl-substituted indolizine derivatives and their use as histamine h3 ligands
01/02/2003EP1268478A2 Phenyl-substituted imidazopyridines
01/02/2003EP1268441A1 An intermediate and process for its synthesis
01/02/2003EP1268425A2 Carbamate caspase inhibitors and uses thereof
01/02/2003EP1268424A1 Method for synthesis of perindopril and its pharmaceutically acceptable salts
01/02/2003EP1268423A1 Indole derivatives as mcp-1 receptor antagonists
01/02/2003EP1268422A1 Indoles for treating diseases that can be treated using thyroid hormones
01/02/2003EP1268421A2 Phenyl-substituted indoles as histamine h3-receptor antagonists
01/02/2003EP1268404A1 Malonamic acids and derivatives thereof as thyroid receptor ligands
01/02/2003EP1268398A2 Novel method for synthesis of n- (s)-1-carboxybutyl]-(s)-alanine esters and use in synthesis of perindopril
01/02/2003EP1268051A2 Dosing form for reagents, use of said dosing form in organic chemical synthesis and production of said dosing form
01/02/2003EP1267878A2 Compounds with 5-ht activity useful for controlling visual field loss
01/02/2003EP1109785B1 Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
01/02/2003EP1083897A4 Hiv integrase inhibitors
01/02/2003EP1053246B1 Beta-sheet mimetics and methods relating to the use thereof
01/02/2003EP0891341B1 1,3,4-oxadiazine derivatives and their use as pesticides
01/02/2003CA2414726A1 Bicyclic lactams and sulfonamides with 5-ht1a-affinity and use thereof for preventing and treating cerebral ischaemia
12/2002
12/31/2002US6500854 Chondrongenesis promotors and indolin-2-one derivatives
12/31/2002US6500853 Enzyme inhibitors such as 4-((1-benzhydryl-5-(((butylamino)-carbonyl)amino)-1h-indol-3-yl)methyl)-3 -methoxybenzoic acid used as antiinflammatory agents for prophylaxis of arthritis, inflammatory bowel disease or asthma
12/31/2002US6500852 Inhibitors of bacterial NAD synthetase
12/31/2002US6500851 Antithrombotic agents